A New Era in Oncology: Tennessee's $20 Million Leap into Radiopharmaceutical Research
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Substrate
Enzyme
Products
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Roquinimex
DB11366
Cytochrome P450 3A4
4-hydroxy-1-methyl-2-oxo-N-phenyl-1,2-dihydroquinoline-3-carboxamide
Details
Roquinimex
DB11366
Cytochrome P450 3A4
4,8-dihydroxy-N,1-dimethyl-2-oxo-N-phenyl-1,2-dihydroquinoline-3-carboxamide
Details
Roquinimex
DB11366
Cytochrome P450 3A4
4,7-dihydroxy-N,1-dimethyl-2-oxo-N-phenyl-1,2-dihydroquinoline-3-carboxamide
Details
Roquinimex
DB11366
Cytochrome P450 3A4
4-hydroxy-N-methyl-2-oxo-N-phenyl-1,2-dihydroquinoline-3-carboxamide
Details
Roquinimex
DB11366
Cytochrome P450 3A4
4-hydroxy-N-(4-hydroxyphenyl)-N,1-dimethyl-2-oxo-1,2-dihydroquinoline-3-carboxamide
Details
Rosiglitazone
DB00412
Cytochrome P450 2C8
/
Cytochrome P450 2C9
N-Desmethylrosiglitazone
Details
Rosiglitazone
DB00412
Cytochrome P450 2C8
/
Cytochrome P450 2C9
ortho-Hydroxyrosiglitazone
Details
Rosiglitazone
DB00412
Not Available
Phenoxyacetic acid derivative of rosiglitazone
Details
Rosiglitazone
DB00412
Cytochrome P450 2C8
/
Cytochrome P450 2C9
para-Hydroxyrosiglitazone
Details
Rosiglitazone
DB00412
Not Available
N-Despyridinyl rosiglitazone
Details
Rosuvastatin
DB01098
Cytochrome P450 2C9
/
Cytochrome P450 2C19
N-Desmethylrosuvastatin
Details
Rosuvastatin
DB01098
Cytochrome P450 2C9
Rosuvastatin 5 S-lactone
Details
Rotigotine
DB05271
Not Available
N-despropyl-rotigotine
Details
Rotigotine
DB05271
Not Available
N-desthienylethyl-rotigotine
Details
Roxadustat
DB04847
Cytochrome P450 2C8
/
UDP-glucuronosyltransferase 1-9
Roxadustat O-glucuronide
Details
Roxadustat
DB04847
Cytochrome P450 2C8
/
UDP-glucuronosyltransferase 1-9
Hydroxy-roxadustat
Details
Roxithromycin
DB00778
Not Available
descladinose roxithromycin
Details
Roxithromycin
DB00778
Not Available
N-mono roxithromycin
Details
Roxithromycin
DB00778
Not Available
N-di-demethyl roxithromycin
Details
RP101075
DBMET03088
Arylamine N-acetyltransferase 2
/
Amine oxidase [flavin-containing] B
CC 112273
/
RP101442
Details
RS-88390 (CVT-2514)
DBMET02242
Not Available
Ranolazine M1
Details
Rucaparib
DB12332
Cytochrome P450 2D6
/
Cytochrome P450 1A2
/
Cytochrome P450 3A4
Rucaparib M309 metabolite
Details
Rucaparib
DB12332
Cytochrome P450 2D6
/
Cytochrome P450 1A2
/
Cytochrome P450 3A4
Rucaparib M337b metabolite
Details
Rucaparib
DB12332
Cytochrome P450 2D6
/
Cytochrome P450 1A2
/
Cytochrome P450 3A4
Rucaparib M323 metabolite
Details
Rucaparib
DB12332
Cytochrome P450 2D6
/
Cytochrome P450 1A2
/
Cytochrome P450 3A4
Rucaparib M324 metabolite
Details
Rucaparib M323 metabolite
DBMET03519
Not Available
Rucaparib M337c metabolite
Details
Rucaparib M323 metabolite
DBMET03519
Not Available
Rucaparib M337a metabolite
Details
Rucaparib M324 metabolite
DBMET03522
UDP-glucuronosyltransferase 1-1
Rucaparib M500 metabolite
Details
Rufinamide
DB06201
Not Available
CGP-47292
Details
Ruxolitinib
DB08877
Cytochrome P450 3A4
/
Cytochrome P450 2C9
Ruxolitinib M16 metabolite
Details
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