| Alteplase | target | Plasminogen | Details |
| Alteplase | target | Fibrinogen alpha chain | Details |
| Sermorelin | target | Growth hormone-releasing hormone receptor | Details |
| Interferon alfa-n1 | enzyme | Cytochrome P450 1A2 | Details |
| Interferon alfa-n1 | target | Interferon alpha/beta receptor 2 | Details |
| Interferon alfa-n1 | target | Interferon alpha/beta receptor 1 | Details |
| Darbepoetin alfa | target | Erythropoietin receptor | Details |
| Urokinase | target | Plasminogen | Details |
| Urokinase | target | Plasminogen activator inhibitor 2 | Details |
| Urokinase | target | Plasminogen activator inhibitor 1 | Details |
| Urokinase | target | Low-density lipoprotein receptor-related protein 2 | Details |
| Urokinase | target | Urokinase plasminogen activator surface receptor | Details |
| Urokinase | target | Nidogen-1 | Details |
| Urokinase | target | Suppressor of tumorigenicity 14 protein | Details |
| Urokinase | target | Plasma serine protease inhibitor | Details |
| Urokinase | enzyme | Macrophage metalloelastase | Details |
| Goserelin | target | Lutropin-choriogonadotropic hormone receptor | Details |
| Goserelin | target | Gonadotropin-releasing hormone receptor | Details |
| Reteplase | target | Plasminogen activator inhibitor 1 | Details |
| Reteplase | target | Fibrinogen alpha chain | Details |
| Reteplase | target | Plasminogen | Details |
| Erythropoietin | target | Erythropoietin receptor | Details |
| Salmon calcitonin | target | Calcitonin receptor | Details |
| Interferon alfa-n3 | enzyme | Cytochrome P450 1A2 | Details |
| Interferon alfa-n3 | target | Interferon alpha/beta receptor 1 | Details |
| Interferon alfa-n3 | target | Interferon alpha/beta receptor 2 | Details |
| Pegfilgrastim | target | Granulocyte colony-stimulating factor receptor | Details |
| Pegfilgrastim | enzyme | Neutrophil elastase | Details |
| Sargramostim | target | Bone marrow proteoglycan | Details |
| Sargramostim | target | Interleukin-3 receptor subunit alpha | Details |