| Tenecteplase | target | Plasminogen | Details |
| Menotropins | target | Follicle-stimulating hormone receptor | Details |
| Menotropins | target | Lutropin-choriogonadotropic hormone receptor | Details |
| Interferon gamma-1b | target | Interferon gamma receptor 1 | Details |
| Interferon gamma-1b | target | Interferon gamma receptor 2 | Details |
| Interferon gamma-1b | enzyme | Cytochrome P450 1A2 | Details |
| Interferon alfa-2a | enzyme | Cytochrome P450 1A2 | Details |
| Interferon alfa-2a | target | Interferon alpha/beta receptor 1 | Details |
| Interferon alfa-2a | target | Interferon alpha/beta receptor 2 | Details |
| Desmopressin | target | Vasopressin V1b receptor | Details |
| Desmopressin | enzyme | Prostaglandin G/H synthase 1 | Details |
| Desmopressin | enzyme | Prostaglandin G/H synthase 2 | Details |
| Desmopressin | target | Vasopressin V1a receptor | Details |
| Desmopressin | target | Vasopressin V2 receptor | Details |
| Coagulation factor VIIa Recombinant Human | target | Coagulation factor X | Details |
| Coagulation factor VIIa Recombinant Human | target | Tissue factor | Details |
| Coagulation factor VIIa Recombinant Human | target | Vitamin K-dependent gamma-carboxylase | Details |
| Coagulation factor VIIa Recombinant Human | target | Coagulation factor VII | Details |
| Coagulation factor VIIa Recombinant Human | target | Tissue factor pathway inhibitor | Details |
| Oprelvekin | target | Interleukin-11 receptor subunit alpha | Details |
| Palifermin | target | Basement membrane-specific heparan sulfate proteoglycan core protein | Details |
| Palifermin | target | Fibroblast growth factor receptor 2 | Details |
| Palifermin | target | Fibroblast growth factor receptor 1 | Details |
| Glucagon | target | Glucagon-like peptide 2 receptor | Details |
| Glucagon | target | Glucagon-like peptide 1 receptor | Details |
| Glucagon | target | Glucagon receptor | Details |
| Aldesleukin | enzyme | Cytosolic phospholipase A2 | Details |
| Aldesleukin | target | Interleukin-2 receptor subunit alpha | Details |
| Aldesleukin | target | Cytokine receptor common subunit gamma | Details |
| Aldesleukin | enzyme | Xanthine dehydrogenase/oxidase | Details |