| DB01365 | Mephentermine | approved | yes | agonist | Details |
| DB00182 | Amphetamine | approved, illicit, investigational | unknown | agonist | Details |
| DB09205 | Moxisylyte | approved, investigational | yes | antagonist | Details |
| DB09229 | Aranidipine | experimental | unknown | agonist | Details |
| DB11577 | Indigotindisulfonic acid | approved, investigational | no | agonist | Details |
| DB13345 | Dihydroergocristine | approved, experimental | yes | antagonistagonist | Details |
| DB01049 | Ergoloid mesylate | approved | yes | antagonistagonist | Details |
| DB11273 | Dihydroergocornine | approved | yes | antagonistagonist | Details |
| DB11278 | DL-Methylephedrine | approved | yes | agonist | Details |
| DB00268 | Ropinirole | approved, investigational | unknown | antagonist | Details |
| DB01069 | Promethazine | approved, investigational | unknown | antagonist | Details |
| DB01576 | Dextroamphetamine | approved, illicit | unknown | inhibitorinducer | Details |