| DB00241 | Butalbital | approved, illicit | yes | potentiator | Details |
| DB00273 | Topiramate | approved | yes | agonist | Details |
| DB00292 | Etomidate | approved | yes | agonist | Details |
| DB00306 | Talbutal | approved, illicit | yes | potentiator | Details |
| DB00312 | Pentobarbital | approved, investigational, vet_approved | yes | potentiator | Details |
| DB00418 | Secobarbital | approved, vet_approved | yes | potentiator | Details |
| DB00463 | Metharbital | withdrawn | yes | potentiator | Details |
| DB00474 | Methohexital | approved | yes | antagonist | Details |
| DB00599 | Thiopental | approved, vet_approved | yes | potentiator | Details |
| DB00794 | Primidone | approved, vet_approved | yes | potentiator | Details |
| DB00837 | Progabide | experimental | yes | agonist | Details |
| DB00849 | Methylphenobarbital | approved | yes | potentiator | Details |
| DB00898 | Ethanol | approved | yes | agonist | Details |
| DB01107 | Methyprylon | approved, illicit, withdrawn | yes | agonist | Details |
| DB01154 | Thiamylal | approved, vet_approved | yes | agonist | Details |
| DB01174 | Phenobarbital | approved, investigational | yes | potentiator | Details |
| DB01205 | Flumazenil | approved | yes | antagonist | Details |
| DB00425 | Zolpidem | approved | yes | agonist | Details |
| DB00466 | Picrotoxin | experimental | yes | antagonist | Details |
| DB00753 | Isoflurane | approved, vet_approved | yes | agonist | Details |
| DB00962 | Zaleplon | approved, illicit, investigational | yes | potentiator | Details |
| DB01028 | Methoxyflurane | approved, investigational, vet_approved, withdrawn | yes | agonist | Details |
| DB01159 | Halothane | approved, vet_approved | unknown | other/unknown | Details |
| DB01355 | Hexobarbital | experimental | yes | potentiator | Details |
| DB01353 | Butobarbital | approved, illicit | yes | potentiator | Details |
| DB00371 | Meprobamate | approved, illicit | yes | agonist | Details |
| DB06470 | Clomethiazole | investigational | unknown | | Details |
| DB00543 | Amoxapine | approved | unknown | antagonist | Details |
| DB00402 | Eszopiclone | approved, investigational | yes | potentiator | Details |
| DB01198 | Zopiclone | approved | yes | potentiator | Details |
| DB01381 | Ginkgo biloba | approved, investigational, nutraceutical | unknown | negative modulator | Details |
| DB01567 | Fludiazepam | experimental, illicit | yes | potentiator | Details |
| DB01341 | Dihydroquinidine barbiturate | experimental | yes | potentiator | Details |
| DB01351 | Amobarbital | approved, illicit | yes | potentiator | Details |
| DB01354 | Heptabarbital | experimental | yes | potentiator | Details |
| DB01352 | Aprobarbital | experimental, illicit | yes | potentiator | Details |
| DB01483 | Barbital | illicit | yes | potentiator | Details |
| DB01496 | Dihydro-2-thioxo-5-((5-(2-(trifluoromethyl)phenyl)-2-furanyl)methyl)-4,6(1H,5H)-pyrimidinedione | experimental, illicit | yes | potentiator | Details |
| DB01437 | Glutethimide | approved, illicit | yes | agonist | Details |
| DB01346 | Quinidine barbiturate | approved | yes | potentiator | Details |
| DB00395 | Carisoprodol | approved | unknown | activatormodulator | Details |
| DB12458 | Muscimol | investigational | unknown | | Details |
| DB00363 | Clozapine | approved | unknown | antagonist | Details |