The Future of Drug Discovery: Tackling the Undruggable with New Biotechnologies
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Drug Name
Type
Name
target
enzyme
carrier
transporter
Clear
3-isobutyl-1-methyl-7H-xanthine
target
Adenosine receptor A1
Details
3-isobutyl-1-methyl-7H-xanthine
target
cGMP-inhibited 3',5'-cyclic phosphodiesterase 3A
Details
3-isobutyl-1-methyl-7H-xanthine
target
Adenosine receptor A2a
Details
3-isobutyl-1-methyl-7H-xanthine
target
3',5'-cyclic-AMP phosphodiesterase 4B
Details
3-isobutyl-1-methyl-7H-xanthine
target
Adenosine receptor A2b
Details
3-isobutyl-1-methyl-7H-xanthine
target
cGMP-specific 3',5'-cyclic phosphodiesterase
Details
3-isobutyl-1-methyl-7H-xanthine
target
3',5'-cyclic-AMP phosphodiesterase 4D
Details
3-isobutyl-1-methyl-7H-xanthine
target
Adenosine receptor A3
Details
(2-BROMOETHYL)(2-'FORMYL-4'-AMINOPHENYL) ACETATE
target
Chymotrypsin-like elastase family member 1
Details
[1-(3-CHLORO-2-FORMYL-PHENYLCARBAMOYL)-2-METHYL-PROPYL]-CARBAMIC ACID TERT-BUTYL ESTER
target
Chymotrypsin-like elastase family member 1
Details
METHYL(2-ACETOXY-2-(2-CARBOXY-4-AMINO-PHENYL))ACETATE
target
Chymotrypsin-like elastase family member 1
Details
(2-CARBAMOYLMETHYL-5-PROPYL-OCTAHYDRO-INDOL-7-YL)ACETIC ACID
target
Group IIE secretory phospholipase A2
Details
3-(1H-BENZIMIDAZOL-2-YL)-1H-INDAZOLE
target
Serine/threonine-protein kinase Chk1
Details
5-ACETAMIDO-5,6-DIHYDRO-4-HYDROXY-6-ISOBUTOXY-4H-PYRAN-2-CARBOXYLIC ACID
target
Sialidase-2
Details
1-(4-Cyano-phenyl)-3-[2-(2,6-dichloro-phenyl)-1-imino-ethyl]-thiourea
target
Gag-Pol polyprotein
Details
METHYL N-[(2',4'-DIFLUORO-4-HYDROXY-5-IODOBIPHENYL-3-YL)CARBONYL]-BETA-ALANINATE
carrier
Transthyretin
Details
N-[(2',4'-DIFLUORO-4-HYDROXY-5-IODOBIPHENYL-3-YL)CARBONYL]-BETA-ALANINE
carrier
Transthyretin
Details
(3S)-4-{[4-(BUT-2-YNYLOXY)PHENYL]SULFONYL}-N-HYDROXY-2,2-DIMETHYLTHIOMORPHOLINE-3-CARBOXAMIDE
target
Disintegrin and metalloproteinase domain-containing protein 17
Details
6-(cyclohexylamino)-9-[2-(4-methylpiperazin-1-yl)-ethyl]-9H-purine-2-carbonitrile
target
Cathepsin K
Details
[4-({4-[(5-cyclopropyl-1H-pyrazol-3-yl)amino]quinazolin-2-yl}amino)phenyl]acetonitrile
target
Proto-oncogene tyrosine-protein kinase Src
Details
9-CYCLOPENTYL-6-[2-(3-IMIDAZOL-1-YL-PROPOXY)-PHENYLAMINO]-9H-PURINE-2-CARBONITRILE
target
Cathepsin K
Details
N-(2-CHLORO-4-FLUOROBENZOYL)-N'-(5-HYDROXY-2-METHOXYPHENYL)UREA
target
Glycogen phosphorylase, liver form
Details
3-[3-(4-methylpiperazin-1-yl)-7-(trifluoromethyl)quinoxalin-5-yl]phenol
target
Hepatocyte growth factor receptor
Details
5-[(2-methyl-5-{[3-(trifluoromethyl)phenyl]carbamoyl}phenyl)amino]pyridine-3-carboxamide
target
Ephrin type-A receptor 7
Details
5-AMINO-2-{4-[(4-AMINOPHENYL)SULFANYL]PHENYL}-1H-ISOINDOLE-1,3(2H)-DIONE
target
Cytochrome P450 130
Details
1-(3-METHYLPHENYL)-1H-BENZIMIDAZOL-5-AMINE
target
Cytochrome P450 130
Details
N-(1-ISOPROPYLPIPERIDIN-4-YL)-1-(3-METHOXYBENZYL)-1H-INDOLE-2-CARBOXAMIDE
target
Coagulation factor X
Details
1-{2-[(4-CHLOROPHENYL)AMINO]-2-OXOETHYL}-N-(1-ISOPROPYLPIPERIDIN-4-YL)-1H-INDOLE-2-CARBOXAMIDE
target
Coagulation factor X
Details
2-({[3,5-DIFLUORO-3'-(TRIFLUOROMETHOXY)BIPHENYL-4-YL]AMINO}CARBONYL)CYCLOPENT-1-ENE-1-CARBOXYLIC ACID
target
Dihydroorotate dehydrogenase (quinone), mitochondrial
Details
3-{[(3-FLUORO-3'-METHOXYBIPHENYL-4-YL)AMINO]CARBONYL}THIOPHENE-2-CARBOXYLIC ACID
target
Dihydroorotate dehydrogenase (quinone), mitochondrial
Details
Displaying targets
22651 - 22680
of
33504
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