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Targets
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Drug Name
Type
Name
target
enzyme
carrier
transporter
Clear
N~4~-methyl-N~4~-(3-methyl-1H-indazol-6-yl)-N~2~-(3,4,5-trimethoxyphenyl)pyrimidine-2,4-diamine
target
Vascular endothelial growth factor receptor 2
Details
1-[4-(PYRIDIN-4-YLOXY)PHENYL]-3-[3-(TRIFLUOROMETHYL)PHENYL]UREA
target
Tyrosine-protein kinase ABL1
Details
ABT-341
target
Dipeptidyl peptidase 4
Details
4-{4-[4-(3-AMINOPROPOXY)PHENYL]-1H-PYRAZOL-5-YL}-6-CHLOROBENZENE-1,3-DIOL
target
Heat shock protein HSP 90-beta
Details
2-chloro-5-[(1S)-1-hydroxy-3-oxo-2H-isoindol-1-yl]benzenesulfonamide
target
Carbonic anhydrase 2
Details
4-[1-allyl-7-(trifluoromethyl)-1H-indazol-3-yl]benzene-1,3-diol
target
Estrogen receptor
Details
4-[1-allyl-7-(trifluoromethyl)-1H-indazol-3-yl]benzene-1,3-diol
target
Nuclear receptor coactivator 2
Details
4-(6-HYDROXY-1H-INDAZOL-3-YL)BENZENE-1,3-DIOL
target
Estrogen receptor
Details
4-(6-HYDROXY-1H-INDAZOL-3-YL)BENZENE-1,3-DIOL
target
Nuclear receptor coactivator 2
Details
7,8-dihydroxy-4-phenyl-2H-chromen-2-one
target
Catechol O-methyltransferase
Details
5-phenyl-2-keto-valeric acid
target
Indole-3-pyruvate decarboxylase
Details
(2R)-4-(2-BENZOYL-1,2-DIAZEPAN-1-YL)-4-OXO-1-(2,4,5-TRIFLUOROPHENYL)BUTAN-2-AMINE
target
Dipeptidyl peptidase 4
Details
PP-121
target
Serine/threonine-protein kinase mTOR
Details
PP-121
target
Platelet-derived growth factor receptor alpha
Details
PP-121
target
Tyrosine-protein kinase ABL1
Details
PP-121
target
Tyrosine-protein kinase HCK
Details
PP-121
target
Vascular endothelial growth factor receptor 2
Details
PP-121
target
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform
Details
PP-121
target
Epidermal growth factor receptor
Details
PP-121
target
Proto-oncogene tyrosine-protein kinase Src
Details
PP-121
target
DNA-dependent protein kinase catalytic subunit
Details
PP-121
target
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform
Details
1-cyclobutyl-3-(3,4-dimethoxyphenyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
target
Proto-oncogene tyrosine-protein kinase Src
Details
1-(1-methylethyl)-3-quinolin-6-yl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
target
Proto-oncogene tyrosine-protein kinase Src
Details
N-(2-chlorophenyl)-5-phenylimidazo[1,5-a]pyrazin-8-amine
target
Tyrosine-protein kinase Lck
Details
N-(2,6-dimethylphenyl)-5-phenylimidazo[1,5-a]pyrazin-8-amine
target
Tyrosine-protein kinase Lck
Details
N-(2-chloro-6-methylphenyl)-8-[(3S)-3-methylpiperazin-1-yl]imidazo[1,5-a]quinoxalin-4-amine
target
Tyrosine-protein kinase Lck
Details
4-[3-(1,4-diazepan-1-ylcarbonyl)-4-fluorobenzyl]phthalazin-1(2H)-one
target
Poly [ADP-ribose] polymerase 1
Details
4-[3-(1,4-diazepan-1-ylcarbonyl)-4-fluorobenzyl]phthalazin-1(2H)-one
target
Protein mono-ADP-ribosyltransferase PARP3
Details
Wortmannin
target
Phosphatidylinositol 3-kinase regulatory subunit alpha
Details
Displaying targets
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