The Future of Drug Discovery: Tackling the Undruggable with New Biotechnologies
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Displaying targets
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Drug Name
Type
Name
target
enzyme
carrier
transporter
Clear
7-{[(CYCLOHEXYLAMINO)CARBONYL]AMINO}HEPTANOIC ACID
target
Bifunctional epoxide hydrolase 2
Details
(1S,2R,3S,4R,5R)-2,3,4-trihydroxy-N-octyl-6-oxa-8-azabicyclo[3.2.1]octane-8-carbothioamide
target
Beta-glucosidase A
Details
2-hydroxy-7-methoxy-5-methyl-naphthalene-1-carboxylic acid meso-2,5-dihydroxy-cyclopent-3-enyl ester
target
Neocarzinostatin
Details
2,6-dicarboxynaphthalene
target
Hemoglobin subunit alpha
Details
2,6-dicarboxynaphthalene
target
Hemoglobin subunit beta
Details
N-(carboxycarbonyl)-D-phenylalanine
target
Hypoxia-inducible factor 1-alpha inhibitor
Details
(1R, 2S)-cis 1,2 dihydroxy-1,2-dihydronaphthalene
target
Naphthalene 1,2-dioxygenase subunit beta
Details
(1R, 2S)-cis 1,2 dihydroxy-1,2-dihydronaphthalene
target
Naphthalene 1,2-dioxygenase subunit alpha
Details
2-(TOLUENE-4-SULFONYL)-2H-BENZO[D][1,2,3]DIAZABORININ-1-OL
target
Enoyl-[acyl-carrier-protein] reductase [NADH] FabI
Details
Methyl [(1E,5R)-5-{3-[(2E,4E)-2,5-dimethyl-2,4-octadienoyl]-2,4-dioxo-3,4-dihydro-2H-pyran-6-yl}hexylidene]carbamate
target
DNA-directed RNA polymerase subunit beta
Details
Methyl [(1E,5R)-5-{3-[(2E,4E)-2,5-dimethyl-2,4-octadienoyl]-2,4-dioxo-3,4-dihydro-2H-pyran-6-yl}hexylidene]carbamate
target
DNA-directed RNA polymerase subunit beta'
Details
Methyl [(1E,5R)-5-{3-[(2E,4E)-2,5-dimethyl-2,4-octadienoyl]-2,4-dioxo-3,4-dihydro-2H-pyran-6-yl}hexylidene]carbamate
target
DNA-directed RNA polymerase subunit alpha
Details
Methyl [(1E,5R)-5-{3-[(2E,4E)-2,5-dimethyl-2,4-octadienoyl]-2,4-dioxo-3,4-dihydro-2H-pyran-6-yl}hexylidene]carbamate
target
RNA polymerase sigma factor SigA
Details
Methyl [(1E,5R)-5-{3-[(2E,4E)-2,5-dimethyl-2,4-octadienoyl]-2,4-dioxo-3,4-dihydro-2H-pyran-6-yl}hexylidene]carbamate
target
DNA-directed RNA polymerase subunit omega
Details
6-amino-4-(2-phenylethyl)-1,7-dihydro-8H-imidazo[4,5-g]quinazolin-8-one
target
Queuine tRNA-ribosyltransferase
Details
6-AMINO-4-[2-(4-METHYLPHENYL)ETHYL]-1,7-DIHYDRO-8H-IMIDAZO[4,5-G]QUINAZOLIN-8-ONE
target
Queuine tRNA-ribosyltransferase
Details
N-(2-AMINOETHYL)-N~2~-{(1S)-1-[4'-(AMINOSULFONYL)BIPHENYL-4-YL]-2,2,2-TRIFLUOROETHYL}-L-LEUCINAMIDE
target
Cathepsin K
Details
N-ISOBUTYL-N-[4-METHOXYPHENYLSULFONYL]GLYCYL HYDROXAMIC ACID
target
Stromelysin-2
Details
N-ISOBUTYL-N-[4-METHOXYPHENYLSULFONYL]GLYCYL HYDROXAMIC ACID
target
Macrophage metalloelastase
Details
N-ISOBUTYL-N-[4-METHOXYPHENYLSULFONYL]GLYCYL HYDROXAMIC ACID
target
Stromelysin-1
Details
N-ISOBUTYL-N-[4-METHOXYPHENYLSULFONYL]GLYCYL HYDROXAMIC ACID
target
Matrix metalloproteinase-20
Details
(4S)-4-(2-NAPHTHYLMETHYL)-D-GLUTAMIC ACID
target
Glutamate racemase
Details
4-HYDROXY-5-IODO-3-NITROPHENYLACETYL-EPSILON-AMINOCAPROIC ACID ANION
target
Immunoglobulin lambda variable 7-43
Details
4-HYDROXY-5-IODO-3-NITROPHENYLACETYL-EPSILON-AMINOCAPROIC ACID ANION
target
Immunoglobulin heavy variable 1-2
Details
6,7,8,9-TETRAHYDRO-4-HYDROXY-3-(1-PHENYLPROPYL)CYCLOHEPTA[B]PYRAN-2-ONE
target
Gag-Pol polyprotein
Details
N-DODECANOYL-L-TYROSINE
target
Long-chain N-acyl amino acid synthase
Details
trifluoro-[hydroxy-[hydroxy-[2-(N-methyl-2-nitro-anilino)ethoxy]phosphoryl]oxy-phosphoryl]oxy-beryllium(1-)
target
Myosin-14
Details
2-(2-CHLORO-4-FLUOROPHENOXY)-2-METHYL-N-[(1R,2S,3S,5S,7S)-5-(METHYLSULFONYL)-2-ADAMANTYL]PROPANAMIDE
target
11-beta-hydroxysteroid dehydrogenase 1
Details
1-(2-cyclopropylethyl)-3-(1,1-dioxo-2H-1,2,4-benzothiadiazin-3-yl)-6-fluoro-4-hydroxy-2(1H)-quinolinone
target
Genome polyprotein
Details
3-{ISOPROPYL[(TRANS-4-METHYLCYCLOHEXYL)CARBONYL]AMINO}-5-PHENYLTHIOPHENE-2-CARBOXYLIC ACID
target
Genome polyprotein
Details
Displaying targets
23161 - 23190
of
33504
in total
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