The Future of Drug Discovery: Tackling the Undruggable with New Biotechnologies
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Drug Name
Type
Name
target
enzyme
carrier
transporter
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2-amino-4-[2,4-dichloro-5-(2-pyrrolidin-1-ylethoxy)phenyl]-N-ethylthieno[2,3-d]pyrimidine-6-carboxamide
target
Heat shock protein HSP 90-alpha
Details
2-CHLORO-N-(3-CYANO-5,6-DIHYDRO-4H-CYCLOPENTA[B]THIOPHEN-2-YL)-5-DIETHYLSULFAMOYL-BENZAMIDE
target
UDP-N-acetylmuramoyl-tripeptide--D-alanyl-D-alanine ligase
Details
N-{2-[(4'-CYANO-1,1'-BIPHENYL-4-YL)OXY]ETHYL}-N'-HYDROXY-N-METHYLUREA
target
Neutrophil collagenase
Details
7A-[(4-cyanophenyl)methyl]-6-(3,5-dichlorophenyl)-5-oxo-2,3,5,7A-tetrahydro-1H-pyrrolo[1,2-A]pyrrole-7-carbonitrile
target
Integrin alpha-L
Details
Bisphenol A
target
Androgen receptor
Details
Bisphenol A
target
Estrogen receptor beta
Details
Bisphenol A
target
Estrogen-related receptor gamma
Details
5-hydroxy-4-(7-methoxy-1,1-dioxido-2H-1,2,4-benzothiadiazin-3-yl)-2-(3-methylbutyl)-6-phenylpyridazin-3(2H)-one
target
Genome polyprotein
Details
1-(5-OXO-2,3,5,9B-TETRAHYDRO-1H-PYRROLO[2,1-A]ISOINDOL-9-YL)-3-(5-PYRROLIDIN-2-YL-1H-PYRAZOL-3-YL)-UREA
target
Cyclin-dependent kinase 2
Details
(2S)-1-{[5-(1H-Indazol-5-yl)-3-pyridinyl]oxy}-3-(7aH-indol-3-yl)-2-propanamine
target
cAMP-dependent protein kinase catalytic subunit alpha
Details
N'-[(1E)-(3,5-dibromo-2,4-dihydroxyphenyl)methylidene]-4-methoxybenzohydrazide
target
3-hydroxyacyl-[acyl-carrier-protein] dehydratase FabZ
Details
5-(dodecylthio)-1H-1,2,3-triazole-4-carboxylic acid
target
2-Hydroxyacid oxidase 1
Details
(2S)-2-(1H-indol-3-yl)hexanoic acid
target
S-phase kinase-associated protein 1
Details
(2S)-2-(1H-indol-3-yl)pentanoic acid
target
S-phase kinase-associated protein 1
Details
(2S)-8-[(tert-butoxycarbonyl)amino]-2-(1H-indol-3-yl)octanoic acid
target
S-phase kinase-associated protein 1
Details
(5-phenyl-7-(pyridin-3-ylmethylamino)pyrazolo[1,5-a]pyrimidin-3-yl)methanol
target
Cyclin-dependent kinase 2
Details
(1R,2R,3R,4S,5R)-4-(Benzylamino)-5-(methylthio)cyclopentane-1,2,3-triol
target
Alpha-mannosidase 2
Details
2-[({4-[2-(trifluoromethyl)phenyl]piperidin-1-yl}carbonyl)amino]benzoic acid
carrier
Retinol-binding protein 4
Details
2-CHLORO-N-[(1R,2R)-1-HYDROXY-2,3-DIHYDRO-1H-INDEN-2-YL]-6H-THIENO[2,3-B]PYRROLE-5-CARBOXAMIDE
target
Glycogen phosphorylase, muscle form
Details
(R)-Atenolol
target
Group IIE secretory phospholipase A2
Details
(R)-Atenolol
target
Lactotransferrin
Details
2-HYDROXY-5-{[(1E)-2-PHENYLETHYLIDENE]AMINO}-L-TYROSINE
target
Phenylethylamine oxidase
Details
{4-[2-BENZYL-3-METHOXY-2-(METHOXYCARBONYL)-3-OXOPROPYL]PHENYL}SULFAMIC ACID
target
Receptor-type tyrosine-protein phosphatase beta
Details
4-[(1E,7E)-8-(2,6-DIOXO-1,2,3,6-TETRAHYDROPYRIMIDIN-4-YL)-3,6-DIOXA-2,7-DIAZAOCTA-1,7-DIEN-1-YL]BENZOIC ACID
target
Uracil-DNA glycosylase
Details
N-[2-methyl-5-(methylcarbamoyl)phenyl]-2-{[(1R)-1-methylpropyl]amino}-1,3-thiazole-5-carboxamide
target
Mitogen-activated protein kinase 14
Details
(3,3-dimethylpiperidin-1-yl)(6-(3-fluoro-4-methylphenyl)pyridin-2-yl)methanone
target
11-beta-hydroxysteroid dehydrogenase 1
Details
(2S,3S)-4-cyclopropyl-3-{(3R,5R)-3-[2-fluoro-4-(methylsulfonyl)phenyl]-1,2,4-oxadiazolidin-5-yl}-1-[(3S)-3-fluoropyrrolidin-1-yl]-1-oxobutan-2-amine
target
Dipeptidyl peptidase 4
Details
(2S,3S)-3-{3-[2-chloro-4-(methylsulfonyl)phenyl]-1,2,4-oxadiazol-5-yl}-1-cyclopentylidene-4-cyclopropyl-1-fluorobutan-2-amine
target
Dipeptidyl peptidase 4
Details
N-({4-[(2-aminopyridin-4-yl)oxy]-3-fluorophenyl}carbamoyl)-2-(4-fluorophenyl)acetamide
target
Hepatocyte growth factor receptor
Details
D-leucyl-N-(4-carbamimidoylbenzyl)-L-prolinamide
target
Prothrombin
Details
Displaying targets
21271 - 21300
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