The Future of Drug Discovery: Tackling the Undruggable with New Biotechnologies
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Displaying targets
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Drug Name
Type
Name
target
enzyme
carrier
transporter
Clear
Sobetirome
target
Thyroid hormone receptor beta
Details
Sobetirome
target
Muscarinic acetylcholine receptor M1
Details
Sobetirome
target
Thyroid hormone receptor, alpha isoform 1 variant
Details
[1-HYDROXY-2-(1,1':3',1''-TERPHENYL-3-YLOXY)ETHANE-1,1-DIYL]BIS(PHOSPHONIC ACID)
target
Ditrans,polycis-undecaprenyl-diphosphate synthase ((2E,6E)-farnesyl-diphosphate specific)
Details
[1-HYDROXY-2-(1,1':3',1''-TERPHENYL-3-YLOXY)ETHANE-1,1-DIYL]BIS(PHOSPHONIC ACID)
target
Farnesyl pyrophosphate synthase
Details
2-[(2-methoxy-5-methylphenoxy)methyl]pyridine
target
Hemoglobin subunit alpha
Details
2-[(2-methoxy-5-methylphenoxy)methyl]pyridine
target
Hemoglobin subunit beta
Details
4-[(5-methoxy-2-methylphenoxy)methyl]pyridine
target
Hemoglobin subunit beta
Details
4-[(5-methoxy-2-methylphenoxy)methyl]pyridine
target
Hemoglobin subunit alpha
Details
2-({[4-bromo-3-(diethylsulfamoyl)phenyl]carbonyl}amino)benzoic acid
target
3-oxoacyl-[acyl-carrier-protein] synthase 3
Details
(10R)-10-methyl-3-(6-methylpyridin-3-yl)-9,10,11,12-tetrahydro-8H-[1,4]diazepino[5',6':4,5]thieno[3,2-f]quinolin-8-one
target
MAP kinase-activated protein kinase 2
Details
(3R)-3-(aminomethyl)-9-methoxy-1,2,3,4-tetrahydro-5H-[1]benzothieno[3,2-e][1,4]diazepin-5-one
target
MAP kinase-activated protein kinase 2
Details
(3R)-3-(aminomethyl)-9-methoxy-1,2,3,4-tetrahydro-5H-[1]benzothieno[3,2-e][1,4]diazepin-5-one
target
Cyclin-dependent kinase 2
Details
[[(3R,4R,5S,6R)-3-(butanoylamino)-4,5-dihydroxy-6-(hydroxymethyl)oxan-2-ylidene]amino] N-phenylcarbamate
target
O-GlcNAcase BT_4395
Details
[[(3R,4R,5S,6R)-3-(butanoylamino)-4,5-dihydroxy-6-(hydroxymethyl)oxan-2-ylidene]amino] N-phenylcarbamate
target
Beta-hexosaminidase
Details
(TERT-BUTYLOXYCARBONYL)-ALANYL-AMINO ETHYL-FORMAMIDE
target
Chymotrypsin-like elastase family member 1
Details
HONH-BENZYLMALONYL-L-ALANYLGLYCINE-P-NITROANILIDE
target
Thermolysin
Details
1,2,3-TRIHYDROXY-1,2,3,4-TETRAHYDROBENZO[A]PYRENE
target
DNA polymerase I
Details
1,2,3-TRIHYDROXY-1,2,3,4-TETRAHYDROBENZO[A]PYRENE
target
DNA polymerase kappa
Details
N-(1-PHENYL-PROPYL)-FORMAMIDE
target
Capsid scaffolding protein
Details
5-Benzylacyclouridine
target
Uridine phosphorylase 1
Details
5-Benzylacyclouridine
target
Uridine phosphorylase
Details
1-((2-HYDROXYETHOXY)METHYL)-5-(3-(BENZYLOXY)BENZYL)-6-HYDROXYPYRIMIDINE-2,4(1H,3H)-DIONE
target
Uridine phosphorylase
Details
4-TERT-BUTYLBENZENESULFONIC ACID
target
Prothrombin
Details
3-{[(9-CYANO-9,10-DIHYDRO-10-METHYLACRIDIN-9-YL)CARBONYL]AMINO}PROPANOIC ACID
target
Immunoglobulin heavy constant gamma 1
Details
3-{[(9-CYANO-9,10-DIHYDRO-10-METHYLACRIDIN-9-YL)CARBONYL]AMINO}PROPANOIC ACID
target
Immunoglobulin kappa constant
Details
(2Z)-N-biphenyl-4-yl-2-cyano-3-hydroxybut-2-enamide
target
Dihydroorotate dehydrogenase (quinone), mitochondrial
Details
(2Z)-N-biphenyl-4-yl-2-cyano-3-hydroxybut-2-enamide
target
Dihydroorotate dehydrogenase (quinone), mitochondrial
Details
6-(3-AMINOPROPYL)-4,9-DIMETHYLPYRROLO[3,4-C]CARBAZOLE-1,3(2H,6H)-DIONE
target
Death-associated protein kinase 1
Details
N'-[(1E)-(3,5-DIBROMO-2,4-DIHYDROXYPHENYL)METHYLENE]NICOTINOHYDRAZIDE
target
3-hydroxyacyl-[acyl-carrier-protein] dehydratase FabZ
Details
Displaying targets
21871 - 21900
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