The Future of Drug Discovery: Tackling the Undruggable with New Biotechnologies
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Displaying targets
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Drug Name
Type
Name
target
enzyme
carrier
transporter
Clear
CIS-(1R,2S)-2-AMINO-1,2,3,4-TETRAHYDRONAPHTHALEN-1-OL
target
Phenylethanolamine N-methyltransferase
Details
2,3,6A,7,8,9-HEXAHYDRO-11H-[1,4]DIOXINO[2,3-G]PYRROLO[2,1-B][1,3]BENZOXAZIN-11-ONE
target
Glutamate receptor 2
Details
[(2-AMINO-ALPHA-METHOXYIMINO-4-THIAZOLYLACETYL)AMINO]METHYLBORONIC ACID
target
Beta-lactamase TEM
Details
4-chloro-6-{5-[(2-morpholin-4-ylethyl)amino]-1,2-benzisoxazol-3-yl}benzene-1,3-diol
target
Heat shock protein HSP 90-alpha
Details
S-{3-[(4-ANILINOQUINAZOLIN-6-YL)AMINO]-3-OXOPROPYL}-L-CYSTEINE
target
Epidermal growth factor receptor
Details
(6AR,11AS,11BR)-10-ACETYL-9-HYDROXY-7,7-DIMETHYL-2,6,6A,7,11A,11B-HEXAHYDRO-11H-PYRROLO[1',2':2,3]ISOINDOLO[4,5,6-CD]INDOL-11-ONE
target
Sarcoplasmic/endoplasmic reticulum calcium ATPase 1
Details
2-({4-[(5-CHLORO-1H-INDOL-2-YL)SULFONYL]PIPERAZIN-1-YL}CARBONYL)THIENO[3,2-B]PYRIDINE 4-OXIDE
target
Coagulation factor X
Details
6-(3,4-DIHYDROXYBENZYL)-3-ETHYL-1-(2,4,6-TRICHLOROPHENYL)-1H-PYRAZOLO[3,4-D]PYRIMIDIN-4(5H)-ONE
target
Cyclin-dependent kinase 2
Details
4-[5-(3-IODO-PHENYL)-2-(4-METHANESULFINYL-PHENYL)-1H-IMIDAZOL-4-YL]-PYRIDINE
target
Mitogen-activated protein kinase 14
Details
N-(5-{[(2S)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1H-indazol-3-yl)benzamide
target
Dual specificity tyrosine-phosphorylation-regulated kinase 1A
Details
N,N-DIMETHYL(5-(PYRIDIN-3-YL)FURAN-2-YL)METHANAMINE
target
Cytochrome P450 2A6
Details
1,2-Dihydroxynaphthalene
target
1,2-dihydroxynaphthalene dioxygenase
Details
DECANE-1-THIOL
target
3-oxoacyl-[acyl-carrier-protein] synthase 3
Details
6-(3-AMINOPHENYL)-N-(TERT-BUTYL)-2-(TRIFLUOROMETHYL)QUINAZOLIN-4-AMINE
target
Cyclin-dependent kinase 2
Details
3-phenyl-5-(1H-pyrazol-3-yl)isoxazole
target
Hematopoietic prostaglandin D synthase
Details
PHENYL-5-(1H-PYRAZOL-3-YL)-1,3-THIAZOLE
target
Hematopoietic prostaglandin D synthase
Details
Tranilast
target
Hematopoietic prostaglandin D synthase
Details
Tranilast
enzyme
Cytochrome P450 3A4
Details
Tranilast
enzyme
Cytochrome P450 2C9
Details
Tranilast
target
Steryl-sulfatase
Details
Tranilast
target
Histamine H1 receptor
Details
4-{[4-(4-fluoro-3-methylphenyl)-1,3-thiazol-2-yl]amino}-2-hydroxybenzoic acid
target
Hematopoietic prostaglandin D synthase
Details
N-METHYL(5-(PYRIDIN-3-YL)FURAN-2-YL)METHANAMINE
target
Cytochrome P450 2A6
Details
2-(4-(AMINOMETHYL)PIPERIDIN-1-YL)-N-(3_CYCLOHEXYL-4-OXO-2,4-DIHYDROINDENO[1,2-C]PYRAZOL-5-YL)ACETAMIDE
target
Cyclin-dependent kinase 2
Details
N-cyclopropyl-N-(trans-4-pyridin-3-ylcyclohexyl)-4-[(1S)-2,2,2-trifluoro-1-hydroxy-1-methylethyl]benzamide
target
11-beta-hydroxysteroid dehydrogenase 1
Details
2-[(2,4-DICHLORO-5-METHYLPHENYL)SULFONYL]-1,3-DINITRO-5-(TRIFLUOROMETHYL)BENZENE
target
Replicase polyprotein 1ab
Details
2-[(2,4-DICHLORO-5-METHYLPHENYL)SULFONYL]-1,3-DINITRO-5-(TRIFLUOROMETHYL)BENZENE
target
Replicase polyprotein 1a
Details
(5-(PYRIDIN-3-YL)FURAN-2-YL)METHANAMINE
target
Cytochrome P450 2A6
Details
(5-(PYRIDIN-3-YL)FURAN-2-YL)METHANAMINE
target
Cytochrome P450 2D6
Details
1-(3-(2,4-DIMETHYLTHIAZOL-5-YL)-4-OXO-2,4-DIHYDROINDENO[1,2-C]PYRAZOL-5-YL)-3-(4-METHYLPIPERAZIN-1-YL)UREA
target
Cyclin-dependent kinase 2
Details
Displaying targets
22111 - 22140
of
33504
in total
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734
735
736
737
738
739
740
741
742
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