The Future of Drug Discovery: Tackling the Undruggable with New Biotechnologies
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Targets
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Drug Name
Type
Name
target
enzyme
carrier
transporter
Clear
Wortmannin
target
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform
Details
Wortmannin
target
Serine/threonine-protein kinase PLK1
Details
Wortmannin
target
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform
Details
Wortmannin
target
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform
Details
4-(2-AMINOPHENYL)-4-OXOBUTANOIC ACID
target
Alanine--glyoxylate aminotransferase
Details
4-[3-(4-CHLOROPHENYL)-1H-PYRAZOL-5-YL]PIPERIDINE
target
Prothrombin
Details
3-(4-CHLOROPHENYL)-5-(METHYLTHIO)-4H-1,2,4-TRIAZOLE
target
Prothrombin
Details
1-BENZYL-3-(4-METHOXYPHENYLAMINO)-4-PHENYLPYRROLE-2,5-DIONE
target
Retinoic acid receptor RXR-alpha
Details
1-BENZYL-3-(4-METHOXYPHENYLAMINO)-4-PHENYLPYRROLE-2,5-DIONE
target
Oxysterols receptor LXR-alpha
Details
N-(3-TERT-BUTYL-1H-PYRAZOL-5-YL)-N'-{4-CHLORO-3-[(PYRIDIN-3-YLOXY)METHYL]PHENYL}UREA
target
Mitogen-activated protein kinase 14
Details
2-(1H-pyrazol-3-yl)-1H-benzimidazole
target
Aurora kinase A
Details
N-[3-(1H-BENZIMIDAZOL-2-YL)-1H-PYRAZOL-4-YL]BENZAMIDE
target
Aurora kinase A
Details
N-[3-(1H-BENZIMIDAZOL-2-YL)-1H-PYRAZOL-4-YL]BENZAMIDE
target
Cyclin-dependent kinase 2
Details
4-[(2-{4-[(CYCLOPROPYLCARBAMOYL)AMINO]-1H-PYRAZOL-3-YL}-1H-BENZIMIDAZOL-6-YL)METHYL]MORPHOLIN-4-IUM
target
Tyrosine-protein kinase JAK2
Details
N-[4-CHLORO-3-(PYRIDIN-3-YLOXYMETHYL)-PHENYL]-3-FLUORO-
target
Mitogen-activated protein kinase 14
Details
4-AMINO-5-(2-METHYLPHENYL)-2,4-DIHYDRO-3H-1,2,4-TRIAZOLE-3-THIONE
target
Metallo-beta-lactamase L1
Details
2-[4-(3-METHYL-1H-PYRAZOL-4-YL)PHENYL]ETHANAMINE
target
cAMP-dependent protein kinase catalytic subunit alpha
Details
2-[4-(3-METHYL-1H-PYRAZOL-4-YL)PHENYL]ETHANAMINE
target
cAMP-dependent protein kinase inhibitor alpha
Details
(2S)-1-methyl-2-[(2S,4R)-2-methyl-4-phenylpentyl]piperidine
target
Probable L-lysine-epsilon aminotransferase
Details
4-(2-AMINOETHOXY)-3,5-DICHLORO-N-[3-(1-METHYLETHOXY)PHENYL]BENZAMIDE
target
Urokinase-type plasminogen activator
Details
(2S)-1-(1H-INDOL-3-YL)-3-{[5-(3-METHYL-1H-INDAZOL-5-YL)PYRIDIN-3-YL]OXY}PROPAN-2-AMINE
target
cAMP-dependent protein kinase inhibitor alpha
Details
(2S)-1-(1H-INDOL-3-YL)-3-{[5-(3-METHYL-1H-INDAZOL-5-YL)PYRIDIN-3-YL]OXY}PROPAN-2-AMINE
target
RAC-alpha serine/threonine-protein kinase
Details
(2S)-1-(1H-INDOL-3-YL)-3-{[5-(3-METHYL-1H-INDAZOL-5-YL)PYRIDIN-3-YL]OXY}PROPAN-2-AMINE
target
RAC-beta serine/threonine-protein kinase
Details
(2S)-1-(1H-INDOL-3-YL)-3-{[5-(3-METHYL-1H-INDAZOL-5-YL)PYRIDIN-3-YL]OXY}PROPAN-2-AMINE
target
Glycogen synthase kinase-3 beta
Details
(2S)-1-(1H-INDOL-3-YL)-3-{[5-(3-METHYL-1H-INDAZOL-5-YL)PYRIDIN-3-YL]OXY}PROPAN-2-AMINE
target
cAMP-dependent protein kinase catalytic subunit alpha
Details
3-(3-Methyl-2-buten-1-yl)-3H-purin-6-amine
target
Biotin carboxylase
Details
4-(2-amino-1,3-thiazol-4-yl)pyrimidin-2-amine
target
Biotin carboxylase
Details
4-[1-(2,6-dichlorobenzyl)-2-methyl-1H-imidazol-4-yl]pyrimidin-2-amine
target
Biotin carboxylase
Details
2-[4-({[(3,5-DICHLOROPHENYL)AMINO]CARBONYL}AMINO)PHENOXY]-2-METHYLPROPANOIC ACID
target
Hemoglobin subunit alpha
Details
2-[4-({[(3,5-DICHLOROPHENYL)AMINO]CARBONYL}AMINO)PHENOXY]-2-METHYLPROPANOIC ACID
target
Hemoglobin subunit beta
Details
Displaying targets
22801 - 22830
of
33504
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