| Anacaulase | enzyme | Cytochrome P450 2C9 | Details |
| Anacaulase | enzyme | Cytochrome P450 2C8 | Details |
| Anacaulase | target | Alpha-1-antichymotrypsin | Details |
| Anacaulase | target | Alpha-2-macroglobulin | Details |
| Pirtobrutinib | enzyme | UDP-glucuronosyltransferase 1-8 | Details |
| Pirtobrutinib | enzyme | Cytochrome P450 1A2 | Details |
| Pirtobrutinib | enzyme | Cytochrome P450 2B6 | Details |
| Pirtobrutinib | enzyme | Cytochrome P450 2C19 | Details |
| Pirtobrutinib | enzyme | Cytochrome P450 3A5 | Details |
| Pirtobrutinib | target | Tyrosine-protein kinase BTK | Details |
| Pirtobrutinib | enzyme | Cytochrome P450 3A4 | Details |
| Pirtobrutinib | enzyme | Cytochrome P450 2C9 | Details |
| Pirtobrutinib | enzyme | UDP-glucuronosyltransferase 1-9 | Details |
| Pirtobrutinib | enzyme | Cytochrome P450 2C8 | Details |
| Pirtobrutinib | enzyme | Cytochrome P450 2D6 | Details |
| Pirtobrutinib | transporter | P-glycoprotein 1 | Details |
| Pirtobrutinib | transporter | ATP-binding cassette sub-family G member 2 | Details |
| Bioymifi | target | Tumor necrosis factor receptor superfamily member 10B | Details |
| Atidarsagene autotemcel | target | Human Arylsulfatase A mRNA | Details |
| KIN-3248 | target | Fibroblast growth factor receptor 2 | Details |
| KIN-3248 | target | Fibroblast growth factor receptor 3 | Details |
| Flotufolastat F-18 | target | Glutamate carboxypeptidase 2 | Details |
| Lotilaner | target | Gaba-gated chloride channel, putative | Details |
| (R)-9b | target | Activated CDC42 kinase 1 | Details |