Unlocking Undruggable Targets: Shifting Paradigms in Modern Drug Discovery
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Displaying targets
25531 - 25560
of
29784
in total
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Drug Name
Type
Name
target
enzyme
carrier
transporter
Clear
Bictegravir
enzyme
Multidrug and toxin extrusion protein 1
Details
Tivozanib
enzyme
Cytochrome P450 3A4
Details
Tivozanib
target
Vascular endothelial growth factor receptor 3
Details
Tivozanib
target
Mast/stem cell growth factor receptor Kit
Details
Tivozanib
transporter
ATP-binding cassette sub-family G member 2
Details
Tivozanib
target
Protein-tyrosine kinase 6
Details
Tivozanib
target
Fibroblast growth factor receptor 1
Details
Tivozanib
target
Vascular endothelial growth factor receptor 1
Details
Tivozanib
target
Vascular endothelial growth factor receptor 2
Details
Tivozanib
target
Platelet-derived growth factor receptor alpha
Details
Tivozanib
target
Angiopoietin-1 receptor
Details
Tivozanib
carrier
Serum albumin
Details
Tivozanib
target
Platelet-derived growth factor receptor beta
Details
Tivozanib
transporter
P-glycoprotein 1
Details
Tivozanib
target
Receptor-type tyrosine-protein kinase FLT3
Details
Tivozanib
target
Hepatocyte growth factor receptor
Details
Saracatinib
enzyme
Cytochrome P450 3A4
Details
Arhalofenate
target
Peroxisome proliferator-activated receptor gamma
Details
Baricitinib
transporter
P-glycoprotein 1
Details
Baricitinib
enzyme
Cytochrome P450 3A4
Details
Baricitinib
target
Tyrosine-protein kinase JAK1
Details
Baricitinib
target
Tyrosine-protein kinase JAK3
Details
Baricitinib
transporter
Solute carrier family 22 member 8
Details
Baricitinib
transporter
ATP-binding cassette sub-family G member 2
Details
Baricitinib
transporter
Multidrug and toxin extrusion protein 2
Details
Baricitinib
target
Tyrosine-protein kinase JAK2
Details
Baricitinib
transporter
Solute carrier family 22 member 6
Details
Baricitinib
transporter
Solute carrier family 22 member 2
Details
Baricitinib
transporter
Solute carrier organic anion transporter family member 1B3
Details
Baricitinib
target
Non-receptor tyrosine-protein kinase TYK2
Details
Displaying targets
25531 - 25560
of
29784
in total
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848
849
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852
853
854
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