From Impossible to Inevitable: Transforming Undruggable Targets
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Targets
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Displaying targets
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of
29784
in total
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Drug Name
Type
Name
target
enzyme
carrier
transporter
Clear
Momelotinib
enzyme
Cytochrome P450 1A2
Details
Momelotinib
enzyme
Cytochrome P450 2B6
Details
Momelotinib
enzyme
UDP-glucuronosyltransferase 1-1
Details
Momelotinib
enzyme
UDP-glucuronosyltransferase 1-9
Details
Momelotinib
transporter
ATP-binding cassette sub-family G member 2
Details
Momelotinib
transporter
Solute carrier organic anion transporter family member 1B3
Details
Momelotinib
target
Tyrosine-protein kinase JAK1
Details
Momelotinib
target
Tyrosine-protein kinase JAK2
Details
Momelotinib
target
Tyrosine-protein kinase JAK3
Details
Momelotinib
target
Non-receptor tyrosine-protein kinase TYK2
Details
Spebrutinib
target
Tyrosine-protein kinase BTK
Details
Sarilumab
target
High affinity immunoglobulin gamma Fc receptor I
Details
Sarilumab
target
Low affinity immunoglobulin gamma Fc region receptor II-a
Details
Sarilumab
enzyme
Cytochrome P450 3A4
Details
Sarilumab
target
Low affinity immunoglobulin gamma Fc region receptor II-b
Details
Sarilumab
target
Low affinity immunoglobulin gamma Fc region receptor III-A
Details
Sarilumab
target
Low affinity immunoglobulin gamma Fc region receptor III-B
Details
Sarilumab
target
Interleukin-6 receptor subunit alpha
Details
Talinolol
transporter
P-glycoprotein 1
Details
Talinolol
transporter
Canalicular multispecific organic anion transporter 1
Details
Talinolol
enzyme
Cytochrome P450 2D6
Details
Tremelimumab
target
Cytotoxic T-lymphocyte protein 4
Details
Pilaralisib
target
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform
Details
Pazufloxacin
enzyme
Cytochrome P450 1A2
Details
Danoprevir
enzyme
Cytochrome P450 3A4
Details
Danoprevir
target
Genome polyprotein
Details
Tosedostat
target
Leukotriene A-4 hydrolase
Details
Tosedostat
target
Puromycin-sensitive aminopeptidase
Details
Anisodamine
enzyme
Cytochrome P450 2D6
Details
Capmatinib
target
Hepatocyte growth factor receptor
Details
Displaying targets
25471 - 25500
of
29784
in total
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846
847
848
849
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851
852
853
854
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