At least one prior systemic therapy

DrugDrug NameDrug Description
DB15568AdagrasibA KRAS inhibitor indicated for the treatment of locally advanced or metastatic KRAS G12C-mutated non-small cell lung cancer in patients who have received at least one prior systemic therapy.
DB15149FutibatinibA kinase inhibitor used to treat intrahepatic cholangiocarcinoma in previously treated adults.
DB06176RomidepsinA histone deacetylase (HDAC) inhibitor used to treat cutaneous T-cell lymphoma.
DrugDrug NameTargetType
DB15568AdagrasibGTPase KRastarget
DB15568AdagrasibCytochrome P450 3A4enzyme
DB15568AdagrasibCytochrome P450 2C8enzyme
DB15568AdagrasibCytochrome P450 1A2enzyme
DB15568AdagrasibCytochrome P450 2B6enzyme
DB15568AdagrasibCytochrome P450 2C9enzyme
DB15568AdagrasibCytochrome P450 2D6enzyme
DB15568AdagrasibP-glycoprotein 1transporter
DB15149FutibatinibCytochrome P450 3A4enzyme
DB15149FutibatinibP-glycoprotein 1transporter
DB15149FutibatinibATP-binding cassette sub-family G member 2transporter
DB15149FutibatinibSerum albumincarrier
DB15149FutibatinibAlpha-1-acid glycoprotein 1carrier
DB15149FutibatinibCytochrome P450 2C9enzyme
DB15149FutibatinibCytochrome P450 2D6enzyme
DB15149FutibatinibFibroblast growth factor receptor 1target
DB15149FutibatinibFibroblast growth factor receptor 2target
DB15149FutibatinibFibroblast growth factor receptor 3target
DB15149FutibatinibFibroblast growth factor receptor 4target
DB06176RomidepsinCytochrome P450 3A4enzyme
DB06176RomidepsinCytochrome P450 3A5enzyme
DB06176RomidepsinP-glycoprotein 1transporter
DB06176RomidepsinSolute carrier organic anion transporter family member 1B3transporter
DB06176RomidepsinCytochrome P450 1A1enzyme
DB06176RomidepsinCytochrome P450 2B6enzyme
DB06176RomidepsinCytochrome P450 2C19enzyme
DB06176RomidepsinHistone deacetylase 1target
DB06176RomidepsinHistone deacetylase 2target
DB06176RomidepsinHistone deacetylase 4target
DB06176RomidepsinHistone deacetylase 6target
DB06176RomidepsinMultidrug resistance-associated protein 1target
DB06176RomidepsinBile salt export pumptransporter
DB06176RomidepsinSolute carrier organic anion transporter family member 1B1transporter
DB06176RomidepsinSolute carrier family 22 member 6transporter
DB06176RomidepsinSolute carrier family 22 member 2transporter
DB06176RomidepsinHistone deacetylasetarget
DrugDrug NamePhaseStatusCount