Adrenergics for Systemic Use

Name
Adrenergics for Systemic Use
Accession Number
DBCAT002232
Description

Not Available

ATC Classification
Drugs
DrugDrug Description
TerbutalineA beta-2 adrenergic agonist used as a bronchodilator and to prevent premature labor.
ProcaterolA beta-2 adrenergic receptor agonist and bronchodilator used for the treatment of asthma and chronic obstructive pulmonary disease (COPD).
BambuterolA long acting beta2-adrenoceptor agonist for the management of lung diseases associated with bronchospasm.
TulobuterolAn inhaled long-acting beta2-adrenergic receptor agonist used as a bronchodilator in the management of asthma and COPD.
MethoxyphenamineNot Annotated
CarbuterolNot Annotated
OrciprenalineA beta-2 adrenergic agonist used to treat bronchospasm, asthma, and COPD.
IsoprenalineA catecholamine non-selective beta-adrenergic agonist typically used to treat bradycardia and heart block.
FenoterolA beta-2 adrenergic agonist and bronchodilator used for the symptomatic treatment of asthma.
PirbuterolA beta-2 adrenergic agonist and bronchodilator used for the symptomatic treatment of asthma.
EphedrineAn alpha and beta-adrenergic agonist indicated to treat hypotension under anesthesia, allergic conditions, bronchial asthma, and nasal congestion.
ClenbuterolA decongestant and bronchodilator used in a variety of respiratory conditions.
HexoprenalineHexoprenaline is a stimulant of beta 2 adrenergic receptors. It is used as a bronchodilator, antiasthmatic, and tocolytic agent.
ReproterolA short-acting β2 adrenoreceptor agonist used to treat various types of asthma including allergic asthma, non-allergic asthma, and exercise-induced asthma.
TretoquinolNot Annotated
AmbroxolA medication indicated for airway secretion clearance therapy.
FormoterolAn inhaled long-acting beta2-adrenergic receptor agonist used as a bronchodilator in the management of asthma and COPD.
IsoetharineFor the treatment of asthma, wheezing, and chronic asthmatic bronchitis.
Drugs & Drug Targets
DrugTargetType
TerbutalineBeta-2 adrenergic receptortarget
TerbutalineCholinesteraseenzyme
TerbutalineBeta-3 adrenergic receptortarget
TerbutalineBeta-1 adrenergic receptortarget
TerbutalineSulfotransferaseenzyme
TerbutalineUDP-glucuronosyltransferases (UGTs)enzyme
TerbutalineSolute carrier family 22 member 5transporter
TerbutalineSolute carrier family 22 member 2transporter
ProcaterolBeta-2 adrenergic receptortarget
BambuterolBeta-2 adrenergic receptortarget
BambuterolCholinesteraseenzyme
BambuterolCholinesterasetarget
TulobuterolBeta-2 adrenergic receptortarget
MethoxyphenamineBeta-2 adrenergic receptortarget
OrciprenalineBeta-2 adrenergic receptortarget
IsoprenalineBeta-1 adrenergic receptortarget
IsoprenalineBeta-2 adrenergic receptortarget
IsoprenalineBeta-3 adrenergic receptortarget
IsoprenalineCytochrome P450 1A1enzyme
IsoprenalineSuperoxide dismutase [Cu-Zn]target
IsoprenalineCytochrome P450 1B1enzyme
IsoprenalineSerum albumincarrier
IsoprenalineCatechol O-methyltransferaseenzyme
IsoprenalineCholinesteraseenzyme
FenoterolBeta-2 adrenergic receptortarget
FenoterolBeta-1 adrenergic receptortarget
FenoterolBeta-3 adrenergic receptortarget
PirbuterolBeta-2 adrenergic receptortarget
PirbuterolBeta-1 adrenergic receptortarget
EphedrineAlpha-1A adrenergic receptortarget
EphedrineSodium-dependent noradrenaline transportertarget
EphedrineCholinesteraseenzyme
EphedrineSerum albumincarrier
EphedrineBeta-1 adrenergic receptortarget
EphedrineBeta-2 adrenergic receptortarget
EphedrineSynaptic vesicular amine transportertransporter
EphedrineAcetylcholinesteraseenzyme
ClenbuterolBeta-2 adrenergic receptortarget
ClenbuterolBeta-nerve growth factortarget
ClenbuterolTumor necrosis factortarget
ClenbuterolBeta-1 adrenergic receptortarget
ClenbuterolBeta-3 adrenergic receptortarget
ClenbuterolCytochrome P450 1A1enzyme
AmbroxolCytochrome P450 3A4enzyme
FormoterolBeta-2 adrenergic receptortarget
FormoterolBeta-1 adrenergic receptortarget
FormoterolBeta-3 adrenergic receptortarget
FormoterolCytochrome P450 2D6enzyme
FormoterolCytochrome P450 2C19enzyme
FormoterolCytochrome P450 2C9enzyme
FormoterolCytochrome P450 2A6enzyme
FormoterolUDP-glucuronosyltransferase 1A1enzyme
FormoterolUDP-glucuronosyltransferase 1-8enzyme
FormoterolUDP-glucuronosyltransferase 1-9enzyme
FormoterolUDP-glucuronosyltransferase 2B7enzyme
FormoterolUDP-glucuronosyltransferase 2B15enzyme
FormoterolSolute carrier family 22 member 1transporter
FormoterolSolute carrier family 22 member 4transporter
FormoterolSolute carrier family 22 member 5transporter
FormoterolSolute carrier family 22 member 3transporter
FormoterolSerum albumincarrier
IsoetharineBeta-1 adrenergic receptortarget
IsoetharineBeta-2 adrenergic receptortarget