The Future of Drug Discovery: Tackling the Undruggable with New Biotechnologies
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Displaying targets
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Drug Name
Type
Name
target
enzyme
carrier
transporter
Clear
Tetrodotoxin
target
Sodium channel protein type 8 subunit alpha
Details
Tetrodotoxin
target
Sodium channel protein type 5 subunit alpha
Details
AP1081
target
Estrogen receptor
Details
LGD2941
target
Androgen receptor
Details
NRP409
target
Thyroid hormone receptor alpha
Details
NRP409
carrier
Transthyretin
Details
NRP409
carrier
Thyroxine-binding globulin
Details
NRP409
target
Ketimine reductase mu-crystallin
Details
Cobimetinib
transporter
Solute carrier organic anion transporter family member 1B3
Details
Cobimetinib
enzyme
Cytochrome P450 3A5
Details
Cobimetinib
carrier
Alpha-1-acid glycoprotein 1
Details
Cobimetinib
target
Dual specificity mitogen-activated protein kinase kinase 1
Details
Cobimetinib
transporter
ATP-dependent translocase ABCB1
Details
Cobimetinib
enzyme
Cytochrome P450 3A4
Details
Cobimetinib
transporter
Solute carrier organic anion transporter family member 1B1
Details
Cobimetinib
transporter
Broad substrate specificity ATP-binding cassette transporter ABCG2
Details
Cobimetinib
enzyme
UDP-glucuronosyltransferase 2B7
Details
Cobimetinib
enzyme
Cytochrome P450 2D6
Details
XL765
target
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform
Details
XL765
target
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform
Details
XL765
target
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform
Details
XL765
target
Serine/threonine-protein kinase mTOR
Details
XL765
target
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform
Details
XL019
target
Tyrosine-protein kinase JAK2
Details
Silver sulfadiazine
target
Dihydropteroate synthase
Details
Silver sulfadiazine
target
DNA
Details
Methsuximide
enzyme
Cytochrome P450 2C19
Details
Methsuximide
target
Voltage-dependent T-type calcium channel subunit alpha-1G
Details
FavId
target
Granulocyte colony-stimulating factor receptor
Details
Fenoxaprop-ethyl
target
Nitric oxide synthase, inducible
Details
Displaying targets
18901 - 18930
of
33504
in total
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