The Future of Drug Discovery: Tackling the Undruggable with New Biotechnologies
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Drug Name
Type
Name
target
enzyme
carrier
transporter
Clear
Nicaraven
target
Poly [ADP-ribose] polymerase 1
Details
Bazedoxifene
target
Estrogen receptor
Details
Bazedoxifene
enzyme
UDP-glucuronosyltransferase 1A4
Details
Bazedoxifene
target
Estrogen receptor beta
Details
Bazedoxifene
enzyme
UDP-glucuronosyltransferase 1A8
Details
Bazedoxifene
enzyme
UDP-glucuronosyltransferase 1A10
Details
Telavancin
target
Neuronal acetylcholine receptor subunit alpha-2
Details
Telavancin
target
Corticotropin-releasing factor receptor 1
Details
Telavancin
target
Neuronal acetylcholine receptor subunit alpha-3
Details
Ambrisentan
enzyme
Cytochrome P450 3A4
Details
Ambrisentan
enzyme
UDP-glucuronosyltransferase 1A9
Details
Ambrisentan
enzyme
UDP-glucuronosyltransferase 1A3
Details
Ambrisentan
transporter
Solute carrier organic anion transporter family member 1B1
Details
Ambrisentan
target
Endothelin receptor type B
Details
Ambrisentan
target
Endothelin-1 receptor
Details
Ambrisentan
enzyme
UDP-glucuronosyltransferase 2B7
Details
Ambrisentan
transporter
Solute carrier organic anion transporter family member 1B3
Details
Ambrisentan
enzyme
Cytochrome P450 3A5
Details
Ambrisentan
enzyme
Cytochrome P450 2C19
Details
Ambrisentan
transporter
ATP-dependent translocase ABCB1
Details
Human C1-esterase inhibitor
target
Plasma kallikrein
Details
Human C1-esterase inhibitor
target
Tissue-type plasminogen activator
Details
Human C1-esterase inhibitor
target
Complement C1r subcomponent
Details
Human C1-esterase inhibitor
target
Complement C1s subcomponent
Details
Human C1-esterase inhibitor
target
Coagulation factor XII
Details
Human C1-esterase inhibitor
target
Prothrombin
Details
Human C1-esterase inhibitor
target
Coagulation factor XI
Details
Idraparinux
target
Coagulation factor X
Details
Taribavirin
target
RNA-directed RNA polymerase L
Details
Taribavirin
target
Inosine-5'-monophosphate dehydrogenase 1
Details
Displaying targets
20221 - 20250
of
33504
in total
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