The Future of Drug Discovery: Tackling the Undruggable with New Biotechnologies
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Drug Name
Type
Name
target
enzyme
carrier
transporter
Clear
Bisegliptin
target
Dipeptidyl peptidase 4
Details
Dimethylcurcumin
target
Androgen receptor
Details
SNS-314
target
Aurora kinase A
Details
SNS-314
target
Aurora kinase C
Details
SNS-314
target
Aurora kinase B
Details
Tirbanibulin
target
Tubulin beta chain
Details
Tirbanibulin
enzyme
Cytochrome P450 2B6
Details
Tirbanibulin
enzyme
Cytochrome P450 2D6
Details
Tirbanibulin
transporter
Solute carrier family 22 member 1
Details
Tirbanibulin
transporter
Solute carrier family 22 member 2
Details
Tirbanibulin
enzyme
Cytochrome P450 2C9
Details
Tirbanibulin
transporter
Multidrug and toxin extrusion protein 2
Details
Tirbanibulin
transporter
Solute carrier organic anion transporter family member 1B1
Details
Tirbanibulin
transporter
Solute carrier organic anion transporter family member 1B3
Details
Tirbanibulin
target
Proto-oncogene tyrosine-protein kinase Src
Details
Tirbanibulin
enzyme
Cytochrome P450 3A4
Details
Tirbanibulin
enzyme
Cytochrome P450 2C8
Details
Tirbanibulin
enzyme
Cytochrome P450 1A2
Details
Tirbanibulin
enzyme
Cytochrome P450 2C19
Details
Tirbanibulin
transporter
Multidrug and toxin extrusion protein 1
Details
IRL-1620
target
Endothelin receptor type B
Details
SUVN-502
target
5-hydroxytryptamine receptor 6
Details
Sertindole
target
Alpha-1A adrenergic receptor
Details
Sertindole
target
Alpha-1B adrenergic receptor
Details
Sertindole
target
Alpha-1D adrenergic receptor
Details
Sertindole
target
5-hydroxytryptamine receptor 6
Details
Sertindole
enzyme
Cytochrome P450 2D6
Details
Sertindole
target
D(2) dopamine receptor
Details
Sertindole
target
Voltage-gated inwardly rectifying potassium channel KCNH2
Details
Sertindole
target
5-hydroxytryptamine receptor 2A
Details
Displaying targets
19681 - 19710
of
33504
in total
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