Coagulants

Name
Coagulants
Accession Number
DBCAT000113
Description

Agents that cause clotting.

Drugs
DrugDrug Description
AdrenaloneNot Annotated
AminaphthoneA medication that inhibits erythrocyte aggregation in capillaries, improving venous return for the treatment of capillary fragility.
Aminocaproic acidAn antifibrinolytic agent used to induce clotting postoperatively.
Andexanet alfaA recombinant Factor Xa used to reverse anticoagulation caused by rivaroxaban and apixaban.
AnivamersenAnivamersen is under investigation in clinical trial NCT01848106 (A Study to Determine the Efficacy and Safety of REG1 Compared to Bivalirudin in Patients Undergoing PCI).
Anti-inhibitor coagulant complexA medication used to control bleeding episodes and prevent bleeding episodes in hemophilia A and B.
Antihemophilic factor humanA Factor VIII replacement therapy used to treat hemophilia A.
AprotininA serine protease inhibitor used to reduce the risk for perioperative blood loss and the need for blood transfusion in high-risk patients during cardiopulmonary bypass for coronary artery bypass graft surgery.
BatroxobinNo approved indications. Batroxobin is a defibrongenating agent which has been observed to reduce fibrinogen levels and thus reduce clot risk when used intravenously.
Beroctocog alfaBeroctocog alfa is indicated for the prevention and control of bleeding in patients with hemophilia A or acquired Factor VIII (FVIII) deficiency. It is also indicated for surgical/invasive procedures in...
Bismuth subgallateA medication used to deodorize flatulence and stools as well as hemostasis in soft tissue surgery.
CarbazochromeIndicated for capillary and parenchymal hemorrhage (trauma, tonsillectomy, during surgery), intestinal bleeding, and thrombocytopenic purpura.
Carbazochrome sulfonic acidA hemostatic agent indicated to treat bleeding in capillary fragility.
DesmopressinA synthetic vasopressin (antidiuretic hormone) analog and $V_2$ receptor agonist used as replacement therapy for central diabetes insipidus, and as a prohemostatic agent to increase Factor VIII and von Willebrand factor levels in patients with Hemophilia A or Type 1 von Willebrand disease.
Dobesilic acidA medication indicated in the treatment of hemorrhoids, venous insufficiency, and other microangiopathies.
EtamsylateA hemostatic agent that acts by restoring capillary resistance and improving platelet adhesion.
Ferric subsulfateFerric subsulfate is a stypic or hemostatic agent that causes agglutination of surface proteins resulting in local hemostasis. It has the chemical formula Fe4(OH)2(SO4)5. It is used after superficial skin...
KallidinogenaseNot Annotated
LypressinNot Annotated
MenadioneThe primary known function of vitamin K is to assist in the normal clotting of blood, but it may also play a role in normal bone calcification.
Menadione bisulfiteNot Annotated
MenaquinoneMenaquinone is under investigation in clinical trial NCT01533441 (Vitamin K2 Intervention in Patients With Vitamin K Antagonists).
Menaquinone 6Menaquinone 6 is under investigation in clinical trial NCT01194778 (Comparison of Efficacy of Different Dosages Vitamin K2).
Menaquinone 7Menaquinone 7 is under investigation in clinical trial NCT00402974 (The Effect of Vitamin K Supplementation on Osteocalcin Carboxylation in Healthy Children).
MenatetrenoneA form of vitamin K2 which is used in the treatment of osteoporosis to stimulate osteogenesis.
NaftazoneA naphthoquinone derivative indicated in the treatment of varicose veins, hemorrhoids, and superficial thrombophlebitis.
OrnipressinNot Annotated
Oxidized celluloseNot Annotated
PhylloquinoneA fat soluble vitamin used to treat hemorrhagic conditions in infants and coumarin overdoses.
PoliglusamPoliglusam, or chitosan, is a linear polysaccharide consisting of D-glucosamine and N-acetyl-D-glucosamine. Naturally-occuring poliglusam is found in the cell walls of fungi, soil and sediments where it is produced from...
Potassium triiodideNot Annotated
ProtamineA heparin antagonist indicated in the treatment of heparin overdoses, to counteract heparins preoperatively, or during cardiac surgery and dialysis.
Rurioctocog alfa pegolA pegylated recombinant human coagulation factor VIII used to treat and prevent bleeding episodes in patients 12 years and above with hemophilia A.
ThrombinA coagulation factor used to stop bleeding during surgery.
Tranexamic acidAn antifibrinolytic used to reduce or prevent hemorrhagic episodes, especially in the context of hyperfibrinolytic disorders.
VasopressinA peptide hormone used to increase blood pressure in patients with vasodilatory shock who are resistant to fluid and catecholamine therapy.
Drugs & Drug Targets
DrugTargetType
AdrenaloneDopamine beta-hydroxylasetarget
Aminocaproic acidPlasminogentarget
Aminocaproic acidTissue-type plasminogen activatortarget
Aminocaproic acidApolipoprotein(a)target
Aminocaproic acidAldehyde oxidaseenzyme
Andexanet alfaTissue factor pathway inhibitortarget
Anti-inhibitor coagulant complexCoagulation factor XIII A chaintarget
Anti-inhibitor coagulant complexCoagulation factor VIItarget
Anti-inhibitor coagulant complexCoagulation factor VIIItarget
Anti-inhibitor coagulant complexCoagulation factor Vtarget
Anti-inhibitor coagulant complexFibrinogen beta chaintarget
Anti-inhibitor coagulant complexFibrinogen alpha chaintarget
Anti-inhibitor coagulant complexProthrombintarget
Anti-inhibitor coagulant complexCoagulation factor Xtarget
Antihemophilic factor humanCoagulation factor Xtarget
Antihemophilic factor humanCoagulation factor IXtarget
Antihemophilic factor humanVitamin K-dependent protein Cenzyme
AprotininPlasma kallikreintarget
AprotininCholinesteraseenzyme
AprotininKallikrein-1target
AprotininPlasminogentarget
AprotininChymotrypsinogen Btarget
AprotininSerine protease 1target
BatroxobinCoagulation factor Xtarget
BatroxobinFibrinogentarget
Beroctocog alfavon Willebrand factorcarrier
Beroctocog alfaCoagulation factor VIIItarget
Bismuth subgallateAlbumincarrier
Bismuth subgallateCoagulation factor XIItarget
CarbazochromeCytochrome P450 3A4enzyme
CarbazochromeRibosyldihydronicotinamide dehydrogenase [quinone]enzyme
CarbazochromeNADPH--cytochrome P450 reductaseenzyme
CarbazochromeGlutathione S-transferase Mu 2enzyme
CarbazochromeGlutathione S-transferase Mu 1enzyme
DesmopressinVasopressin V1a receptortarget
DesmopressinOxytocin receptortarget
DesmopressinProstaglandin G/H synthase 2enzyme
DesmopressinProstaglandin G/H synthase 1enzyme
DesmopressinVasopressin V1b receptortarget
DesmopressinVasopressin V2 receptortarget
Dobesilic acidVascular endothelial growth factor receptor 2target
Dobesilic acidSpike glycoproteintarget
EtamsylateFibroblast growth factor 2target
KallidinogenaseKininogen-1target
LypressinATP-binding cassette sub-family C member 2transporter
LypressinVasopressin V1b receptortarget
LypressinVasopressin V2 receptortarget
LypressinVasopressin V1a receptortarget
MenadioneCytochrome P450 2C9enzyme
MenadioneCytochrome P450 2C19enzyme
MenadioneCytochrome P450 2D6enzyme
MenadioneCytochrome P450 2C8enzyme
MenadioneCytochrome P450 2B6enzyme
MenadioneCytochrome P450 1B1enzyme
MenadioneCytochrome P450 2A6enzyme
MenadioneCytochrome P450 3A5enzyme
MenadioneOsteocalcintarget
MenadioneCytochrome P450 1A1enzyme
MenadioneCytochrome P450 3A4enzyme
MenadioneMethylenetetrahydrofolate reductase (NADPH)enzyme
MenadioneAldehyde oxidaseenzyme
MenadioneXanthine dehydrogenase/oxidaseenzyme
MenadioneVitamin K epoxide reductase complex subunit 1-like protein 1target
MenadioneRibosyldihydronicotinamide dehydrogenase [quinone]target
MenadioneNAD(P)H dehydrogenase [quinone] 1target
MenadioneCytochrome P450 2E1enzyme
MenadioneAldehyde oxidasetarget
MenadioneVitamin K-dependent protein Starget
MenadioneVitamin K-dependent protein Ctarget
MenadioneVitamin K-dependent gamma-carboxylasetarget
MenadioneCoagulation factor IXtarget
MenadioneVitamin K epoxide reductase complex subunit 1target
MenadioneProthrombintarget
MenadioneCytochrome P450 3A7enzyme
MenadioneCytochrome P450 1A2enzyme
Menadione bisulfiteCarbonyl reductases (CBRs)enzyme
Menadione bisulfiteCarbonyl reductase [NADPH] 1enzyme
MenaquinoneSuccinate dehydrogenaseenzyme
MenaquinoneSulfide-quinone reductaseenzyme
Menaquinone 6Cruzipaintarget
Menaquinone 7Nuclear factor NF-kappa-Btarget
MenatetrenoneCruzipaintarget
NaftazoneUDP-glucuronosyltransferase 1A6enzyme
OrnipressinVasopressin V1a receptortarget
PhylloquinoneProthrombintarget
PhylloquinoneVitamin K epoxide reductase complex subunit 1enzyme
PhylloquinoneUbiA prenyltransferase domain-containing protein 1enzyme
PhylloquinoneCytochrome P450 4F2enzyme
PhylloquinoneOsteocalcintarget
PhylloquinoneVitamin K-dependent gamma-carboxylasetarget
Potassium triiodideThymidylate synthasetarget
ProtamineExtracellular calcium-sensing receptortarget
ProtamineTryptase beta-2target
ProtamineHeparan sulfatetarget
ProtamineProthrombintarget
ProtamineTissue factortarget
ProtamineCoagulation factor VIItarget
ProtamineLaminin subunit alpha-3enzyme
Rurioctocog alfa pegolCoagulation factor VIIItarget
Rurioctocog alfa pegolvon Willebrand factortarget
ThrombinFibrinogen alpha chaintarget
ThrombinFibrinogen beta chaintarget
ThrombinFibrinogen gamma chaintarget
ThrombinCoagulation factor Vtarget
ThrombinCoagulation factor VIIItarget
ThrombinCoagulation factor XIII A chaintarget
ThrombinCoagulation factor XItarget
ThrombinCoagulation factor XIII B chaintarget
ThrombinProteinase-activated receptor 4target
ThrombinProteinase-activated receptor 1target
Tranexamic acidPlasminogentarget
VasopressinVasopressin V2 receptortarget
VasopressinOxytocin receptortarget
VasopressinATP-binding cassette sub-family C member 2transporter
VasopressinVasopressin V1a receptortarget
VasopressinVasopressin V1b receptortarget