Chelating Agents

Name
Chelating Agents
Accession Number
DBCAT000624
Description

Chemicals that bind to and remove ions from solutions. Many chelating agents function through the formation of COORDINATION COMPLEXES with METALS.

Drugs
DrugDrug Description
1,10-PhenanthrolineNot Available
2,3-Dimercapto-1-propanesulfonic acidNot Annotated
ActeosideActeoside is under investigation in clinical trial NCT02662283 (Validity and Security of Reh-acteoside Therapy for Patients of IgA Nephropathy).
AlanosineInvestigated for use/treatment in brain cancer and cancer/tumors (unspecified).
Ammonium tetrathiomolybdateNot Annotated
Calcium acetateA phosphate binder used in patients with end-stage renal disease (ESRD) to prevent elevated phosphate levels and resulting ectopic calcification and secondary hyperparathyroidism.
CefiderocolA cephalosporin antibiotic used in complicated urinary tract infections.
Citric acidAn anti-chelation additive used in blood collection tubes and as a flavoring and preservative agent in various cosmetic and pharmaceutical products.
DeferasiroxAn iron chelator used to treat chronic iron overload caused by blood transfusions. Also used in patients with non-transfusion-dependent thalassemia syndromes, and in patients with elevated liver iron concentration and serum ferritin.
DeferiproneAn iron chelator used to treat patients with transfusional iron overload caused by thalassemia syndromes.
DeferoxamineA chelating agent used to treat iron or aluminum toxicity and some blood transfusion dependent anemias.
DimercaprolA chelating agent used as an antidote to arsenic, gold, and mercury poisoning, as well as acute lead poisoning in combination with edetate calcium disodium.
Dimercaptosuccinic acidNot Annotated
Dipicolinic acidNot Available
DitiocarbA chelating agent that has been used to mobilize toxic metals from the tissues of man and experimental animals. It is the main metabolite of DISULFIRAM.
Ditiocarb zincDitiocarb Zinc is approved for use within allergenic epicutaneous patch tests which are indicated for use as an aid in the diagnosis of allergic contact dermatitis (ACD) in persons 6...
Edetate calcium disodium anhydrousA chelating agent used to treat lead poisoning.
Edetate disodium anhydrousA polyvalent ion chelator indicated for emergency treatment of hypercalcemia and digitalis toxicity associated ventricular arrhythmias.
Edetic acidA chelating agent used to treat mercury and lead toxicity and some blood transfusion dependent anemias.
Egtazic acidEgtazic acid is a small molecule drug. Egtazic acid has a monoisotopic molecular weight of 380.14 Da.
EmeramideEmeramide has been used in trials studying the treatment of Mercury Poisoning.
Gadoteric acidA gadolinium-based contrast agent (GBCA) used with contrasted magnetic resonance imaging (MRI) to detect and visualize lesions and abnormal vascularity.
Gluconic AcidAn electrolyte supplement used in total parenteral nutrition.
L-tartaric acidTartaric Acid is primarily indicated in conditions like Antiscorbutic, Antiseptic.
Nitrilotriacetic acidNitrilotriacetic acid is a derivative of acetic acid, N(CH2COOH)3. It is a complexing (sequestering) agent that forms stable complexes with Zn2+. (From Miall's Dictionary of Chemistry, 5th ed.)
PenicillamineA chelator used to treat Wilson's disease, cystinuria, and rheumatoid arthritis.
Pentetic acidDTPA is widely used in industry and medicine. As a medical agent, it is approved for its use in medical imaging and for the decorporation of internally deposited radionuclides. It...
Picolinic acidInvestigated for use/treatment in acne, herpes labialis infections (cold sores), and venereal disease.
PoliglusamPoliglusam, or chitosan, is a linear polysaccharide consisting of D-glucosamine and N-acetyl-D-glucosamine. Naturally-occuring poliglusam is found in the cell walls of fungi, soil and sediments where it is produced from...
SevelamerA phosphate binder used to treat hyperphosphatemia.
SuccimerA mercaptodicarboxylic acid heavy metal chelator used in the treatment of heavy metal poisoning.
TagatoseIntended for use as a therapeutic adjunct in the treatment of type II diabetes.
TetrathiomolybdateInvestigated for use/treatment in liver disease and pulmonary fibrosis.
ThenoyltrifluoroacetoneThenoyltrifluoroacetone is a chelating agent and inhibitor of cellular respiration.
Thiosulfuric acidA sulfur donor used sequentially with sodium nitrite for the reversal of life-threatening acute cyanide poisoning. Also used to reduce the risk of ototoxicity associated with cisplatin.
TolevamerA potassium-binding resin used in the treatment of hyperkalemia.
TriethylenetetramineA copper chelating agent used for the management of Wilson's disease in cases where penicillamine therapy is clinically inappropriate.
Drugs & Drug Targets
DrugTargetType
1,10-PhenanthrolineMetallo-beta-lactamase L1 type 3target
1,10-PhenanthrolineMethyl-accepting chemotaxis protein IItarget
2,3-Dimercapto-1-propanesulfonic acidDelta-aminolevulinic acid dehydratasetarget
2,3-Dimercapto-1-propanesulfonic acidAngiotensin-converting enzymetarget
2,3-Dimercapto-1-propanesulfonic acidAngiotensin-converting enzymeenzyme
2,3-Dimercapto-1-propanesulfonic acidNa(+)/dicarboxylate cotransporter 3transporter
2,3-Dimercapto-1-propanesulfonic acidDelta-aminolevulinic acid dehydrataseenzyme
2,3-Dimercapto-1-propanesulfonic acidATP-binding cassette sub-family C member 2transporter
2,3-Dimercapto-1-propanesulfonic acidOrganic anion transporter 3transporter
2,3-Dimercapto-1-propanesulfonic acidSolute carrier family 22 member 6transporter
ActeosideProtein kinase C alpha typetarget
AlanosineCystine/glutamate transportertransporter
AlanosineAdenylosuccinate synthetase isozyme 1target
AlanosineAdenylosuccinate synthetase isozyme 2target
AlanosineAspartate carbamoyltransferase catalytic subunittarget
Ammonium tetrathiomolybdateSuperoxide dismutase [Cu-Zn]target
Calcium acetatePhosphatetarget
CefiderocolPenicillin-binding proteintarget
CefiderocolOuter membrane ferric siderophore receptortransporter
CefiderocolColicin I receptortransporter
CefiderocolCatecholate siderophore receptor Fiutransporter
CefiderocolAlbumincarrier
CefiderocolMexAB-OprM efflux systemtransporter
CefiderocolD-alanyl-D-alanine carboxypeptidase DacBtarget
CefiderocolPeptidoglycan D,D-transpeptidase MrdAtarget
CefiderocolPenicillin-binding protein 1Btarget
CefiderocolPenicillin-binding protein 1Atarget
CefiderocolPeptidoglycan D,D-transpeptidase FtsItarget
Citric acidSAR-endolysintarget
Citric acidLanosterol 14-alpha demethylasetarget
Citric acidTransient receptor potential cation channel subfamily V member 4target
Citric acidMetallo-beta-lactamase type 2target
Citric acidSolute carrier organic anion transporter family member 2B1transporter
Citric acidPyruvate decarboxylasetarget
Citric acid3-carboxy-cis,cis-muconate cycloisomerasetarget
Citric acidGlycerol uptake operon antiterminator-related proteintarget
Citric acidInosine triphosphate pyrophosphatasetarget
Citric acidGMP synthase [glutamine-hydrolyzing]target
Citric acidRibose-5-phosphate isomerase Atarget
Citric acidPeptidoglycan editing factor PgeFtarget
Citric acidGlyoxalase family proteintarget
Citric acidGlucose-1-phosphate thymidylyltransferasetarget
Citric acidMetallo-beta-lactamase type 2target
Citric acidAldo-keto reductase family 1 member B1target
Citric acidCitrate synthase, mitochondrialtarget
Citric acidProto-oncogene tyrosine-protein kinase Srctarget
Citric acidRibonuclease pancreatictarget
Citric acidIsocitrate dehydrogenase [NADP]target
Citric acidEosinophil cationic proteintarget
Citric acidBeta-lactamasetarget
Citric acidFumarate hydratase class IItarget
Citric acid6-phosphogluconolactonasetarget
Citric acidL-amino-acid oxidasetarget
Citric acidCarboxy-terminal domain RNA polymerase II polypeptide A small phosphatase 1target
Citric acidCytochrome c peroxidasetarget
Citric acidHepatocyte growth factor-regulated tyrosine kinase substratetarget
Citric acidInvasintarget
Citric acidIntron-associated endonuclease 1target
Citric acidShort tail fiber protein gp12target
Citric acidMalate dehydrogenase, mitochondrialtarget
Citric acidN5-carboxyaminoimidazole ribonucleotide mutasetarget
Citric acidLarge ribosomal subunit protein uL4target
Citric acidCarboxypeptidase Btarget
Citric acidHexon proteintarget
Citric acidRiboflavin biosynthesis proteintarget
Citric acidBeta-fructosidasetarget
Citric acidStringent starvation protein Atarget
Citric acidCitrate synthasetarget
Citric acidRNA 3'-terminal phosphate cyclasetarget
Citric acidU6 snRNA-associated Sm-like protein LSm6target
Citric acidPleckstrin homology domain-containing family A member 1target
Citric acidFe(3+)-binding periplasmic proteintarget
Citric acidSignal recognition particle receptor FtsYtarget
Citric acidNicotinate-nucleotide adenylyltransferasetarget
Citric acidTranscription antitermination protein NusBtarget
Citric acidComplement component C8 gamma chaintarget
Citric acidRibonucleoside-diphosphate reductase subunit betatarget
Citric acidGlutamine synthetase 1target
Citric acid2-methylcitrate synthasetarget
Citric acid9,11-endoperoxide prostaglandin H2 reductasetarget
Citric acidAdenine phosphoribosyltransferasetarget
DeferasiroxUDP-glucuronosyltransferase 1A1enzyme
DeferasiroxCytochrome P450 3A4enzyme
DeferasiroxCytochrome P450 1A2enzyme
DeferasiroxUDP-glucuronosyltransferase 1A9enzyme
DeferasiroxCytochrome P450 2C8enzyme
DeferasiroxIrontarget
DeferasiroxUDP-glucuronosyltransferase 1A3enzyme
DeferiproneIrontarget
DeferiproneUDP-glucuronosyltransferase 1A6enzyme
DeferoxamineXanthine dehydrogenase/oxidaseenzyme
DeferoxamineIrontarget
DeferoxamineAluminumtarget
DeferoxamineAmyloid-beta precursor proteintarget
DimercaprolLeadtarget
DimercaprolMercurytarget
DimercaprolCadmiumtarget
DimercaprolArsenictarget
Dimercaptosuccinic acidMercurytarget
Dimercaptosuccinic acidArsenictarget
Dipicolinic acid4-hydroxy-tetrahydrodipicolinate reductasetarget
Dipicolinic acid4-hydroxy-tetrahydrodipicolinate reductasetarget
DitiocarbCytochrome P450 2E1enzyme
DitiocarbCytochrome P450 3A4enzyme
DitiocarbCytochrome P450 3A5enzyme
DitiocarbDopamine beta-hydroxylasetarget
DitiocarbSuperoxide dismutase [Cu-Zn]target
DitiocarbTyrosinasetarget
DitiocarbCytochrome P450 2A6enzyme
DitiocarbCatalasetarget
Ditiocarb zincSuperoxide dismutase [Cu-Zn]target
Ditiocarb zincDopamine beta-hydroxylasetarget
Ditiocarb zincCytochrome P450 2A6target
Ditiocarb zincCytochrome P450 2E1target
Ditiocarb zincMetal regulatory transcription factor 1target
Edetate calcium disodium anhydrousSerum paraoxonase/arylesterase 1enzyme
Edetate calcium disodium anhydrousCytochrome P450 3A4enzyme
Edetate calcium disodium anhydrousAromataseenzyme
Edetate calcium disodium anhydrousSerum paraoxonase/lactonase 3enzyme
Edetate calcium disodium anhydrousAdenosine deaminaseenzyme
Edetate calcium disodium anhydrousLeadtarget
Edetate calcium disodium anhydrousIrontarget
Edetate calcium disodium anhydrousManganese cationtarget
Edetate disodium anhydrousLeadtarget
Edetate disodium anhydrousIrontarget
Edetate disodium anhydrousManganese cationtarget
Edetate disodium anhydrousAdenosine deaminaseenzyme
Edetate disodium anhydrousSerum paraoxonase/lactonase 3enzyme
Edetate disodium anhydrousAromataseenzyme
Edetate disodium anhydrousCytochrome P450 3A4enzyme
Edetate disodium anhydrousSerum paraoxonase/arylesterase 1enzyme
Edetic acidSerum paraoxonase/lactonase 3enzyme
Edetic acidLeadtarget
Edetic acidIrontarget
Edetic acidManganese cationtarget
Edetic acidAdenosine deaminaseenzyme
Edetic acidAromataseenzyme
Egtazic acidCalcium ionstarget
EmeramideMercurytarget
Gadoteric acidE3 ubiquitin-protein ligase XIAPtarget
Gluconic AcidAldo-keto reductase family 1 member B1target
Gluconic AcidQuinoprotein glucose dehydrogenase Benzyme
L-tartaric acidBeta-glucuronidasetarget
L-tartaric acidProstatic acid phosphatasetarget
Nitrilotriacetic acidLactotransferrintarget
PenicillamineSolute carrier organic anion transporter family member 1B1transporter
PenicillamineCoppertarget
PenicillamineCystinetarget
Pentetic acidAlpha-1-antitrypsincarrier
Pentetic acidTransuranium elementstarget
Picolinic acidE3 ubiquitin-protein ligase UBR4target
Picolinic acidZinc finger Y-chromosomal proteintarget
SevelamerPhosphatetarget
SuccimerLeadtarget
SuccimerMercurytarget
SuccimerCadmiumtarget
SuccimerArsenictarget
TagatoseD-galactose/methyl-galactoside binding periplasmic protein MglBtransporter
TetrathiomolybdateSuperoxide dismutase [Cu-Zn]target
TetrathiomolybdateAmyloid-beta precursor proteintarget
ThenoyltrifluoroacetoneLiver carboxylesterase 1target
ThenoyltrifluoroacetoneSuccinate dehydrogenase [ubiquinone] flavoprotein subunit, mitochondrialtarget
Thiosulfuric acidThiosulfate sulfurtransferasetarget
Thiosulfuric acid3-mercaptopyruvate sulfurtransferaseenzyme
Thiosulfuric acidCytochrome P450 1A1enzyme
Thiosulfuric acidCytochrome P450 2B6enzyme
Thiosulfuric acidThiosulfate sulfurtransferaseenzyme
Thiosulfuric acidThiosulfate:glutathione sulfurtransferaseenzyme
Thiosulfuric acidSolute carrier family 13 member 4transporter
TolevamerPotassiumtarget
TolevamerToxin Atarget
TolevamerToxin Btarget
TriethylenetetramineCarbonic anhydrase 14target
TriethylenetetramineDiamine acetyltransferase 1enzyme