At least one prior therapy

DrugDrug NameDrug Description
DB08889CarfilzomibA proteasome inhibitor used either alone or in conjunction with a chemotherapy regimen to treat patients with relapsed or refractory multiple myeloma.
DB08904Certolizumab pegolA tumor necrosis factor (TNF) blocker used to treat a variety of autoimmune and autoinflammatory conditions like Crohn's disease, rheumatoid arthritis, active psoriatic arthritis, ankylosing spondylitis, axial spondyloarthritis, and plaque psoriasis.
DB00002CetuximabAn endothelial growth factor receptor binding fragment used to treat colorectal cancer as well as squamous cell carcinoma of the head and neck.
DB09331DaratumumabA CD38-directed cytolytic antibody used alone or as an adjunct drug in the treatment of multiple myeloma and light chain amyloidosis.
DB16581DarvadstrocelA mesenchymal stem cell advanced therapy used to treat complex perianal fistulas in adults with non-active or mildly active luminal Crohn’s disease after an inadequate response to at least one standard treatments.
DB00997DoxorubicinA medication used to treat various cancers, including AIDS-associated Kaposi's Sarcoma and metastatic cancers.
DB09053IbrutinibAn antineoplastic agent used to treat chronic lymphocytic leukemia, mantle cell lymphoma, and Waldenstrom's Macroglobulinemia.
DB09035NivolumabA PD-1 blocking antibody used to treat melanoma, non small-cell lung cancer, renal cell cancer, head and neck cancer, and Hodgkin lymphoma.
DB12240Polatuzumab vedotinA CD79b antibody conjugate indicated to treat different types of large B-cell lymphoma.
DB11942SelinexorSelinexor is indicated in combination with bortezomib and dexamethasone for the treatment of multiple myeloma in adult patients who have received at least one prior therapy. Selinexor is also indicated...
DB15035ZanubrutinibA kinase inhibitor used to treat mantle cell lymphoma, a type of B-cell non-Hodgkin lymphoma, in adults who previously received therapy.
DrugDrug NameTargetType
DB08889CarfilzomibP-glycoprotein 1transporter
DB08889CarfilzomibProteasome subunit beta type-5target
DB08889CarfilzomibProteasome subunit beta type-9target
DB08889CarfilzomibProteasome subunit beta type-10target
DB08889CarfilzomibProteasome subunit beta type-8target
DB08889CarfilzomibProteasome subunit beta type-1target
DB08889CarfilzomibProteasome subunit beta type-2target
DB08904Certolizumab pegolTumor necrosis factortarget
DB08904Certolizumab pegolAlcohol dehydrogenase [NADP(+)]enzyme
DB00002CetuximabEpidermal growth factor receptortarget
DB00002CetuximabLow affinity immunoglobulin gamma Fc region receptor III-Btarget
DB00002CetuximabComplement C1q subcomponent subunit Atarget
DB00002CetuximabComplement C1q subcomponent subunit Btarget
DB00002CetuximabComplement C1q subcomponent subunit Ctarget
DB00002CetuximabLow affinity immunoglobulin gamma Fc region receptor III-Atarget
DB00002CetuximabHigh affinity immunoglobulin gamma Fc receptor Itarget
DB00002CetuximabLow affinity immunoglobulin gamma Fc region receptor II-atarget
DB09331DaratumumabADP-ribosyl cyclase 1target
DB00997DoxorubicinDNA topoisomerase 2-alphatarget
DB00997DoxorubicinDNAtarget
DB00997DoxorubicinCytochrome P450 3A4enzyme
DB00997DoxorubicinCytochrome P450 2D6enzyme
DB00997DoxorubicinCytochrome P450 2B6enzyme
DB00997DoxorubicinP-glycoprotein 1transporter
DB00997DoxorubicinCanalicular multispecific organic anion transporter 2transporter
DB00997DoxorubicinMultidrug resistance-associated protein 6transporter
DB00997DoxorubicinMultidrug resistance-associated protein 1transporter
DB00997DoxorubicinMultidrug resistance-associated protein 7transporter
DB00997DoxorubicinATP-binding cassette sub-family G member 2transporter
DB00997DoxorubicinBile salt export pumptransporter
DB00997DoxorubicinSolute carrier family 22 member 16transporter
DB00997DoxorubicinATP-binding cassette sub-family B member 8, mitochondrialtransporter
DB00997DoxorubicinCytochrome P450 1B1enzyme
DB00997DoxorubicinCarbonyl reductase [NADPH] 1enzyme
DB00997DoxorubicinCarbonyl reductase [NADPH] 3enzyme
DB00997DoxorubicinAlcohol dehydrogenase [NADP(+)]enzyme
DB00997DoxorubicinAldo-keto reductase family 1 member C3enzyme
DB00997DoxorubicinNAD(P)H dehydrogenase [quinone] 1enzyme
DB00997DoxorubicinXanthine dehydrogenase/oxidaseenzyme
DB00997DoxorubicinNitric oxide synthase, endothelialenzyme
DB00997DoxorubicinNitric oxide synthase, inducibleenzyme
DB00997DoxorubicinNitric oxide synthase, brainenzyme
DB00997DoxorubicinNADH dehydrogenase [ubiquinone] iron-sulfur protein 2, mitochondrialenzyme
DB00997DoxorubicinNADH dehydrogenase [ubiquinone] iron-sulfur protein 3, mitochondrialenzyme
DB00997DoxorubicinNADH dehydrogenase [ubiquinone] iron-sulfur protein 7, mitochondrialenzyme
DB00997DoxorubicinNADPH--cytochrome P450 reductaseenzyme
DB00997DoxorubicinRalA-binding protein 1transporter
DB00997DoxorubicinCanalicular multispecific organic anion transporter 1transporter
DB00997DoxorubicinSerum albumincarrier
DB00997DoxorubicinNucleolar and coiled-body phosphoprotein 1target
DB00997DoxorubicinDNA topoisomerase 1target
DB00997DoxorubicinDNA topoisomerase 2-betatarget
DB00997DoxorubicinAldose reductaseenzyme
DB00997DoxorubicinAldo-keto reductase family 1 member B10enzyme
DB00997DoxorubicinAldo-keto reductase family 1 member C4enzyme
DB09053IbrutinibTyrosine-protein kinase BTKtarget
DB09053IbrutinibCytochrome P450 3A4enzyme
DB09053IbrutinibCytochrome P450 3A5enzyme
DB09053IbrutinibSerum albumincarrier
DB09053Ibrutinibalpha1-acid glycoproteincarrier
DB09053IbrutinibCytochrome P450 2D6enzyme
DB09035NivolumabProgrammed cell death protein 1target
DB09035NivolumabProgrammed cell death 1 ligand 1target
DB12240Polatuzumab vedotinCytochrome P450 3A4enzyme
DB12240Polatuzumab vedotinB-cell antigen receptor complex-associated protein beta chaintarget
DB12240Polatuzumab vedotinP-glycoprotein 1transporter
DB12240Polatuzumab vedotinCytochrome P450 3A5enzyme
DB11942SelinexorCytochrome P450 3A4enzyme
DB11942SelinexorSolute carrier organic anion transporter family member 1B3transporter
DB11942SelinexorExportin-1target
DB15035ZanubrutinibCytochrome P450 3A4enzyme
DB15035ZanubrutinibP-glycoprotein 1transporter
DB15035ZanubrutinibCytochrome P450 2B6enzyme
DB15035ZanubrutinibTyrosine-protein kinase BTKtarget
DB15035ZanubrutinibEpidermal growth factor receptortarget
DB15035ZanubrutinibReceptor tyrosine-protein kinase erbB-2target
DB15035ZanubrutinibReceptor tyrosine-protein kinase erbB-4target
DB15035ZanubrutinibTyrosine-protein kinase ITK/TSKtarget
DB15035ZanubrutinibCytoplasmic tyrosine-protein kinase BMXtarget
DB15035ZanubrutinibTyrosine-protein kinase JAK2target
DB15035ZanubrutinibTyrosine-protein kinase Tectarget
DB15035ZanubrutinibTyrosine-protein kinase Blktarget
DB15035ZanubrutinibTyrosine-protein kinase JAK3target
DB15035ZanubrutinibProtein-tyrosine kinase 6target
DB15035ZanubrutinibTyrosine-protein kinase Fgrtarget
DB15035ZanubrutinibTyrosine-protein kinase FRKtarget
DB15035ZanubrutinibTyrosine-protein kinase Lcktarget
DB15035ZanubrutinibTyrosine-protein kinase TXKtarget
DB15035ZanubrutinibCytochrome P450 3A Subfamilyenzyme
DrugDrug NamePhaseStatusCount