Vasoconstrictor Agents

Name
Vasoconstrictor Agents
Accession Number
DBCAT000165
Description

Drugs used to cause constriction of the blood vessels.

Drugs
DrugDrug Description
AdrenaloneNot Annotated
Angiotensin IIA peptide hormone of the RAAS system used to raise blood pressure in septic or other forms of shock.
AngiotensinamideNot Annotated
AzepexoleAzepexole is a small molecule drug. Azepexole has a monoisotopic molecular weight of 181.12 Da.
Calyculin ANot Available
CirazolineCirazoline acts on a number of α adrenergic receptors. It is an agonist of α1A, partial agonist of α1B and α1D, and a nonselective antagonist of α2. It is believed...
CocaineAn ester local anesthetic used during diagnostic procedures and surgeries in or through the nasal cavities.
DihydroergotamineAn ergot alkaloid used in the acute treatment of migraine headache and cluster headache.
EphedrineAn alpha and beta-adrenergic agonist indicated to treat hypotension under anesthesia, allergic conditions, bronchial asthma, and nasal congestion.
EpinephrineA hormone and neurotransmitter used to treat allergic reactions, to restore cardiac rhythm, and to control mucosal congestion, glaucoma, and asthma.
ErgotamineAn alpha-1 selective adrenergic agonist vasoconstrictor used to treat migraines with or without aura and cluster headaches.
EtilefrineAn adrenergic agonist primarily of α1 and β1 receptors used as an anti-hypotensive.
FelypressinFor use as an alternative to adrenaline as a localising agent, provided that local ischaemia is not essential.
LevonordefrinA topical sympathomimetic amine found in local anesthetic products that is used for nasal decongestion or vasoconstriction during dental procedures.
LypressinNot Annotated
MephentermineA sympathomimetic agent used in the treatment of hypotension.
MetaraminolFor the treatment and prevention of hypotension due to hemorrhage, spinal anesthesia, and shock associated with brain damage
MethoxamineAn alpha adrenergic agonist used to treat hypotension.
MethysergideAn ergot alkaloid used for the prophylaxis of migraine and cluster headaches.
MidodrineAn alpha-adrenergic agonist used to treat orthostatic hypotension.
NaphazolineA sympathomimetic vasoconstrictor used for the symptomatic relief of redness and itching of the eye, and nasal congestion.
NaratriptanA 5-HT1B/1D receptor agonist used to treat migraines.
NorepinephrineA sympathomimetic used in the control of blood pressure during various hypotensive states and as an adjunct treatment during cardiac arrest.
OctopamineOctopamine is structurally similar to norepinephrine. It has been used as a nootropic, and therefore it and all of its enantiomer are prohibited by the World Anti-doping Agency (WADA) as...
OrnipressinNot Annotated
OxymetazolineAn alpha-1A adrenoceptor agonist used to treat nasal congestion, allergic reactions of the eye, and facial erythema associated with rosacea.
PhenylephrineAn alpha-1 adrenergic agonist used in the management of hypotension, generally in the surgical setting associated with the use of anesthetics.
PhenylpropanolamineA sympathomimetic that was previously used in nasal decongestants and weight loss products, but has been withdrawn by the FDA due to safety risks and lack of efficacy.
PseudoephedrineAn alpha and beta adrenergic agonist used to treat nasal and sinus congestion, as well as allergic rhinitis.
RacepinephrineA bronchodilator used to treat intermittent asthma.
S-EthylisothioureaS-Ethylisothiourea is a nitric oxide synthase inhibitor.
SumatriptanA serotonin receptor agonist used to treat migraines and cluster headaches.
SynephrineSynephrine, also referred to as, p-synephrine, is naturally occurring alkaloid. It is present in approved drug products as neo-synephrine, its m-substituted analog. p-synephrine and m-synephrine are known for their longer...
TerlipressinA drug used to treat bleeding caused by esophageal varices.
TetryzolineAn alpha-adrenergic agonist used in the temporary symptomatic relief of discomfort and redness of the eyes due to minor irritations, as well as alleviate nasal congestion.
UlobetasolA lipocortin corticosteroid used to treat inflammatory and pruritic corticosteroid-responsive dermatoses.
VasopressinA peptide hormone used to increase blood pressure in patients with vasodilatory shock who are resistant to fluid and catecholamine therapy.
XylometazolineA direct-acting alpha-adrenergic agonist used for the symptomatic treatment of nasal congestion and minor inflammation due to allergies or colds.
Drugs & Drug Targets
DrugTargetType
AdrenaloneDopamine beta-hydroxylasetarget
Angiotensin IIType-2 angiotensin II receptortarget
Angiotensin IIType-1 angiotensin II receptortarget
AngiotensinamideType-1 angiotensin II receptortarget
AngiotensinamideATP-dependent translocase ABCB1transporter
AngiotensinamideReplicase polyprotein 1abtarget
AzepexoleAlpha-2 adrenergic receptorstarget
Calyculin ASolute carrier family 12 member 1target
Calyculin ASerine/threonine-protein phosphatase PP1-gamma catalytic subunittarget
CirazolineAlpha-2C adrenergic receptortarget
CirazolineAlpha-2 adrenergic receptorstarget
CirazolineAlpha-1D adrenergic receptortarget
CirazolineAlpha-1B adrenergic receptortarget
CirazolineAlpha-1A adrenergic receptortarget
CocaineSodium-dependent noradrenaline transportertarget
CocaineSodium channel proteintarget
CocaineSodium-dependent serotonin transportertarget
CocaineSodium-dependent dopamine transportertarget
CocaineCytochrome P450 3A4enzyme
CocaineMuscarinic acetylcholine receptor M1target
CocaineMuscarinic acetylcholine receptor M2target
CocaineCytochrome P450 2D6enzyme
CocaineSolute carrier family 22 member 2transporter
CocaineCytochrome P450 2C8enzyme
CocaineSigma non-opioid intracellular receptor 1target
CocaineLiver carboxylesterase 1target
CocaineCholinesteraseenzyme
CocaineSodium-dependent dopamine transportertransporter
Cocainealpha1-acid glycoproteincarrier
CocaineLiver carboxylesterase 1enzyme
CocaineVoltage-gated sodium channel alpha subunittarget
DihydroergotamineBeta-3 adrenergic receptortarget
Dihydroergotamine5-hydroxytryptamine receptor 4target
DihydroergotamineCytochrome P450 3A4enzyme
Dihydroergotamine5-hydroxytryptamine receptor 1Btarget
Dihydroergotamine5-hydroxytryptamine receptor 1Dtarget
Dihydroergotamine5-hydroxytryptamine receptor 2Btarget
DihydroergotamineATP-dependent translocase ABCB1transporter
Dihydroergotamine5-hydroxytryptamine receptor 1Atarget
Dihydroergotamine5-hydroxytryptamine receptor 1Etarget
Dihydroergotamine5-hydroxytryptamine receptor 2Atarget
DihydroergotamineD(2) dopamine receptortarget
Dihydroergotamine5-hydroxytryptamine receptor 2Ctarget
DihydroergotamineAlpha-1 adrenergic receptorstarget
DihydroergotamineAlpha-2 adrenergic receptorstarget
DihydroergotamineD(3) dopamine receptortarget
DihydroergotamineD(4) dopamine receptortarget
Dihydroergotamine5-hydroxytryptamine receptor 1Ftarget
DihydroergotamineAlpha-2A adrenergic receptortarget
EphedrineBeta-2 adrenergic receptortarget
EphedrineSynaptic vesicular amine transportertransporter
EphedrineAcetylcholinesteraseenzyme
EphedrineD(2) dopamine receptortarget
EphedrineBeta-1 adrenergic receptortarget
EphedrineAlbumincarrier
EphedrineCholinesteraseenzyme
EphedrineSodium-dependent noradrenaline transportertarget
EphedrineAlpha-1A adrenergic receptortarget
EpinephrineMonoamine oxidaseenzyme
EpinephrineCatechol O-methyltransferaseenzyme
EpinephrineAlpha-1A adrenergic receptortarget
EpinephrineBeta-1 adrenergic receptortarget
EpinephrineBeta-2 adrenergic receptortarget
EpinephrineSolute carrier family 22 member 2transporter
EpinephrineSolute carrier family 22 member 1transporter
EpinephrineCytochrome P450 2C9enzyme
EpinephrineCytochrome P450 3A4enzyme
EpinephrineAlpha-1B adrenergic receptortarget
EpinephrineAlpha-1D adrenergic receptortarget
EpinephrineAlpha-2A adrenergic receptortarget
EpinephrineAlpha-2B adrenergic receptortarget
EpinephrineTumor necrosis factortarget
ErgotamineAlpha-1A adrenergic receptortarget
Ergotamine5-hydroxytryptamine receptor 1Dtarget
ErgotamineAlpha adrenergic receptortarget
ErgotamineAlpha-2C adrenergic receptortarget
Ergotamine5-hydroxytryptamine receptor 2Btarget
Ergotamine5-hydroxytryptamine receptor 2Ctarget
Ergotamine5-hydroxytryptamine receptor 1Btarget
Ergotamine5-hydroxytryptamine receptor 2Atarget
ErgotamineAlpha-2A adrenergic receptortarget
Ergotamine5-hydroxytryptamine receptor 1Ftarget
Ergotamine5-hydroxytryptamine receptor 1Atarget
ErgotamineD(1) dopamine receptortarget
ErgotamineATP-dependent translocase ABCB1transporter
ErgotamineD(2) dopamine receptortarget
ErgotamineCytochrome P450 3A4enzyme
ErgotamineAlpha-1B adrenergic receptortarget
ErgotamineAlpha-1D adrenergic receptortarget
EtilefrineAlpha adrenergic receptortarget
EtilefrineAlpha-1D adrenergic receptortarget
EtilefrineSolute carrier family 22 member 3transporter
FelypressinVasopressin V1a receptortarget
LevonordefrinAlpha-2 adrenergic receptorstarget
LevonordefrinAlpha-1D adrenergic receptortarget
LevonordefrinAlpha-1B adrenergic receptortarget
LevonordefrinAlpha-1A adrenergic receptortarget
LypressinVasopressin V1b receptortarget
LypressinVasopressin V2 receptortarget
LypressinVasopressin V1a receptortarget
LypressinATP-binding cassette sub-family C member 2transporter
MephentermineAlpha adrenergic receptortarget
MephentermineBeta adrenergic receptortarget
MephentermineD(2) dopamine receptortarget
MetaraminolAlpha-1A adrenergic receptortarget
MetaraminolD(2) dopamine receptortarget
MetaraminolAlpha-1 adrenergic receptorstarget
MethoxamineAlpha-1 adrenergic receptorstarget
MethoxamineAlpha-1D adrenergic receptortarget
MethoxamineAlpha-1A adrenergic receptortarget
MethoxamineAlpha-1B adrenergic receptortarget
Methysergide5-hydroxytryptamine receptor 2Atarget
Methysergide5-hydroxytryptamine receptor 1Atarget
Methysergide5-hydroxytryptamine receptor 7target
Methysergide5-hydroxytryptamine receptor 2Ctarget
Methysergide5-hydroxytryptamine receptor 2Btarget
Methysergide5-hydroxytryptamine receptor 1Btarget
Methysergide5-hydroxytryptamine receptor 1Ftarget
Methysergide5-hydroxytryptamine receptor 1Etarget
MethysergideCytochrome P450 3A4enzyme
MidodrineAlpha-1A adrenergic receptortarget
MidodrineAlpha-1B adrenergic receptortarget
MidodrineCytochrome P450 2D6enzyme
MidodrineSolute carrier family 15 member 1transporter
MidodrineAlpha-1D adrenergic receptortarget
MidodrineAlpha-1 adrenergic receptorstarget
NaphazolineAlpha adrenergic receptortarget
NaphazolineD(2) dopamine receptortarget
NaphazolineAlpha-2A adrenergic receptortarget
NaphazolineAlpha-1A adrenergic receptortarget
NaratriptanAmine oxidase [flavin-containing] Aenzyme
Naratriptan5-hydroxytryptamine receptor 1Atarget
Naratriptan5-hydroxytryptamine receptor 1Ftarget
Naratriptan5-hydroxytryptamine receptor 1Btarget
Naratriptan5-hydroxytryptamine receptor 1Dtarget
NorepinephrineAlpha-2B adrenergic receptortarget
NorepinephrineAlpha-2C adrenergic receptortarget
NorepinephrineBeta-1 adrenergic receptortarget
NorepinephrineBeta-2 adrenergic receptortarget
NorepinephrineBeta-3 adrenergic receptortarget
NorepinephrineSolute carrier family 22 member 2transporter
NorepinephrineSolute carrier family 22 member 3transporter
NorepinephrineOrganic cation/carnitine transporter 2transporter
NorepinephrineAlpha-2A adrenergic receptortarget
NorepinephrineSolute carrier family 22 member 1transporter
NorepinephrinePOU domain, class 5, transcription factor 1transporter
NorepinephrineSodium-dependent noradrenaline transportertransporter
NorepinephrineSynaptic vesicular amine transportertarget
NorepinephrineChromaffin granule amine transportertarget
NorepinephrinePhenylalanine-4-hydroxylasetarget
NorepinephrineAlpha-1A adrenergic receptortarget
NorepinephrineAlpha-1B adrenergic receptortarget
NorepinephrineAlpha-1D adrenergic receptortarget
OctopamineCoagulation factor Xtarget
OrnipressinVasopressin V1a receptortarget
OxymetazolineAlpha-1A adrenergic receptortarget
OxymetazolineAlpha adrenergic receptortarget
OxymetazolineCytochrome P450 2C19enzyme
OxymetazolineUDP-glucuronosyltransferase 1A9enzyme
Oxymetazoline5-hydroxytryptamine receptor 2Ctarget
Oxymetazoline5-hydroxytryptamine receptor 1Dtarget
Oxymetazoline5-hydroxytryptamine receptor 1Btarget
Oxymetazoline5-hydroxytryptamine receptor 1Atarget
OxymetazolineAlpha-2A adrenergic receptortarget
OxymetazolineAlpha-2C adrenergic receptortarget
OxymetazolineAlpha-2B adrenergic receptortarget
OxymetazolineAlpha-1B adrenergic receptortarget
OxymetazolineAlpha-1D adrenergic receptortarget
PhenylephrineAmine oxidase [flavin-containing] Aenzyme
PhenylephrineAlpha-1D adrenergic receptortarget
PhenylephrineCytochrome P450 1A2enzyme
PhenylephrineSulfotransferase 1A3enzyme
PhenylephrineAmine oxidase [flavin-containing] Benzyme
PhenylephrineD(2) dopamine receptortarget
PhenylephrineAlpha-1 adrenergic receptorstarget
PhenylephrineAlpha-1B adrenergic receptortarget
PhenylephrineAlpha-1A adrenergic receptortarget
PhenylpropanolamineAmine oxidase [flavin-containing] Aenzyme
PhenylpropanolamineD(1A) dopamine receptortarget
PhenylpropanolamineBeta-1 adrenergic receptortarget
PhenylpropanolamineBeta-2 adrenergic receptortarget
PhenylpropanolamineAlpha-2 adrenergic receptorstarget
PhenylpropanolamineTelomerase reverse transcriptasetarget
PhenylpropanolamineAlpha-1A adrenergic receptortarget
PhenylpropanolamineSodium-dependent noradrenaline transportertarget
PseudoephedrineAlpha-1A adrenergic receptortarget
PseudoephedrineSodium-dependent dopamine transportertransporter
PseudoephedrineBeta-2 adrenergic receptortarget
PseudoephedrineAmine oxidase [flavin-containing] Aenzyme
PseudoephedrineBeta-1 adrenergic receptortarget
PseudoephedrineSodium-dependent dopamine transportertarget
PseudoephedrineSodium-dependent noradrenaline transportertarget
PseudoephedrineSodium-dependent serotonin transportertarget
PseudoephedrineNuclear factor of activated T-cells, cytoplasmic 1target
PseudoephedrineTumor necrosis factortarget
PseudoephedrineNuclear factor NF-kappa-B p105 subunittarget
Pseudoephedrineactivator protein 1target
PseudoephedrineInterleukin-2target
PseudoephedrineAlbumincarrier
PseudoephedrineSodium-dependent noradrenaline transportertransporter
PseudoephedrineAlpha-2A adrenergic receptortarget
PseudoephedrineSodium-dependent serotonin transportertransporter
PseudoephedrineD(2) dopamine receptortarget
RacepinephrineBeta-2 adrenergic receptortarget
RacepinephrineAlpha-1D adrenergic receptortarget
RacepinephrineBeta-3 adrenergic receptortarget
RacepinephrineAlpha-2C adrenergic receptortarget
RacepinephrineAlpha-2B adrenergic receptortarget
RacepinephrineAlpha-2A adrenergic receptortarget
RacepinephrineAlpha-1B adrenergic receptortarget
RacepinephrineAlpha-1A adrenergic receptortarget
RacepinephrineBeta-1 adrenergic receptortarget
S-EthylisothioureaNitric oxide synthase oxygenasetarget
S-EthylisothioureaNitric oxide synthase, inducibletarget
S-EthylisothioureaNitric oxide synthase 3target
SumatriptanSolute carrier organic anion transporter family member 1B1transporter
SumatriptanBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
SumatriptanATP-dependent translocase ABCB1transporter
SumatriptanSolute carrier organic anion transporter family member 1A2transporter
Sumatriptan5-hydroxytryptamine receptor 1Atarget
SumatriptanAmine oxidase [flavin-containing] Aenzyme
Sumatriptan5-hydroxytryptamine receptor 1Ftarget
Sumatriptan5-hydroxytryptamine receptor 1Btarget
Sumatriptan5-hydroxytryptamine receptor 1Dtarget
SynephrineAlpha-1 adrenergic receptorstarget
TerlipressinVasopressin V2 receptortarget
TerlipressinVasopressin V1a receptortarget
TerlipressinVasopressin V1b receptortarget
TetryzolineAlpha-1 adrenergic receptorstarget
TetryzolineAlpha-2 adrenergic receptorstarget
TetryzolineAlpha-2C adrenergic receptortarget
TetryzolineAlpha adrenergic receptortarget
UlobetasolEstrogen-related receptor gammatarget
UlobetasolSteroid hormone receptor ERR2target
UlobetasolSteroid hormone receptor ERR1target
UlobetasolGlucocorticoid receptortarget
UlobetasolCorticosteroid-binding globulincarrier
VasopressinVasopressin V1a receptortarget
VasopressinVasopressin V2 receptortarget
VasopressinVasopressin V1b receptortarget
VasopressinATP-binding cassette sub-family C member 2transporter
VasopressinOxytocin receptortarget
XylometazolineAlpha-2A adrenergic receptortarget
XylometazolineAlpha-1A adrenergic receptortarget
XylometazolineAlpha-1B adrenergic receptortarget
XylometazolineAlpha-1D adrenergic receptortarget
XylometazolineAlpha-2B adrenergic receptortarget
XylometazolineAlpha-2C adrenergic receptortarget
XylometazolineAlpha adrenergic receptortarget