Cardiotonic Agents

Name
Cardiotonic Agents
Accession Number
DBCAT000589
Description

Agents that have a strengthening effect on the heart or that can increase cardiac output. They may be CARDIAC GLYCOSIDES; SYMPATHOMIMETICS; or other drugs. They are used after MYOCARDIAL INFARCT; CARDIAC SURGICAL PROCEDURES; in SHOCK; or in congestive heart failure (HEART FAILURE).

Drugs
DrugDrug Description
AcetyldigitoxinUsed for fast digitalization in congestive heart failure.
AcetyldigoxinNot Annotated
AcrihellinAcrihellin is a small molecule drug. Acrihellin has a monoisotopic molecular weight of 498.26 Da.
AdrenomedullinAdrenomedullin is under investigation in clinical trial NCT06072118 (Adrenomedullin for CADASIL).
AlifedrineAlifedrine is a small molecule drug. The usage of the INN stem '-drine' in the name indicates that Alifedrine is a sympathomimetic. Alifedrine has a monoisotopic molecular weight of 289.2...
AminophyllineA bronchodilator consisting of theophylline that is used for the treatment of bronchospasm due to asthma, emphysema and chronic bronchitis.
AmrinoneA positive inotropic agent and phosphodiesterase inhibitor used in the management of treatment of congestive heart failure.
ArbutamineUsed to elicit acute cardiovascular responses (cardiac stumulant), similar to those produced by exercise, in order to aid in diagnosing the presence or absence of coronary artery disease (CAD) in...
BimakalimBimakalim is a small molecule drug. The usage of the INN stem '-kalim' in the name indicates that Bimakalim is a potassium channel activator, antihypertensive. Bimakalim has a monoisotopic molecular...
BufogeninBufogenin is a small molecule drug. Bufogenin has a monoisotopic molecular weight of 384.23 Da.
CanertinibInvestigated for use/treatment in breast cancer and lung cancer.
CarbamoylcholineA direct acting miotic agent administered ophthalmically to decrease intraocular pressure after cataract surgery, and to induce miosis during surgery.
ColforsinPotent activator of the adenylate cyclase system and the biosynthesis of cyclic AMP. From the plant Coleus forskohlii. Has antihypertensive, positive inotropic, platelet aggregation inhibitory, and smooth muscle relaxant activities;...
CymarinNot Annotated
DenopamineDenopamine is a small molecule drug. Denopamine has a monoisotopic molecular weight of 317.16 Da.
DeslanosideFor the treatment and management of Congestive cardiac insufficiency, arrhythmias and heart failure.
DexrazoxaneA cytoprotective drug used to prevent and improve cardiomyopathy associated with doxorubicin treatment for metastatic breast cancer.
DigitoxinA cardiac glycoside used in the treatment and management of congestive cardiac insufficiency, arrhythmias and heart failure.
DigoxinA cardiac glycoside used in the treatment of mild to moderate heart failure and for ventricular response rate control in chronic atrial fibrillation.
DobutamineA beta-1 agonist used to treat cardiac decompensation in patients with organic heart disease or from cardiac surgery.
DopamineA catecholamine neurotransmitter used to treat hemodynamic imbalances, poor perfusion of vital organs, low cardiac output, and hypotension.
EnoximoneA selective phosphodiesterase inhibitor indicated in the short term treatment of congestive heart failure.
EtilefrineAn adrenergic agonist primarily of α1 and β1 receptors used as an anti-hypotensive.
HigenamineHigenamine is under investigation in clinical trial NCT01451229 (Pharmacokinetics and Pharmacodynamics of Higenamine in Chinese Healthy Subjects).
IbopamineA sympathomimetic, indicated in the induction of mydriasis and treatment of pos-surgical ocular hypotonia.
ImazodanImazodan is a small molecule drug. The usage of the INN stem '-dan' in the name indicates that Imazodan is a cardiac stimulant, pimobendan derivative. Imazodan has a monoisotopic molecular...
IsoprenalineA catecholamine non-selective beta-adrenergic agonist typically used to treat bradycardia and heart block.
LevosimendanA calcium sensitizer indicated to treat acutely decompensated severe chronic heart failure.
LisinoprilAn ACE inhibitor used to treat hypertension, heart failure, and acute myocardial infarction.
MetildigoxinA digitalis glycoside indicated in the treatment of acute and chronic heart failure.
MilrinoneA PDE-III inhibitor with inotropic, lusitropic, and vasodilatory properties used for the short-term treatment of acute decompensated heart failure.
OlprinoneNot Annotated
OuabainFor the treatment of atrial fibrillation and flutter and heart failure
OxyfedrineNot Annotated
PeruvosideNot Annotated
PhenylephrineAn alpha-1 adrenergic agonist used in the management of hypotension, generally in the surgical setting associated with the use of anesthetics.
PhosphocreatineA cardioprotective agent indicated for use in cardiac surgery.
PimobendanNot Annotated
PirbuterolA beta-2 adrenergic agonist and bronchodilator used for the symptomatic treatment of asthma.
PiroximonePiroximone is a small molecule drug. Piroximone has a monoisotopic molecular weight of 217.09 Da.
PlumbaginPlumbagin is a compound investigated for its anticancer activity. It has been found that it inactivates the Akt/NF-kB, MMP-9 and VEGF pathways.
PrenalterolNot Annotated
ProscillaridinProscillaridin is a cardiac glycoside that is derived from plants of the genus Scilla and in Drimia maritima (Scilla maritima). Studies suggest the potential cytotoxic and anticancer property of proscillaridin,...
SimendanNot Annotated
TedisamilInvestigated for use/treatment in arrhythmia, atrial fibrillation, and angina.
VesnarinoneVesnarinone has been used in trials studying the treatment of HIV Infections and Sarcoma, Kaposi.
ZatebradineZatebradine is a small molecule drug. The usage of the INN stem '-bradine' in the name indicates that Zatebradine is a bradycardic agent. Zatebradine has a monoisotopic molecular weight of...
Drugs & Drug Targets
DrugTargetType
AcetyldigitoxinSodium/potassium-transporting ATPase subunit alpha-1target
AcetyldigoxinSodium/Potassium Transporting ATPasetarget
AdrenomedullinNeprilysinenzyme
AdrenomedullinCalcitonin gene-related peptide type 1 receptortarget
AminophyllinecGMP-inhibited 3',5'-cyclic phosphodiesterase 3Atarget
AminophyllineAdenosine receptor A3target
AminophyllineAdenosine receptor A1target
AminophyllineCytochrome P450 1A2enzyme
AminophyllineCytochrome P450 2E1enzyme
AminophyllineCytochrome P450 3A4enzyme
AminophyllineHistone deacetylase 2target
AminophyllineAdenosine receptortarget
AminophyllinePhosphodiesterase 3target
AminophyllinePhosphodiesterase 4target
AmrinonecAMP-specific 3',5'-cyclic phosphodiesterase 4 (PDE4)target
AmrinonecGMP-inhibited 3',5'-cyclic phosphodiesterase 3Btarget
AmrinonecGMP-inhibited 3',5'-cyclic phosphodiesterase 3Atarget
AmrinoneTumor necrosis factortarget
ArbutamineBeta-1 adrenergic receptortarget
ArbutamineBeta-2 adrenergic receptortarget
ArbutamineBeta-3 adrenergic receptortarget
BimakalimATP-sensitive potassium channeltarget
BimakalimATP-binding cassette sub-family C member 9target
BimakalimATP-sensitive inward rectifier potassium channel 11target
BufogeninVascular endothelial growth factor receptor 2target
BufogeninSodium/potassium-transporting ATPase subunit alpha-1target
BufogeninSodium/Potassium Transporting ATPasetarget
CanertinibEpidermal growth factor receptortarget
CanertinibReceptor tyrosine-protein kinase erbB-2target
CanertinibReceptor tyrosine-protein kinase erbB-4target
CanertinibRAC-alpha serine/threonine-protein kinasetarget
CarbamoylcholineMuscarinic acetylcholine receptor M1target
CarbamoylcholineMuscarinic acetylcholine receptor M2target
CarbamoylcholineNeuronal acetylcholine receptor subunit alpha-2target
CarbamoylcholineCytosolic phospholipase A2enzyme
CarbamoylcholineMuscarinic acetylcholine receptor M3target
CarbamoylcholineMuscarinic acetylcholine receptor M4target
CarbamoylcholineAcetylcholinesteraseenzyme
ColforsinATP-dependent translocase ABCB1transporter
ColforsinAdenylate cyclase type 2target
ColforsinGuanine nucleotide-binding protein G(s) subunit alpha isoforms shorttarget
ColforsinAdenylate cyclase type 5target
ColforsinCystic fibrosis transmembrane conductance regulatortarget
ColforsinAdenylate cyclasetarget
ColforsinCalcium-activated potassium channeltarget
ColforsinCREB-binding proteintarget
ColforsinExtracellular signal-regulated kinase (ERK)target
ColforsinMucin-2target
ColforsinPlasminogen activator inhibitor 1target
CymarinPeroxisome proliferator-activated receptor alphatarget
DenopamineD(2) dopamine receptortarget
DeslanosideSodium/potassium-transporting ATPase subunit alpha-1target
DexrazoxaneDNA topoisomerase 2target
DexrazoxaneDNA topoisomerase 2-betatarget
DexrazoxaneDNA topoisomerase 2-alphatarget
DigitoxinSodium/potassium-transporting ATPase subunit beta-3target
DigitoxinSodium/potassium-transporting ATPase subunit alpha-1target
DigitoxinAlbumincarrier
DigitoxinCholesterol side-chain cleavage enzyme, mitochondrialenzyme
DigitoxinCytochrome P450 3A4enzyme
DigitoxinSolute carrier organic anion transporter family member 1A2transporter
DigitoxinSolute carrier organic anion transporter family member 4C1transporter
DigitoxinATP-dependent translocase ABCB1transporter
DigitoxinSodium/potassium-transporting ATPase subunit alpha-2target
DigitoxinSodium/potassium-transporting ATPase subunit alpha-3target
DigitoxinSodium/potassium-transporting ATPase subunit beta-1target
DigitoxinSodium/potassium-transporting ATPase subunit beta-2target
DigoxinSolute carrier organic anion transporter family member 4C1target
DigoxinSodium/potassium-transporting ATPase subunit beta-3target
DigoxinSodium/potassium-transporting ATPase subunit alpha-1target
DigoxinCholesterol side-chain cleavage enzyme, mitochondrialenzyme
DigoxinSodium/potassium-transporting ATPase subunit beta-2target
DigoxinSodium/potassium-transporting ATPase subunit beta-1target
DigoxinSodium/potassium-transporting ATPase subunit alpha-3target
DigoxinSodium/potassium-transporting ATPase subunit alpha-2target
DigoxinSolute carrier organic anion transporter family member 1B1transporter
DigoxinOrganic solute transporter subunit betatransporter
DigoxinOrganic solute transporter subunit alphatransporter
DigoxinSolute carrier organic anion transporter family member 1A2transporter
DigoxinBile salt export pumptransporter
DigoxinSolute carrier organic anion transporter family member 4C1transporter
DigoxinATP-dependent translocase ABCB1transporter
DobutamineBeta-1 adrenergic receptortarget
DobutamineCatechol O-methyltransferaseenzyme
DobutamineBeta-2 adrenergic receptortarget
DobutamineAlpha-1 adrenergic receptorstarget
DobutamineEstrogen receptortarget
DopamineDopamine beta-hydroxylasetarget
Dopamine5-hydroxytryptamine receptor 3Btarget
DopamineAmine oxidase [flavin-containing] Aenzyme
DopamineAmine oxidase [flavin-containing] Benzyme
DopamineCatechol O-methyltransferaseenzyme
DopamineSodium-dependent serotonin transportertarget
Dopamine5-hydroxytryptamine receptor 3Atarget
DopamineD(1A) dopamine receptortarget
DopamineSuperoxide dismutase [Cu-Zn]target
DopamineSynaptic vesicular amine transportertarget
DopamineBeta-1 adrenergic receptortarget
DopamineSolute carrier family 22 member 2transporter
DopamineSolute carrier family 22 member 1transporter
DopamineSolute carrier family 22 member 3transporter
DopamineOrganic cation/carnitine transporter 2transporter
DopaminePOU domain, class 5, transcription factor 1transporter
DopamineD(1B) dopamine receptortarget
DopamineD(2) dopamine receptortarget
DopamineD(3) dopamine receptortarget
DopamineD(4) dopamine receptortarget
DopamineSodium-dependent noradrenaline transportertarget
DopamineD(1) dopamine receptortarget
Dopamine5-hydroxytryptamine receptor 7target
Dopamine5-hydroxytryptamine receptor 1Atarget
DopamineDopamine beta-hydroxylaseenzyme
DopamineSodium-dependent dopamine transportertarget
EnoximonecGMP-inhibited 3',5'-cyclic phosphodiesterase 3Atarget
EnoximonePhosphodiesterase 3target
EtilefrineAlpha adrenergic receptortarget
EtilefrineAlpha-1D adrenergic receptortarget
EtilefrineSolute carrier family 22 member 3transporter
HigenamineBeta-2 adrenergic receptortarget
HigenamineBeta-1 adrenergic receptortarget
HigenamineLysine-specific histone demethylase 1Atarget
ImazodancGMP-inhibited 3',5'-cyclic phosphodiesterase 3Atarget
ImazodancGMP-dependent 3',5'-cyclic phosphodiesterasetarget
ImazodancGMP-specific 3',5'-cyclic phosphodiesterasetarget
IsoprenalineBeta-1 adrenergic receptortarget
IsoprenalineBeta-2 adrenergic receptortarget
IsoprenalineBeta-3 adrenergic receptortarget
IsoprenalineCytochrome P450 1A1enzyme
IsoprenalineSuperoxide dismutase [Cu-Zn]target
IsoprenalineCytochrome P450 1B1enzyme
IsoprenalineAlbumincarrier
IsoprenalineCatechol O-methyltransferaseenzyme
IsoprenalineCholinesteraseenzyme
IsoprenalineInterleukin-12 subunit betatarget
IsoprenalineBeta adrenergic receptortarget
LevosimendanTroponin C, slow skeletal and cardiac musclestarget
LevosimendanATP-sensitive inward rectifier potassium channel 11target
LevosimendanATP-sensitive inward rectifier potassium channel 8target
LevosimendancGMP-inhibited 3',5'-cyclic phosphodiesterase 3Atarget
LevosimendanPhosphodiesterase 3target
LisinoprilAngiotensin-converting enzymetarget
LisinoprilSolute carrier family 15 member 1transporter
LisinoprilSolute carrier family 15 member 2transporter
LisinoprilRenintarget
MetildigoxinSodium/Potassium Transporting ATPasetarget
MilrinonecGMP-inhibited 3',5'-cyclic phosphodiesterase 3Atarget
OlprinonecGMP-inhibited 3',5'-cyclic phosphodiesterase 3Atarget
OlprinonePhosphodiesterase 3target
OuabainSodium/potassium-transporting ATPase subunit alpha-3target
OuabainSodium/potassium-transporting ATPase subunit alpha-2target
OuabainSolute carrier organic anion transporter family member 1C1transporter
OuabainSolute carrier organic anion transporter family member 1B3transporter
OuabainSolute carrier organic anion transporter family member 1B1transporter
OuabainOrganic anion transporter 3transporter
OuabainSolute carrier organic anion transporter family member 4C1transporter
OuabainSolute carrier organic anion transporter family member 1A2transporter
OuabainSodium/potassium-transporting ATPase subunit alpha-1target
OxyfedrineBeta adrenergic receptortarget
OxyfedrineAldehyde dehydrogenase 1A1target
OxyfedrineAldehyde dehydrogenase family 3 member A2target
PeruvosideProto-oncogene tyrosine-protein kinase Srctarget
PhenylephrineAlpha-1A adrenergic receptortarget
PhenylephrineAlpha-1B adrenergic receptortarget
PhenylephrineAmine oxidase [flavin-containing] Aenzyme
PhenylephrineAlpha-1D adrenergic receptortarget
PhenylephrineCytochrome P450 1A2enzyme
PhenylephrineSulfotransferase 1A3enzyme
PhenylephrineAmine oxidase [flavin-containing] Benzyme
PhenylephrineD(2) dopamine receptortarget
PhenylephrineAlpha-1 adrenergic receptorstarget
PhosphocreatineGuanidinoacetate N-methyltransferasetarget
PhosphocreatineSodium- and chloride-dependent creatine transporter 1target
PhosphocreatineCreatine kinase M-typetarget
PhosphocreatineCreatine kinase U-type, mitochondrialtarget
PhosphocreatineCreatine kinase S-type, mitochondrialtarget
PhosphocreatineCreatine kinase B-typetarget
PimobendanCytochrome P450 1A2enzyme
PimobendanPhosphodiesterase 3target
PirbuterolBeta-2 adrenergic receptortarget
PirbuterolBeta-1 adrenergic receptortarget
PiroximoneCyclic nucleotide phosphodiesterasetarget
PiroximonePhosphodiesterase 3target
PlumbaginDihydroorotate dehydrogenase (quinone), mitochondrialtarget
PrenalterolBeta-3 adrenergic receptortarget
ProscillaridinAcetylcholinesterasetarget
TedisamilVoltage-gated Potassium Channelstarget
VesnarinoneVoltage-gated inwardly rectifying potassium channel KCNH2target
VesnarinonecGMP-inhibited 3',5'-cyclic phosphodiesterase 3Atarget
ZatebradinePotassium voltage-gated channel subfamily A member 5target