| Cromoglicic acid | A medication used to treat asthma, allergic reactions of the eyes and nose, as well as other mast cell reactions. |
| Hesperetin | For lowering cholesterol and, possibly, otherwise favorably affecting lipids. In vitro research also suggests the possibility that hesperetin might have some anticancer effects and that it might have some anti-aromatase... |
| Flavoxate | A muscarinic antagonist and spasmolytic used for the symptomatic relief of conditions associated with lack of muscle control in the bladder, such as dysuria, urgency, and nocturia. |
| Genistein | Currently Genistein is being studied in clinical trials as a treatment for prostate cancer. |
| Rutin | A flavonol glycoside found in many plants, including buckwheat; tobacco; forsythia; hydrangea; viola, etc. It has been used therapeutically to decrease capillary fragility. |
| Daidzin | Not Available |
| Myricetin | Not Available |
| Naringenin | Not Available |
| Alvocidib | Investigated for use/treatment in esophageal cancer, leukemia (lymphoid), lung cancer, liver cancer, and lymphoma (unspecified). |
| Epigallocatechin | Not Available |
| Quercetin | Quercetin is a flavonol widely distributed in plants. It is an antioxidant, like many other phenolic heterocyclic compounds. Glycosylated forms include RUTIN and quercetrin. |
| 4'-Hydroxyflavanone | Not Available |
| Hesperidin | A bioflavonoid found in a variety of nutritional supplements that is touted to have various beneficial effects on blood vessel disorders and various other conditions. |
| Idronoxil | Intended for the treatment of various forms of cancer. |
| Crofelemer | An antidiarrheal agent used for the symptomatic relief of drug-induced non-infectious diarrhea in adult patients with HIV/AIDS receiving antiretroviral therapy. |
| Elafibranor | Investigated for use/treatment in atherosclerosis and diabetes mellitus type 2. |
| Sofalcone | Investigated for use/treatment in gastroenteritis and ulcers. |
| Triphendiol | Investigated for use/treatment in cancer/tumors (unspecified). |
| beta-Naphthoflavone | β-Naphthoflavone, also known as 5,6-benzoflavone, is a potent agonist of the aryl hydrocarbon receptor and induces cytochromes P450 (CYPs) and uridine 5'-diphospho-glucuronosyltransferases (UGTs). It may be a chemopreventive agent. |
| Apigenin | Not Available |
| Flavone | Not Available |
| Diosmin | Diosmin is a semisynthetic drug indicated for the treatment of venous disease. Diosmin is a flavone that can be found in the plant Teucrium gnaphalodes. Diosmin is available as a... |
| Diosmetin | Diosmetin is an O-methylated flavone and the aglycone part of the flavonoid glycosides diosmin that occurs naturally in citrus fruits . Pharmacologically, diosmetin is reported to exhibit anticancer, antimicrobial, antioxidant,... |
| Rotenone | Rotenone is an isoflavone compound that naturally occurs in the jicama vine plant as well as many Fabaceae plants. It has broad spectrum insecticide and pesticide activity and is also... |
| Equol | Equol has been used in trials studying the treatment of Breast Cancer. |
| Epicatechin | Epicatechin has been used in trials studying the treatment of Pre-diabetes. |
| Icariin | Icariin has been investigated for the basic science of the Pharmacokinetic Profile of Icariin in Humans. |
| Recoflavone | Recoflavone has been used in trials studying the treatment of Acute Gastritis, Dry Eye Syndrome, and Chronic Gastritis. |
| Epigallocatechin gallate | Epigallocatechin gallate has been investigated for the treatment of Hypertension and Diabetic Nephropathy. |
| Puerarin | Puerarin has been investigated for the treatment of Alcohol Abuse. |
| Isoquercetin | Isoquercetin has been used in trials studying the treatment of Kidney Cancer, Renal cell carcinoma, Advanced Renal Cell Carcinoma, Thromboembolism of Vein in Pancreatic Cancer, and Thromboembolism of Vein VTE... |
| Icaritin | Icaritin has been used in trials studying the treatment of Solid Tumors, Metastatic Breast Cancer, and Hepatocellular Carcinoma (HCC). |
| ME-344 | ME-344 has been used in trials studying the treatment of Solid Tumors. |
| Troxerutin | Troxerutin has been used in trials studying the treatment of Chronic Venous Insufficiency. |
| Daidzein | Not Annotated |
| Efloxate | Not Annotated |
| Dimefline | Not Annotated |
| Hidrosmin | Not Annotated |
| Ipriflavone | Not Annotated |
| Hispidulin | Hispidulin (4',5,7-trihydroxy-6-methoxyflavone) is a potent benzodiazepine (BZD) receptor ligand with positive allosteric properties . |
| Cianidanol | An antioxidant flavonoid, occurring especially in woody plants as both (+)-catechin and (-)-epicatechin (cis) forms. |
| Dihydroxymethoxychalcone | Cardamonin (also known as Dihydroxymethoxychalcone), as shown by the increasing number of publications, has received growing attention from the scientific community due to the expectations toward its benefits to human... |
| Citrus bioflavonoids | Not Annotated |
| Taxifolin | Not Available |
| Isoliquiritigenin | Isoliquiritigenin is a precursor to several flavonones in many plants. |
| Fisetin | Not Available |
| Silibinin | Currently being tested as a treatment of severe intoxications with hepatotoxic substances, such as death cap (Amanita phalloides) poisoning. |
| Biochanin A | Biochanin A is under investigation in clinical trial NCT02174666 (Isoflavone Treatment for Postmenopausal Osteopenia.). |
| Formononetin | Formononetin is under investigation in clinical trial NCT02174666 (Isoflavone Treatment for Postmenopausal Osteopenia.). |
| Xanthohumol | Xanthohumol is under investigation in clinical trial NCT01367431 (Xanthohumol and Metabolic Syndrome). |
| Resveratrol | Being investigated for the treatment of Herpes labialis infections (cold sores). |
| Chrysin | Not Annotated |
| Luteolin | Not Annotated |
| Phloretin | Phloretin is a natural dihydrochalcone found in apples and many other fruits. |
| Tricetin | Not Available |
| alpha-Naphthoflavone | Not Available |
| Sakuranetin | Not Available |
| Dihydromyricetin | Dihydromyricetin is under investigation in clinical trial NCT03606694 (Effect of Dihydromirycetin on Glycemic Control, Insulin Sensitivity and Insulin Secretion in Type 2 Diabetes Mellitus). |
| Maritime pine extract | Not Annotated |