Histamine H1 Antagonists

DBCAT000665Therapeutic category

Drugs that selectively bind to but do not activate histamine H1 receptors, thereby blocking the actions of endogenous histamine. Included here are the classical antihistaminics that antagonize or prevent the action of histamine mainly in... A DrugBank category of 101 drugs. 89 of them are approved.

Also known as
Antagonists, Histamine H1 · Antagonists, Histamine H1 Receptor · Antihistamines, Classical · Antihistamines, Sedating · Antihistaminics, Classical

What you can answer from here — as of May 25, 2021

101DrugsEach linked to its full drug card
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119Drug targetsEvery drug–target pair in the class, with bond type
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39,792Marketed productsAcross the regions we cover, with dosage forms and routes
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22Routes of administrationHow the drugs in this class are given
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1SubcategoryNarrower classes within this one
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Which targets do Histamine H1 Antagonists share, and which companies have late-stage candidates in this class?

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