Antibacterials for Systemic Use

Name
Antibacterials for Systemic Use
Accession Number
DBCAT002130
Description

Not Available

ATC Classification
Drugs
DrugDrug Description
DaptomycinA cyclic lipopeptide antibiotic used to treat complicated skin and skin structure infections by susceptible Gram-positive bacteria and bacteremia due to Staphylococcus aureus.
AzithromycinA macrolide antibiotic used to treat a variety of bacterial infections.
CefotiamA cephalosporin antibiotic used to treat a variety of bacterial infections.
DoxycyclineA tetracycline antibiotic used to treat a wide variety of bacterial infections.
LymecyclineA tetracycline antibiotic used for the treatment of acne vulgaris and other susceptible infections.
CefmenoximeUsed to treat female gynecologic and obstetric infections caused by susceptible aerobic (including the gonococcus) and anaerobic bacteria.
CefmetazoleA cephalosporin antibiotic used to treat a variety of bacterial infections.
FlucloxacillinA narrow spectrum penicillin antibiotic that exerts specific activity against Gram positive organisms in skin and soft tissue infections, except those caused by methicillin resistant staphylococcus aureus (MRSA).
ErtapenemA carbapenem antibiotic used for the treatment of moderate to severe infections caused by susceptible bacteria.
PiperacillinA penicillin antibiotic combined with tazobactam to treat piperacillin-resistant, piperacillin/tazobactam­ susceptible, β-lactamase generating strains of several bacteria.
AztreonamA beta-lactam antibiotic used to treat select aztreonam sensitive gram negative bacteria.
SulfadiazineA sulfonamide antibiotic used in a variety of infections, such as urinary tract infections, trachoma, and chancroid.
GrepafloxacinA fluoroquinolone antibiotic used to treat various gram positive and gram negative bacterial infections.
AmpicillinA penicillin derivative used for the treatment of a variety of infections caused by gram-positive and gram-negative bacteria as well as some anaerobes.
PhenoxymethylpenicillinA penicillin antibiotic used to prevent and treat mild to moderately severe infections in the respiratory tract, skin, and soft tissues.
CefpiramideFor treatment of severe infections caused by susceptible bacteria such as P. aeruginosa.
CeftazidimeAn injected broad-spectrum third-generation cephalosporin beta-lactam antibiotic used to treat or prevent a variety of bacterial infections, including pneumonia, gynecological infections, bone and joint infections, and septicemia, among others.
TrimethoprimAn antifolate antibiotic often used in combination with sulfamethoxazole to treat a number of infections, including those of the urinary tract, respiratory tract, and gastrointestinal tract.
LoracarbefUsed to treat upper respiratory tract bacterial infections, chronic bronchitis, pneumonia, sinusitis, pharyntitis and tonsillitis, skin absceses, urinary tract infections and pyelonephritis caused by E. coli, S. pyogenes, S. aureus,...
ClomocyclineFor the treatment and management of Brucellosis, mycoplasma infection, acne vulgaris, chlamydial infection;Chronic bronchitis
CefalotinA broad-spectrum cephalosporin antibiotic used for the treatment of serious bacterial infections in various locations, such as the urinary tract, skin, bone, and lower respiratory tract.
EnoxacinFor the treatment of adults (≥18 years of age) with the following infections caused by susceptible strains of the designated microorganisms: (1) uncomplicated urethral or cervical gonorrhea due to Neisseria...
AmikacinAn aminoglycoside used to treat infections caused by more resistant strains of Gram negative bacteria and some Gram positive bacteria.
DicloxacillinA penicillin used to treat penicillinase-producing bacterial infections that are susceptible to the drug.
PefloxacinAn antibiotic used to treat a variety of bacterial infections.
CefotaximeA third generation cephalosporin used to treat susceptible Gram negative and Gram positive bacterial infections.
VancomycinA glycopeptide antibiotic used to treat severe but susceptible bacterial infections such as MRSA (methicillin-resistant Staphylococcus aureus) infections.
CefdinirA third generation cephalosporin used to treat susceptible Gram negative and Gram positive bacterial infections.
CiprofloxacinA second generation fluoroquinolone used to treat various susceptible bacterial infections.
TigecyclineA glycylcycline antibiotic used to treat a number of susceptible bacterial infections.
CephalexinA first generation cephalosporin used to treat certain susceptible bacterial infections.
CarbenicillinFor the treatment of acute and chronic infections of the upper and lower urinary tract and in asymptomatic bacteriuria due to susceptible strains of bacteria.
LinezolidAn oxazolidinone antibiotic used to treat infections by susceptible strains of aerobic Gram-positive bacteria.
NafcillinA penicillin derivative antibiotic used to treat susceptible staphylococcal infections.
CefiximeA third generation cephalosporin used to treat susceptible Gram-negative and Gram-positive bacterial infections.
TobramycinAn aminoglycoside antibiotic used to treat cystic fibrosis-associated bacterial, lower respiratory tract, urinary tract, eye, skin, bone, and skin structure infections.
TrovafloxacinAn antibiotic used to treat gonorrhea and chlamydia.
NitrofurantoinAn antibiotic used to treat urinary tract infections.
OxacillinA penicillin antibiotic used to treat a number of susceptible bacterial infections.
HetacillinHetacillin is a beta-lactam antibiotic prodrug used to treat bacterial infections. In the body it gets converted to ampicillin.
TetracyclineAn antibiotic used to treat a wide variety of susceptible infections.
MeropenemA carbapenem antibiotic used to treat a wide variety of infections in the body.
RoxithromycinAn antibiotic used to treat a variety of susceptible bacterial infections.
Nalidixic acidA quinolone antibiotic used to treat urinary tract infections.
GentamicinAn aminoglycoside used to treat a wide variety of aerobic infections in the body.
ColistinA polymyxin antibiotic used to treat bacterial infections caused by susceptible Gram negative bacteria.
RosoxacinFor the treatment of bacterial infection of respiratory tract, urinary tract, GI, CNS and immuno compromised patients.
CinoxacinFor the treatment of initial and recurrent urinary tract infections in adults caused by the following susceptible microorganisms: Escherichia coli, Proteus mirabilis, Proteus vulgaris, Klebsiella species (including K. pneumoniae), and...
FosfomycinA broad spectrum antibiotic used to treat uncomplicated urinary tract infections.
CefaclorA second generation cephalosporin used to treat a wide variety of infections in the body.
SulfapyridineA sulfonamide antibiotic used to treat dermatitis herpetiformis, benign mucous membrane pemphigoid and pyoderma gangrenosum.
Benzylpenicilloyl polylysineA penicillin derivative used to determine penicillin allergies.
MetronidazoleA nitroimidazole used to treat trichomoniasis, amebiasis, inflammatory lesions of rosacea, and bacterial infections, as well as prevent postoperative infections.
SpectinomycinAn aminocyclitol antibiotic used to treat susceptible strains of Neisseria gonorrhoeae.
CeforanideFor the treatment of infections caused by susceptible organisms.
MetacyclineFor the treatment of acute bacterial exacerbations of chronic bronchitis
MezlocillinUsed to treat serious gram–negative infections of the lungs, urinary tract, and skin.
DirithromycinAn antibiotic used to treat a variety of respiratory, skin, and other infections.
NetilmicinAn aminoglycoside used to treat a wide variety of infections in the body.
TelithromycinAn ketolide used to treat community acquired pneumonia of mild to moderate severity.
CyclacillinFor the treatment of bacterial infections caused by susceptible organisms.
MinocyclineA tetracycline analog used to treat a wide variety of infections in the body.
GatifloxacinA fourth generation fluoroquinolone used to treat a wide variety of infections in the body.
NorfloxacinA broad-spectrum fluoroquinolone antibiotic with variable activity against gram-positive and gram-negative bacteria. Typically reserved for the treatment of UTIs due to accumulation in the urine.
AmoxicillinA penicillin derivative used for the treatment of infections caused by gram-positive bacteria, in particular streptococcal bacteria causing upper respiratory tract infections.
AzlocillinFor the treatment of infections caused by Pseudomonas aeruginosa, Escherichia coli, and Haemophilus influenzae.
CefditorenA broad-spectrum third-generation cephalosporin antibiotic typically used to treat bacterial infections of the skin and respiratory tract.
CefuroximeA cephalosporin indicated for the treatment of a variety of infections including acute bacterial otitis media, several upper respiratory tract infections, skin infections, urinary tract infections, gonorrhea, early Lyme disease, and impetigo.
LevofloxacinA fluoroquinolone antibiotic used to treat infections caused by susceptible bacteria of the upper respiratory tract, skin and skin structures, urinary tract, and prostate, as well as for post-exposure treatment of inhaled anthrax and the plague.
CefapirinA first generation cephalosporin indicated in the treatment of susceptible bacterial infections.
CefadroxilA cephalosporin antibiotic used in the treatment of various bacterial infections, such as urinary tract infections, skin and skin structure infections, and tonsillitis.
CloxacillinAn antibiotic agent used for the treatment of beta-hemolytic streptococcal and pneumococcal infections as well as staphylococcal infections.
CefprozilA cephalosporin antibiotic used in the treatment of various bacterial infections, such as pharyngitis, tonsillitis, otitis media, and uncomplicated skin infections.
GemifloxacinA quinolone antibacterial agent used for the treatment of acute bacterial exacerbation of chronic bronchitis and mild to moderate community-acquired pneumonia caused by susceptible bacteria.
AmdinocillinUsed in the treatment of urinary tract infections caused by some strains of E. coli and klebsiella and enterobacter species. Used mainly against Gram negative organisms.
OfloxacinAn antibacterial agent used for the treatment of bacterial infections in many parts of the body, including the respiratory tract, kidney, skin, soft tissue, and urinary tract.
SparfloxacinA fluoroquinolone antibiotic used to treat bacterial respiratory infections and sinusitis.
CeftriaxoneA broad-spectrum cephalosporin antibiotic used for the treatment of bacterial infections in various locations, such as in the respiratory tract, skin, soft tissue, and urinary tract.
RolitetracyclineA broad-spectrum tetracycline antibiotic used in cases needing high concentrations or when oral administration is impractical.
JosamycinA macrolide antibiotic used for the treatment of various susceptible bacterial infections.
CefamandoleA beta-lactam antibiotic used in the treatment of various infections caused by susceptible strains of bacteria, such as lower respiratory infections, urinary tract infections, skin infections, and bone and joint infections.
CefazolinA broad-spectrum cephalosporin antibiotic mainly used for the treatment of skin bacterial infections and other moderate to severe bacterial infections in the lung, bone, joint, stomach, blood, heart valve, and urinary tract.
CefonicidFor the treatment of bacterial infections caused by susceptible microorganisms.
CefoperazoneA broad-spectrum cephalosporin antibiotic used for the treatment of bacterial infections in various locations, including the respiratory tract, abdomen, skin, and female genital tracts.
CefotetanAn antibiotic medication used for the prophylaxis and treatment of various bacterial infections, including urinary tract infections, bone and joint infection, and lower respiratory tract infections.
CefoxitinA semi-synthetic, broad-spectrum antibiotic for parenteral administration used for the treatment of serious bacterial infections, such as urinary tract infection, blood infection, bone and joint infection, and lower respiratory tract infection.
CeftizoximeA third-generation cephalosporin antibiotic used in the treatment of various bacterial infections, including lower respiratory tract infection, urinary tract infection, and gonorrhea.
CefradineA first-generation cephalosporin antibiotic used in the treatment of bacterial infections of the respiratory and urinary tracts and of the skin and soft tissues.
TemafloxacinFor the treatment of lower respiratory tract infections, genital and urinary infections like prostatitis, and skin infections.
CefepimeA fourth-generation cephalosporin antibiotic used in the treatment of infections caused by susceptible bacteria, such as pneumonia, urinary tract infections, and skin infections.
CefacetrileA broad-spectrum first-generation cephalosporin used for the treatment of susceptible bacterial infections.
CeftibutenA third-generation cephalosporin antibiotic commonly used in the treatment of acute bacterial exacerbations of chronic bronchitis (ABECB), acute bacterial otitis media, pharyngitis, and tonsillitis.
CefpodoximeA third-generation cephalosporin antibiotic used in the treatment of various bacterial infections, including gonorrhea, community acquired pneumonia, and sinusitis.
NitroxolineNitroxoline is an antibiotic agent.
SulfamerazineAn antibacterial agent used in the treatment of various bacterial infections, such as bronchitis, prostatitis, and urinary tract infections.
ImipenemA carbapenem antibiotic normally administered with cilastatin to treat a variety of infections.
BacampicillinAn ampicillin prodrug used to treat various susceptible bacterial infections in the body, such as respiratory infections and skin and subcutaneous tissue infections.
MeticillinUsed to treat infections caused by susceptible Gram-positive bacteria, particularly beta-lactamase-producing organisms such as Staphylococcus aureus that would otherwise be resistant to most penicillins.
PivampicillinAn ampicillin prodrug used to treat a variety of infections.
PivmecillinamA prodrug of the beta lactam antibiotic mecillinam, indicated for the treatment of uncomplicated urinary tract infections (UTIs).
TazobactamA beta lactamase inhibitor administered with antibiotics such as piperacillin and ceftolozane to prevent their degradation, resulting in increased efficacy.
TicarcillinA beta lactam antibiotic used to treat a variety of infections in the body.
LincomycinAn antibiotic indicated only for the treatment of serious infections and is typically reserved for use in cases of penicillin allergy or where penicillin is inappropriate.
RibostamycinA broad spectrum aminoglycoside antibiotic on the list of WHO critical antimicrobials for human medicine.
LatamoxefLatamoxef is an oxacephem antibiotic usually grouped with the cephalosporins. It is used to treat bacterial infections. Latamoxef is primarily indicated in conditions like Bone and joint infection, GI infections,...
FleroxacinFleroxacin is a broad-spectrum antimicrobial fluoroquinolone.
OritavancinAn antibacterial agent used to treat acute bacterial skin and skin structure infections caused by susceptible Gram-positive bacteria.
SpiramycinA macrolide antimicrobial agent used in the treatment of various bacterial infections.
TeicoplaninA glycopeptide antibiotic with a similar mechanism of action and spectrum of activity to vancomycin used to treat various infections caused by gram-positive bacteria.
SulfadimethoxineFor use in the treatment of infections.
GarenoxacinInvestigated for use/treatment in bacterial infection.
DoripenemAn antibiotic of the penem class used to treat complicated intra-abdominal and urinary tract infections.
DalbavancinAn antibacterial used to treat acute bacterial skin and skin structure infections (ABSSSI) caused by susceptible strains of Gram-positive bacteria.
IclaprimInvestigated for use/treatment in bacterial infection, skin infections/disorders, obesity, liver disease, kidney disease, and pneumonia.
TelavancinAn antibacterial agent used in the treatment of complicated skin and skin structure infections and types of hospital-acquired bacterial pneumonia.
Ceftaroline fosamilAn antibacterial agent used to treat various bacterial infections, such as acute bacterial skin and skin structure infections and community-acquired bacterial pneumonia.
NemonoxacinInvestigated for use/treatment in bacterial infection and pneumonia.
ArbekacinArbekacin is used for the short term treatment of multi-resistant bacterial infections, such as methicillin-resistant Staphylococcus aureus (MRSA).
MethenamineA urinary tract antiseptic and antibacterial drug used for the prophylaxis and treatment of frequently recurring urinary tract infections requiring a long-term therapy.
SulfameterLong acting sulfonamide used in leprosy, urinary, and respiratory tract infections.
ThiamphenicolA semisynthetic derivative of chloramphenicol with a broad spectrum of antibacterial activity.
AzidocillinFor treatment of infection (Respiratory, GI, UTI and meningitis) due to E. coli, P. mirabilis, enterococci, Shigella, S. typhosa and other Salmonella, nonpenicillinase-producing N. gononhoeae, H. influenzae, staphylococci, streptococci including...
SulfamoxoleFor the treatment of bacterial infection.
FlumequineFlumequine is a synthetic chemotherapeutic antibiotic of the fluoroquinolone drug class used to treat bacterial infections.
CefaloridineCephaloridine or cefaloridine is a first generation semisynthetic cephalosporin. It is derived from cephalosporin C and is a zwitterion at physiological pH.
CefminoxCefminox (INN) is a second generation cephalosporin antibiotic. It is approved for use in Japan.
CarindacillinA penicillin antibiotic used to treat a variety of infections, but is no longer marketed in the USA.
Procaine benzylpenicillinA local anesthetic and antibiotic combination for intramuscular injection to treat a variety of bacterial infections while reducing pain from a deep intramuscular injection.
SulbactamAn beta-lactamase inhibitor antibiotic combined with other antibiotics to treat a variety of susceptible bacterial infections.
CefroxadineWas used for the treatment of bacterial infections.
OleandomycinOleandomycin is a macrolide antibiotic, though it is less effective than erythromycin. It is synthesized from strains of Streptomyces antibioticus.
PazufloxacinPazufloxacin is under investigation in clinical trial NCT02592096 (Pazufloxacin Mesilate Ear Drops Clinical Trial Protocol).
PrulifloxacinA broad-spectrum fluoroquinolone antibiotic used to treat a variety of susceptible bacterial infections.
FlomoxefFlomoxef has been used in trials studying the treatment of Urinary Tract Infection.
SultamicillinA mutual prodrug of ampicillin and sulbactam useful in the treatment of infections caused by beta-lactamase-producing bacteria.
FaropenemFaropenem has been used in trials studying the treatment of Tuberculosis, Pulmonary Tuberculosis, and Community Acquired Pneumonia.
TemocillinTemocillin has been investigated in Infection, Liver Dysfunction, and Urinary Tract Infection.
SisomicinSisomicin has been used in trials studying the treatment of Pyoderma.
SecnidazoleA nitroimidazole antibiotic used to treat bacterial vaginosis.
OrnidazoleA nitroimidazole agent indicated in the treatment of infections such as trichomoniasis, amebiasis, and giardiasis.
BiapenemA carbapenem antibiotic indicated in the treatment of bacterial infections.
TroleandomycinFor the treatment of bacterial infection.
ClofoctolAn antibacterial agent indicated in the treatment of respiratory infections; or prevention of infections after ear, nose, and throat surgery.
SitafloxacinA fluoroquinolone antibiotic indicated in the treatment of susceptible bacterial infections.
PenimepicyclinePenimepicycline is a tetracycline-class antibiotic. It is mentioned on List A produced by the Government of Canada, which is a list of antimicrobial active pharmaceutical ingredients . In the classification...
CefatrizineNot Annotated
DibekacinDibekacin is an aminoglycoside antibiotic marketed in Japan .
SulfaisodimidineSulfaisodimidine also called sulfisomidine is an antibacterial product that has been studied for the treatment of urinary tract infections in the 1950s, however, it is unclear whether this drug has...
MiocamycinMiocamycin is a macrolide type antimicrobial . This drug may be marketed in Japan for clinical use as it is listed in the Japanese pharmacopeia . It has shown to...
EpicillinNot Annotated
SulfaperinNot Annotated
PheneticillinPheneticillin (or phenethicillin) is a penicillin antibiotic which is approved for use internationally.
FlurithromycinNot Annotated
RokitamycinNot Annotated
MidecamycinA macrolide antibiotic used to treat a variety of infections caused by susceptible bacteria.
CefcapeneNot Annotated
CefodizimeA broad-spectrum, third-generation cephalosporin used to treat serious infections caused by susceptible bacteria.
FurazidinNot Annotated
SulfametomidineNot Annotated
CefsulodinNot Annotated
CefetametNot Annotated
IsepamicinNot Annotated
CarumonamNot Annotated
SulfamazoneNot Annotated
Oxolinic acidNot Annotated
CefbuperazoneNot Annotated
PropicillinNot Annotated
CefozopranNot Annotated
BekanamycinAn aminoglycoside antibiotic indicated in the treatment of eye infections.
CefpiromeAn antibiotic indicated in the treatment of a wide variety of infections in the body.
ClometocillinNot Annotated
SulbenicillinNot Annotated
SulfathioureaNot Annotated
PristinamycinNot Annotated
XibornolA lipophilic antiseptic indicated as an adjunct in the treatment of susceptible oral infections.
NifurtoinolNot Annotated
PenamecillinNot Annotated
Piromidic acidNot Annotated
RufloxacinA fluoroquinolone antibiotic indicated in the treatment of susceptible respiratory infections and uncomplicated cystitis.
SulfamethoxypyridazineA sulphonamide antibiotic indicated in the treatment of gonorrhea, inflammation, urinary tract ulcers, and bronchitis.
CefazedoneNot Annotated
BrodimoprimNot Annotated
TalampicillinNot Annotated
AspoxicillinNot Annotated
CeftezoleNot Annotated
Pipemidic acidA quinolone antibiotic indicated in the treatment of susceptible urinary tract infections.
MetampicillinMetampicillin is a penicillin antibiotic prepared by the reaction of ampicillin with formaldehyde. It is hydrolysed in aqueous solution to form ampicillin. Hydrolysis is rapid under acid conditions like the...
ErythromycinA macrolide antibiotic used to treat and prevent a variety of bacterial infections.
MoxifloxacinA fluoroquinolone antibiotic used to treat various bacterial infections.
SulfanilamideA sulfonamide anti-infective used to treat vulvovaginal candidiasis caused by Candida albicans.
SulfisoxazoleA sulfonamide antibiotic used with other antibiotics to prevent and treat a variety of bacterial infections.
ChloramphenicolA broad spectrum antibiotic that is effective against a variety of susceptible and serious bacterial infections but is not frequently used because of its high risk of bone marrow toxicity.
SulfamethizoleA sulfonamide antibiotic used to treat a wide variety of susceptible bacterial infections.
OxytetracyclineA tetracycline antibiotic used to treat a wide variety of susceptible bacterial infections.
DemeclocyclineA tetracycline antibiotic used to treat a wide variety of susceptible bacterial infections.
BacitracinA cyclic polypeptide antibiotic used to prevent wound infections, treat pneumonia and empyema in infants, and to treat skin and eye infections.
SulfametopyrazineAn antibiotic used in the treatment or prevention of bacterial infections and malaria.
TinidazoleA nitroimidazole used to treat trichomoniasis, giardiasis, amebiasis, and bacterial vaginosis.
LomefloxacinA fluoroquinolone used to prevent and treat a wide variety of infections in the body.
NeomycinAn aminoglycoside antibiotic agent used orally and topically to treat a wide variety of infections in the body.
SulfamethoxazoleAn oral sulfonamide antibiotic, given in combination with trimethoprim, used to treat a variety of infections of the urinary tract, respiratory system, and gastrointestinal tract.
BenzylpenicillinA penicillin used for the treatment of infections caused by gram-positive cocci, in particular streptococcal infections. This form of penicillin is typically used in intravenous or long-acting injectable formulations due to poor oral absorption.
StreptomycinAn aminoglycoside antibiotic indicated to treat multi-drug resistant mycobacterium tuberculosis and various non-tuberculosis infections.
KanamycinAn aminoglycoside antibiotic agent used in the treatment of various infections caused by susceptible bacteria.
ClindamycinA lincosamide antibiotic used to treat serious infections caused by susceptible anaerobic, streptococcal, staphylococcal, and pneumococcal bacteria.
ClarithromycinA macrolide antibiotic used for the treatment of a wide variety of bacterial infections such as acute otitis, pharyngitis, tonsillitis, respiratory tract infections, uncomplicated skin infections, and helicobacter pylori infection.
SulfamethazineAn antibacterial agent used in the treatment of various bacterial infections, such as bronchitis, prostatitis, and urinary tract infections.
Fusidic acidA topical antibacterial agent used to prevent and treat mild to moderate skin infections caused by susceptible bacteria.
SulfathiazoleSulfathiazole is effective against a wide range of gram positive and gram negative pathogenic microorganisms. Although no longer used in humans, it is used in cattle.
SulfaphenazoleFor the treatment bacterial infections.
ChlortetracyclineThe first tetracycline antibiotic most commonly used for veterinary purposes.
Mandelic acidMandelic acid is an approved aromatic, alpha hydroxy acid . Mandelic acid is used as an ingredient in cosmetics and drug products applied topically.
TedizolidAn oxazolidinone class antibiotic that inhibits bacterial protein synthesis and is proven to be effective in the treatment of certain Gram-positive bacterial infections.
SarecyclineA tetracycline antibiotic used to treat inflammatory lesions of non-nodular moderate to severe acne vulgaris.
OmadacyclineA tetracycline antibiotic used to treat community acquired bacterial pneumonia.
Ceftobiprole medocarilA cephalosporin indicated in the treatment of pneumonia.
SolithromycinInvestigated for the treatment of community-acquired pneumonia (CAP).
DelafloxacinA fluoroquinolone antibiotic used to treat skin and skin structure infections.
VaborbactamA beta lactamase inhibitor used to treat complicated urinary tract infections.
EravacyclineA tetracycline antibiotic used to treat complicated intra-abdominal infections.
Polymyxin BA polymyxin antibiotic used to treat a wide variety of infections in the body.
PlazomicinAn aminoglycoside antibiotic used to treat complicated urinary tract infections.
LefamulinA pleuromutilin antibacterial used to treat community-acquired bacterial pneumonia (CABP).
SulfametroleAn antibiotic indicated in combination intravenous products for various bacterial infections.
TetroxoprimNot Annotated
Tebipenem pivoxilNot Annotated
TosufloxacinNot Annotated
RelebactamA beta-lactamase inhibitor used to prevent hydrolysis of beta-lactam antibiotics, leading to increased effectiveness.
CefiderocolA cephalosporin antibiotic used in complicated urinary tract infections.
LevonadifloxacinLevonadifloxacin is under investigation in clinical trial NCT03405064 (Comparative Study of Levonadifloxacin (IV and Oral) With Linezolid (IV and Oral) in Acute Bacterial Skin and Skin Structure Infections (ABSSSI)).
Drugs & Drug Targets
DrugTargetType
DaptomycinCytoplasmic membranetarget
DaptomycinSerum albumincarrier
DaptomycinAlpha-1-acid glycoprotein 1carrier
DaptomycinAlpha-1-antitrypsincarrier
DaptomycinLow-density lipoprotein receptorcarrier
DaptomycinSex hormone-binding globulincarrier
DaptomycinHemopexincarrier
DaptomycinP-glycoprotein 1transporter
Azithromycin23S ribosomal RNAtarget
AzithromycinP-glycoprotein 1transporter
AzithromycinCytochrome P450 3A4enzyme
AzithromycinProtein-arginine deiminase type-4target
AzithromycinCanalicular multispecific organic anion transporter 1transporter
CefotiamPenicillin-binding protein 1Atarget
CefotiamSolute carrier family 22 member 6transporter
CefotiamSolute carrier family 22 member 8transporter
DoxycyclineSolute carrier family 22 member 6transporter
DoxycyclineCytochrome P450 3A4enzyme
DoxycyclineATP-binding cassette sub-family B member 5transporter
DoxycyclineSerum albumincarrier
Doxycycline30S ribosomal proteintarget
Lymecycline30S ribosomal protein S4target
CefmenoximePenicillin-binding protein 1Atarget
CefmenoximePeptidoglycan synthase FtsItarget
CefmetazolePenicillin binding protein 2atarget
CefmetazoleSerum albumincarrier
CefmetazoleSolute carrier family 15 member 1transporter
CefmetazoleSolute carrier family 15 member 2transporter
CefmetazolePenicillin-binding protein 1Atarget
CefmetazolePenicillin-binding protein 1Btarget
CefmetazolePeptidoglycan synthase FtsItarget
CefmetazoleD-alanyl-D-alanine carboxypeptidase DacAtarget
CefmetazoleD-alanyl-D-alanine carboxypeptidase DacCtarget
FlucloxacillinPenicillin-binding protein 1Atarget
FlucloxacillinCytochrome P450 3A4enzyme
FlucloxacillinBile salt export pumptransporter
ErtapenemPenicillin-binding protein 2target
ErtapenemPeptidoglycan synthase FtsItarget
ErtapenemPenicillin-binding protein 1Atarget
ErtapenemD-alanyl-D-alanine carboxypeptidase DacCtarget
ErtapenemD-alanyl-D-alanine carboxypeptidase DacBtarget
ErtapenemPenicillin-binding protein 1Btarget
ErtapenemPeptidoglycan synthase FtsItarget
ErtapenemPenicillin-binding protein 2target
ErtapenemSerum albumincarrier
ErtapenemDipeptidase 1enzyme
PiperacillinSolute carrier family 22 member 6transporter
PiperacillinPenicillin-binding protein 3target
PiperacillinPenicillin-binding protein 2Btarget
PiperacillinPenicillin-binding protein 2atarget
PiperacillinPenicillin-binding protein 1btarget
PiperacillinSolute carrier family 22 member 8transporter
AztreonamPenicillin-binding protein 3target
AztreonamBeta-lactamasetarget
AztreonamBeta-lactamase Toho-1target
SulfadiazineCytochrome P450 2C9enzyme
SulfadiazineDihydropteroate synthetasetarget
SulfadiazineCytochrome P450 2C8enzyme
SulfadiazineCytochrome P450 3A4enzyme
GrepafloxacinDNA gyrase subunit Atarget
GrepafloxacinDNA topoisomerase 4 subunit Atarget
GrepafloxacinCytochrome P450 3A4enzyme
GrepafloxacinCytochrome P450 1A2enzyme
GrepafloxacinSolute carrier family 22 member 2transporter
GrepafloxacinSolute carrier family 22 member 5transporter
GrepafloxacinCanalicular multispecific organic anion transporter 1transporter
GrepafloxacinP-glycoprotein 1transporter
GrepafloxacinMultidrug resistance-associated protein 1transporter
GrepafloxacinSolute carrier family 22 member 6transporter
AmpicillinSerum albumincarrier
AmpicillinSolute carrier family 22 member 5transporter
AmpicillinSolute carrier family 15 member 1transporter
AmpicillinSolute carrier family 15 member 2transporter
AmpicillinPenicillin-binding protein 2atarget
AmpicillinPenicillin-binding protein 1btarget
AmpicillinPenicillin-binding protein 3target
AmpicillinPenicillin-binding protein 1Atarget
AmpicillinPenicillin-binding protein 2Btarget
AmpicillinMonocarboxylate transporter 1transporter
AmpicillinSolute carrier family 15 member 1target
AmpicillinSolute carrier family 15 member 2target
AmpicillinAngiopoietin-1 receptortarget
PhenoxymethylpenicillinPenicillin-binding protein 1Atarget
PhenoxymethylpenicillinMecA PBP2' (penicillin binding protein 2')target
PhenoxymethylpenicillinD-alanyl-D-alanine carboxypeptidase DacBtarget
PhenoxymethylpenicillinPenicillin acylasetarget
PhenoxymethylpenicillinSolute carrier family 15 member 1target
CefpiramidePenicillin binding protein 2atarget
CefpiramideSerum albumincarrier
CefpiramidePeptidoglycan synthase FtsItarget
CefpiramidePenicillin-binding protein 1Btarget
CefpiramidePenicillin-binding protein 1Atarget
CefpiramidePenicillin-binding protein 1Btarget
CefpiramideD-alanyl-D-alanine carboxypeptidase DacCtarget
CefpiramidePenicillin-binding protein 1Atarget
CeftazidimeSolute carrier family 22 member 6transporter
CeftazidimePeptidoglycan synthase FtsItarget
CeftazidimePenicillin-binding protein 1Atarget
CeftazidimePenicillin-binding protein 1Btarget
CeftazidimePenicillin-binding protein 2target
CeftazidimeSerum albumincarrier
CeftazidimeBeta-lactamase Toho-1target
TrimethoprimDihydrofolate reductasetarget
TrimethoprimCytochrome P450 2C8enzyme
TrimethoprimCytochrome P450 3A4enzyme
TrimethoprimP-glycoprotein 1transporter
TrimethoprimCytochrome P450 2C9enzyme
TrimethoprimCytochrome P450 1A2enzyme
TrimethoprimMultidrug and toxin extrusion protein 1transporter
TrimethoprimMultidrug and toxin extrusion protein 2transporter
LoracarbefPenicillin-binding protein 1Atarget
LoracarbefSolute carrier family 15 member 1transporter
LoracarbefSolute carrier family 15 member 2transporter
LoracarbefPenicillin-binding protein 3target
Clomocycline30S ribosomal protein S4target
Clomocycline30S ribosomal protein S9target
Clomocycline16S ribosomal RNAtarget
CefalotinPenicillin-binding protein 1Atarget
CefalotinD-alanyl-D-alanine carboxypeptidasetarget
CefalotinBeta-lactamasetarget
CefalotinSolute carrier family 22 member 5transporter
CefalotinSolute carrier family 15 member 1transporter
CefalotinSolute carrier family 15 member 2transporter
CefalotinSolute carrier family 22 member 6transporter
CefalotinSolute carrier family 22 member 8transporter
CefalotinSolute carrier family 22 member 11transporter
CefalotinSolute carrier family 22 member 7transporter
CefalotinPenicillin-binding protein 1Atarget
CefalotinPenicillin-binding protein 1btarget
CefalotinPenicillin-binding protein 3target
CefalotinPenicillin-binding protein 2atarget
CefalotinPenicillin-binding protein 2Btarget
CefalotinSerum albumincarrier
EnoxacinDNA gyrase subunit Atarget
EnoxacinDNA topoisomerase 4 subunit Atarget
EnoxacinDNA topoisomerase 2-alphatarget
EnoxacinCytochrome P450 1A2enzyme
Amikacin30S ribosomal protein S12target
DicloxacillinSolute carrier family 15 member 1transporter
DicloxacillinSolute carrier family 15 member 2transporter
DicloxacillinPenicillin-binding protein 3target
DicloxacillinPenicillin-binding protein 1btarget
DicloxacillinPenicillin-binding protein 2atarget
DicloxacillinPenicillin-binding protein 3target
DicloxacillinPenicillin-binding protein 1Atarget
DicloxacillinPenicillin-binding protein 2Btarget
DicloxacillinCytochrome P450 3A4enzyme
DicloxacillinSerum albumincarrier
PefloxacinDNA gyrase subunit Atarget
PefloxacinDNA topoisomerase 4 subunit Atarget
PefloxacinDNA topoisomerase 2-alphatarget
PefloxacinCytochrome P450 1A2enzyme
PefloxacinDNA topoisomerase 1target
CefotaximePenicillin-binding protein 3target
CefotaximeSolute carrier family 15 member 1transporter
CefotaximeSolute carrier family 15 member 2transporter
CefotaximeSolute carrier family 22 member 6transporter
CefotaximeSolute carrier family 22 member 8transporter
CefotaximeSolute carrier family 22 member 11transporter
CefotaximeSolute carrier family 22 member 7transporter
CefotaximePenicillin-binding protein 1btarget
CefotaximePenicillin-binding protein 2atarget
CefotaximePenicillin-binding protein 1Atarget
CefotaximePenicillin-binding protein 2Btarget
CefotaximeSolute carrier family 22 member 6target
CefotaximeSolute carrier family 22 member 8target
CefotaximeSolute carrier family 22 member 11target
CefotaximeSolute carrier family 22 member 7target
CefotaximeSolute carrier family 15 member 1target
CefotaximeSerum albumintarget
CefotaximeBeta-lactamasetarget
CefotaximeSolute carrier family 15 member 2target
VancomycinD-Ala-D-Ala moiety of NAM/NAG peptide subunits of peptidoglycantarget
VancomycinSerum albumincarrier
Vancomycinalpha1-acid glycoproteincarrier
VancomycinHistamine H1 receptorcarrier
CefdinirMyeloperoxidasetarget
CefdinirPenicillin-binding protein 2target
CefdinirPBP3target
CefdinirSolute carrier family 22 member 5transporter
CefdinirSolute carrier family 15 member 1transporter
CefdinirSolute carrier family 15 member 2transporter
CefdinirSolute carrier family 22 member 6transporter
CefdinirSolute carrier family 22 member 8transporter
CefdinirPeptidoglycan transpeptidasetarget
CiprofloxacinDNA gyrase subunit Atarget
CiprofloxacinDNA topoisomerase 4 subunit Atarget
CiprofloxacinDNA topoisomerase 2-alphatarget
CiprofloxacinCytochrome P450 1A2enzyme
CiprofloxacinCytochrome P450 3A4enzyme
CiprofloxacinCytochrome P450 3A5enzyme
CiprofloxacinCytochrome P450 3A7enzyme
CiprofloxacinP-glycoprotein 1transporter
CiprofloxacinPotassium voltage-gated channel subfamily H member 2target
CiprofloxacinDNA gyrase subunit Atarget
CiprofloxacinDNA topoisomerase 4 subunit Atarget
CiprofloxacinDNA topoisomerase 4 subunit Btarget
CiprofloxacinDNA gyrase subunit Atarget
CiprofloxacinMultidrug resistance protein MdtKtarget
CiprofloxacinGyrase Atarget
CiprofloxacinDNA gyrase subunit Atarget
CiprofloxacinMultidrug and toxin extrusion protein 1transporter
CiprofloxacinMultidrug and toxin extrusion protein 2transporter
CiprofloxacinSerum albumincarrier
Tigecycline30S ribosomal protein S9target
Tigecycline16S ribosomal RNAtarget
Tigecycline30S ribosomal protein S14target
Tigecycline30S ribosomal protein S13target
Tigecycline30S ribosomal protein S19target
Tigecycline30S ribosomal protein S12target
CephalexinSerum albumincarrier
CephalexinSolute carrier family 22 member 5transporter
CephalexinSolute carrier family 15 member 1transporter
CephalexinSolute carrier family 15 member 2transporter
CephalexinSolute carrier family 22 member 6transporter
CephalexinSolute carrier family 22 member 8transporter
CephalexinMultidrug and toxin extrusion protein 1transporter
CephalexinPenicillin-binding protein 3target
CephalexinPenicillin-binding protein 2atarget
CephalexinPenicillin-binding protein 1btarget
CephalexinPenicillin-binding protein 1Atarget
CephalexinPenicillin-binding protein 2Btarget
CarbenicillinSolute carrier family 22 member 6transporter
CarbenicillinPenicillin-binding proteintarget
CarbenicillinCytosolic phospholipase A2enzyme
CarbenicillinBeta-lactamase Toho-1target
Linezolid23S ribosomal RNAtarget
LinezolidAmine oxidase [flavin-containing] Aenzyme
LinezolidAmine oxidase [flavin-containing] Benzyme
LinezolidSerum albumincarrier
LinezolidSolute carrier family 22 member 6transporter
LinezolidSolute carrier family 22 member 8transporter
NafcillinCytochrome P450 1A2enzyme
NafcillinCytochrome P450 3A4enzyme
NafcillinSolute carrier family 22 member 6transporter
NafcillinPenicillin-binding protein 1btarget
NafcillinPenicillin-binding protein 2Btarget
NafcillinPenicillin-binding protein 2atarget
NafcillinPenicillin-binding protein 3target
NafcillinPenicillin-binding protein 1Atarget
NafcillinSerum albumincarrier
CefiximePenicillin-binding protein 2target
CefiximeSolute carrier family 22 member 5transporter
CefiximeSolute carrier family 15 member 1transporter
CefiximeSolute carrier family 15 member 2transporter
Tobramycin16S ribosomal RNAtarget
TobramycinBacterial outer membranetarget
TobramycinCytoplasmic membranetarget
Tobramycin23S ribosomal RNAtarget
TrovafloxacinDNA gyrase subunit Atarget
TrovafloxacinDNA topoisomerase 4 subunit Atarget
TrovafloxacinDNA topoisomerase 2-alphatarget
TrovafloxacinCytochrome P450 1A2enzyme
Nitrofurantoin30S ribosomal protein S10target
NitrofurantoinOxygen-insensitive NADPH nitroreductasetarget
NitrofurantoinProbable pyruvate-flavodoxin oxidoreductasetarget
NitrofurantoinATP-binding cassette sub-family G member 2transporter
NitrofurantoinNADPH--cytochrome P450 reductaseenzyme
NitrofurantoinBile salt export pumptransporter
NitrofurantoinP-glycoprotein 1transporter
NitrofurantoinCanalicular multispecific organic anion transporter 1transporter
OxacillinPenicillin-binding protein 1Atarget
OxacillinSolute carrier family 15 member 1transporter
OxacillinSolute carrier family 15 member 2transporter
OxacillinPenicillin-binding protein 3target
OxacillinPenicillin-binding protein 2atarget
OxacillinPenicillin-binding protein 1Atarget
OxacillinPenicillin-binding protein 2Btarget
OxacillinPenicillin-binding protein 1btarget
OxacillinSolute carrier family 15 member 1target
OxacillinPenicillin-binding protein 2target
OxacillinSolute carrier family 15 member 2target
OxacillinBeta-lactamase Toho-1target
HetacillinPenicillin-binding protein 2atarget
HetacillinPenicillin-binding protein 1btarget
HetacillinPenicillin-binding protein 3target
HetacillinPenicillin-binding protein 1Atarget
HetacillinPenicillin-binding protein 2Btarget
Tetracycline16S ribosomal RNAtarget
TetracyclineMajor prion proteintarget
TetracyclineSerum albumincarrier
TetracyclineCytochrome P450 3A4enzyme
TetracyclineSolute carrier family 22 member 6transporter
TetracyclineSolute carrier family 22 member 8transporter
TetracyclineSolute carrier family 22 member 11transporter
TetracyclineSolute carrier family 22 member 7transporter
Tetracycline30S ribosomal protein S3target
Tetracycline30S ribosomal protein S8target
Tetracycline30S ribosomal protein S19target
Tetracycline30S ribosomal protein S14target
Tetracycline30S ribosomal protein S7target
TetracyclineMultidrug translocase MdfAtarget
TetracyclineProtein-arginine deiminase type-4target
TetracyclineSolute carrier organic anion transporter family member 2B1transporter
MeropenemD-alanyl-D-alanine carboxypeptidase DacBtarget
MeropenemBeta-lactamase OXA-10enzyme
MeropenemDipeptidase 1enzyme
Roxithromycin50S ribosomal protein L10target
RoxithromycinP-glycoprotein 1target
RoxithromycinCytochrome P450 3A4enzyme
RoxithromycinCytochrome P450 2B6enzyme
Nalidixic acidDNAtarget
Nalidixic acidSolute carrier family 22 member 6transporter
Nalidixic acidTryptophan 2,3-dioxygenaseenzyme
Nalidixic acidCytochrome P450 1A2enzyme
Gentamicin30S ribosomal protein S12target
Gentamicin16S ribosomal RNAtarget
GentamicinNH(3)-dependent NAD(+) synthetasetarget
GentamicinDihydrofolate reductasetarget
Gentamicin23S ribosomal RNAtarget
GentamicinBacterial outer membranetarget
GentamicinCytoplasmic membranetarget
GentamicinLow-density lipoprotein receptor-related protein 2transporter
GentamicinSolute carrier family 22 member 2transporter
GentamicinCanalicular multispecific organic anion transporter 1transporter
ColistinBacterial outer membranetarget
RosoxacinDNA topoisomerase 4 subunit Atarget
RosoxacinDNA gyrase subunit Btarget
RosoxacinCytochrome P450 1A2enzyme
CinoxacinDNAtarget
CinoxacinDNA gyrase subunit Atarget
CinoxacinSolute carrier family 22 member 6transporter
CinoxacinCytochrome P450 1A2enzyme
FosfomycinUDP-N-acetylglucosamine 1-carboxyvinyltransferasetarget
CefaclorPenicillin-binding protein 1Atarget
CefaclorSolute carrier family 15 member 1transporter
CefaclorSolute carrier family 15 member 2transporter
CefaclorPenicillin-binding protein 3target
CefaclorMyeloperoxidaseenzyme
CefaclorSolute carrier family 22 member 8transporter
CefaclorBile salt export pumptransporter
SulfapyridineDihydropteroate synthase type-1target
SulfapyridineCytochrome P450 2C9enzyme
Benzylpenicilloyl polylysineHigh affinity immunoglobulin epsilon receptor subunit gammatarget
Benzylpenicilloyl polylysineHigh affinity immunoglobulin epsilon receptor subunit alphatarget
MetronidazoleOxygen-insensitive NADPH nitroreductasetarget
MetronidazoleCytochrome P450 2C9enzyme
MetronidazoleCytochrome P450 3A4enzyme
MetronidazoleCytochrome P450 2C8enzyme
MetronidazoleUDP-glucuronosyltransferase 1-1enzyme
MetronidazoleAnaerobic bacterial DNAtarget
MetronidazoleProtozoal DNAtarget
MetronidazoleP-glycoprotein 1transporter
MetronidazoleCytochrome P450 2A6enzyme
MetronidazoleCytochrome P450 3A5enzyme
MetronidazoleCytochrome P450 3A7enzyme
Spectinomycin30S ribosomal protein S12target
CeforanidePenicillin-binding protein 2target
MetacyclineSerum albumincarrier
Metacycline16S ribosomal RNAtarget
MezlocillinPenicillin-binding protein 1Atarget
MezlocillinPenicillin-binding protein 2target
MezlocillinPenicillin-binding protein 3target
Dirithromycin23S ribosomal RNAtarget
DirithromycinCytochrome P450 3A4enzyme
Netilmicin30S ribosomal protein S12target
Netilmicin16S ribosomal RNAtarget
Telithromycin23S ribosomal RNAtarget
TelithromycinCytochrome P450 3A4enzyme
TelithromycinSolute carrier organic anion transporter family member 1B1transporter
TelithromycinSolute carrier organic anion transporter family member 1B3transporter
CyclacillinSolute carrier family 22 member 5transporter
CyclacillinSolute carrier family 15 member 1transporter
CyclacillinSolute carrier family 15 member 2transporter
CyclacillinPenicillin-binding protein 1Atarget
CyclacillinPenicillin-binding protein 3target
CyclacillinPenicillin binding protein 2atarget
CyclacillinPenicillin-binding proteintarget
Minocycline30S ribosomal protein S4target
Minocycline30S ribosomal protein S9target
Minocycline16S ribosomal RNAtarget
MinocyclineInterleukin-1 betatarget
MinocyclineArachidonate 5-lipoxygenasetarget
MinocyclineMatrix metalloproteinase-9target
MinocyclineVascular endothelial growth factor Atarget
MinocyclineCaspase-1target
MinocyclineCaspase-3target
MinocyclineCytochrome ctarget
MinocyclineSolute carrier family 22 member 6transporter
MinocyclineSolute carrier family 22 member 7transporter
MinocyclineOuter membrane protein Ftransporter
MinocyclineOuter membrane porin Ctransporter
MinocyclineMitogen-activated Protein Kinasestarget
MinocyclineNitric oxide synthase, inducibletarget
GatifloxacinSerum albumincarrier
GatifloxacinDNA gyrase subunit Atarget
GatifloxacinDNA gyrase subunit Btarget
GatifloxacinDNA topoisomerase 4 subunit Atarget
GatifloxacinDNA topoisomerase 4 subunit Btarget
GatifloxacinCytochrome P450 1A2enzyme
NorfloxacinDNA gyrase subunit Atarget
NorfloxacinDNA topoisomerase 4 subunit Atarget
NorfloxacinDNA topoisomerase 2-alphatarget
NorfloxacinCytochrome P450 1A2enzyme
NorfloxacinCytochrome P450 3A4enzyme
NorfloxacinSolute carrier family 22 member 5transporter
NorfloxacinSolute carrier family 22 member 6transporter
NorfloxacinCytochrome P450 1A1enzyme
NorfloxacinCytochrome P450 3A7enzyme
NorfloxacinDNA gyrase subunit Atarget
NorfloxacinDNA topoisomerase 2target
NorfloxacinDNA topoisomerase 4 subunit Atarget
AmoxicillinSolute carrier family 15 member 1transporter
AmoxicillinSolute carrier family 15 member 2transporter
AmoxicillinSolute carrier family 22 member 6transporter
AmoxicillinCytochrome P450 2C8enzyme
AmoxicillinSerum albumincarrier
AmoxicillinBeta-lactamase 2enzyme
AmoxicillinPenicillin binding proteintarget
AzlocillinPenicillin-binding protein 1Atarget
CefditorenPenicillin-binding protein 1Atarget
CefditorenPenicillin-binding protein 2Btarget
CefuroximePenicillin-binding protein 1Atarget
CefuroximeSolute carrier family 15 member 1transporter
CefuroximeSolute carrier family 15 member 2transporter
LevofloxacinDNA gyrase subunit Atarget
LevofloxacinDNA topoisomerase 4 subunit Atarget
LevofloxacinSolute carrier family 22 member 2transporter
LevofloxacinP-glycoprotein 1transporter
LevofloxacinSolute carrier family 22 member 4transporter
LevofloxacinMultidrug and toxin extrusion protein 1transporter
LevofloxacinMultidrug and toxin extrusion protein 2transporter
LevofloxacinCytochrome P450 2C9enzyme
LevofloxacinSerum albumincarrier
LevofloxacinSolute carrier organic anion transporter family member 4C1transporter
LevofloxacinSolute carrier family 22 member 1transporter
LevofloxacinSolute carrier organic anion transporter family member 1A2transporter
CefapirinPenicillin-binding protein 1Atarget
CefadroxilSolute carrier family 22 member 5transporter
CefadroxilSolute carrier family 15 member 1transporter
CefadroxilSolute carrier family 15 member 2transporter
CefadroxilSolute carrier family 22 member 6transporter
CefadroxilSolute carrier family 22 member 8transporter
CefadroxilPenicillin-binding protein 3target
CefadroxilPenicillin-binding protein 1Atarget
CefadroxilPenicillin-binding protein 1btarget
CefadroxilPenicillin-binding protein 2Btarget
CloxacillinSerum albumincarrier
CloxacillinSolute carrier family 15 member 1transporter
CloxacillinSolute carrier family 15 member 2transporter
CloxacillinD-alanyl-D-alanine carboxypeptidase DacAtarget
CloxacillinSolute carrier family 22 member 8transporter
CloxacillinPenicillin-binding protein 2Xtarget
CloxacillinPenicillin-binding protein 1Atarget
CefprozilPenicillin-binding protein 1Atarget
CefprozilPenicillin-binding protein 2xtarget
CefprozilPenicillin-binding protein 2Btarget
GemifloxacinDNA gyrase subunit Atarget
GemifloxacinDNA topoisomerase 4 subunit Atarget
GemifloxacinCytochrome P450 1A2enzyme
AmdinocillinPenicillin-binding protein 2target
AmdinocillinPenicillin-binding protein 2atarget
AmdinocillinPenicillin-binding protein 3target
AmdinocillinPenicillin-binding protein 1Atarget
AmdinocillinPenicillin-binding protein 2Btarget
AmdinocillinPenicillin-binding protein 1btarget
OfloxacinDNA gyrase subunit Atarget
OfloxacinDNA topoisomerase 4 subunit Atarget
OfloxacinDNA topoisomerase 2-alphatarget
OfloxacinCytochrome P450 1A2enzyme
OfloxacinSolute carrier family 22 member 5transporter
OfloxacinMultidrug resistance-associated protein 1transporter
OfloxacinSolute carrier family 22 member 6transporter
OfloxacinCanalicular multispecific organic anion transporter 1transporter
OfloxacinSolute carrier family 22 member 4transporter
OfloxacinBile salt export pumptransporter
SparfloxacinDNA gyrase subunit Atarget
SparfloxacinDNA topoisomerase 4 subunit Atarget
SparfloxacinDNA topoisomerase 2-alphatarget
SparfloxacinSolute carrier family 22 member 5transporter
SparfloxacinCanalicular multispecific organic anion transporter 1transporter
SparfloxacinP-glycoprotein 1transporter
SparfloxacinCytochrome P450 1A2enzyme
CeftriaxoneSerum albumincarrier
CeftriaxoneSolute carrier family 15 member 1transporter
CeftriaxoneSolute carrier family 15 member 2transporter
CeftriaxoneSolute carrier family 22 member 6transporter
CeftriaxoneSolute carrier family 22 member 8transporter
CeftriaxoneSolute carrier family 22 member 11transporter
CeftriaxonePenicillin-binding protein 2Btarget
CeftriaxoneGlutamine synthetaseenzyme
CeftriaxoneSolute carrier family 22 member 11target
CeftriaxoneSolute carrier family 22 member 6target
CeftriaxoneSolute carrier family 22 member 8target
CeftriaxoneSolute carrier family 15 member 1target
CeftriaxoneP-glycoprotein 1transporter
Rolitetracycline30S ribosomal protein S9target
Rolitetracycline16S ribosomal RNAtarget
Josamycin50S ribosomal protein L4target
CefamandoleSolute carrier family 22 member 6transporter
CefamandoleSolute carrier family 22 member 8transporter
CefamandoleSolute carrier family 22 member 11transporter
CefamandoleSolute carrier family 22 member 7transporter
CefamandolePenicillin-binding protein 2target
CefazolinSerum paraoxonase/arylesterase 1target
CefazolinSerum albumincarrier
CefazolinSolute carrier family 22 member 6transporter
CefazolinSolute carrier family 22 member 8transporter
CefazolinSolute carrier family 22 member 11transporter
CefazolinPenicillin-binding protein 1Atarget
CefazolinPenicillin-binding protein 1Btarget
CefazolinPenicillin-binding protein 2target
CefazolinPenicillin-binding protein 1Ctarget
CefazolinPeptidoglycan synthase FtsItarget
CefazolinMultidrug resistance-associated protein 4transporter
CefazolinThiopurine S-methyltransferaseenzyme
CefazolinInterleukin-15target
CefazolinInterleukin-2target
CefonicidSerum albumincarrier
CefonicidPenicillin-binding protein 1Atarget
CefonicidPeptidoglycan synthase FtsItarget
CefonicidPenicillin-binding protein 1Btarget
CefonicidD-alanyl-D-alanine carboxypeptidase DacBtarget
CefonicidPenicillin-binding protein 2target
CefoperazoneSerum albumincarrier
CefoperazoneSolute carrier family 22 member 6transporter
CefoperazoneSolute carrier family 22 member 8transporter
CefoperazoneSolute carrier family 22 member 11transporter
CefoperazoneSolute carrier family 22 member 7transporter
CefoperazonePeptidoglycan synthase FtsItarget
CefoperazonePenicillin-binding protein 1Btarget
CefoperazonePenicillin-binding protein 2target
CefoperazonePenicillin-binding protein 1Atarget
CefoperazoneD-alanyl-D-alanine carboxypeptidase DacCtarget
CefoperazoneD-alanyl-D-alanine carboxypeptidase DacAtarget
CefoperazoneD-alanyl-D-alanine carboxypeptidase DacBtarget
CefoperazonePenicillin-binding protein 1Atarget
CefoperazonePenicillin-binding protein 1Btarget
CefotetanSerum albumincarrier
CefotetanPenicillin-binding protein 3target
CefoxitinPenicillin-binding protein 1Atarget
CefoxitinPenicillin-binding protein 1Btarget
CefoxitinPeptidoglycan synthase FtsItarget
CefoxitinD-alanyl-D-alanine carboxypeptidase DacAtarget
CefoxitinD-alanyl-D-alanine carboxypeptidase DacBtarget
CefoxitinD-alanyl-D-alanine carboxypeptidase DacCtarget
CefoxitinD-alanyl-D-alanine endopeptidasetarget
CefoxitinBeta-lactamaseenzyme
CefoxitinPenicillin-binding protein 3target
CefoxitinPenicillin-binding protein 1btarget
CefoxitinPenicillin-binding protein 2atarget
CefoxitinPenicillin-binding protein 1Atarget
CefoxitinPenicillin-binding protein 2Btarget
CeftizoximeSolute carrier family 15 member 1transporter
CeftizoximePenicillin-binding protein 1Atarget
CeftizoximePenicillin-binding protein 1Btarget
CeftizoximeSolute carrier family 22 member 6transporter
CeftizoximeSolute carrier family 22 member 8transporter
CeftizoximePeptidoglycan transpeptidasetarget
CeftizoximeD-alanyl-D-alanine carboxypeptidase DacCtarget
CefradineSolute carrier family 22 member 5transporter
CefradineSolute carrier family 15 member 1transporter
CefradineSolute carrier family 15 member 2transporter
CefradineSolute carrier family 22 member 6transporter
CefradinePenicillin-binding protein 1Atarget
CefradineCytochrome P450 3A4enzyme
CefradineMultidrug and toxin extrusion protein 1transporter
TemafloxacinDNA gyrase subunit Atarget
TemafloxacinDNA topoisomerase 4 subunit Atarget
TemafloxacinCytochrome P450 1A2enzyme
CefepimeSolute carrier family 22 member 5transporter
CefepimeSolute carrier family 15 member 1transporter
CefepimeSolute carrier family 15 member 2transporter
CefepimePenicillin-binding protein 2target
CefepimePeptidoglycan synthase FtsItarget
CefepimePenicillin-binding protein 3target
CefepimePenicillin-binding protein 2target
CefepimePenicillin-binding protein 1Atarget
CefepimePenicillin-binding protein 1Btarget
CefepimePenicillin-binding protein 1Btarget
CefacetrilePenicillin-binding protein 1Atarget
CefacetrilePenicillin-binding protein 1Btarget
CefacetrileSolute carrier family 22 member 6transporter
CefacetrileSolute carrier family 22 member 8transporter
CeftibutenSolute carrier family 15 member 1transporter
CeftibutenSolute carrier family 15 member 2transporter
CeftibutenPeptidoglycan synthase FtsItarget
CeftibutenPenicillin-binding protein 1Atarget
CeftibutenPenicillin-binding protein 1Btarget
CeftibutenPenicillin-binding protein 2target
CeftibutenSolute carrier family 22 member 6transporter
CeftibutenSolute carrier family 22 member 8transporter
CefpodoximePeptidoglycan synthase FtsItarget
NitroxolineMethionine aminopeptidase 2target
NitroxolineMagnesium cationtarget
NitroxolineManganese cationtarget
SulfamerazineDihydropteroate synthasetarget
SulfamerazineSerum albumincarrier
ImipenemPenicillin-binding protein 1Atarget
ImipenemPenicillin-binding protein 1Btarget
ImipenemPenicillin-binding protein 2target
ImipenemPenicillin-binding protein 3target
ImipenemDipeptidase 1enzyme
ImipenemPenicillin-binding protein 4target
ImipenemBeta-lactamase SHV-1enzyme
ImipenemBeta-lactamase TEMenzyme
ImipenemBeta-lactamase CTX-Menzyme
ImipenemBeta-lactamase (KPC-2)enzyme
ImipenemBeta-lactamasetarget
BacampicillinPenicillin-binding proteintarget
MeticillinMecA PBP2' (penicillin binding protein 2')target
MeticillinPenicillin-binding protein 2atarget
MeticillinPenicillin-binding protein 1btarget
MeticillinPenicillin-binding protein 2Btarget
MeticillinPenicillin-binding protein 3target
MeticillinPenicillin-binding protein 1Atarget
PivampicillinPenicillin-binding protein 1Atarget
PivmecillinamPenicillin-binding protein 1Atarget
TazobactamBeta-lactamase TEMtarget
TazobactamSolute carrier family 22 member 6transporter
TazobactamSolute carrier family 22 member 8transporter
TazobactamBeta-lactamase Ohio-1target
TazobactamBeta-lactamase SHV-1target
TicarcillinPenicillin binding protein 2atarget
Lincomycin23S ribosomal RNAtarget
LincomycinAlpha-1-acid glycoprotein 1carrier
RibostamycinProtein disulfide-isomerasetarget
Ribostamycin30S ribosomal protein S12target
RibostamycinAminoglycoside N(6')-acetyltransferase type 1target
RibostamycinAminoglycoside 2'-N-acetyltransferasetarget
RibostamycinAminoglycoside 2'-N-acetyltransferaseenzyme
LatamoxefPenicillin-binding protein 3target
LatamoxefPenicillin-binding protein 1Atarget
LatamoxefPenicillin-binding protein 1Btarget
LatamoxefD-alanyl-D-alanine carboxypeptidase DacBtarget
FleroxacinDNA topoisomerase 2-alphatarget
FleroxacinDNA gyrase subunit Atarget
FleroxacinDNA topoisomerase 4 subunit Atarget
OritavancinCytochrome P450 3A4enzyme
OritavancinCytochrome P450 2D6enzyme
OritavancinCytochrome P450 2C9enzyme
OritavancinCytochrome P450 2C19enzyme
OritavancinSerum albumincarrier
OritavancinPeptidoglycan precursorstarget
OritavancinBacterial cell wall peptide bridging segmentstarget
OritavancinPentaglycyl bridging segmenttarget
Spiramycin50S ribosomal protein L3target
TeicoplaninD-Ala-D-Ala moiety of NAM/NAG peptide subunits of peptidoglycantarget
SulfadimethoxineCytochrome P450 2C9enzyme
SulfadimethoxineSerum albumincarrier
GarenoxacinCytochrome P450 1A2enzyme
DoripenemDipeptidase 1enzyme
DoripenemPenicillin-binding protein 1Atarget
DoripenemPenicillin-binding protein 1Btarget
DoripenemPenicillin-binding protein 2target
DoripenemPenicillin-binding protein 3target
DoripenemPenicillin-binding protein 4target
DoripenemSolute carrier family 22 member 8transporter
DalbavancinD-Ala-D-Ala moiety of NAM/NAG peptide subunits of peptidoglycantarget
IclaprimDihydrofolate reductasetarget
NemonoxacinCytochrome P450 1A2enzyme
Arbekacin30S ribosomal protein S12target
SulfameterDihydropteroate synthasetarget
ThiamphenicolDr hemagglutinin structural subunittarget
AzidocillinPenicillin-binding protein 2atarget
AzidocillinPenicillin-binding protein 1btarget
AzidocillinPenicillin-binding protein 3target
AzidocillinPenicillin-binding protein 1Atarget
AzidocillinPenicillin-binding protein 2Btarget
AzidocillinSolute carrier family 22 member 5transporter
AzidocillinSolute carrier family 15 member 1transporter
AzidocillinSolute carrier family 15 member 2transporter
SulfamoxoleDihydropteroate synthetasetarget
SulfamoxoleCytochrome P450 2C9enzyme
FlumequineCytochrome P450 1A2enzyme
CefaloridineSolute carrier family 22 member 6transporter
CefaloridineSolute carrier family 22 member 8transporter
CarindacillinPenicillin-binding proteintarget
SulbactamBeta-lactamasetarget
CefroxadineBeta-lactamaseenzyme
CefroxadinePenicillin-binding protein 1Btarget
OleandomycinCytochrome P450 3A4enzyme
PazufloxacinCytochrome P450 1A2enzyme
PrulifloxacinCytochrome P450 1A2enzyme
SecnidazoleCytochrome P450 3A4enzyme
SecnidazoleCytochrome P450 3A5enzyme
SecnidazoleCytochrome P450 2C19enzyme
TroleandomycinCytochrome P450 3A5enzyme
TroleandomycinCytochrome P450 3A43enzyme
Troleandomycin50S ribosomal protein L4target
Troleandomycin50S ribosomal protein L32target
TroleandomycinP-glycoprotein 1transporter
TroleandomycinCytochrome P450 2C8enzyme
TroleandomycinCytochrome P450 3A4enzyme
TroleandomycinNuclear receptor subfamily 1 group I member 2target
TroleandomycinCytochrome P450 3A7enzyme
SitafloxacinCytochrome P450 1A2enzyme
MiocamycinCytochrome P450 3A4enzyme
FlurithromycinCytochrome P450 3A4enzyme
RokitamycinCytochrome P450 3A4enzyme
MidecamycinCytochrome P450 3A4enzyme
RufloxacinCytochrome P450 1A2enzyme
Pipemidic acidCytochrome P450 1A2enzyme
Erythromycin23S ribosomal RNAtarget
ErythromycinCytochrome P450 3A4enzyme
ErythromycinCytochrome P450 3A7enzyme
ErythromycinP-glycoprotein 1transporter
ErythromycinSolute carrier organic anion transporter family member 1B1transporter
ErythromycinMotilin receptortarget
ErythromycinPotassium voltage-gated channel subfamily H member 2target
ErythromycinCytochrome P450 3A5enzyme
ErythromycinSolute carrier organic anion transporter family member 1B3transporter
ErythromycinBile salt export pumptransporter
ErythromycinCanalicular multispecific organic anion transporter 1transporter
ErythromycinSolute carrier organic anion transporter family member 1A2transporter
MoxifloxacinDNA gyrase subunit Atarget
MoxifloxacinDNA topoisomerase 4 subunit Atarget
MoxifloxacinDNA topoisomerase 2-alphatarget
MoxifloxacinCytochrome P450 1A2enzyme
MoxifloxacinSerum paraoxonase/arylesterase 1target
SulfanilamideDihydropteroate synthasetarget
SulfisoxazoleDihydropteroate synthasetarget
SulfisoxazoleCytochrome P450 2C9enzyme
ChloramphenicolComplement decay-accelerating factortarget
ChloramphenicolDr hemagglutinin structural subunittarget
ChloramphenicolCytochrome P450 2C19enzyme
ChloramphenicolCytochrome P450 3A4enzyme
ChloramphenicolCytochrome P450 3A5enzyme
ChloramphenicolCytochrome P450 3A7enzyme
ChloramphenicolSolute carrier family 22 member 6transporter
Chloramphenicol50S ribosomal protein L16target
ChloramphenicolChloramphenicol acetyltransferase 3enzyme
ChloramphenicolChloramphenicol acetyltransferaseenzyme
ChloramphenicolChloramphenicol 3-O phosphotransferaseenzyme
SulfamethizoleDihydropteroate synthasetarget
SulfamethizoleSerum albumincarrier
SulfamethizoleCytochrome P450 2C9enzyme
Oxytetracycline30S ribosomal protein S4target
Oxytetracycline30S ribosomal protein S9target
Oxytetracycline16S ribosomal RNAtarget
OxytetracyclineSolute carrier family 22 member 6transporter
OxytetracyclineSolute carrier family 22 member 8transporter
OxytetracyclineSolute carrier family 22 member 11transporter
OxytetracyclineSolute carrier family 22 member 7transporter
OxytetracyclineSerum albumincarrier
Demeclocycline30S ribosomal proteintarget
DemeclocyclineVasopressin V2 receptortarget
BacitracinAlpha-2-macroglobulintarget
BacitracinInsulin-degrading enzymetarget
BacitracinC55-isoprenyl pyrophosphatetarget
BacitracinBacitracin transport ATP-binding protein BcrAtransporter
BacitracinBacitracin transport permease protein BCRBtransporter
BacitracinBacitracin transport permease protein BcrCtransporter
SulfametopyrazineDihydropteroate synthetasetarget
TinidazoleCytochrome P450 3A4enzyme
TinidazoleDNAtarget
TinidazoleBile salt export pumptransporter
LomefloxacinDNA gyrase subunit Atarget
LomefloxacinDNA topoisomerase 4 subunit Atarget
LomefloxacinDNA topoisomerase 2-alphatarget
LomefloxacinCytochrome P450 1A2enzyme
LomefloxacinSolute carrier family 22 member 5transporter
LomefloxacinCanalicular multispecific organic anion transporter 1transporter
Neomycin30S ribosomal protein S12target
Neomycin16S ribosomal RNAtarget
NeomycinExtracellular calcium-sensing receptortarget
SulfamethoxazoleCytochrome P450 2C9enzyme
SulfamethoxazoleSerum albumincarrier
SulfamethoxazoleArylamine N-acetyltransferase 1enzyme
SulfamethoxazoleArylamine N-acetyltransferase 2enzyme
SulfamethoxazoleDihydropteroate synthasetarget
SulfamethoxazoleCytochrome P450 3A4enzyme
SulfamethoxazoleBile salt export pumptransporter
BenzylpenicillinSolute carrier family 22 member 5transporter
BenzylpenicillinSolute carrier family 15 member 1transporter
BenzylpenicillinSolute carrier family 15 member 2transporter
BenzylpenicillinSolute carrier family 22 member 6transporter
BenzylpenicillinSolute carrier family 22 member 8transporter
BenzylpenicillinSolute carrier family 22 member 4transporter
BenzylpenicillinSolute carrier family 22 member 11transporter
BenzylpenicillinSolute carrier organic anion transporter family member 2B1transporter
BenzylpenicillinSolute carrier organic anion transporter family member 4A1transporter
BenzylpenicillinSolute carrier organic anion transporter family member 3A1transporter
BenzylpenicillinSolute carrier organic anion transporter family member 1B1transporter
BenzylpenicillinPenicillin-binding protein 3target
BenzylpenicillinSolute carrier family 22 member 8target
BenzylpenicillinSolute carrier family 15 member 1target
BenzylpenicillinSolute carrier family 15 member 2target
BenzylpenicillinBeta-lactamase TEMenzyme
BenzylpenicillinSerum albumincarrier
Streptomycin30S ribosomal protein S12target
Streptomycin16S ribosomal RNAtarget
StreptomycinProtein-arginine deiminase type-4target
Streptomycin23S ribosomal RNAtarget
StreptomycinBacterial outer membranetarget
StreptomycinCytoplasmic membranetarget
Kanamycin30S ribosomal protein S12target
Kanamycin16S ribosomal RNAtarget
KanamycinAminoglycoside 2'-N-acetyltransferaseenzyme
KanamycinKanamycin nucleotidyltransferaseenzyme
KanamycinAminoglycoside 3'-phosphotransferaseenzyme
ClindamycinCytochrome P450 3A4enzyme
ClindamycinCytochrome P450 3A5enzyme
ClindamycinAlpha-1-acid glycoprotein 1carrier
ClindamycinP-glycoprotein 1transporter
Clindamycin50S ribosomal protein L1target
Clarithromycin50S ribosomal protein L10target
ClarithromycinCytochrome P450 3A4enzyme
ClarithromycinCytochrome P450 3A5enzyme
ClarithromycinP-glycoprotein 1transporter
ClarithromycinSolute carrier family 22 member 7transporter
ClarithromycinPotassium voltage-gated channel subfamily H member 2target
ClarithromycinSolute carrier organic anion transporter family member 1B1target
ClarithromycinSolute carrier organic anion transporter family member 1B3target
ClarithromycinBile salt export pumptransporter
ClarithromycinSolute carrier organic anion transporter family member 1B1transporter
ClarithromycinSolute carrier organic anion transporter family member 1B3transporter
SulfamethazineDihydropteroate synthasetarget
SulfamethazineSerum albumincarrier
SulfamethazineArylamine N-acetyltransferaseenzyme
Fusidic acidChloramphenicol acetyltransferase 3target
Fusidic acidChloramphenicol acetyltransferasetarget
Fusidic acidBile salt export pumptransporter
Fusidic acidCanalicular multispecific organic anion transporter 1transporter
Fusidic acidElongation factor Gtarget
Fusidic acidCytochrome P450 2D6enzyme
Fusidic acidCytochrome P450 3A4enzyme
Fusidic acidUDP-glucuronosyltransferase 1-1enzyme
Fusidic acidATP-binding cassette sub-family G member 2transporter
Fusidic acidSolute carrier organic anion transporter family member 1B1transporter
SulfathiazoleDihydropteroate synthetasetarget
SulfathiazoleCytochrome P450 19A1enzyme
SulfaphenazoleCytochrome P450 2C9enzyme
SulfaphenazoleCytochrome P450 2B6enzyme
SulfaphenazoleCytochrome P450 2C8enzyme
SulfaphenazoleCytochrome P450 2D6enzyme
SulfaphenazoleDihydropteroate synthasetarget
Chlortetracycline16S ribosomal RNAtarget
ChlortetracyclineSerum albumincarrier
Chlortetracycline30S ribosomal protein S3target
Chlortetracycline30S ribosomal protein S8target
Chlortetracycline30S ribosomal protein S19target
Chlortetracycline30S ribosomal protein S14target
Chlortetracycline30S ribosomal protein S7target
ChlortetracyclineADP-ribosylation factor 1target
ChlortetracyclineCatalasetarget
ChlortetracyclineEphrin type-B receptor 1target
ChlortetracyclinePancreatic triacylglycerol lipasetarget
ChlortetracyclineProtein-arginine deiminase type-4target
Tedizolid23S ribosomal RNAtarget
TedizolidAmine oxidase [flavin-containing] Aenzyme
TedizolidAmine oxidase [flavin-containing] Benzyme
SarecyclineP-glycoprotein 1transporter
OmadacyclineP-glycoprotein 1transporter
Omadacycline30S ribosomal protein S3target
Omadacycline30S ribosomal protein S7target
Omadacycline30S ribosomal protein S8target
Omadacycline30S ribosomal protein S19target
Omadacycline30S ribosomal protein S14target
Omadacycline16S ribosomal RNAtarget
OmadacyclineSerum albumincarrier
SolithromycinCytochrome P450 3A4enzyme
DelafloxacinUDP-glucuronosyltransferase 1-1enzyme
DelafloxacinUDP-glucuronosyltransferase 1-3enzyme
DelafloxacinUDP-glucuronosyltransferase 2B15enzyme
DelafloxacinDNA topoisomerase 4 subunit Atarget
DelafloxacinDNA gyrase subunit Atarget
DelafloxacinCytochrome P450 2E1enzyme
DelafloxacinCytochrome P450 2C9enzyme
DelafloxacinCytochrome P450 3A4enzyme
DelafloxacinATP-binding cassette sub-family B member 5transporter
DelafloxacinATP-binding cassette sub-family G member 2transporter
DelafloxacinSerum albumincarrier
VaborbactamBeta-lactamasetarget
VaborbactamCarbapenem-hydrolyzing beta-lactamase KPCtarget
VaborbactamBeta-lactamase (KPC-2)target
VaborbactamBeta-lactamase CTX-Mtarget
VaborbactamBeta-lactamase (blaSHV)target
VaborbactamBeta-lactamase SHV-1target
VaborbactamBeta-lactamase TEMtarget
VaborbactamBeta-lactamase (MIR-1)target
VaborbactamBeta-lactamasetarget
EravacyclineCytochrome P450 3A4enzyme
EravacyclineAmine oxidase [flavin-containing] Aenzyme
Eravacycline30S ribosomal protein S4target
Polymyxin BBacterial outer membranetarget
Polymyxin BSolute carrier family 15 member 2transporter
PlazomicinMultidrug and toxin extrusion protein 1transporter
PlazomicinMultidrug and toxin extrusion protein 2transporter
Plazomicin30S ribosomal protein S14target
Plazomicin30S ribosomal protein S11target
LefamulinCytochrome P450 3A4enzyme
Lefamulin50S ribosomal protein L22target
LefamulinP-glycoprotein 1transporter
RelebactamSolute carrier family 22 member 8transporter
RelebactamSolute carrier family 22 member 11transporter
RelebactamMultidrug and toxin extrusion protein 1transporter
RelebactamMultidrug and toxin extrusion protein 2transporter
RelebactamBeta-lactamase TEMtarget
RelebactamBeta-lactamase SHV-1target
RelebactamBeta-lactamase CTX-Mtarget
RelebactamBeta-lactamase (KPC-2)target
RelebactamBeta-lactamasetarget
CefiderocolPenicillin-binding protein 3target
CefiderocolPenicillin-binding protein 1Atarget
CefiderocolPenicillin-binding protein 1Btarget
CefiderocolPenicillin-binding protein 2target
CefiderocolD-alanyl-D-alanine carboxypeptidase DacBtarget
CefiderocolMexAB-OprM efflux systemtransporter
CefiderocolSerum albumincarrier
CefiderocolCatecholate siderophore receptor Fiutransporter
CefiderocolColicin I receptortransporter
CefiderocolPutative outer membrane ferric siderophore receptortransporter