Cytochrome P-450 CYP3A Substrates

Accession Number

DBCAT003919

Description

Not Available

Drugs

Drug	Drug Description
Indinavir	A protease inhibitor used to treat HIV infection.
Lovastatin	An HMG-CoA reductase inhibitor used to lower LDL cholesterol and reduce the risk of cardiovascular disease and associated conditions, including myocardial infarction and stroke.
Diltiazem	A calcium channel blocker used to treat hypertension and to manage chronic stable angina.
Amlodipine	A calcium channel blocker used to treat hypertension and angina.
Nisoldipine	A calcium channel blocker used as monotherapy or combined with other drugs for the treatment of hypertension.
Alprazolam	A triazolobenzodiazepine with intermediate onset commonly used to treat panic disorders and generalized anxiety in addition to anxiety associated with depression.
Quinine	An alkaloid used to treat uncomplicated Plasmodium falciparum malaria.
Buspirone	An anxiolytic agent used for short-term treatment of generalized anxiety and second-line treatment of depression.
Vincristine	A vinca alkaloid used to treat acute leukemia, malignant lymphoma, Hodgkin's disease, acute erythraemia, and acute panmyelosis.
Cisapride	A medication used to treat heartburn associated with GERD.
Imatinib	A tyrosine kinase inhibitor used to treat a number of leukemias, myelodysplastic/myeloproliferative disease, systemic mastocytosis, hypereosinophilic syndrome, dermatofibrosarcoma protuberans, and gastrointestinal stromal tumors.
Astemizole	A second generation antihistamine used to treat allergy symptoms.
Simvastatin	An HMG-CoA reductase inhibitor used to lower lipid levels and reduce the risk of cardiovascular events including myocardial infarction and stroke.
Tamoxifen	A selective estrogen receptor modulator used to treat estrogen receptor positive breast cancer, reduce the risk of invasive breast cancer following surgery, or reduce the risk of breast cancer in high risk women.
Midazolam	A short-acting benzodiazepine with rapid onset that is commonly used in seizures, anesthesia and anxiety disorders.
Alfentanil	An opioid agonist used to induce and maintain anesthesia, as well as an analgesic.
Tadalafil	A phosphodiesterase 5 inhibitor used to treat erectile dysfunction, benign prostatic hyperplasia, and pulmonary arterial hypertension.
Diazepam	A long-acting benzodiazepine with rapid onset commonly used to treat panic disorders, severe anxiety, alcohol withdrawal, and seizures.
Vardenafil	A phosphodiesterase 5 inhibitor used to treat erectile dysfunction.
Tacrolimus	A calcineurin inhibitor used to prevent organ transplant rejection and to treat moderate to severe atopic dermatitis.
Sirolimus	An mTOR inhibitor immunosuppressant used to prevent organ transplant rejections, treat lymphangioleiomyomatosis, and treat adults with perivascular epithelioid cell tumors.
Triazolam	A benzodiazepine used for short term treatment of insomnia.
Telithromycin	An ketolide used to treat community acquired pneumonia of mild to moderate severity.
Felodipine	A calcium channel blocker used to treat hypertension.
Nitrendipine	A dihydropyridine calcium channel blocker indicated in the treatment of arterial hypertension.
Atorvastatin	An HMG-CoA reductase inhibitor used to lower lipid levels and reduce the risk of cardiovascular disease including myocardial infarction and stroke.
Pimozide	An antipsychotic used to manage debilitating motor and phonic tics in patients with Tourette's Disorder.
Chlorpheniramine	A histamine-H1 receptor antagonist indicated for the management of symptoms associated with upper respiratory allergies.
Nifedipine	A dihydropyridine calcium channel blocker indicated for the management of several subtypes of angina pectoris, and hypertension.
Clarithromycin	A macrolide antibiotic used for the treatment of a wide variety of bacterial infections such as acute otitis, pharyngitis, tonsillitis, respiratory tract infections, uncomplicated skin infections, and helicobacter pylori infection.
Saquinavir	An HIV protease inhibitor used in combination with other antiretroviral agents for the treatment of HIV-1 with advanced immunodeficiency.
Aripiprazole	An atypical antipsychotic used in the treatment of a wide variety of mood and psychotic disorders, such as schizophrenia, bipolar I, major depressive disorder, irritability associated with autism, and Tourette's syndrome.
Erythromycin	A macrolide antibiotic used to treat and prevent a variety of bacterial infections.
Carbamazepine	An anticonvulsant used to treat various types of seizures and pain resulting from trigeminal neuralgia.
Sildenafil	A phosphodiesterase inhibitor used for the treatment of erectile dysfunction.
Quinidine	A medication used to restore normal sinus rhythm, treat atrial fibrillation and flutter, and treat ventricular arrhythmias.
Trazodone	A serotonin uptake inhibitor used to treat major depressive disorder.
Cyclosporine	A steroid-sparing immunosuppressant used in organ and bone marrow transplants as well as inflammatory conditions such as ulcerative colitis, rheumatoid arthritis, and atopic dermatitis.
Verapamil	A non-dihydropyridine calcium channel blocker used in the treatment of angina, arrhythmia, and hypertension.
Haloperidol	An antipsychotic agent used to treat schizophrenia and other psychoses, as well as symptoms of agitation, irritability, and delirium.
Azithromycin	A macrolide antibiotic used to treat a variety of bacterial infections.
Rosuvastatin	An HMG-CoA reductase inhibitor used to lower lipid levels and reduce the risk of cardiovascular disease including myocardial infarction and stroke.
Telaprevir	An NS3/4A viral protease inhibitor used in combination with other antivirals for the curative treatment of chronic Hepatitis C Virus infections.
Boceprevir	A hepatitis C virus NS3/4A protease inhibitor used in combination with other medications to treat chronic hepatitis C genotype 1 infection. Boceprevir is not indicated as monotherapy.
Ritonavir	An HIV protease inhibitor used in combination with other antivirals in the treatment of HIV infection.
Amiodarone	A class III antiarrhythmic indicated for the treatment of recurrent hemodynamically unstable ventricular tachycardia and recurrent ventricular fibrillation.
Isavuconazole	Indicated for patients 18 years of age and older for the treatment of invasive aspergillosis [FDA Label]. Indicated for patients 18 years of age and older for the treatment of...
Atazanavir	An antiviral protease inhibitor used in combination with other antiretrovirals for the treatment of HIV.
Etravirine	A non-nucleoside reverse transcriptase inhibitor (NNRTI) used in the treatment of HIV-1 infections in combination with other antiretroviral agents.
Amprenavir	A protease inhibitor used to treat HIV infection.
Nelfinavir	A viral protease inhibitor used in the treatment of HIV infection.
Fosamprenavir	An antiretroviral agent used for the treatment and postexposure prophylaxis of human immunodeficiency virus (HIV-1) infection.
Nefazodone	An antidepressant used in the treatment of depression.
Riociguat	A stimulator of soluble guanylate cyclase indicated for the management of persistent or recurrent chronic thromboembolic pulmonary hypertension and pulmonary arterial hypertension.
Simeprevir	A direct-acting antiviral agent that inhibits HCV NS3/4A protease to treat chronic hepatitis C virus (HCV) infection in adults with HCV genotype 1 or 4.
Temsirolimus	A antineoplastic agent used in the treatment of renal cell carcinoma (RCC) that works by inhibiting mTOR.
Asunaprevir	An NS3 protease inhibitor used to treat hepatitis C genotype 1b.
Amitriptyline	A tricyclic antidepressant indicated in the treatment of depressive illness, either endogenous or psychotic, and to relieve depression associated anxiety.
Clomipramine	A tricyclic antidepressant used in the treatment of obsessive-compulsive disorder and disorders with an obsessive-compulsive component, such as depression, schizophrenia, and Tourette’s disorder.
Cyclobenzaprine	A skeletal muscle relaxant that works on the brainstem to treat muscle spasms of local origin.
Doxepin	A psychotropic agent used for the treatment of depression, anxiety, manic-depressive disorder, and insomnia.
Imipramine	A tricyclic antidepressant indicated for the treatment of depression and to reduce childhood enuresis.
Nortriptyline	A tricyclic antidepressant used in the treatment of depression.
Avanafil	A phosphodiesterase-5 (PDE5) inhibitor used to treat erectile dysfunction.
Conivaptan	An antidiuretic hormone inhibitor used to raise serum sodium levels.
Darifenacin	An M3 muscarinic receptor blocker used to treat urinary incontinence.
Darunavir	A HIV protease inhibitor used in the treatment of human immunodeficiency virus (HIV) infection in patients with history of prior antiretroviral therapies.
Ebastine	A second generation H1-receptor antagonist useful in the treatment of allergic rhinitis and urticaria.
Everolimus	A mammalian target of rapamycin (mTOR) kinase inhibitor used to treat various types of malignancies.
Ibrutinib	An antineoplastic agent used to treat chronic lymphocytic leukemia, mantle cell lymphoma, and Waldenstrom's Macroglobulinemia.
Lomitapide	A microsomal triglyceride transfer protein inhibitor used to lower cholesterol associated with homozygous familial hypercholesterolemia (HoFH), reducing risk of cardiovascular events such as myocardial infarction and stroke.
Naloxegol	A peripherally-selective opioid antagonist used to treat opioid-induced constipation (OIC) in adult patients with chronic non-cancer pain.
Budesonide	A corticosteroid used to treat Crohn's disease, asthma, COPD, hay fever and allergies, and ulcerative colitis.
Dasatinib	A tyrosine kinase inhibitor used for the treatment of Philadelphia chromosome-positive acute lymphoblastic leukemia or chronic myeloid leukemia.
Dronedarone	An antiarrhythmic agent used in the reduce the risk of hospitalization in patients with paroxysmal or persistent atrial fibrillation.
Eletriptan	A triptan used for the treatment of migraines.
Eplerenone	An aldosterone receptor antagonist used to improve survival of patients with symptomatic heart failure and to reduce blood pressure.
Lurasidone	An atypical antipsychotic used to treat schizophrenia and depressive episodes associated with bipolar I disorder.
Maraviroc	A CCR5 co-receptor antagonist used with other antiretroviral medications to treat CCR5-tropic HIV-1 infection.
Quetiapine	An atypical antipsychotic agent used for the management of bipolar disorder, schizophrenia, and major depressive disorder.
Ticagrelor	A P2Y12 platelet inhibitor used in patients with a history of myocardial infarction or with acute coronary syndrome (ACS) to prevent future myocardial infarction, stroke and cardiovascular death.
Tolvaptan	A selective vasopressin V2-receptor antagonist to slow kidney function decline in patients at risk for rapidly progressing autosomal dominant polycystic kidney disease (ADPKD). Also used to treat hypervolemic and euvolemic hyponatremia.
Aprepitant	A substance P/neurokinin 1 receptor antagonist used to treat nausea and vomiting caused by chemotherapy and surgery.
Colchicine	An alkaloid used to treat gout and Familial Mediterranean Fever as well as prevent major cardiovascular events.
Eliglustat	A glucosylceramide synthase used to treat type 1 Gaucher disease in patients who are CYP2D6 extensive, intermediate, or poor metabolizers.
Rilpivirine	A non-nucleoside reverse transcriptase inhibitor (NNRTI) used in combination with other antiretrovirals to specifically treat human immunodeficiency virus type 1 (HIV-1).
Rivaroxaban	A factor Xa inhibitor used to treat deep vein thrombosis (DVT) and pulmonary embolism (PE). May also be used as thrombosis prophylaxis in specific situations.
Methysergide	An ergot alkaloid used for the prophylaxis of migraine and cluster headaches.
Tianeptine	An atypical tricyclic antidepressant with antidepressant and anxiolytic effects primarily used to treat major depressive disorder.
Estradiol	An estrogenic steroid used to treat vasomotor symptoms of vulvar and vaginal atrophy in menopause, hypoestrogenism, prevention of postmenopausal osteoporosis, treatment of breast cancer, and advanced androgen-dependent carcinoma of the prostate.
Estradiol cypionate	An estradiol prodrug used to treat vasomotor symptoms and hypoestrogenisms from hypogonadism.
Estradiol valerate	An estradiol prodrug used to treat some effects of menopause, hypoestrogenism, androgen dependant carcinoma of the prostate, and in combination products for endometriosis and contraception.
Ethinylestradiol	An estradiol used as a contraceptive.
Mestranol	A synthetic estradiol found in oral contraceptive pills for contraception and the treatment of other conditions in the female reproductive system, such as dysmenorrhea and dysfunctional uterine bleeding.
Aminophylline	A bronchodilator consisting of theophylline that is used for the treatment of bronchospasm due to asthma, emphysema and chronic bronchitis.
Theophylline	A xanthine used to manage the symptoms of asthma, COPD, and other lung conditions caused by reversible airflow obstruction.
Bromocriptine	A dopamine D2 receptor agonist used for the treatment of galactorrhea due to hyperprolactinemia and other prolactin-related conditions, as well as in early Parkinsonian Syndrome.
Cabergoline	A dopamine receptor agonist used for the treatment of hyperprolactinemic conditions due to various causes.
Dihydroergocornine	A nootropic with an unknown mechanism of action indicated in individuals over sixty who manifest signs and symptoms of an idiopathic decline in mental capacity.
Dihydroergocristine	An ergot alkaloid used to delay progressive mental decline in conditions like Alzheimer's.
Dihydroergocryptine	A dopamine agonist indicated in the treatment of cerebrovascular diseases and atherosclerosis.
Dihydroergotamine	An ergot alkaloid used in the acute treatment of migraine headache and cluster headache.
Ergoloid mesylate	A nootropic with an unknown mechanism of action indicated in individuals over sixty who manifest signs and symptoms of an idiopathic decline in mental capacity.
Ergometrine	An ergot alkaloid used for the treatment of postpartum haemorrhage and post abortion hemorrhage in patients with uterine atony.
Ergotamine	An alpha-1 selective adrenergic agonist vasoconstrictor used to treat migraines with or without aura and cluster headaches.
Lisuride	For the management of Parkinson's Disease
Lysergic acid diethylamide	Debate continues over the nature and causes of chronic flashbacks. Explanations in terms of LSD physically remaining in the body for months or years after consumption have been discounted by...
Methylergometrine	An ergot alkaloid used to prevent and control uterine atony and hemorrhage before and after delivery.
Terguride	Not Annotated
Triamcinolone	A glucocorticoid used to treat a wide variety of inflammatory conditions of organ systems and tissues.
Voriconazole	A triazole compound used to treat fungal infections.
Esomeprazole	A proton pump inhibitor used to treat GERD, reduce the risk of NSAID associated gastric ulcers, eradicate H. pylori, and to treat conditions causing gastric acid hypersecretion.
Omeprazole	A proton pump inhibitor used to treat GERD associated conditions such as heartburn and gastric acid hypersecretion, and to promote healing of tissue damage and ulcers caused by gastric acid and H. pylori infection.
Propafenone	A Class 1C antiarrhythmic agent used in the management of paroxysmal atrial fibrillation/flutter and ventricular arrhythmias.
Lopinavir	An HIV-1 protease inhibitor used in combination with ritonavir to treat human immunodeficiency virus (HIV) infection.
Tipranavir	A protease inhibitor used to treat HIV-1 resistant to more than 1 protease inhibitor.
Phenprocoumon	An anticoagulant drug used for the prevention of thrombosis.
Teniposide	A cytotoxic drug used as an adjunct for chemotherapy induction in the treatment of refractory childhood acute lymphoblastic leukemia.
Ulipristal	A selective progesterone receptor modulator used for emergency contraception after unprotected intercourse or in a situation where a planned method of contraception has failed.
Disopyramide	A class 1A antiarrhythmic agent used to treat life-threatening ventricular arrhythmias.
Methadone	An opioid analgesic indicated for management of severe pain that is not responsive to alternative treatments. Also used to aid in detoxification and maintenance treatment of opioid addiction.
Alfuzosin	An alpha-1 adrenergic antagonist used in the symptomatic management of benign prostatic hypertrophy (BPH).
Buprenorphine	A partial opioid agonist used for management of severe pain that is not responsive to alternative treatments. Also used for maintenance treatment of opioid addiction.
Fostamatinib	A spleen tyrosine kinase inhibitor used to treat chronic immune thrombocytopenia after attempting one other treatment.
Udenafil	A PDE5 inhibitor used to treat erectile dysfunction.
Prednisone	A corticosteroid used to treat inflammation or immune-mediated reactions and to treat endocrine or neoplastic diseases.
Fluticasone	A corticosteroid indicated in the treatment of corticosteroid responsive dermatoses, asthma, and COPD.
Pantoprazole	A proton pump inhibitor used to treat erosive esophagitis, gastric acid hypersecretion, and to promote healing of tissue damage caused by gastric acid.
Lansoprazole	A proton pump inhibitor used to help gastrointestinal ulcers heal, to treat symptoms of gastroesophageal reflux disease (GERD), to eradicate Helicobacter pylori, and to treat hypersecretory conditions such as Zollinger-Ellison Syndrome.
Dexlansoprazole	A proton pump inhibitor used to treat erosive esophagitis, heartburn, and gastroesophageal reflux disease (GERD).
Rabeprazole	A proton pump inhibitor used to help gastrointestinal ulcers heal, to treat symptoms of gastroesophageal reflux disease (GERD), to eradicate Helicobacter pylori, and to treat hypersecretory conditions such as Zollinger-Ellison Syndrome.
Lacidipine	A lipophilic dihydropyridine calcium channel blocker with a slow onset of action used to treat hypertension.
Allylestrenol	A steroid used to prevent premature labour in pregnant women.
Betamethasone	A systemic corticosteroid used to relieve inflammation in various conditions, including but not limited to allergic states, dermatologic disorders, gastrointestinal diseases, and hematological disorders.
Ciclesonide	A glucocorticoid used in the symptomatic relief of nasal symptoms associated with seasonal and perennial allergic rhinitis in adults and adolescents.
Cortisone acetate	A steroid hormone used for the relief of the inflammatory and pruritic manifestations of corticosteroid-responsive dermatoses and endocrine disorders associated with inadequate production of steroid hormones.
Deflazacort	A corticosteroid used to treat Duchenne muscular dystrophy.
Dienogest	An oral progestin used for the treatment of endometriosis as monotherapy or contraception in combination with ethinylestradiol.
Dexamethasone	A glucocorticoid available in various modes of administration that is used for the treatment of various inflammatory conditions, including bronchial asthma, as well as endocrine and rheumatic disorders.
Dexamethasone isonicotinate	Dexamethasone isonicotinate is an anti-inflammatory, anti-allergic glucocorticoid that can be administered orally, by inhalation, topically, and parenterally. Its unintended mineralocorticoid action may cause salt and water retention.
Drospirenone	A progestin used in oral contraceptive pills for the prevention of pregnancy and other conditions.
Estrone	An estrogen used to treat perimenopausal and postmenopausal symptoms.
Estrone sulfate	An estrogen used as monotherapy or in several combination hormone replacement products for managing menopause symptoms and hormone disorders.
Etonogestrel	A long-acting synthetic derived progestin contraceptive used in various devices such as contraceptive rings and intradermal implants.
Flunisolide	An inhaled corticosteroid used as a prophylactic therapy in the maintenance treatment of asthma.
Fluocortolone	A glucocorticoid used topically for localized skin reactions and also orally for systemic use.
Fluorometholone	An ophthalmic corticosteroid used for the relief of inflammation located in both the palpebral and bulbar conjunctiva, the cornea, and the anterior segment of the globe of the eye.
Fluticasone furoate	An inhaled corticosteroid that can be used as maintenance treatment of asthma and/or chronic obstructive pulmonary disease (COPD) depending on the product. Also available as a nasal spray to manage symptoms of allergic rhinitis.
Fluticasone propionate	A glucocorticoid used to treat asthma, inflammatory pruritic dermatoses, and nonallergic rhinitis.
Hydrocortisone	A glucocorticoid used to treat corticosteroid-responsive dermatoses, endocrine disorders, immune conditions, and allergic disorders.
Hydrocortisone aceponate	For the relief of the inflammatory and pruritic manifestations of corticosteroid-responsive dermatoses. Also used to treat endocrine (hormonal) disorders (adrenal insufficiency, Addisons disease). It is also used to treat many...
Hydrocortisone acetate	A corticosteroid used to treat inflammatory and pruritic corticosteroid-responsive dermatoses and ulcerative colitis.
Hydrocortisone butyrate	A corticosteroid used to treat inflammatory and pruritic corticosteroid-responsive dermatoses.
Hydrocortisone cypionate	For the relief of the inflammatory and pruritic manifestations of corticosteroid-responsive dermatoses. Also used to treat endocrine (hormonal) disorders (adrenal insufficiency, Addisons disease). It is also used to treat many...
Hydrocortisone phosphate	A corticosteroid used to treat congenital adrenal hyperplasia, for emergency asthma treatment, hypersensitivity, and inflammation.
Hydrocortisone probutate	A corticosteroid used to treat inflammatory and pruritic corticosteroid-responsive dermatoses.
Hydrocortisone valerate	A corticosteroid used to treat inflammatory and pruritic corticosteroid-responsive dermatoses.
Hydroxyprogesterone caproate	A synthetic progestin used for the prevention of spontaneous preterm births in singleton pregnancies in women who have previously had a spontaneous preterm birth.
Levonorgestrel	A progestin found in oral and IUD contraceptives and at higher doses in emergency contraceptives.
Medroxyprogesterone acetate	A progestin used as a contraceptive and in the treatment of secondary amenorrhea, abnormal uterine bleeding, pain from endometriosis, endometrial and renal carcinomas, paraphilia in males, and GnRH-dependent precocious puberty.
Methylprednisolone	A corticosteroid used to treat inflammation or immune reactions across a variety of organ systems, endocrine conditions, and neoplastic diseases.
Norethisterone	A synthetic second-generation progestin used for contraception, prevention of endometrial hyperplasia in hormone replacement therapy, and in the treatment of other hormone-mediated illnesses such as endometriosis.
Norgestimate	A progesterone used as a contraceptive and to treat acne vulgaris.
Norgestrel	A progestin used in combination with ethinyl estradiol for oral contraception and prevention of pregnancy in women.
Paramethasone	For the treatment of all conditions in which corticosteroid therapy is indicated except adrenal-deficiency states for which its lack of sodium-retaining properties makes it less suitable than hydrocortisone with supplementary...
Prasterone	A steroid formulated as a vaginal insert indicated for the treatment of moderate to severe dyspareunia associated with menopausal vulvar and vaginal atrophy.
Prednisolone	A glucocorticoid used to treat adrenocortical insufficiency, inflammatory conditions, and some cancers.
Progesterone	A hormone used for a variety of functions, including contraception, control of abnormal uterine bleeding, maintenance of pregnancy, and prevention of endometrial hyperplasia.
Ramelteon	A melatonin receptor agonist used to treat insomnia.
Zolpidem	A sedative hypnotic used for the short-term treatment of insomnia to improve sleep latency.
Zidovudine	A dideoxynucleoside used in the treatment of HIV infection.
Diethylstilbestrol	Used in the treatment of prostate cancer. Previously used in the prevention of miscarriage or premature delivery in pregnant women prone to miscarriage or premature delivery.
Dapsone	A sulfone drug used to treat acne vulgaris, Hansen's disease, and dermatitis herpetiformis.
Morphine	An opioid agonist used for the relief of moderate to severe acute and chronic pain.
Acenocoumarol	An anticoagulant drug used in the prevention of thromboembolic diseases in infarction and transient ischemic attacks, as well as management of deep vein thrombosis and myocardial infarction.
Diphenadione	Not Annotated
Ethyl biscoumacetate	Ethyl biscoumacetate is a courmarin that is used as an anticoagulant. It has actions similar to those of Warfarin. (From Martindale, The Extra Pharmacopoeia, 30th ed, p226)
Warfarin	A vitamin K antagonist used to treat venous thromboembolism, pulmonary embolism, thromboembolism with atrial fibrillation, thromboembolism with cardiac valve replacement, and thromboembolic events post myocardial infarction.
Azelnidipine	For the treatment of hypertension.
Barnidipine	A calcium channel blocker used to treat various forms of hypertension.
Bencyclane	A vasodilator agent found to be effective in a variety of peripheral circulation disorders. It has various other potentially useful pharmacological effects. Its mechanism may involve block of calcium channels.
Benidipine	A synthetic dihydropyridine calcium channel blocker used to treat hypertension and angina pectoris.
Bepridil	For the treatment of hypertension, and chronic stable angina (classic effort-associated angina).
Bioallethrin	Bioallethrin was used for lice and scabies infestation. Other pyrethroids are now used in place of bioallethrin.
Carboxyamidotriazole	Carboxyamidotriazole has been used in trials studying the treatment of Lymphoma, Lung Cancer, Breast Cancer, Kidney Cancer, and Ovarian Cancer, among others.
Caroverine	A calcium channel blocker indicated in the treatment of smooth muscle spasms, alcohol and drug withdrawal, and tinnitus.
Cilnidipine	A dihydropyridine calcium channel blocker with action on both N- and L-type calcium channels used to treat hypertension.
Cinnarizine	A drug used for the management of labyrinthine disorder symptoms, including vertigo, tinnitus, nystagmus, nausea, and vomiting.
Clevidipine	A dihydropyridine L-type calcium channel blocker used to lower blood pressure when oral antihypertensive therapy is not feasible or not desirable.
Cyclandelate	A vasodilator used for the treatment of various blood vessel diseases, such as claudication and arteriosclerosis.
Darodipine	Darodipine is a calcium channel blocker.
Dexniguldipine	Not Annotated
Dexverapamil	Not Annotated
Dotarizine	A calcium antagonist used to treat and prevent migraines.
Efonidipine	For the treatment of hypertension.
Emopamil	Prevents renal injury after warm & cold ischemia.
Eperisone	An antispasmodic that functions through voltage-gated channel blockade, notably with little to no sedation, effective in relaxing skeletal muscles and vascular smooth muscles.
Ethosuximide	An anticonvulsant used to treat petit mal seizures.
Fendiline	Fendiline is a coronary vasodilator which inhibits calcium function in muscle cells in excitation-contraction coupling. It has been proposed as an antiarrhythmic and antianginal agent. Fendiline is non-selective.
Fish oil	A source of essential fatty acids used as a source of calories in parenteral nutrition and as a dietary supplement.
Flunarizine	A selective calcium-entry blocker used as migraine prophylaxis in patients with severe and frequent episodes who have not responded adequately to more common treatments.
Fluspirilene	An antipsychotic agent used in the treatment of schizophrenia.
Gallopamil	Gallopamil has been used in trials studying the treatment of Asthma.
Isradipine	A dihydropyridine calcium channel blocker used for the treatment of hypertension.
Lercanidipine	A calcium channel blocker for the management of hypertension.
Lidoflazine	Not Annotated
Lomerizine	Lomerizine is a diphenylmethylpiperazine calcium channel blocker[A245378, A245383] with relatively selective central nervous system (CNS) effects. This drug is used to prophylactically treat migraines[A245368, A245373] and is also being investigated...
Loperamide	A long acting antidiarrheal used to control nonspecific diarrhea and chronic diarrhea caused by inflammatory bowel disease, or gastroenteritis.
Manidipine	A dihydropyridine calcium channel blocker used to treat hypertension.
Levomenthol	An organic compound used to treat mild to moderate muscle and joint pain.
Mibefradil	For the treatment of angina and high blood pressure.
Naftopidil	Naftopidil has been investigated for the treatment of Disorder of Urinary Stent.
Nicardipine	A calcium channel blocker used for the short-term treatment of hypertension and chronic stable angina.
Niludipine	Niludipine is a calcium channel blocker.
Nilvadipine	A calcium channel blocker used to manage arterial hypertension.
Nimesulide	A cyclooxygenase 2 inhibitor used to treat acute pain and primary dysmenorrhea.
Nimodipine	A calcium channel blocker used to improve neurological outcomes in patients with subarachnoid hemorrhage due to a ruptured intracranial aneurysm.
Nylidrin	A vasodilator used to treat patients with peripheral vascular disorders, and elderly patients with symptoms associated with organic mental disorders.
Niguldipine	Niguldipine is a calcium channel blocker drug (CCB) with a1-adrenergic antagonist properties.
Otilonium	A spasmolytic medication used to treat irritable bowel syndrome (IBS).
Penfluridol	Not Annotated
Perhexiline	For the management of severe angina pectoris.
Pinaverium	A spasmolytic agent used for the symptomatic treatment of irritable bowel syndrome (IBS) and functional disorders of the biliary tract.
Prenylamine	Prenylamine was withdrawn from the Canadian, US, and UK markets in 1988 due to concerns regarding cardiac arrhythmias.
Terodiline	Not Annotated
Tetrahydropalmatine	Tetrahydropalmatine is under investigation in clinical trial NCT02118610 (Treatment of Schizophrenia With L-tetrahydropalmatine (l-THP): a Novel Dopamine Antagonist With Anti-inflammatory and Antiprotozoal Activity).
Tetrandrine	Not Annotated
Tolfenamic acid	In the information for tolfenamic acid, it is stated that this drug, being an NSAID, is effective in treating the pain associated with the acute attack of migraines in adults.
Tranilast	For the treatment of bronchial asthma, keloid and hypertrophic scar, and allergic disorders such as asthma, allergic rhinitis and atopic dermatitis.
Trimebutine	A spasmolytic agent used for the symptomatic treatment of irritable bowel syndrome (IBS) and treatment of postoperative paralytic ileus following abdominal surgery.
Trimethadione	An anticonvulsant agent indicated for the control of treatment-refractory petit mal seizures.
Seletracetam	Investigated for use/treatment in epilepsy.
Vinpocetine	A synthetic derivative of a vinca alkaloid used to treat neurological symptoms of cerebrovascular disease.
WIN 55212-2	WIN 55,212-2 is a chemical described as an aminoalkylindole derivative, which produces effects similar to those of cannabinoids such as tetrahydrocannabinol (THC) but has an entirely different chemical structure. It...
Zonisamide	A sulfonamide anticonvulsant used to treat partial seizures.
Ivermectin	An anti parasite medication used to treat head lice, onchocerciasis, strongyloidiasis, ascariasis, trichuriasis, and enterobiasis.
Ixabepilone	A microtubule inhibitor administered in combination with capecitabine or alone in the treatment of metastatic or locally advanced breast cancer that has shown inadequate response to taxanes and anthracyclines.
Rifabutin	An antibiotic used to treat mycobacterium avium complex disease in patients with HIV.
Rifapentine	An antibiotic agent used in the treatment of pulmonary tuberculosis.
Rifaximin	A rifamycin-based non-systemic antibiotic used for the treatment of gastrointestinal bacterial infections, such as traveler's diarrhea and irritable bowel syndrome, and reduction of overt hepatic encephalopathy recurrence in adults.
Regorafenib	A kinase inhibitor used to treat patients with metastatic colorectal cancer, unresectable, locally advanced, or metastatic gastrointestinal stromal tumors, and hepatocellular carcinoma.
Ivabradine	A HCN channel blocker used to reduce the risk of hospitalization for worsening heart failure in adult patients and for treatment of stable symptomatic heart failure as a result of dilated cardiomyopathy in pediatric patients.
Vemurafenib	A kinase inhibitor used to treat patients with Erdheim-Chester Disease who have the BRAF V600 mutation, and melanoma in patients who have the BRAF V600E mutation.
Vortioxetine	A serotonin modulating antidepressant indicated for the treatment of major depressive disorder (MDD).
Pazopanib	An antineoplastic agent used in the treatment of advanced renal cell cancer and advanced soft tissue sarcoma in patients with prior chemotherapy.
Perampanel	A non-competitive AMPA glutamate receptor antagonist used to treat partial-onset seizures with or without secondarily generalized seizures, and as adjunctive treatment of primary generalized tonic-clonic seizures in patients with epilepsy.
Crizotinib	A receptor tyrosine kinase inhibitor used to treat metastatic non-small cell lung cancer (NSCLC) where the tumors have been confirmed to be anaplastic lymphoma kinase (ALK), or ROS1-positive.
Cabozantinib	A tyrosine kinase inhibitor used to treat advanced renal cell carcinoma, hepatocellular carcinoma, and medullary thyroid cancer.
Isavuconazonium	A triazole antifungal used for the treatment of invasive aspergillosis and mucormycosis.
Axitinib	An oral VEGFR and kinase inhibitor used for the treatment of advanced renal cell carcinoma after failure of one prior systemic therapy.
Codeine	An opioid analgesic used to treat moderate to severe pain when the use of an opioid is indicated.
Apixaban	An anticoagulant used for the prophylaxis of stroke and systemic embolism in nonvalvular atrial fibrillation, and deep vein thrombosis(DVT) leading to pulmonary embolism(PE), including in patients after a hip or knee replacement surgery.
Pioglitazone	A thiazolidinedione used adjunctively with diet and exercise to normalize glycemic levels in adults with type 2 diabetes mellitus.
Lapatinib	An antineoplastic agent and tyrosine kinase inhibitor used for the treatment of advanced or metastatic HER-positive breast cancer in patients who received prior chemotherapeutic treatments.
Icotinib	Icotinib hydrochloride is a novel epidermal growth factor receptor (EGFR)–tyrosine kinase inhibitor, exhibits encouraging efficacy and tolerability in patients with advanced non-small-cell lung cancer (NSCLC) who failed previous chemotherapy.
Cevimeline	A muscarinic agonist with parasympathomimetic activities that is used for the symptomatic treatment of dry mouth in patients with Sjögren's Syndrome.
Bortezomib	A proteasome inhibitor used to treat multiple myeloma in patients who have not been successfully treated with at least two previous therapies.
Dofetilide	A class III antiarrhythmic drug used for the maintenance of normal sinus rhythm and cardioversion in cases of atrial fibrillation and atrial flutter.
Reboxetine	A drug used for the acute treatment of major depression and for maintenance therapy of depression.
Ranolazine	An anti-anginal drug used for the treatment of chronic angina.
Ziprasidone	An atypical antipsychotic used to manage schizophrenia, bipolar mania, and agitation in patients with schizophrenia.
Conjugated estrogens	A mixture of estrogens used in estrogen replacement therapy for menopause and hypoestrogenism, used in the treatment of various malignancies, and used in the treatment of postmenopausal osteoporosis.
Bupivacaine	A local anesthetic used in a wide variety of superficial and invasive procedures.
Bexarotene	A retinoid drug used for cutaneous manifestations of T-cell lymphoma in patients who have not responded well to previous systemic therapy.
Vindesine	A vinca alkaloid derived from vinblastine used for various types of malignancies, but mainly acute lymphocytic leukemia (ALL).
Gefitinib	A tyrosine kinase inhibitor used as first-line therapy to treat non-small cell lung carcinoma (NSCLC) that meets certain genetic mutation criteria.
Terfenadine	An antihistamine for the treatment of allergy symptoms.
Vinorelbine	A vinca alkaloid used in the treatment of metastatic non-small cell lung carcinoma (NSLC) and in conjunction with other drugs in locally advanced NSCLC.
Grepafloxacin	A fluoroquinolone antibiotic used to treat various gram positive and gram negative bacterial infections.
Mirtazapine	A tetracyclic antidepressant used in the treatment of major depression and is used off-label as a drug for insomnia and to increase appetite.
Sorafenib	A kinase inhibitor used to treat unresectable liver carcinoma, advanced renal carcinoma, and differentiated thyroid carcinoma.
Eszopiclone	A sedative-hypnotic used in the treatment of insomnia, improving both the latency phase and the maintenance phase of sleep.
Prochlorperazine	A phenothiazine derivative used in the treatment of schizophrenia and anxiety and to relieve severe nausea and vomiting.
Loratadine	A second generation antihistamine used to manage the symptoms of allergic rhinitis.
Dronabinol	A synthetic delta-9-THC used in the treatment of anorexia and weight loss in HIV patients as well as nausea and vomiting in cancer chemotherapy.
Montelukast	A leukotriene receptor antagonist used as part of an asthma therapy regimen, to prevent exercise induced bronchoconstriction, and to treat seasonal allergic rhinitis.
Albendazole	A benzimidazole anthelmintic used to treat parenchymal neurocysticercosis and other helminth infections.
Erlotinib	An EGFR tyrosine kinase inhibitor used to treat certain small cell lung cancers or advanced metastatic pancreatic cancers.
Rofecoxib	A COX-2 inhibitor NSAID used to treat osteoarthritis, rheumatoid arthritis, acute pain, primary dysmenorrhea, and migraine attacks.
Toremifene	A first generation nonsteroidal selective estrogen receptor modulator used to treat certain breast cancers.
Bosentan	A dual endothelin receptor antagonist used to treat pulmonary arterial hypertension.
Vinblastine	A vinca alkaloid used to treat breast cancer, testicular cancer, neuroblastoma, Hodgkin's and non-Hodgkins lymphoma, mycosis fungoides, histiocytosis, and Kaposi's sarcoma.
Testosterone	A hormone used to treat hypogonadism, breast carcinoma in women, or the vasomotor symptoms of menopause.
Efavirenz	A non-nucleoside reverse transcriptase inhibitor used to treat HIV infection or prevent the spread of HIV.
Clofibrate	A fibric acid derivative used to treat hypertriglyceridemia and high cholesterol.
Galantamine	A cholinesterase inhibitor used to manage mild to moderate dementia associated with Alzheimer's Disease.
Losartan	An angiotensin receptor blocker used to treat hypertension and diabetic nephropathy, and is used to reduce the risk of stroke.
Delavirdine	A non-nucleoside reverse transcriptase inhibitor used to treat HIV infection.
Nateglinide	A meglitinide used to treat non insulin dependent diabetes mellitus.
Zileuton	A leukotriene synthesis inhibitor used in the prophylaxis and treatment of chronic asthma.
Modafinil	A stimulant used to improve wakefulness in patients with sleep apnea, narcolepsy, or shift work disorder.
Dolasetron	An antinauseant and antiemetic used in chemotherapy and postoperatively.
Clopidogrel	An antiplatelet agent used to prevent blood clots in peripheral vascular disease, coronary artery disease, and cerebrovascular disease.
Irinotecan	A topoisomerase inhibitor used to treat metastatic carcinoma of the colon or rectum and pancreatic adenocarcinoma.
Etoposide	A podophyllotoxin derivative used to treat testicular and small cell lung tumors.
Roxithromycin	An antibiotic used to treat a variety of susceptible bacterial infections.
Fentanyl	An opioid analgesic used in anesthesia, for breakthrough cancer pain, or round the clock pain management.
Mifepristone	A cortisol receptor blocker used to treat Cushing's syndrome, and to terminate pregnancies up to 70 days gestation.
Donepezil	An acetylcholinesterase inhibitor used to treat the behavioral and cognitive effects of Alzheimer's Disease and other types of dementia.
Granisetron	A 5HT3 antagonist used to treat nausea and vomiting in cancer therapy and postoperatively.
Ondansetron	A serotonin 5-HT3 receptor antagonist used to prevent nausea and vomiting in cancer chemotherapy and postoperatively.
Tiagabine	An antiepileptic used to treat partial seizures.
Cocaine	An ester local anesthetic used during diagnostic procedures and surgeries in or through the nasal cavities.
Paricalcitol	A vitamin D analog used to treat hyperparathyroidism associated with stage 3 or greater chronic kidney disease.
Tinidazole	A nitroimidazole used to treat trichomoniasis, giardiasis, amebiasis, and bacterial vaginosis.
Almotriptan	A 5-HT1B/1D receptor agonist used to treat migraines.
Salmeterol	A long-acting beta-2 adrenergic receptor agonist used to treat asthma and COPD.
Hydrocodone	An opioid agonist used as an analgesic and antitussive agent.
Zaleplon	A sedative used for short term treatment of insomnia in adults.
Exemestane	An aromatase inhibitor used to treat breast cancer in postmenopausal women after treatment with tamoxifen.
Doxorubicin	A medication used to treat various cancers, including AIDS-associated Kaposi's Sarcoma and metastatic cancers.
Levobupivacaine	A drug used for nerve block and anesthesia.
Letrozole	An aromatase inhibitor used to treat breast cancer in postmenopausal women.
Busulfan	An alkylating agent used to treat chronic myelogenous leukemia.
Cinacalcet	A calcium sensing receptor agonist used to treat secondary hyperparathyroidism in chronic kidney disease and hypercalcemia in parathyroid carcinoma.
Ketoconazole	A broad spectrum antifungal used to treat seborrheic dermatitis and fungal skin infections.
Oxybutynin	An antimuscarinic agent that reduces detrusor muscle activity, relaxing the bladder and preventing the urge to void.
Clonazepam	A long-acting benzodiazepine with intermediate onset commonly used to treat panic disorders, severe anxiety, and seizures.
Sibutramine	A norepinephrine, serotonin and dopamine reuptake inhibitor indicated to assist with weight loss in obesity.
Dutasteride	An antiandrogenic compound that is used for the treatment of symptomatic benign prostatic hyperplasia (BPH) in adult males by inhibiting 5-alpha reductase.
Cilostazol	An antiplatelet agent and vasodilator used for the symptomatic relief of intermittent claudication.
Itraconazole	A triazole antifungal agent used to treat various fungal infections, such as blastomycosis and onychomycosis.
Escitalopram	A selective serotonin re-uptake inhibitor used in the treatment of major depressive disorder (MDD), generalized anxiety disorder (GAD), and other select psychiatric disorders such as obsessive-compulsive disorder (OCD).
Domperidone	A dopamine receptor antagonist used as a peristaltic stimulant and anti-emetic agent for dyspepsia, indigestion, epigastric pain, nausea, and vomiting.
Clindamycin	A lincosamide antibiotic used to treat serious infections caused by susceptible anaerobic, streptococcal, staphylococcal, and pneumococcal bacteria.
Estazolam	A benzodiazepine used for the short-term management of insomnia.
Finasteride	An antiandrogenic compound that is used for the treatment of symptomatic benign prostatic hyperplasia (BPH) and male pattern hair loss in adult males by inhibiting Type II 5-alpha reductase.
Halofantrine	An antimalarial used for the treatment of severe malaria.
Levacetylmethadol	For the treatment and management of opiate dependence. It is sometimes used to treat severe pain in terminal patients.
Paclitaxel	A taxoid chemotherapeutic agent used as first-line and subsequent therapy for the treatment of advanced carcinoma of the ovary, and other various cancers including breast and lung cancer.
Retapamulin	A topical antibiotic agent used for the treatment of impetigo caused by methicillin-susceptible Staphylococcus aureus or Streptococcus pyogenes.
Sitagliptin	An oral dipeptidyl peptidase-4 (DPP-4) inhibitor used for the management of type 2 diabetes mellitus.
Sunitinib	A receptor tyrosine kinase inhibitor and chemotherapeutic agent used for the treatment of renal cell carcinoma (RCC) and imatinib-resistant gastrointestinal stromal tumor (GIST).
Posaconazole	A triazole antifungal drug that is used to treat invasive infections by Candida species and Aspergillus species in severely immunocompromised patients.
Alosetron	A 5-HT3 antagonist used to treat diarrhea-predominant IBS.
Tiotropium	A long-acting bronchodilator used in the management of chronic obstructive pulmonary disease (COPD).
Solifenacin	A muscarinic antagonist with antispasmodic properties used to treat urge urinary incontinence, urgency, and urinary frequency associated with an overactive bladder.
Palonosetron	A serotonin antagonist used in the prophylaxis or management of vomiting that results from emetogenic chemotherapy, and for the management of postoperative nausea and vomiting.
Valdecoxib	A COX-2 inhibitor used to treat osteoarthritis and dysmenorrhoea.
Sertindole	An atypical antipsychotic indicated in the treatment of schizophrenia.
Tesmilifene	Intended for the treatment of various forms of cancer.
Etoricoxib	A selective COX-2 inhibitor used to relieve moderate post-surgical dental pain as a short-term treatment and inflammatory and painful symptoms of various forms of arthritis.
Rimonabant	For use in conjunction with diet and exercise for patients with a body mass index greater than 30 kg/m2, or patients wih a BMI greater than 27 kg/m2 with associated...
Vicriviroc	Investigated for use/treatment in HIV infection and viral infection.
Laquinimod	Investigated for use/treatment in multiple sclerosis.
Fluvastatin	An HMG-CoA reductase inhibitor used to lower lipid levels and reduce the risk of cardiovascular disease including myocardial infarction and stroke.
Rotigotine	A non-selective dopamine agonist used for the treatment of Parkinson's Disease and Restless Leg Syndrome.
Cerivastatin	A statin (or HMG CoA reductase inhibitor) used with dietary changes to decrease lipid levels and reduce the risk of cardiovascular events.
Risperidone	A second-generation antipsychotic medication used to treat a number of mental health disorders including schizophrenia, bipolar mania, psychosis, or as an adjunct in severe depression.
Selegiline	A monoamine oxidase inhibitor used to treat major depressive disorder and Parkinson's.
Halothane	A general inhalation anesthetic used for the induction and maintenance of general anesthesia.
Ifosfamide	An alkylating and immunosuppressive agent used in chemotherapy for the treatment of cancers, including testicular cancer, ovarian cancer, cervical cancer, osteocarcinoma, bladder cancer, small cell lung cancer, and non-Hodgkin's lymphoma.
Meloxicam	An NSAID used to treat osteoarthritis in adults, rheumatoid arthritis in adults, and juvenile rheumatoid arthritis in pediatrics.
Citalopram	A selective serotonin reuptake inhibitor (SSRI) used in the treatment of depression.
Fluoxetine	A selective serotonin reuptake inhibitor used to treat major depressive disorder, bulimia, OCD, premenstrual dysphoric disorder, panic disorder, and bipolar I.
Sertraline	A selective serotonin reuptake inhibitor (SSRI) indicated to treat major depressive disorder, social anxiety disorder and many other psychiatric conditions.
Mianserin	A tetracyclic antidepressant with therapeutic activity similar to amitriptyline used to treat depression and anxiety.
Antipyrine	An antipyretic agent used for the symptomatic treatment of acute otitis media, most commonly in combination with benzocaine.
Cyclophosphamide	A nitrogen mustard used to treat lymphomas, myelomas, leukemia, mycosis fungoides, neuroblastoma, ovarian adenocarcinoma, retinoblastoma, and breast carcinoma.
Trabectedin	An alkylating agent approved for the treatment of unresectable or metastatic soft tissue sarcoma (liposarcoma or leiomyosarcoma).
Venlafaxine	A selective serotonin and norepinephrine reuptake inhibitor (SNRI) used for the treatment of major depression, generalized or social anxiety disorder, and panic disorder.
Terbinafine	An allylamine antifungal used to treat dermatophyte infections of toenails and fingernails as well as other fungal skin infections.
Azelastine	A histamine H1-receptor antagonist used intranasally to treat allergic and vasomotor rhinitis and in an ophthalmic solution to treat allergic conjunctivitis.
Caffeine	A stimulant present in tea, coffee, cola beverages, analgesic drugs, and agents used to increase alertness. It is also used in to prevent and treat pulmonary complications of premature birth.
Dextromethorphan	An NMDA receptor antagonist used to treat cases of dry cough.
Docetaxel	A taxoid antineoplastic agent used in the treatment of various cancers, such as locally advanced or metastatic breast cancer, metastatic prostate cancer, gastric adenocarcinoma, and head and neck cancer.
Lidocaine	A local anesthetic used in a wide variety of superficial and invasive procedures.
Propranolol	A non-selective beta adrenergic antagonist used to treat hypertension, angina, atrial fibrillation, myocardial infarction, migraine, essential tremor, hypertrophic subaortic stenosis, and pheochromocytoma.
Ambrisentan	A selective type A endothelin receptor antagonist used to treat primary pulmonary arterial hypertension and pulmonary arterial hypertension based on diagnostic classifications.
Benzphetamine	A sympathomimetic used to manage exogenous obesity short term.
Bisoprolol	A beta-1 adrenergic blocking agent used to prevent myocardial infarction and heart failure and to treat mild to moderate hypertension.
Calcitriol	An active metabolite of vitamin D that is used to treat hyperparathyroidism and is also used in dialysis patients to combat hypocalcemia.
Chlordiazepoxide	A benzodiazepine used to treat the withdrawal symptoms of acute alcoholism, to treat preoperative anxiety, and to treat anxiety over a short term period.
Chloroquine	An antimalarial drug used to treat susceptible infections with P. vivax, P. malariae, P. ovale, and P. falciparum. It is also used for second line treatment for rheumatoid arthritis.
Clobazam	A benzodiazepine used as adjunct treatment in seizures associated with Lennox-Gastaut syndrome.
Clorazepic acid	A benzodiazepine used to treat anxiety, partial seizures, and alcohol withdrawal.
Digitoxin	A cardiac glycoside used in the treatment and management of congestive cardiac insufficiency, arrhythmias and heart failure.
Felbamate	An anticonvulsant used to treat severe epilepsy.
Fesoterodine	An antimuscarinic agent used in the treatment of overactive bladder with symptoms of urge urinary incontinence, urgency, and frequency.
Flurazepam	A long-acting benzodiazepine with a rapid onset of action that is commonly used to treat insomnia.
Flutamide	An antiandrogen used for locally confined stage B2-C and D-2 metastatic prostate carcinoma.
Guanfacine	An alpha-2A adrenergic receptor agonist used to treat ADHD.
Mefloquine	An antimalarial agent used in the prophylaxis and treatment of malaria caused by Plasmodium falciparum and Plasmodium vivax.
Nilotinib	A kinase inhibitor used for the chronic phase treatment of Chronic Myeloid Leukemia (CML) that is Philadelphia chromosome positive and for the treatment of CML that is resistant to therapy containing imatinib.
Oxycodone	An opioid used in the management of moderate to severe pain.
Pipotiazine	An antipsychotic indicated for the management of chronic, non-agitated schizophrenic patients.
Praziquantel	An anthelmintic medication used to treat parasitic worm infections such as schistosomiasis, clonorchiasis, and opisthorchiasis
Primaquine	An antimalarial indicated to prevent relapse of vivax malaria.
Dextropropoxyphene	An opioid analgesic used to treat mild to moderate pain.
Repaglinide	A antihyperglycemic used to improve glycemic control in diabetes.
Romidepsin	A histone deacetylase (HDAC) inhibitor used to treat cutaneous T-cell lymphoma.
Silodosin	An alpha-1 adrenergic receptor antagonist used to treat symptoms associated with benign prostatic hyperplasia (BPH).
Tamsulosin	An alpha-1A and alpha-1B adrenergic receptor antagonist used to treat benign prostatic hyperplasia, ureteral stones, prostatitis, and female voiding dysfunction.
Tetracycline	An antibiotic used to treat a wide variety of susceptible infections.
Tolterodine	A muscarinic receptor antagonist used to treat overactive bladder with urinary incontinence, urgency, and frequency.
Tramadol	A centrally-acting opioid agonist and SNRI (serotonin/norepinephrine reuptake inhibitor) used for the management of moderate to severe pain in adults.
Trimethoprim	An antifolate antibiotic often used in combination with sulfamethoxazole to treat a number of infections, including those of the urinary tract, respiratory tract, and gastrointestinal tract.
Zopiclone	A nonbenzodiazepine hypnotic used for the short-term management of insomnia.
Phenytoin	An anticonvulsant drug used in the prophylaxis and control of various types of seizures.
Ketamine	A rapid-acting general anesthetic and NMDA receptor antagonist used for induction of anesthesia diagnostic and surgical procedures typically in combination with a muscle relaxant.
Saxagliptin	An DPP-4 inhibitor used for the management of type 2 diabetes mellitus.
Sufentanil	An opioid used to induce and maintain anesthesia, to act as an analgesic in labor and delivery, and to treat severe, acute pain.
Bicalutamide	An androgen receptor inhibitor used to treat Stage D2 metastatic carcinoma of the prostate.
Aminophenazone	An analgesic drug used to treat acute migraine attacks in combination with ergotamine and caffeine.
Clozapine	An atypical or second-generation antipsychotic drug used in treatment-resistant schizophrenia and to decrease suicide risk in schizophrenic patients.
Promazine	A phenothiazine used to manage schizophrenia.
Carvedilol	A non selective beta-adrenergic antagonist used to treat mild to severe chronic heart failure, hypertension, and left ventricular dysfunction following myocardial infarction in clinically stable patients.
Diclofenac	An NSAID used to treat the signs and symptoms of osteoarthritis and rheumatoid arthritis.
Celecoxib	An NSAID used to treat osteoarthritis, rheumatoid arthritis, acute pain, menstrual symptoms, and to reduce polyps is familial adenomatous polyposis.
Glyburide	A sulfonylurea used in the treatment of non insulin dependent diabetes mellitus.
Sulfinpyrazone	A platelet inhibitory and uricosuric agent used to inhibit thrombotic and embolic processes and to manage the chronic phases of gout .
Seratrodast	Seratrodast (INN) is a thromboxane receptor antagonist used primarily in the treatment of asthma.
Ketobemidone	For the treatment of all types of severe pain, such as postoperative, cancer, kidney stones and fractures.
Adinazolam	For the treatment of anxiety and status epilepticus.
Temazepam	A short-acting benzodiazepine commonly used to treat panic disorders, severe anxiety, and insomnia.
Vanoxerine	An investigational dopamine transporter antagonist suggested to be beneficial in the treatment of cocaine addiction.
Cholecalciferol	A form of Vitamin D used in the treatment of specific medical conditions such as refractory rickets, hypoparathyroidism, and familial hypophosphatemia, as well as osteoporosis and chronic kidney disease.
Oxymorphone	An opioid analgesic used in the management of moderate-to-severe pain and for analgesic therapies.
Orphenadrine	A muscarinic antagonist used as an adjunct for the symptomatic relief of musculoskeletal pain and discomfort.
Cabazitaxel	An antineoplastic agent used in combination with corticosteroids to treat metastatic castration-resistant prostate cancer in patients previously treated with a docetaxel-containing treatment regimen.
Desvenlafaxine	An antidepressant agent and SNRI used for the treatment of major depressive disorders in adults.
Artemether	An antimalarial agent used in combination with lumefantrine for the treatment of acute uncomplicated malaria caused by Plasmodium falciparum.
Lumefantrine	An antimalarial agent used in combination with artemether for the treatment of acute uncomplicated malaria caused by Plasmodium falciparum.
Ambroxol	A medication indicated for airway secretion clearance therapy.
Argatroban	A synthetic direct thrombin inhibitor used for the prevention and treatment of thrombosis related to heparin use.
Bezafibrate	A lipid-lowering fibrate used in the management of primary and secondary hyperlipidaemia, when there is a lack of clinical improvement following lifestyle modifications or correction of the underlying disorder.
Brinzolamide	A carbonic anhydrase inhibitor used for the reduction of elevated intraocular pressure in patients with ocular hypertension or open-angle glaucoma.
Cephalexin	A first generation cephalosporin used to treat certain susceptible bacterial infections.
Chlorpromazine	A phenothiazine antipsychotic used to treat nausea, vomiting, preoperative anxiety, schizophrenia, bipolar disorder, and severe behavioral problems in children.
Chlorzoxazone	A drug with muscle relaxant properties that is used as an adjunct to physical therapy and analgesics to treat stiffness and pain caused by a variety of musculoskeletal conditions.
Clomethiazole	Investigated for use/treatment in strokes.
Clotiazepam	A thienodiazepine used to manage anxiety disorders and insomnia.
Cytarabine	A pyrimidine nucleoside analogue used to treat acute non-lymphocytic leukemia, lymphocytic leukemia, and the blast phase of chronic myelocytic leukemia.
Daunorubicin	An anthracycline aminoglycoside used to induce remission of nonlymphocytic leukemia and acute lymphocytic leukemia.
Dihydrocodeine	An opioid analgesic agent used for the management of pain severe enough to require an opioid analgesic and for which alternative treatments are inadequate.
Disulfiram	A carbamate derivative used to treat alcohol addiction.
Epinastine	An H1 receptor antagonist used to prevent itching in allergic conjunctivitis.
Estramustine	An antineoplastic agent used for the management of metastatic and/or progressive prostate cancer in palliative setting.
Ethanol	For therapeutic neurolysis of nerves or ganglia for the relief of intractable chronic pain in such conditions as inoperable cancer and trigeminal neuralgia (tic douloureux), in patients for whom neurosurgical...
Ethylmorphine	An opioid analgesic and antitussive agent used to reduce coughs caused by colds and lung infections in combination with codeine.
Fenofibrate	A peroxisome proliferator receptor alpha activator used to lower LDL-C, total-C, triglycerides, and Apo B, while increasing HDL-C in hypercholesterolemia, dyslipidemia, and hypertriglyceridemia.
Flunitrazepam	A benzodiazepine used to manage anxiety disorders and insomnia.
Fulvestrant	An estrogen receptor antagonist used to treat HR+ breast cancer that may also be HER2-.
Imiquimod	A toll-like receptor 7 agonist used to treat non hyperkeratotic, non hypertrophic actinic keratosis, basal cell carcinoma, genital or perianal warts, and condyloma acuminata.
Quinacrine	For the treatment of giardiasis and cutaneous leishmaniasis and the management of malignant effusions.
Methaqualone	For the treatment of insomnia, and as a sedative and muscle relaxant.
Methoxyflurane	For use in the induction and maintenance of general anesthesia
Methyltestosterone	A synthetic anabolic steroid used for the replacement therapy in conditions associated with testosterone deficiencies in males, such as hypogonadism, and treatment of advancing inoperable metastatic breast cancer in females.
Mexiletine	A class 1B antiarrhythmic agent used in the treatment of documented ventricular arrhythmias that warrant treatment.
Nicotine	A stimulatory alkaloid found in tobacco products that is often used for the relief of nicotine withdrawal symptoms and as an aid to smoking cessation.
Nitrazepam	A long-acting benzodiazepine with intermediate onset commonly used to treat panic disorders, severe anxiety, insomnia, and seizures.
Olopatadine	A histamine H1 antagonist used to treat allergic conjunctivitis and rhinitis.
Acetaminophen	An analgesic drug used alone or in combination with opioids for pain management, and as an antipyretic agent.
Perphenazine	A phenothiazine used to treat schizophrenia as well as nausea and vomiting.
Meperidine	An opioid agonist with analgesic and sedative properties used to manage severe pain.
Phenacetin	Used principally as an analgesic.
Prazepam	A benzodiazepine used to manage more severe forms of anxiety disorders.
Quazepam	A long-acting benzodiazepine used to manage insomnia.
Ropivacaine	An amide-type local anesthetic used for local or regional anesthesia during surgery and for short-term management of acute pain.
Sevoflurane	A inhalation anaesthetic agent used for induction and maintenance of general anesthesia during surgical procedures.
Sulfadiazine	A sulfonamide antibiotic used in a variety of infections, such as urinary tract infections, trachoma, and chancroid.
Tasosartan	Tasosartan is infrequently in the treatment of hypertension and heart failure.
Thiotepa	An alkylating agent used to prevent graft rejection in stem cell transplantation and to treat a variety of malignancies including certain types of adenocarcinoma and superficial bladder carcinomas.
Troleandomycin	For the treatment of bacterial infection.
Yohimbine	An alpha-2-adrenergic blocker and sympatholytic found in supplements used to.
Zomepirac	Zomepirac was indicated for the management of mild to severe pain.
Ketazolam	A long-acting benzodiazepine used to manage anxiety and insomnia.
Paramethadione	Used for the control of absence (petit mal) seizures that are refractory to treatment with other medications.
Tretinoin	A vitamin A derivative used to treat acne vulgaris and certain types of promyelocytic leukemia, as well as various skin conditions in over-the-counter medications.
Iloperidone	An atypical antipsychotic agent used to treat schizophrenia and manic or mixed episodes associated with bipolar I disorder in adults.
Vilazodone	An antidepressant agent used for the treatment of major depressive disorder that targets the 5-HT transporter and 5-HT1A receptors.
Clonidine	An alpha-2 adrenergic agonist used to treat hypertension and severe cancer pain, among other conditions, and to treat withdrawal symptoms from various substances. It is also used to aid in the diagnosis of pheochromocytoma and to prevent migraines.
Indapamide	A thiazide diuretic used to treat hypertension as well as edema due to congestive heart failure.
Ivacaftor	A cystic fibrosis transmembrane conductance regulator (CFTR) potentiator used alone or in combination products to treat cystic fibrosis in patients who have specific genetic mutations that are responsive to the medication.
Banoxantrone	For the treatment of various forms of cancer.
Indacaterol	An inhaled long-acting beta-2 adrenergic agonist used to relax bronchial smooth muscle and improve symptoms and airflow obstruction caused by Chronic Obstructive Pulmonary Disease (COPD) and moderate to severe asthma.
Chenodeoxycholic acid	A bile acid used for the treatment of primary biliary cirrhosis.
Pinacidil	Pinacidil is a cyanoguanidine drug that acts by opening ATP-sensitive potassium channels, leading to peripheral vasodilatation of arterioles and decreasing peripheral vascular resistance. The above processes result in reduced blood...
Pimecrolimus	A topical calcineurin inhibitor used in the treatment of mild-moderate atopic dermatitis who are not candidates for other types of therapy due to previous lack of response or other reasons.
Vismodegib	A hedgehog pathway inhibitor used to treat patients with locally advanced or metastatic basal cell carcinoma.
Prasugrel	A P2Y12 platelet inhibitor used to reduce risk of thrombotic cardiovascular events in unstable angina or non-ST-elevation myocardial infarction (NSTEMI), and in patients with STEMI when managed with either primary or delayed PCI.
Asenapine	An atypical antipsychotic used to treat patients with bipolar I disorder and patients with schizophrenia.
Brentuximab vedotin	A CD30-directed antibody-drug conjugate used to treat various types of lymphoma.
Lorcaserin	A serotonin 2C receptor agonist used in conjunction with physical activity and calorie restriction for weight loss in obese patients with a body mass index (BMI) of 30 and above, and in overweight patients with weight-related comorbidities.
Vandetanib	An antineoplastic kinase inhibitor used to treat symptomatic or progressive medullary thyroid cancer in patients with unresectable locally advanced or metastatic disease.
Ruxolitinib	A kinase inhibitor used to treat various types of myelofibrosis, polycythemia vera in patients who have not responded to or cannot tolerate hydroxyurea, and to treat graft-versus-host disease in cases that are refractory to steroid treatment.
Abiraterone	An antiandrogen used in the treatment of metastatic castration-resistant prostate cancer and metastatic high-risk castration-sensitive prostate cancer.
Mirabegron	A beta-3 adrenergic agonist used to treat overactive bladder and neurogenic detrusor overactivity.
Enzalutamide	A second-generation androgen receptor inhibitor used to treat castration-resistant prostate cancer and metastatic castration-sensitive prostate cancer.
Tofacitinib	A Janus kinase (JAK) inhibitor used to treat rheumatic conditions, such as rheumatoid arthritis and ankylosing spondylitis, and ulcerative colitis.
Bosutinib	An antineoplastic agent used for the treatment of chronic, accelerated, or blast phase Philadelphia chromosome-positive (Ph+) chronic myelogenous leukemia (CML) in adults with inadequate clinical response to other treatments.
Ponatinib	A kinase inhibitor used to treat patients with various types of chronic myeloid leukemia (CML).
Bedaquiline	A diarylquinoline antimycobacterial used in combination with other antibacterials to treat pulmonary multidrug resistant tuberculosis (MDR-TB).
Canagliflozin	A sodium-glucose co-transporter 2 (SGLT2) inhibitor used to manage hyperglycemia in type 2 diabetes mellitus (DM). Also used to reduce the risk of major cardiovascular events in patients with established cardiovascular disease and type 2 DM.
Alogliptin	A dipeptidyl peptidase-4 (DPP-4) inhibitor used to treat hyperglycemia in patients with type 2 diabetes mellitus.
Ospemifene	A non-hormonal estrogen receptor modulator (SERM) used to treat moderate to severe dyspareunia, a symptom of vulvar and vaginal atrophy, due to menopause.
Pomalidomide	A thalidomide analogue used in combination with dexamethasone to treat patients with multiple myeloma.
Dabrafenib	A kinase inhibitor used to treat patients with specific types of melanoma, non-small cell lung cancer, and thyroid cancer.
Trastuzumab emtansine	An antineoplastic agent and antibody-drug conjugate used to treat HER2-overexpressing breast cancer.
Taurochenodeoxycholic acid	Taurochenodeoxycholic acid is likely indicated as a choleretic and cholagogue. It is also being investigated for its role in inflammation and cancer therapy.
Mycophenolate mofetil	An inosine monophosphate dehydrogenase inhibitor used to prevent the rejection of kidney, heart, or liver transplants.
Levomilnacipran	A selective serotonin and norepinephrine reuptake inhibitor (SNRI) used to treat major depressive disorder (MDD) in adults.
Macitentan	An endothelin receptor antagonist used to manage pulmonary arterial hypertension to delay disease progression.
Dapagliflozin	A sodium-glucose cotransporter 2 inhibitor used in the management of type 2 diabetes mellitus.
Apremilast	A non-steroidal medication used for the treatment of inflammatory conditions such as psoriasis and psoriatic arthritis.
Olaparib	A poly (ADP-ribose) polymerase (PARP) inhibitor used to treat ovarian cancer, breast cancer, pancreatic cancer, and prostate cancer.
Palbociclib	An endocrine-based chemotherapeutic agent used in combination with other antineoplastic agents to treat HER2-negative and HR-positive advanced or metastatic breast cancer.
Vilanterol	A long-acting beta2-adrenergic agonist used in combination with other bronchodilators for the management of chronic obstructive pulmonary disease (COPD), including chronic bronchitis and/or emphysema.
Aliskiren	A direct renin inhibitor used to manage hypertension.
Elvitegravir	An antiretroviral agent used in combination with other antiretrovirals for the treatment of HIV-1 infection in antiretroviral treatment-experienced adults.
Cariprazine	An atypical antipsychotic used to treat schizophrenia and acute manic or mixed episodes due to bipolar I disorder.
Parecoxib	A selective COX-2 inhibitor and NSAID used for the short-term management of perioperative pain.
Brexpiprazole	A serotonin–dopamine activity modulator used in the treatment of major depressive disorder as an adjunct, schizophrenia, and agitation associated with dementia due to Alzheimer’s disease.
Rolapitant	A neurokinin-1 (NK-1) receptor antagonist used in combination with other antiemetics for the prevention of delayed nausea and vomiting associated with emetogenic chemotherapy.
Flibanserin	A 5-HT receptor modulator used for the treatment of selected premenopausal women with acquired, generalized hypoactive sexual desire disorder (HSDD).
Daclatasvir	A direct-acting antiviral agent used to treat specific hepatitis C virus (HCV) infections in combination with other antiviral agents.
Sonidegib	An antineoplastic agent used for the treatment of locally advanced recurrent basal cell carcinoma (BCC) following surgery and radiation therapy, or in cases where surgery or radiation therapy are not appropriate.
Panobinostat	A non-selective histone deacetylase inhibitor used to treat multiple myeloma in combination with other antineoplastic agents.
Ixazomib	A proteasome inhibitor used with other medications to treat multiple myeloma in patients who have received one other therapy already.
Selexipag	A non prostanoid IP prostacyclin receptor agonist used to treat pulmonary arterial hypertension.
Dasabuvir	A direct-acting antiviral agent used to treat specific hepatitis C virus (HCV) infections in combination with other antiviral agents.
Paritaprevir	A direct acting antiviral agent used in combination with other antiviral agents for the treatment of Hepatitis C Virus (HCV) infections.
Synthetic Conjugated Estrogens, A	A mixture of estrogens used to treat a variety of postmenopausal symptoms, including vaginal atrophy and dyspareunia.
Synthetic Conjugated Estrogens, B	A mixture of estrogens used to treat a variety of postmenopausal symptoms, including vaginal dryness.
Venetoclax	A BCL-2 inhibitor used to treat chronic lymphocytic leukemia, small lymphocytic lymphoma, or acute myeloid leukemia.
Esterified estrogens	A female hormone used to treat conditions related to estrogen deficiency and moderate to severe vasomotor menopausal symptoms in women.
Rucaparib	A poly (ADP-ribose) polymerase (PARP) inhibitor used to treat recurrent ovarian and prostate cancers in previously treated adults.
Safinamide	A MAO-B inhibitor used as an add-on treatment to levodopa/carbidopa for Parkinson's disease during "off" episodes.
Deutetrabenazine	A vesicular monoamine transporter 2 inhibitor used for the symptomatic treatment of tardive dyskinesia and chorea associated with Huntington's disease.
Dexchlorpheniramine maleate	A first generation antihistamine used to treat allergic and vasomotor rhinitis, allergic conjunctivitis, and mild urticaria and angioedema.
Velpatasvir	A NS5A inhibitor used to treat chronic hepatitis C infections in patients without cirrhosis or with compensated cirrhosis.
Brivaracetam	An anticonvulsant used for the treatment of partial-onset seizures that functions by binding to synaptic vesicle glycoprotein 2A (SV2A) in the brain.
Valbenazine	A vesicular monoamine transporter 2 inhibitor used to treat tardive dyskinesia and chorea associated with Huntington's disease.
Odanacatib	Investigated for use/treatment in osteoporosis .
Grazoprevir	An antiviral and NS3/4A protease inhibitor used to treat hepatitis C infections.
Perospirone	For the treatment of schizophrenia and acute cases of bipolar mania.
Etizolam	A thienodiazepine derivative used to treat anxiety and insomnia.
Rupatadine	A selective histamine H1 receptor antagonist and platelet activating factor (PAF) antagonist used to treat allergic rhinitis.
Imidafenacin	An antispasmodic with anticholinergic effects used to reduce urinary frequency.
Neratinib	A protein kinase inhibitor used to treat breast cancer that over expresses the HER2 receptor.
Voxilaprevir	A nonstructural protein 3 and 4a protease inhibitor used to treat Hepatitis C infections.
Enasidenib	An isocitrate dehydrogenase-2 inhibitor used to treat relapsed or refractory acute myeloid leukemia with an isocitrate dehydrogenase-2 mutation.
Midostaurin	An antineoplastic agent used to treat high-risk acute myeloid leukemia (AML) with specific mutations, aggressive systemic mastocytosis (ASM), systemic mastocytosis with associated hematologic neoplasm (SM-AHN), or mast cell leukemia (MCL).
Elbasvir	An antiviral and NS5A inhibitor used to treat hepatitis C infections.
Copanlisib	A PI3K inhibitor used to treat relapsed follicular lymphoma in adults.
Abemaciclib	A medication used to treat HR+ HER2- advanced or metastatic breast cancer.
Brigatinib	An anaplastic lymphoma kinase inhibitor used to treat anaplastic lymphoma kinase positive metastatic non small cell lung cancer.
Baricitinib	A Janus kinase inhibitor used to treat moderate to severe rheumatoid arthritis that has responded poorly to at least one TNF antagonist.
Macimorelin	A medication used to treat adult growth hormone deficiency.
Blonanserin	Used for the treatment of schizophrenia .
Cannabidiol	An active cannabinoid used as an adjunctive treatment for the management of seizures associated with Lennox-Gastaut syndrome or Dravet syndrome and symptomatic relief of moderate to severe neuropathic pain or other painful conditions, like cancer.
Testosterone cypionate	An androgen used to treat low or absent testosterone.
Testosterone enanthate	An androgen used to treat low or absent testosterone.
Testosterone undecanoate	An androgen indicated for testosterone replacement therapy in adult males with primary hypogonadism and hypogonadotropic hypogonadism.
Estradiol acetate	An estrogen used to treat vasomotor symptoms and moderate to severe vulvar and vaginal atrophy from menopause.
Estradiol benzoate	An estrogen indicated in combination with progesterone for the treatment of irregular menstruation.
Estradiol dienanthate	An estrogen used in some combined hormonal oral contraceptives.
Piperaquine	For the treatment of uncomplicated Plasmodium falciparum infection in adults, children, and infants aged 6 months and up weighing over 5 kg [FDA Label]. Used in combination with DB11638.
Testosterone propionate	A slow-release anabolic steroid no longer used commonly for the treatment of androgen deficiency or promotion of anabolic effects on muscles.
Bictegravir	An integrase inhibitor used to treat HIV infections.
Apalutamide	An androgen receptor inhibitor used to treat non-metastatic castration-resistant and metastatic castration-sensitive prostate cancer.
Zotepine	Zotepine, like other atypical antipsychotics, is considered as the first-line treatment in newly diagnosed schizophrenia. It is usually thought to be an option of choice for managing acute schizophrenic episodes...
Pitolisant	An antagonist and inverse agonist at the histamine H3 receptor that is used to treat narcolepsy in adults.
Tezacaftor	A medication used to treat homozygous or heterozygous F508del mutation cystic fibrosis.
Opium	A medication used to treat moderate to severe pain.
Tocopherol	Tocopherol can be used as a dietary supplement for patients with a deficit of vitamin E; this is mainly prescribed in the alpha form. Vitamin E deficiency is rare, and...
alpha-Tocopherol acetate	A form of vitamin E used to treat and prevent vitamin deficiencies.
Propiverine	An antimuscarinic agent used to treat urinary incontinence or increased urinary frequency or urgency.
Nabiximols	In Canada, Sativex has received a Notice of Compliance (NOC) for use as an as adjunctive treatment for symptomatic relief of spasticity in patients with multiple sclerosis (MS) who have...
Medical Cannabis	The use of the plant species Cannabis sativa and Cannabis indica, popularly known as marijuana, has gained popularity in recent years for the management of a wide variety of medical...
Vinflunine	A vinca alkaloid used to treat advanced or metastatic transitional cell carcinoma of the urothelial tract after a platinum containing treatment has failed.
Tocofersolan	A derivative of alpha tocopherol used to treat vitamin E deficiencies.
Delamanid	An antibiotic used to treat multidrug resistant tuberculosis.
Fosnetupitant	A medication used in combination with others to prevent chemotherapy associated nausea and vomiting.
Dihydro-alpha-ergocryptine	A nootropic with an unknown mechanism of action indicated in individuals over sixty who manifest signs and symptoms of an idiopathic decline in mental capacity.
Ipecac	An emetic agent used to induce vomiting in poisoning.
Midecamycin	A macrolide antibiotic used to treat a variety of infections caused by susceptible bacteria.
Aripiprazole lauroxil	An antipsychotic used to treat schizophrenia in adults.
Encorafenib	A kinase inhibitor used to treat unresectable or metastatic melanoma with specific mutations.
Segesterone acetate	Segesterone acetate in combination with ethinyl estradiol is indicated for use by females of reproductive potential to prevent pregnancy as a combination hormonal contraceptive (CHC). It induces contraception for thirteen...
Fosphenytoin	An antiepileptic agent used for the management of generalized convulsive status epilepticus and prevention and treatment of seizures occurring during neurosurgery.
Cobicistat	A CYP3A inhibitor used to increase the systemic exposure of atazanavir or darunavir in combination with other antiretroviral agents in the treatment of HIV-1 infection.
Dapoxetine	A selective serotonin reuptake inhibitor used in the treatment of premature ejaculation.
Linagliptin	A dipeptidyl peptidase-4 (DPP-4) inhibitor used to manage hyperglycemia in patients with type 2 diabetes mellitus.
Cobimetinib	An antineoplastic agent and selective inhibitor of the mitogen-activated extracellular kinase (MEK) pathway used to treat unresectable or metastatic melanoma.
Osimertinib	A tyrosine kinase inhibitor used in the treatment of certain types of non-small cell lung carcinoma.
Netupitant	An antiemetic agent used in combination with palonosetron to prevent acute and delayed vomiting and nausea caused by chemotherapy.
Ceritinib	An antineoplastic kinase inhibitor used to treat anaplastic lymphoma kinase (ALK)-positive metastatic non-small cell lung cancer (NSCLC) in patients with inadequate clinical response or intolerance to crizotinib.
Ribociclib	A kinase inhibitor used to treat HR+, HER2- advanced or metastatic breast cancer.
Nintedanib	A triple angiokinase inhibitor indicated for the treatment of idiopathic pulmonary fibrosis, systemic sclerosis-associated interstitial lung disease, and in combination with docetaxel for non-small cell lung cancer.
Roflumilast	A selective phosphodiesterase-4 inhibitor indicated to decrease the risk of exacerbations in patients with severe chronic obstructive pulmonary disease (COPD) and to treat skin conditions such as plaque psoriasis and atopic dermatitis.
Suvorexant	A orexin receptor antagonist used to treat insomnia that is characterized by difficulties with sleep onset and/or sleep maintenance.
Tasimelteon	A melatonin receptor agonist used to treat Non- 24-Hour Sleep-Wake Disorder.
Vorapaxar	A platelet aggregation inhibitor used to reduce thrombotic cardiovascular events in patients with a history of myocardial infarction (MI) or peripheral arterial disease (PAD).
Zuclopenthixol	An antipsychotic indicated for the management of schizophrenia. The acuphase formulation is indicated for initial treatment of acute psychosis or exacerbation of psychosis, while the depot formulation is best for maintenance.
Idelalisib	An antineoplastic kinase inhibitor used to treat chronic lymphocytic leukemia (CLL), relapsed follicular B-cell non-Hodgkin lymphoma (FL), and relapsed small lymphocytic lymphoma (SLL).
Lacosamide	An antiepileptic drug used to treat partial-onset seizures and primary generalized tonic-clonic seizures.
Pranlukast	A leukotriene receptor antagonist for the treatment of allergic rhinitis and asthma symptoms.
Eravacycline	A tetracycline antibiotic used to treat complicated intra-abdominal infections.
Fosaprepitant	An antiemetic drug used in combination with other antiemetic agents for the prevention of acute and delayed nausea and vomiting caused by chemotherapy.
Cethromycin	A ketolide antibiotic with broad-spectrum activity against Gram-positive, Gram-negative, and atypical bacteria that may be useful for treating several conditions including community-acquired pneumonia, inhalation anthrax, plague, and tularemia.
Tegafur	An antineoplastic agent used in combination with other anticancer medications to treat advanced gastric and colorectal cancers.
Doravirine	A non-nucleoside reverse transcriptase inhibitor used in combination with other antiretrovirals to treat HIV-1 infections.
Duvelisib	An inhibitor of phosphatidylinositol 3-kinase delta and gamma used to treat relapsed or refractory chronic lymphocytic leukemia or small lymphocytic lymphoma.
Nevirapine	A non-nucleoside reverse transcriptase inhibitor used as part of a management regimen for HIV-1 virus infection.
(R)-warfarin	Warfarin consists of a racemic mixture of two active enantiomers—R- and S- forms—each of which is cleared by different pathways. S-warfarin is 2-5 times more potent than the R-isomer in...
Ivosidenib	An isocitrate dehydrogenase-1 inhibitor used to treat acute myeloid leukemia and cholangiocarcinoma in adults with a susceptible IDH1 mutation.
3,5-diiodothyropropionic acid	DITPA has been investigated in Congestive Heart Failure.
5-androstenedione	5-androstenedione is a prohormone of testosterone. In the United States, the Controlled Substance Act is inclusive to anabolic steroids and their precursors. Thus 5-androstenedione is a controlled substance, and its...
Alclometasone	A topical corticosteroid used to relieve the symptoms of corticosteroid-responsive dermatoses.
Aldosterone	A hormone secreted by the adrenal cortex that regulates electrolyte and water balance by increasing the renal retention of sodium and the excretion of potassium.
Amcinonide	A topical corticosteroid used in the treatment of inflammation and pruritus due to a variety of dermatoses.
Androstenedione	A delta-4 C19 steroid that is produced not only in the testis, but also in the ovary and the adrenal cortex. Depending on the tissue type, androstenedione can serve as...
Beclomethasone dipropionate	An inhaled corticosteroid used as maintenance treatment in the prophylaxis of asthma attacks.
Clobetasol	Clobetasol is under investigation for the treatment of Scleroderma. Clobetasol has been investigated for the prevention of Psoriasis and Cutaneous Atrophy Due to Corticosteroids.
Clobetasol propionate	A corticosteroid used to treat corticosteroid-responsive dermatoses and plaque psoriasis.
Clobetasone	A corticosteroid used to treat dry eyes, eczema, and dermatitis.
Corticosterone	An adrenocortical steroid that has modest but significant activities as a mineralocorticoid and a glucocorticoid. (From Goodman and Gilman's The Pharmacological Basis of Therapeutics, 8th ed, p1437)
Corticotropin	A diagnostic agent used in the screening of patients presumed to have adrenocortical insufficiency.
Cyproterone acetate	A steroid used in combination with ethinyl estradiol to treat women with severe acne and symptoms of androgenization. Also used alone at much higher doses for palliative treatment of patients with prostate cancer
Nomegestrol	Nomegestrol is an ingredient in the EMA-authorised product Zoely.
Nomegestrol acetate	Nomegestrol acetate, also known as NOMAC, is a progestin used in oral contraceptives, menopausal hormone therapy, and for the treatment of gynecological disorders.
Desogestrel	A synthetic progestin used in contraception, often in combination with ethinyl estradiol.
Desonide	A topical corticosteroid used for the symptomatic treatment of inflammatory and pruritic manifestations of corticosteroid responsive dermatoses.
Desoxycorticosterone acetate	Not Annotated
Desoxycorticosterone pivalate	Examined for treatment of adrenocortical insufficiency especially in multiple sclerosis, congenital cerebral palsy, polyarteritis nodosa, and rheumatoid arthritis. Currently only approved in treating cats and dogs for the treatment of...
Difluocortolone	A topical corticosteroid used for the symptomatic treatment of inflammatory skin disorders like eczema, seborrheic eczema, lichen planus and psoriasis.
Difluprednate	A topical corticosteroid used for the symptomatic treatment of inflammation and pain associated with ocular surgery.
Dydrogesterone	A synthetic progesterone for menstrual cycle regulation, infertility treatment, prevention of miscarriage, and other conditions.
Equilenin	Equilenin is an estrogenic steroid produced by horses. It has a total of five double bonds in the A- and B-ring. High concentration of equilenin is found in the urine...
Equilin	For the treatment of moderate to severe vasomotor symptoms associated with the menopause, atrophic vaginitis, osteoporosis, hypoestrogenism due to hypogonadism, castration, primary ovarian failure, breast cancer (for palliation only), and...
Etynodiol	Etynodiol (INN), or ethynodiol (BAN) is a steroidal progestin related to norethisterone which was never marketed. While etynodiol is sometimes used as a synonym for etynodiol diacetate, it usually refers...
Ethynodiol diacetate	An oral contraceptive used to prevent pregnancy.
Fludrocortisone	A mineralocorticoid used to treat adrenocortical insufficiency and salt-losing adrenogenital syndrome.
Flumethasone	A corticosteroid used to treat contact dermatitis, atopic dermatitis, eczema, psoriasis, diaper rash, and other skin conditions.
Fluocinolone acetonide	A corticosteroid used to treat skin conditions, eczematous otitis externa, diabetic macular edema, and non-infectious uveitis of the posterior segment of the eye.
Fluocinonide	A high potency corticosteroid commonly used topically for a number of inflammatory skin conditions.
Fluprednidene	Fluprednidene is a corticosteroid.
Fluprednisolone	A synthetic glucocorticoid with anti-inflammatory properties.
Flurandrenolide	A corticosteroid used to treat corticosteroid-responsive dermatoses.
Gestodene	Gestodene is a progestogen hormonal contraceptive. Products containing gestoden include Meliane, which contains 20 mcg of ethinylestradiol and 75 mcg of gestodene; and Gynera, which contains 30 mcg of ethinylestradiol...
Halcinonide	A corticosteroid used for the management and symptomatic relief of the inflammatory and pruritic manifestations of corticosteroid-responsive dermatoses.
HE3286	For the treatment of rheumatoid arthritis and type 2 diabetes.
Hydrocortisone succinate	A corticosteroid used to treat severe allergic reactions, dermatologic diseases, endocrine disorders, gastrointestinal diseases, hematological disorders, neoplastic diseases, nervous system conditions, ophthalmic diseases, renal diseases, respiratory diseases, and rheumatic disorders.
Hydroxyprogesterone	Not Annotated
Liotrix	May be used to treat primary, secondary or tertiary hypothyroidism. May also be used to suppress thyroid stimulating hormone (TSH) secretion in patients with simple (nontoxic) goiter, subacute or chronic...
Loteprednol etabonate	A corticosteroid used to treat allergic conjunctivitis as well as inflammation and pain after ocular surgery.
Lynestrenol	A progestin used for contraception and in the treatment of menstrual disorders.
Medrogestone	A progestin used as an adjunct to control secondary amenorrhea and dysfunctional bleeding in adolescent and adult females, and treat endometrial shedding in menopausal women.
Medrysone	A topical glucocorticoid applied ophthalmically for the treatment of various ocular inflammatory or allergic conditions.
Megestrol acetate	A progestin that is administered orally to treat anorexia and cachexia or serious unexplained weight loss and is also used as an antineoplastic agent to treat certain types of malignancy.
Melengestrol	Melengestrol is a steroidal progestin and antineoplastic agent which was never marketed. An acylated derivative, melengestrol acetate, is used as a growth promoter in animals.
Meprednisone	Not Annotated
Mometasone	A corticosteroid with no indications.
Mometasone furoate	A corticosteroid used to treat asthma, allergic rhinitis, nasal congestion, nasal polyps, dermatitis, and pruritus.
Norelgestromin	A progestin used for the prevention of pregnancy in women who elect to use a transdermal patch as a method of contraception.
Norethynodrel	A synthetic progestational hormone with actions and uses similar to those of PROGESTERONE. It has been used in the treatment of functional uterine bleeding and endometriosis. As a contraceptive, it...
Prednicarbate	A medium potency topical corticosteroid used to manage pruritus and inflammation associated with responsive skin conditions.
Prednylidene	Prednylidene is an experimental systemic glucocorticoid.
Pregnenolone	A 21-carbon steroid, derived from cholesterol and found in steroid hormone-producing tissues. Pregnenolone is the precursor to gonadal steroid hormones and the adrenal corticosteroids.
Promegestone	Not Annotated
Rimexolone	A glucocorticoid used to treat inflammation of the eye.
Atovaquone	An antimicrobial indicated for the prevention and treatment of Pneumocystis jirovecii pneumonia (PCP) and for the prevention and treatment of Plasmodium falciparum malaria.
Gestrinone	Endometriosis with or without accompanying sterility. Treatment is limited to a single course of 6 months duration per lifetime [L1699, L1700].
Chlormadinone	A progestin indicated in combination with an estrogen for oral combined hormonal contraceptive therapy.
Quingestanol	Not Annotated
Demegestone	Demegestone is a progesterone receptor agonist that was previously used to treat luteal insufficiency. It was previously marketed in France as Lutionex, but has since been discontinued.
(S)-Warfarin	Warfarin consists of a racemic mixture of two active enantiomers—R- and S- forms—each of which is cleared by different pathways. S-warfarin is 2-5 times more potent than the R-isomer in...
Thiamylal	Used for the production of complete anaesthesia of short duration, for the induction of general anaesthesia, and for inducing a hypnotic state.
Agmatine	Agmatine is being studied experimentally for several indications such as cardioprotection, diabetes, decreased kidney function, neuroprotection (stroke, severe CNS injuries, epilepsy, glaucoma, and neuropathic pain), and psychiatric conditions (depression, anxiety,...
Gemfibrozil	A lipid regulator that is used in the reduction of serum triglyceride levels in high-risk patients with hyperlipidemia.
Balaglitazone	Balaglitazone has been used in trials studying the treatment of Diabetes Mellitus, Type 2.
Ciglitazone	Developed by Takeda Pharmaceuticals in the early 1980s, it is considered the prototypical compound for the thiazolidinedione class. Ciglitazone was never used as a medication, but it sparked interest in...
Lobeglitazone	Lobeglitazone was approved by the Ministry of Food and Drug Safety (South Korea) in 2013, and is being monitored by postmarketing surveillance until 2019. Lobeglitazone is not approved for use...
Netoglitazone	Netoglitazone (MCC-555) is a hypoglycemic agent.
Rivoglitazone	Rivoglitazone (INN) is a thiazolidinedione undergoing research for use in the treatment of type 2 diabetes. It is being developed by Daiichi Sankyo Co.
Rosiglitazone	A thiazolidinedione indicated as an adjunct to diet and exercise to maintain glycemic control in type 2 diabetes.
Paliperidone	An atypical antipsychotic used in the treatment of schizophrenia and other schizoaffective or delusional disorders.
6-O-benzylguanine	6-O-benzylguanine has been used in trials studying the treatment of HIV Infection, Adult Gliosarcoma, Adult Glioblastoma, Stage I Adult Hodgkin Lymphoma, and Stage II Adult Hodgkin Lymphoma, among others.
Fluvoxamine	A selective serotonin-reuptake inhibitor used to treat obsessive-compulsive disorder.
Indalpine	Indalpine was one of the first selective serotonin reuptake inhibitors to reach the American market. It was initially marketed by Pharmuka. However, after the emergence of widespread concern regarding adverse...
Milnacipran	A selective serotonin and norepinephrine reuptake inhibitor (SNRI) used for the treatment of fibromyalgia and a short-term treatment of major depressive disorder.
Fusidic acid	A topical antibacterial agent used to prevent and treat mild to moderate skin infections caused by susceptible bacteria.
Aranidipine	Aranidipine has been used for many years to treat angina pectoris and hypertension.
Lenvatinib	A receptor tyrosine kinase inhibitor used for the treatment of metastatic thyroid cancer, advanced renal cell carcinoma in combination with everolimus, and unresectable hepatocellular carcinoma.
Lorpiprazole	In 2016, lorpiprazole was classified in the "Chemical structure-related drug-like criteria of global approved drugs" as an antipsychotic and anxiolytic. An antipsychotic is a medication used to treat a state...
Propacetamol	Propacetamol is a paracetamol prodrug of intravenous administration used to control fever and pain of perioperative period in multimodal analgesia therapy.
Valproic acid	An anticonvulsant used to control complex partial seizures and both simple and complex absence seizures.
Pentamidine	An antifungal agent used to treat Pneumocystis pneumonia in patients infected with HIV.
St. John's Wort	An herbal ingredient used in non-prescription therapeutic products for the short-term treatment of minor skin irritations, insomnia, depression, and anxiety.
9-aminocamptothecin	Aminocamptothecin has been used in trials studying the treatment of Lymphoma, Gastric Cancer, Ovarian Cancer, Esophageal Cancer, and Ovarian Neoplasms, among others.
Methylprednisone	Methylprednisone has been used in trials studying the treatment of Leukemia, Rheumatoid Arthritis, Renal Transplantation, Kidney Transplantation, and Acute Lymphocytic Leukemia, among others.
Dacomitinib	A medication used to treat non small cell lung cancer with EGFR exon 19 deletion of exon 21 L858R substitution.
Nebivolol	A beta blocking agent used to treat hypertension and aid in the management of heart failure.
Larotrectinib	A kinase inhibitor used to treat solid tumors with neurotrophic receptor tyrosine kinase gene fusion, are metastatic, high risk for surgery, or have no alternative treatments.
Lorlatinib	An anaplastic lymphoma kinase inhibitor used to treat anaplastic lymphoma kinase positive metastatic non small cell lung cancer.
Gilteritinib	An AXL receptor tyrosine kinase inhibitor used to treat relapsed or refractory acute myeloid leukemia.
1,2-Benzodiazepine	Benzodiazepine is under investigation for the prevention of Delirium and C.Surgical Procedure; Cardiac. Benzodiazepine has been investigated for the treatment of Obesity, Sleep Apnea, Obstructive, and Disorders of Gallbladder, Biliary...
Brotizolam	A benzodiazepine analogue with sedative-hypnotic properties used for short-term treatment of severe or debilitating insomnia.
Vitamin D	An ingredient found in a variety of supplements and vitamins.
Doxazosin	An alpha-1 adrenergic receptor used to treat mild to moderate hypertension and urinary obstruction due to benign prostatic hyperplasia.
SN-38	Investigated for use/treatment in colorectal cancer.
Prucalopride	A 5-HT4 receptor agonist indicated to treat adults with chronic idiopathic constipation.
Glasdegib	A sonic hedgehog receptor inhibitor used to treat newly diagnosed acute myeloid leukemia in patients over 75 years who cannot receive intense chemotherapy.
Phentermine	A sympathomimetic anorectic agent used as a short-term adjunct therapy that is included in a regimen of weight reduction in cases of exogenous obesity.
Metoprolol	A beta-blocker used in the treatment of hypertension and angina, and used to reduce mortality due to myocardial infarction.
Esketamine	A NMDA receptor antagonist used for treatment-resistant depression.
Siponimod	A medication used to treat relapsing multiple sclerosis.
Erdafitinib	A fibroblast growth factor receptor tyrosine kinase inhibitor used to treat locally advanced or metastatic urothelial carcinoma.
Tenofovir alafenamide	A nucleoside analog reverse transcriptase inhibitor used for the treatment of chronic hepatitis B virus infection in adults with compensated liver disease.
Alpelisib	Alpelisib is indicated in combination with fulvestrant to treat postmenopausal women, and men, with advanced or metastatic breast cancer. This cancer must be hormone receptor (HR)-positive, human epidermal growth factor...
Selinexor	Selinexor is indicated in combination with bortezomib and dexamethasone for the treatment of multiple myeloma in adult patients who have received at least one prior therapy. Selinexor is also indicated...
Metronidazole	A nitroimidazole used to treat trichomoniasis, amebiasis, inflammatory lesions of rosacea, and bacterial infections, as well as prevent postoperative infections.
Clotrimazole	A topical broad-spectrum antifungal agent used for the treatment of a wide variety of dermatophyte infections and candidiasis.
Triclabendazole	An anthelmintic drug used to treat fascioliasis.
Vitamin E	An antioxidant vitamin used in many skin creams and multivitamin preparations.
Isotretinoin	A retinoid used to treat severe recalcitrant acne.
Paroxetine	A selective serotonin reuptake inhibitor used to treat major depressive disorder, panic disorder, OCD, social phobia, generalized anxiety disorder, the vasomotor symptoms of menopause, and premenstrual dysphoric disorder.
Levocetirizine	An H1-receptor antagonist used to treat symptoms associated with chronic allergic rhinitis and uncomplicated cases of chronic idiopathic urticaria.
Butyrfentanyl	A methylated fentanyl analog with no clinical indications but is commonly used as a recreational drug.
Pexidartinib	An antitumor agent that is used for the treatment of rare disease tenosynovial giant cell tumors (TGCT) by inhibiting colony-stimulating factor 1 and its receptor.
Bimatoprost	A prostaglandin analog used to treat hypotrichosis of the eyelashes and intraocular pressure in open angle glaucoma or ocular hypertension.
Pretomanid	Part of a three-drug regimen used for the treatment of extensively drug-resistant and multidrug-resistant pulmonary tuberculosis.
Hydroxychloroquine	An antimalarial medication used to treat uncomplicated cases of malaria and for chemoprophylaxis in specific regions. Also a disease modifying anti-rheumatic drug (DMARD) indicated for treatment of rheumatoid arthritis and lupus erythematosus.
Entrectinib	Entrectinib is indicated for the treatment of metastatic ROS1-positive non-small cell lung cancer in adults. Entrectinib is also indicated in adults and children over 12 years old for the treatment...
Fedratinib	Fedratinib is indicated for the treatment of adult patients with intermediate-2 or high-risk primary or secondary (post-polycythemia vera or post-essential thrombocythemia) myelofibrosis.[L8090,L47016]
Lefamulin	A pleuromutilin antibacterial used to treat community-acquired bacterial pneumonia (CABP).
Sulfamethoxazole	An oral sulfonamide antibiotic, given in combination with trimethoprim, used to treat a variety of infections of the urinary tract, respiratory system, and gastrointestinal tract.
Istradefylline	A selective adenoside A2A receptor antagonist indicated in adjunct to levodopa and carbidopa for the treatment of Parkinson's Disease.
Zafirlukast	A leukotriene receptor antagonist used for prophylaxis and chronic treatment of asthma.
Ibuprofen	An NSAID and non-selective COX inhibitor used to treat mild-moderate pain, fever, and inflammation.
Flucloxacillin	A narrow spectrum penicillin antibiotic that exerts specific activity against Gram positive organisms in skin and soft tissue infections, except those caused by methicillin resistant staphylococcus aureus (MRSA).
Mexazolam	A benzodiazepine indicated to treat anxiety with or without psychoneurotic conditions.
Metoclopramide	An antiemetic agent and dopamine D2 antagonist used in the treatment of gastroesophageal reflux disease, prevention of nausea and vomiting, and to stimulate gastric emptying.
Dexloxiglumide	For the treatment of Irritable Bowel Syndrome (IBS) and Gastroesophageal Reflux Disease (GERD).
Calanolide A	For use in combination treatment of HIV infection (AIDS).
Plitidepsin	Intended for the treatment of various forms of cancer.
Rifalazil	Investigated for use/treatment in atherosclerosis, bacterial infection, and peripheral vascular disease.
Azimilide	Investigated for use/treatment in arrhythmia and atrial fibrillation.
Capravirine	Investigated for use/treatment in acquired immune deficiency syndrome (AIDS) and aids-related infections and HIV infection.
Polatuzumab vedotin	A CD79b antibody conjugate indicated to treat different types of large B-cell lymphoma.
Levamlodipine	A calcium channel blocker used to treat hypertension.
Fluprednisolone acetate	Not Annotated
Baloxavir marboxil	A polymerase acidic endonuclease inhibitor used to treat uncomplicated influenza.
Tenapanor	An NHE3 inhibitor indicated for the treatment of constipation-predominant irritable bowel syndrome (IBS-C) and chronic kidney disease,
Anastrozole	A competitive, selective, non-steroidal aromatase inhibitor used as adjuvant therapy for the treatment of hormone receptor-positive breast cancer in postmenopausal women.
Trifarotene	A topical retinoid indicated for the treatment of acne vulgaris.
Elexacaftor	A small molecule CFTR corrector used in combination with tezacaftor and ivacaftor for the treatment of cystic fibrosis patients with one F508del-CFTR mutation.
Prednisolone acetate	A glucocorticoid used to treat a wide variety of endocrine, inflammatory, and immune conditions as well as for palliation of neoplastic conditions.
Hydroxyzine	An antihistamine used to treat anxiety and tension associated with psychoneuroses, as well as allergic conditions such as pruritus and chronic urticaria.
Zanubrutinib	A kinase inhibitor used to treat mantle cell lymphoma, a type of B-cell non-Hodgkin lymphoma, in adults who previously received therapy.
Voxelotor	A drug used to inhibit the polymerization of hemoglobin S, preventing the painful and sometimes lethal vaso-occlusive crises associated with sickle cell disease.
Cenobamate	A small molecule drug indicated to treat partial onset seizures in adults.
Enfortumab vedotin	An antibody-drug conjugate comprised of a fully human monoclonal antibody and microtubule-disrupting chemotherapeutic agent used in the treatment of advanced or metastatic urothelial cancer.
Trastuzumab deruxtecan	An antibody used to treat certain types of unresectable or metastatic HER2 positive breast cancer.
Lemborexant	A dual orexin antagonist indicated for the treatment of sleep-onset and/or sleep maintenance insomnia.
Darolutamide	An androgen receptor antagonist used for castration-resistant, non-metastatic prostate cancer and metastatic hormone-sensitive prostate cancer.
Upadacitinib	An oral Janus kinase (JAK)1-selective inhibitor used in the treatment of moderate to severe rheumatoid arthritis, active psoriatic arthritis, ankylosing spondylitis, and severe atopic dermatitis, including in patients who did not respond well to other therapies.
Lumateperone	A novel 2nd generation antipsychotic used to manage both positive and negative symptoms in patients with schizophrenia.
Ubrogepant	An oral CGRP antagonist used in the acute treatment of migraine with or without aura.
Avapritinib	A selective tyrosine kinase inhibitor being investigated for the treatment of multidrug resistant gastrointestinal tumors.
Tazemetostat	A methyltransferase inhibitor indicated to treat patients 16 years and older with metastatic or locally advanced epithelioid sarcoma not eligible for complete resection.
Rimegepant	An oral CGRP receptor antagonist used for the acute treatment of migraines with or without aura in adults.
Umifenovir	A dual direct-acting antiviral/host-targeting agent used in the treatment and prophylaxis of influenza and other respiratory viruses.
Osilodrostat	An oral inhibitor of cortisol synthesis used to treat Cushing's disease by normalizing hypercortisolism.
Norethindrone enanthate	A synthetic progestogen indicated for contraceptive therapy.
Ozanimod	A sphingosine 1-phosphate receptor modulator being studied to treat Multiple Sclerosis (MS) and inflammatory bowel disease (IBD).
Methotrexate	An antineoplastic agent used the treatment of a wide variety of cancers as well as severe psoriasis, severe rheumatoid arthritis, and juvenile rheumatoid arthritis.
Selumetinib	A MEK 1/2 inhibitor used in pediatric patients to treat neurofibromatosis type 1 (NF1) accompanied by symptomatic, inoperable plexiform neurofibromas (PN).
Prednisolone phosphate	A corticosteroid used to treat inflammation, immune reactions, as well as endocrine or neoplastic conditions.
Tucatinib	A kinase inhibitor used to treat certain types of unresectable/metastatic HER-2 positive breast cancer.
Pemigatinib	A kinase inhibitor used to treat locally advanced or metastatic, unresectable cholangiocarcinoma in previously treated adult patients.
Remdesivir	A nucleoside analog used to treat RNA virus infections including COVID-19.
Acalabrutinib	A Bruton tyrosine kinase inhibitor used to treat mantle cell lymphoma, chronic lymphocytic leukemia, and small lymphocytic lymphoma.
Capmatinib	A kinase inhibitor targeting c-Met receptor tyrosine kinase in the treatment of non-small cell lung cancer with MET exon 14 skipping.
Alectinib	A kinase inhibitor used to treat anaplastic lymphoma kinase positive metastatic non small cell lung cancer.
Belinostat	A histone deacetylase (HDAC) inhibitor used for the treatment of patients with relapsed or refractory peripheral T-cell lymphoma (PTCL).
Selpercatinib	A RET receptor tyrosine kinase inhibitor for the treatment of RET-driven non-small cell lung cancer, medullary thyroid cancer, and thyroid cancer in appropriate patient populations.
Ripretinib	A kinase inhibitor used to treat advanced gastrointestinal stromal tumor (GIST).
Apomorphine	A morphine derivative D2 dopamine agonist used to treat hypomobile "off" episodes of advanced Parkinson's disease.
Betamethasone phosphate	A fast acting ester prodrug of a corticosteroid used to treat inflammatory conditions.
Lurbinectedin	A chemotherapeutic DNA alkylating agent used in the treatment of metastatic small-cell lung cancer.
Dexamethasone acetate	Commonly known as decadron, dexamethasone acetate is a glucocorticosteroid previously marketed in the USA for the treatment of inflammatory respiratory, allergic, autoimmune, and other conditions.[T797,L10695,L14348] Developed in 1957, dexamethasone is...
Fenfluramine	Fenfluramine is a phenethylamine that is structurally similar to serotonin. Due to its ability to increase extracellular serotonin levels, modulate serotonergic and other neurologic receptors, and control neurotransmission, it is effective in treating pharmacoresistant seizures.
Fostemsavir	An antiretroviral HIV-1 attachment inhibitor targeted against the gp120 subunit within the HIV-1 gp160 envelope glycoprotein.
Risdiplam	An oral mRNA splicing modifier used in the treatment of spinal muscular atrophy (SMA).
Oliceridine	A biased opioid agonist indicated for the management of severe acute pain in adult patients. Through preferential activation of G-protein-coupled signalling pathways, oliceridine provides analgesic effect with a comparable or improved safety profile over conventional opioid agonists.
Pralsetinib	A RET receptor tyrosine kinase inhibitor for the treatment of metastatic RET-driven non-small cell lung cancer.
Lonafarnib	A potent farnesyl transferase inhibitor used to reduce mortality associated with Hutchinson-Gilford progeria syndrome (HGPS) and other progeroid laminopathies.
Tirbanibulin	A tyrosine kinase and tubulin inhibitor used to treat actinic keratosis on the face or scalp.
Vibegron	A beta-3 adrenergic agonist the treatment of overactive bladder (OAB) with symptoms of urge urinary incontinence, urgency, and urinary frequency in adults.
Relugolix	An oral GnRH receptor antagonist for androgen deprivation therapy in the treatment of advanced prostate cancer.
Tepotinib	An oral tyrosine kinase inhibitor targeted against MET for the treatment of metastatic non-small cell lung cancer in patients exhibiting MET exon 14 skipping mutations.
Voclosporin	A calcineurin inhibitor for the treatment of lupus nephritis (LN) in patients diagnosed with systemic lupus erythematosus (SLE).
Scopolamine	A belladonna alkaloid with anticholinergic effects indicated for the treatment of nausea and vomiting associated with motion sickness and postoperative nausea and vomiting (PONV).
Umbralisib	A kinase inhibitor used to treat rare forms of refractory lymphoma.
Tivozanib	A kinase inhibitor to treat adult patients with renal cell carcinoma (RCC) who have failed prior systemic therapies or experienced relapsed disease.
Ponesimod	A sphingosine 1-phosphate receptor modulator indicated to treat relapsing multiple sclerosis.
Pimavanserin	A second generation atypical antipsychotic used for the treatment of hallucinations and delusions caused by Parkinson's Disease.
Glycopyrronium	An anticholinergic agent used to treat hyperhidrosis, severe drooling, COPD, used with other medications to treat ulcers, and used in anesthesia.
Estetrol	An estrogen used in combination with drospirenone for oral contraception.
Loncastuximab tesirine	An antibody-drug conjugate used for the treatment of relapsed and refractory B-cell lymphomas.
Naloxone	An opioid receptor antagonist used to rapidly reverse an opioid overdose. Also included in some drug formulations as an abuse deterrent to prevent injection.
Sotorasib	An experimental KRAS inhibitor being investigated for the treatment of KRAS G12C mutant non small cell lung cancer, colorectal cancer, and appendix cancer.
Infigratinib	An FGFR inhibitor used to treat locally advanced or metastatic cholangiocarcinoma in adults with a fibroblast growth factor receptor 2 (FGFR2) rearrangement.
Ibrexafungerp	A triterpene antifungal indicated in the treatment of vulvovaginal candidiasis and prevention of recurrent vulvovaginal candidiasis in post-menarchal patients.
Samidorphan	A novel opioid-system modulator, similar to naltrexone, that functions primarily as a μ-opioid receptor antagonist in vivo and is used primarily in combination with antipsychotics to reduce their metabolic dysfunction-associated adverse effects.
Finerenone	A nonsteroidal mineralocorticoid receptor antagonist indicated to lower the risk of eGFR decline, end stage kidney disease, cardiovascular death, heart attack, and hospitalization for heart failure in chronic kidney disease associated with type 2 diabetes.
Belumosudil	An oral inhibitor of rho-associated coiled-coil-containing protein kinases (ROCK) used in the treatment of chronic graft-versus-host disease (GVHD).
Belzutifan	An inhibitor of hypoxia-inducible factor 2α used as an antineoplastic in the treatment of certain cancers associated with von Hippel-Lindau (VHL) disease.
Fexinidazole	An orally bioavailable 2-substituted 5-nitroimidazole used to treat early- and late-stage human African trypanosomiasis caused by Trypanosoma brucei gambiense.
Tisotumab vedotin	A tissue factor-directed antibody drug conjugate that is used to treat adults with recurrent or metastatic cervical cancer with disease progression on or after chemotherapy.
Mobocertinib	An oral kinase inhibitor targeted against EGFR and used in the treatment of NSCLC with EGFR exon 20 insertion mutations.
Atogepant	An oral CGRP antagonist used for the preventative therapy of episodic migraine headaches.
Avacopan	An orally bioavailable complement 5a receptor (C5aR) antagonist for the treatment of severe anti-neutrophil cytoplasmic (auto)antibody (ANCA)-associated vasculitis.
Asciminib	An inhibitor of ABL/BCR-ABL1 tyrosine kinase for the treatment of patients with Philadelphia chromosome-positive CML, including those with the T315I mutation.
Maribavir	A cytomegalovirus (CMV) pUL97 kinase inhibitor used for the treatment of refractory post-transplant CMV infection.
Nirmatrelvir	An oral protease inhibitor with emergency use authorization for the treatment of mild-to-moderate COVID-19.
Levoketoconazole	One of two enantiomeric forms of racemic ketoconazole that strongly inhibits multiple steroidogenic enzymes and is used for the symptomatic treatment of endogenous Cushing's syndrome.
Daridorexant	A dual orexin receptor antagonist used to treat insomnia in adults.
Sotagliflozin	An orally administered dual SGLT1/2 inhibitor used alongside insulin to improve glycemic control in patients with type 1 diabetes mellitus.
Abrocitinib	A kinase inhibitor used to treat moderate-to-severe atopic dermatitis in adults.
Palovarotene	A selective agonist of retinoic acid receptor gamma (RARγ) used to reduce heterotopic ossification in patients with Fibrodysplasia Ossificans Progressiva (FOP).
Mitapivat	A pyruvate kinase activator used to treat hemolytic anemia in adults with pyruvate kinase (PK) deficiency.
Secnidazole	A nitroimidazole antibiotic used to treat bacterial vaginosis.
Nabilone	A synthetic delta-9-THC used in the treatment of anorexia and weight loss in HIV patients as well as nausea and vomiting in cancer chemotherapy.
Cannabinol	Cannabinol (CBN) is a physiologically inactive constituent of Cannabis sativa.
Nalmefene	An opioid antagonist used to reduce alcohol consumption in adults with alcohol dependence and treat and prevent opioid overdose.
Pacritinib	A kinase inhibitor used for the treatment of primary and secondary myelofibrosis in adult patients with significantly reduced platelet counts.
Ganaxolone	A neuroactive steroid GABA-A receptor modulator used for the treatment of seizures associated with CDKL5 deficiency disorder (CDD).
Thalidomide	A medication used to treat cancers, particularly newly diagnosed multiple myeloma, and erythema nodosum leprosum.
Mavacamten	A myosin inhibitor used to treat obstructive hypertrophic cardiomyopathy.
Tapinarof	A therapeutic aryl hydrocarbon receptor-modulating agent (TAMA) indicated for the treatment of adult psoriasis.
Mycophenolic acid	An immunosuppressant used to prevent organ transplant rejections.
Stiripentol	An antiepileptic agent used in combination with other anticonvulsants to treat seizures associated with Dravet syndrome.
Lenacapavir	A first-in-class capsid inhibitor being investigated for use in HIV-1 treatment.
Futibatinib	A kinase inhibitor used to treat intrahepatic cholangiocarcinoma in previously treated adults.
Linzagolix	A selective gonadotropin-releasing hormone (GnRH) receptor antagonist used for the symptomatic treatment of uterine fibroids.
Vonoprazan	A potassium-competitive acid blocker used in the treatment of acid-related disorders and as an adjunct to Helicobacter pylori eradication.
Mirvetuximab soravtansine	A folate receptor alpha-directed antibody and microtubule inhibitor conjugate used to treat folate receptor alpha positive, platinum-resistant epithelial ovarian, fallopian tube, or primary peritoneal cancer.
Olutasidenib	An isocitrate dehydrogenase-1 (IDH1) inhibitor indicated for the treatment of patients with relapsed or refractory acute myeloid leukemia with a susceptible IDH1 mutation as detected by an FDA-approved test.
Adagrasib	A KRAS inhibitor indicated for the treatment of locally advanced or metastatic KRAS G12C-mutated non-small cell lung cancer in patients who have received at least one prior systemic therapy.
Bexagliflozin	A sodium-glucose co-transporter 2 inhibitor used to improve glycemic control in patients with type 2 diabetes mellitus.
Elacestrant	An estrogen receptor antagonist used to treat ER-positive, HER2-negative, ESR1-mutated advanced or metastatic breast cancer with disease progression following at least one line of endocrine therapy.
Pirtobrutinib	A kinase inhibitor used to treat relapsed or refractory mantle cell lymphoma (MCL) after at least two lines of systemic therapy.
Daprodustat	A small-molecule hypoxia-inducible factor prolyl hydroxylase inhibitor used for the treatment of anemia in patients with chronic kidney disease.
Sparsentan	An endothelin and angiotensin II receptor antagonist indicated to reduce proteinuria in adults with primary immunoglobulin A nephropathy at risk of rapid disease progression.
Omaveloxolone	A semisynthetic triterpenoid used to treat Friedreich’s ataxia in adults and adolescents 16 years and older.
Zavegepant	A calcitonin gene-related peptide receptor antagonist indicated for the acute treatment of migraine with or without aura.
Trametinib	A kinase inhibitor used alone or in combination with dabrafenib to treat patients with cancers with specific BRAF mutations, such as melanoma and non-small cell lung cancer.
Leniolisib	A phosphoinositide 3-kinase-delta inhibitor that is used to treat activated phosphoinositide 3-kinase delta syndrome.
Momelotinib	A Janus Kinase inhibitor used to treat intermediate or high-risk myelofibrosis.
Quizartinib	A FLT3 inhibitor used in combination with cytarabine and anthracycline to treat acute myeloid leukemia with FLT3 internal tandem duplication
Ritlecitinib	A kinase inhibitor used to treat severe alopecia areata in adults and adolescents 12 years and older.
Zuranolone	A neuroactive steroid drug used to treat postpartum depression
Gepirone	A serotonin receptor agonist used to treat major depressive disorder in adults
Etrasimod	An S1P receptors modulator used to treat moderate to severely active ulcerative colitis in adults
Vamorolone	A synthetic glucocorticoid used as an anti-inflammatory and immunosuppressant in the management of Duchenne muscular dystrophy (DMD).
Capivasertib	A serine/threonine kinase inhibitor used to treat hormone receptor-positive, HER2-negative, locally advanced or metastatic breast cancer
Repotrectinib	A tyrosine kinase inhibitor used to treat locally active or metastatic non-small cell lung cancer
Fruquintinib	A VEGF receptor inhibitor used to treat metastatic colorectal cancer.
Nirogacestat	A gamma-secretase inhibitor used to treat desmoid tumors
Avatrombopag	A thrombopoietin receptor agonist used pre-operatively to treat thrombocytopenia in patients with chronic liver disease and in patients with chronic refractory thrombocytopenia.
Tovorafenib	A type II RAF inhibitor used to treat pediatric low-grade glioma with BRAF gene mutations.
Mavorixafor	A CXC chemokine receptor 4 antagonist used to treat WHIM syndrome.
Deuruxolitinib	A Janus Kinase inhibitor used to treat severe alopecia areata in adults.
Sofpironium	A topical anticholinergic used to treat primary axillary hyperhidrosis.
Seladelpar	A PPAR-delta agonist used to treat primary biliary cholangitis alone or in combination with ursodeoxycholic acid in adults.
Vorasidenib	A isocitrate dehydrogenase type 1 (IDH1) and 2 (IDH2) inhibitor used to treat Grade 2 astrocytoma or oligodendroglioma with a susceptible IDH1 or IDH2 mutation.
Lazertinib	A tyrosine kinase inhibitor used in combiantion with amivantamab to treat non-small cell lung cancer with EGFR mutations.

Drugs & Drug Targets

Drug	Target	Type
Indinavir	Pol polyprotein	target
Indinavir	Cytochrome P450 3A4	enzyme
Indinavir	Cytochrome P450 3A5	enzyme
Indinavir	Cytochrome P450 3A7	enzyme
Indinavir	ATP-dependent translocase ABCB1	transporter
Indinavir	Solute carrier family 22 member 1	transporter
Indinavir	Multidrug resistance-associated protein 1	transporter
Indinavir	Solute carrier organic anion transporter family member 1A2	transporter
Indinavir	Solute carrier organic anion transporter family member 1B1	transporter
Indinavir	ATP-binding cassette sub-family C member 2	transporter
Indinavir	Cytochrome P450 2D6	enzyme
Indinavir	UDP-glucuronosyltransferase 1A1	enzyme
Indinavir	Solute carrier organic anion transporter family member 2B1	transporter
Indinavir	Bile salt export pump	transporter
Indinavir	Gag-Pol polyprotein	target
Lovastatin	3-hydroxy-3-methylglutaryl-coenzyme A reductase	target
Lovastatin	Cytochrome P450 3A4	enzyme
Lovastatin	Cytochrome P450 2C8	enzyme
Lovastatin	Integrin alpha-L	target
Lovastatin	Histone deacetylase 2	target
Lovastatin	Serum paraoxonase/lactonase 3	enzyme
Lovastatin	ATP-dependent translocase ABCB1	transporter
Lovastatin	Solute carrier organic anion transporter family member 1A2	transporter
Lovastatin	Solute carrier organic anion transporter family member 1B1	transporter
Lovastatin	UDP-glucuronosyltransferase 1A1	enzyme
Lovastatin	UDP-glucuronosyltransferase 1A3	enzyme
Lovastatin	UDP-glucuronosyltransferase 2B7	enzyme
Lovastatin	ATP-binding cassette sub-family C member 2	transporter
Lovastatin	Bile salt export pump	transporter
Lovastatin	Albumin	carrier
Lovastatin	Cytochrome P450 2C19	enzyme
Lovastatin	Solute carrier organic anion transporter family member 2B1	transporter
Lovastatin	Solute carrier organic anion transporter family member 1B3	transporter
Diltiazem	Voltage-dependent calcium channel gamma-1 subunit	target
Diltiazem	Cytochrome P450 3A4	enzyme
Diltiazem	Cytochrome P450 2C19	enzyme
Diltiazem	Cytochrome P450 2D6	enzyme
Diltiazem	Cytochrome P450 3A5	enzyme
Diltiazem	Cytochrome P450 3A7	enzyme
Diltiazem	ATP-dependent translocase ABCB1	transporter
Diltiazem	Cytochrome P450 2C8	enzyme
Diltiazem	Albumin	carrier
Diltiazem	Alpha-1-acid glycoprotein 1	carrier
Diltiazem	Voltage-dependent L-type calcium channel subunit alpha-1C	target
Diltiazem	Voltage-dependent calcium channel subunit alpha-2/delta-1	target
Amlodipine	Carbonic anhydrase 1	target
Amlodipine	Cytochrome P450 3A4	enzyme
Amlodipine	Voltage-dependent L-type calcium channel subunit alpha-1C	target
Amlodipine	Cytochrome P450 1A1	enzyme
Amlodipine	Cytochrome P450 2B6	enzyme
Amlodipine	Voltage-dependent N-type calcium channel subunit alpha-1B	target
Amlodipine	Voltage-dependent L-type calcium channel subunit beta-1	target
Amlodipine	Voltage-dependent calcium channel subunit alpha-2/delta-3	target
Amlodipine	Cytochrome P450 3A5	enzyme
Amlodipine	ATP-dependent translocase ABCB1	transporter
Amlodipine	Cytochrome P450 2C8	enzyme
Amlodipine	Cytochrome P450 2D6	enzyme
Amlodipine	Sphingomyelin phosphodiesterase	target
Amlodipine	Voltage-dependent T-type calcium channel subunit alpha-1I	target
Amlodipine	Voltage-dependent N-type calcium channel	target
Amlodipine	Cytochrome P450 2C19	enzyme
Amlodipine	Cytochrome P450 2C9	enzyme
Amlodipine	Voltage-dependent calcium channel subunit alpha-2/delta-1	target
Nisoldipine	Cytochrome P450 3A4	enzyme
Nisoldipine	Voltage-dependent L-type calcium channel subunit alpha-1D	target
Nisoldipine	Voltage-dependent L-type calcium channel subunit alpha-1S	target
Nisoldipine	Voltage-dependent L-type calcium channel subunit alpha-1C	target
Nisoldipine	Voltage-dependent calcium channel subunit alpha-2/delta-1	target
Nisoldipine	Voltage-dependent L-type calcium channel subunit beta-2	target
Nisoldipine	Cytochrome P450 3A5	enzyme
Nisoldipine	Cytochrome P450 3A7	enzyme
Nisoldipine	ATP-dependent translocase ABCB1	transporter
Alprazolam	Cytochrome P450 3A4	enzyme
Alprazolam	Cytochrome P450 2C9	enzyme
Alprazolam	Cytochrome P450 3A5	enzyme
Alprazolam	Cytochrome P450 3A7	enzyme
Alprazolam	GABA(A) Receptor	target
Alprazolam	Albumin	carrier
Alprazolam	alpha1-acid glycoprotein	carrier
Alprazolam	GABA(A) Receptor Benzodiazepine Binding Site	target
Quinine	Platelet glycoprotein IX	target
Quinine	Intermediate conductance calcium-activated potassium channel protein 4	target
Quinine	Cytochrome P450 3A4	enzyme
Quinine	Cytochrome P450 3A5	enzyme
Quinine	Cytochrome P450 1A1	enzyme
Quinine	Cytochrome P450 2D6	enzyme
Quinine	Cytochrome P450 1A2	enzyme
Quinine	Cytochrome P450 2C8	enzyme
Quinine	Cytochrome P450 2C9	enzyme
Quinine	Cytochrome P450 2C19	enzyme
Quinine	Cytochrome P450 2E1	enzyme
Quinine	Cytochrome P450 3A7	enzyme
Quinine	Solute carrier family 22 member 2	transporter
Quinine	Solute carrier family 22 member 1	transporter
Quinine	Organic cation/carnitine transporter 2	transporter
Quinine	ATP-dependent translocase ABCB1	transporter
Quinine	Solute carrier organic anion transporter family member 1A2	transporter
Quinine	Solute carrier family 22 member 4	transporter
Quinine	Fe(II)-protoporphyrin IX	target
Quinine	Solute carrier organic anion transporter family member 1B1	transporter
Buspirone	5-hydroxytryptamine receptor 1A	target
Buspirone	D(2) dopamine receptor	target
Buspirone	Cytochrome P450 3A4	enzyme
Buspirone	Cytochrome P450 3A5	enzyme
Buspirone	Cytochrome P450 3A7	enzyme
Buspirone	ATP-dependent translocase ABCB1	transporter
Buspirone	Cytochrome P450 2D6	enzyme
Buspirone	Albumin	carrier
Buspirone	Alpha-1-acid glycoprotein 1	carrier
Buspirone	D(3) dopamine receptor	target
Buspirone	D(4) dopamine receptor	target
Buspirone	Alpha-1 adrenergic receptors	target
Vincristine	Tubulin beta chain	target
Vincristine	Cytochrome P450 3A4	enzyme
Vincristine	Cytochrome P450 3A5	enzyme
Vincristine	Cytochrome P450 3A7	enzyme
Vincristine	ATP-dependent translocase ABCB1	transporter
Vincristine	ATP-binding cassette sub-family C member 3	transporter
Vincristine	Solute carrier family 22 member 3	transporter
Vincristine	Multidrug resistance-associated protein 1	transporter
Vincristine	ATP-binding cassette sub-family C member 10	transporter
Vincristine	ATP-binding cassette sub-family C member 2	transporter
Vincristine	Bile salt export pump	transporter
Vincristine	Broad substrate specificity ATP-binding cassette transporter ABCG2	transporter
Vincristine	Tubulin alpha-4A chain	target
Vincristine	RalA-binding protein 1	transporter
Vincristine	Solute carrier organic anion transporter family member 1B1	transporter
Vincristine	Solute carrier organic anion transporter family member 1B3	transporter
Cisapride	5-hydroxytryptamine receptor 4	target
Cisapride	5-hydroxytryptamine receptor 3A	target
Cisapride	Potassium voltage-gated channel subfamily H member 2	target
Cisapride	5-hydroxytryptamine receptor 2A	target
Cisapride	Cytochrome P450 3A4	enzyme
Cisapride	Cytochrome P450 3A5	enzyme
Cisapride	Cytochrome P450 3A7	enzyme
Cisapride	Cytochrome P450 2A6	enzyme
Cisapride	Cytochrome P450 2B6	enzyme
Cisapride	Cytochrome P450 2C19	enzyme
Cisapride	Cytochrome P450 2C8	enzyme
Cisapride	Cytochrome P450 2C9	enzyme
Cisapride	Cytochrome P450 2D6	enzyme
Imatinib	Platelet-derived growth factor receptor beta	target
Imatinib	Tyrosine-protein kinase ABL1	target
Imatinib	Mast/stem cell growth factor receptor Kit	target
Imatinib	Proto-oncogene tyrosine-protein kinase receptor Ret	target
Imatinib	High affinity nerve growth factor receptor	target
Imatinib	Macrophage colony-stimulating factor 1 receptor	target
Imatinib	Platelet-derived growth factor receptor alpha	target
Imatinib	Epithelial discoidin domain-containing receptor 1	target
Imatinib	Cytochrome P450 3A4	enzyme
Imatinib	Breakpoint cluster region protein	target
Imatinib	Cytochrome P450 1A2	enzyme
Imatinib	Cytochrome P450 2D6	enzyme
Imatinib	Cytochrome P450 2C9	enzyme
Imatinib	Cytochrome P450 2C19	enzyme
Imatinib	Cytochrome P450 3A5	enzyme
Imatinib	Cytochrome P450 3A7	enzyme
Imatinib	Solute carrier family 22 member 1	transporter
Imatinib	ATP-dependent translocase ABCB1	transporter
Imatinib	Solute carrier family 22 member 2	transporter
Imatinib	Broad substrate specificity ATP-binding cassette transporter ABCG2	transporter
Imatinib	Phospholipid-transporting ATPase ABCA3	transporter
Imatinib	Albumin	carrier
Imatinib	Alpha-1-acid glycoprotein 1	carrier
Imatinib	Bile salt export pump	transporter
Imatinib	Cytochrome P450 2C8	enzyme
Imatinib	ATP-binding cassette sub-family C member 2	transporter
Imatinib	Multidrug resistance-associated protein 1	transporter
Imatinib	Organic cation/carnitine transporter 2	transporter
Imatinib	Solute carrier organic anion transporter family member 1B3	transporter
Imatinib	ATP-binding cassette sub-family C member 4	transporter
Imatinib	Solute carrier organic anion transporter family member 1A2	transporter
Imatinib	Discoidin domain-containing receptor 2	target
Imatinib	Induced myeloid leukemia cell differentiation protein Mcl-1	target
Astemizole	Histamine H1 receptor	target
Astemizole	Potassium voltage-gated channel subfamily H member 2	target
Astemizole	Cytochrome P450 3A4	enzyme
Astemizole	Cytochrome P450 3A5	enzyme
Astemizole	Cytochrome P450 3A7	enzyme
Astemizole	ATP-dependent translocase ABCB1	transporter
Astemizole	Cytochrome P450 2D6	enzyme
Astemizole	Cytochrome P450 2J2	enzyme
Astemizole	Potassium voltage-gated channel subfamily H member 1	target
Astemizole	Microtubule-associated protein tau	target
Astemizole	Bile salt export pump	transporter
Simvastatin	3-hydroxy-3-methylglutaryl-coenzyme A reductase	target
Simvastatin	Cytochrome P450 3A4	enzyme
Simvastatin	Cytochrome P450 2C8	enzyme
Simvastatin	Cytochrome P450 2C9	enzyme
Simvastatin	Cytochrome P450 3A5	enzyme
Simvastatin	ATP-dependent translocase ABCB1	transporter
Simvastatin	Solute carrier organic anion transporter family member 1A2	transporter
Simvastatin	Solute carrier organic anion transporter family member 1B1	transporter
Simvastatin	Cytochrome P450 2B6	enzyme
Simvastatin	Cytochrome P450 2D6	enzyme
Simvastatin	UDP-glucuronosyltransferase 1A1	enzyme
Simvastatin	UDP-glucuronosyltransferase 1A3	enzyme
Simvastatin	UDP-glucuronosyltransferase 2B7	enzyme
Simvastatin	ATP-binding cassette sub-family C member 2	transporter
Simvastatin	Integrin alpha-L	target
Simvastatin	Bile salt export pump	transporter
Simvastatin	Cytochrome P450 2C19	enzyme
Simvastatin	Solute carrier organic anion transporter family member 2B1	transporter
Simvastatin	Solute carrier organic anion transporter family member 1B3	transporter
Simvastatin	Histone deacetylase 2	target
Simvastatin	Cocaine esterase	enzyme
Simvastatin	Liver carboxylesterase 1	enzyme
Tamoxifen	Estrogen receptor	target
Tamoxifen	Estrogen receptor beta	target
Tamoxifen	Cytochrome P450 2C9	enzyme
Tamoxifen	Cytochrome P450 3A4	enzyme
Tamoxifen	Cytochrome P450 2D6	enzyme
Tamoxifen	Cytochrome P450 2C8	enzyme
Tamoxifen	Cytochrome P450 2B6	enzyme
Tamoxifen	Liver carboxylesterase 1	enzyme
Tamoxifen	Cytochrome P450 3A5	enzyme
Tamoxifen	Cytochrome P450 1A1	enzyme
Tamoxifen	Cytochrome P450 1B1	enzyme
Tamoxifen	Cytochrome P450 2C19	enzyme
Tamoxifen	Flavin-containing monooxygenase 1	enzyme
Tamoxifen	Flavin-containing monooxygenase 3	enzyme
Tamoxifen	Cytochrome P450 3A7	enzyme
Tamoxifen	ATP-dependent translocase ABCB1	transporter
Tamoxifen	Broad substrate specificity ATP-binding cassette transporter ABCG2	transporter
Tamoxifen	Aromatase	enzyme
Tamoxifen	Cytochrome P450 2A6	enzyme
Tamoxifen	Cytochrome P450 2E1	enzyme
Tamoxifen	UDP-glucuronosyltransferase 1A10	enzyme
Tamoxifen	Sulfotransferase 1A1	enzyme
Tamoxifen	ATP-binding cassette sub-family C member 2	transporter
Tamoxifen	3-beta-hydroxysteroid-Delta(8),Delta(7)-isomerase	target
Tamoxifen	Protein kinase C	target
Tamoxifen	Androgen receptor	target
Tamoxifen	Potassium voltage-gated channel subfamily H member 2	target
Tamoxifen	Nuclear receptor subfamily 1 group I member 2	target
Tamoxifen	Estrogen-related receptor gamma	target
Tamoxifen	Sex hormone-binding globulin	target
Tamoxifen	Bile salt export pump	transporter
Tamoxifen	Thyroxine-binding globulin	carrier
Tamoxifen	Sulfotransferase 2A1	enzyme
Tamoxifen	Cytochrome P450 1A2	enzyme
Tamoxifen	UDP-glucuronosyltransferase 2B7	enzyme
Tamoxifen	UDP-glucuronosyltransferase 2B17	enzyme
Tamoxifen	Sulfotransferase 1E1	enzyme
Tamoxifen	Phospholipid-transporting ATPase ABCA1	transporter
Tamoxifen	Mitogen-activated protein kinase 8	target
Tamoxifen	Albumin	carrier
Midazolam	Cytochrome P450 3A4	enzyme
Midazolam	Cytochrome P450 3A5	enzyme
Midazolam	UDP-glucuronosyltransferase 1A4	enzyme
Midazolam	Cytochrome P450 3A7	enzyme
Midazolam	GABA(A) Receptor	target
Midazolam	GABA(A) Receptor Benzodiazepine Binding Site	target
Midazolam	ATP-dependent translocase ABCB1	transporter
Midazolam	Albumin	carrier
Midazolam	Alpha-1-acid glycoprotein 1	carrier
Midazolam	Adenosine receptor A2a	target
Midazolam	Excitatory amino acid transporter 2	transporter
Midazolam	UDP-glucuronosyltransferase 2B7	enzyme
Midazolam	UDP-glucuronosyltransferase 2B4	enzyme
Alfentanil	Mu-type opioid receptor	target
Alfentanil	Cytochrome P450 3A4	enzyme
Alfentanil	Cytochrome P450 3A5	enzyme
Alfentanil	Alpha-1-acid glycoprotein 1	carrier
Alfentanil	Albumin	carrier
Alfentanil	Cytochrome P450 3A7	enzyme
Alfentanil	ATP-dependent translocase ABCB1	transporter
Tadalafil	cGMP-specific 3',5'-cyclic phosphodiesterase	target
Tadalafil	Cytochrome P450 3A4	enzyme
Tadalafil	Dual 3',5'-cyclic-AMP and -GMP phosphodiesterase 11A	target
Tadalafil	Retinal rod rhodopsin-sensitive cGMP 3',5'-cyclic phosphodiesterase subunit gamma	target
Diazepam	Cytochrome P450 3A4	enzyme
Diazepam	Albumin	carrier
Diazepam	Cytochrome P450 2C9	enzyme
Diazepam	Cytochrome P450 2C19	enzyme
Diazepam	Cytochrome P450 3A5	enzyme
Diazepam	Cytochrome P450 3A7	enzyme
Diazepam	ATP-dependent translocase ABCB1	transporter
Diazepam	Cytochrome P450 2B6	enzyme
Diazepam	Prostaglandin G/H synthase 1	enzyme
Diazepam	Cytochrome P450 2C18	enzyme
Diazepam	Cytochrome P450 2C8	enzyme
Diazepam	GABA(A) Receptor	target
Diazepam	GABA(A) Receptor Benzodiazepine Binding Site	target
Vardenafil	cGMP-specific 3',5'-cyclic phosphodiesterase	target
Vardenafil	Cytochrome P450 3A4	enzyme
Vardenafil	Retinal rod rhodopsin-sensitive cGMP 3',5'-cyclic phosphodiesterase subunit gamma	target
Vardenafil	Retinal cone rhodopsin-sensitive cGMP 3',5'-cyclic phosphodiesterase subunit gamma	target
Vardenafil	Cytochrome P450 3A5	enzyme
Vardenafil	ATP-dependent translocase ABCB1	transporter
Vardenafil	Cytochrome P450 2C9	enzyme
Vardenafil	Cytochrome P450 2C8	enzyme
Vardenafil	Cytochrome P450 2C19	enzyme
Vardenafil	Cytochrome P450 2D6	enzyme
Tacrolimus	Peptidyl-prolyl cis-trans isomerase FKBP1A	target
Tacrolimus	Cytochrome P450 3A4	enzyme
Tacrolimus	Cytochrome P450 3A5	enzyme
Tacrolimus	ATP-dependent translocase ABCB1	transporter
Tacrolimus	Cholesterol transporter ABCA5	transporter
Tacrolimus	Albumin	carrier
Tacrolimus	Alpha-1-acid glycoprotein 1	carrier
Tacrolimus	Solute carrier organic anion transporter family member 1B1	transporter
Tacrolimus	Protein phosphatase 3 catalytic subunit alpha	target
Sirolimus	Cytochrome P450 3A4	enzyme
Sirolimus	Serine/threonine-protein kinase mTOR	target
Sirolimus	Cytochrome P450 3A5	enzyme
Sirolimus	Cytochrome P450 3A7	enzyme
Sirolimus	ATP-dependent translocase ABCB1	transporter
Sirolimus	Solute carrier organic anion transporter family member 1B1	transporter
Sirolimus	Multidrug and toxin extrusion protein 1	transporter
Sirolimus	Albumin	carrier
Sirolimus	Alpha-1-acid glycoprotein 1	carrier
Sirolimus	Apolipoproteins	carrier
Triazolam	Cytochrome P450 3A4	enzyme
Triazolam	Cytochrome P450 3A5	enzyme
Triazolam	Cytochrome P450 3A7	enzyme
Triazolam	Cytochrome P450 2C8	enzyme
Triazolam	GABA(A) Receptor Benzodiazepine Binding Site	target
Triazolam	GABA(A) Receptor	target
Telithromycin	23S ribosomal RNA	target
Telithromycin	Cytochrome P450 3A4	enzyme
Telithromycin	Solute carrier organic anion transporter family member 1B1	transporter
Telithromycin	Solute carrier organic anion transporter family member 1B3	transporter
Felodipine	Voltage-dependent calcium channel subunit alpha-2/delta-1	target
Felodipine	Cytochrome P450 3A4	enzyme
Felodipine	Voltage-dependent L-type calcium channel subunit alpha-1C	target
Felodipine	Voltage-dependent L-type calcium channel subunit beta-2	target
Felodipine	Cytochrome P450 2C8	enzyme
Felodipine	Dual specificity calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1B	target
Felodipine	Dual specificity calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1A	target
Felodipine	Voltage-dependent T-type calcium channel subunit alpha-1H	target
Felodipine	Voltage-dependent calcium channel subunit alpha-2/delta-2	target
Felodipine	Troponin C, skeletal muscle	target
Felodipine	Troponin C, slow skeletal and cardiac muscles	target
Felodipine	Mineralocorticoid receptor	target
Felodipine	Voltage-dependent L-type calcium channel subunit alpha-1D	target
Felodipine	Voltage-dependent L-type calcium channel subunit alpha-1S	target
Felodipine	Cytochrome P450 3A5	enzyme
Felodipine	Cytochrome P450 3A7	enzyme
Felodipine	ATP-dependent translocase ABCB1	transporter
Felodipine	Cytochrome P450 2C9	enzyme
Felodipine	Cytochrome P450 2D6	enzyme
Felodipine	Bile salt export pump	transporter
Felodipine	Calmodulin	target
Nitrendipine	Cytochrome P450 3A4	enzyme
Nitrendipine	Voltage-dependent T-type calcium channel subunit alpha-1H	target
Nitrendipine	Voltage-dependent calcium channel subunit alpha-2/delta-2	target
Nitrendipine	Voltage-dependent L-type calcium channel subunit alpha-1D	target
Nitrendipine	Voltage-dependent L-type calcium channel subunit alpha-1S	target
Nitrendipine	Voltage-dependent L-type calcium channel subunit alpha-1C	target
Nitrendipine	Voltage-dependent calcium channel subunit alpha-2/delta-1	target
Nitrendipine	Voltage-dependent L-type calcium channel subunit beta-2	target
Nitrendipine	Cytochrome P450 3A5	enzyme
Nitrendipine	Cytochrome P450 3A7	enzyme
Nitrendipine	ATP-dependent translocase ABCB1	transporter
Nitrendipine	Bile salt export pump	transporter
Nitrendipine	Voltage-dependent L-type calcium channel	target
Nitrendipine	Calcium-activated potassium channel	target
Atorvastatin	3-hydroxy-3-methylglutaryl-coenzyme A reductase	target
Atorvastatin	Cytochrome P450 3A4	enzyme
Atorvastatin	Dipeptidyl peptidase 4	target
Atorvastatin	Cytochrome P450 2D6	enzyme
Atorvastatin	Cytochrome P450 2C9	enzyme
Atorvastatin	Cytochrome P450 2C19	enzyme
Atorvastatin	Cytochrome P450 3A5	enzyme
Atorvastatin	Cytochrome P450 3A7	enzyme
Atorvastatin	ATP-dependent translocase ABCB1	transporter
Atorvastatin	Solute carrier organic anion transporter family member 1A2	transporter
Atorvastatin	Solute carrier organic anion transporter family member 1B1	transporter
Atorvastatin	ATP-binding cassette sub-family C member 4	transporter
Atorvastatin	ATP-binding cassette sub-family C member 5	transporter
Atorvastatin	Multidrug resistance-associated protein 1	transporter
Atorvastatin	Cytochrome P450 2B6	enzyme
Atorvastatin	Cytochrome P450 2C8	enzyme
Atorvastatin	Aryl hydrocarbon receptor	target
Atorvastatin	Solute carrier organic anion transporter family member 2B1	transporter
Atorvastatin	Solute carrier organic anion transporter family member 1B3	transporter
Atorvastatin	UDP-glucuronosyltransferase 1A1	enzyme
Atorvastatin	UDP-glucuronosyltransferase 1A3	enzyme
Atorvastatin	ATP-binding cassette sub-family C member 2	transporter
Atorvastatin	Bile salt export pump	transporter
Atorvastatin	Albumin	carrier
Atorvastatin	Histone deacetylase 2	target
Atorvastatin	Nuclear receptor subfamily 1 group I member 3	target
Pimozide	D(2) dopamine receptor	target
Pimozide	Potassium voltage-gated channel subfamily H member 2	target
Pimozide	Cytochrome P450 3A4	enzyme
Pimozide	Cytochrome P450 1A2	enzyme
Pimozide	Cytochrome P450 3A5	enzyme
Pimozide	Cytochrome P450 3A7	enzyme
Pimozide	ATP-dependent translocase ABCB1	transporter
Pimozide	D(3) dopamine receptor	target
Pimozide	Cytochrome P450 2D6	enzyme
Pimozide	Calmodulin	target
Chlorpheniramine	Histamine H1 receptor	target
Chlorpheniramine	Cytochrome P450 3A4	enzyme
Chlorpheniramine	Cytochrome P450 2D6	enzyme
Chlorpheniramine	Sodium-dependent serotonin transporter	target
Chlorpheniramine	Sodium-dependent noradrenaline transporter	target
Chlorpheniramine	Sodium-dependent dopamine transporter	target
Chlorpheniramine	Cytochrome P450 3A5	enzyme
Chlorpheniramine	Cytochrome P450 3A7	enzyme
Chlorpheniramine	Solute carrier family 22 member 2	transporter
Chlorpheniramine	Solute carrier family 22 member 1	transporter
Nifedipine	Cytochrome P450 3A4	enzyme
Nifedipine	Cytochrome P450 2E1	enzyme
Nifedipine	Cytochrome P450 2D6	enzyme
Nifedipine	Voltage-dependent L-type calcium channel subunit alpha-1D	target
Nifedipine	Voltage-dependent L-type calcium channel subunit alpha-1S	target
Nifedipine	Voltage-dependent L-type calcium channel subunit alpha-1C	target
Nifedipine	Voltage-dependent L-type calcium channel subunit beta-2	target
Nifedipine	A-type voltage-gated potassium channel KCND3	target
Nifedipine	Voltage-dependent T-type calcium channel	target
Nifedipine	Cytochrome P450 1A2	enzyme
Nifedipine	Cytochrome P450 2A6	enzyme
Nifedipine	Cytochrome P450 2C8	enzyme
Nifedipine	ATP-binding cassette sub-family C member 3	transporter
Nifedipine	ATP-dependent translocase ABCB1	transporter
Nifedipine	ATP-binding cassette sub-family C member 2	transporter
Nifedipine	Cytochrome P450 1A1	enzyme
Nifedipine	Cytochrome P450 2B6	enzyme
Nifedipine	Nuclear receptor subfamily 1 group I member 2	target
Nifedipine	Solute carrier organic anion transporter family member 1B1	transporter
Nifedipine	Bile salt export pump	transporter
Nifedipine	Cytochrome P450 2C9	enzyme
Nifedipine	Albumin	carrier
Nifedipine	alpha1-acid glycoprotein	carrier
Nifedipine	Cytochrome P450 3A5	enzyme
Nifedipine	Calmodulin	target
Clarithromycin	50S ribosomal protein L10	target
Clarithromycin	Cytochrome P450 3A4	enzyme
Clarithromycin	Cytochrome P450 3A5	enzyme
Clarithromycin	ATP-dependent translocase ABCB1	transporter
Clarithromycin	Solute carrier family 22 member 7	transporter
Clarithromycin	Potassium voltage-gated channel subfamily H member 2	target
Clarithromycin	Solute carrier organic anion transporter family member 1B1	target
Clarithromycin	Solute carrier organic anion transporter family member 1B3	target
Clarithromycin	Bile salt export pump	transporter
Clarithromycin	Solute carrier organic anion transporter family member 1B1	transporter
Clarithromycin	Solute carrier organic anion transporter family member 1B3	transporter
Saquinavir	Pol polyprotein	target
Saquinavir	Cytochrome P450 3A4	enzyme
Saquinavir	Cytochrome P450 3A5	enzyme
Saquinavir	Alpha-1-acid glycoprotein 1	carrier
Saquinavir	Albumin	carrier
Saquinavir	Cytochrome P450 3A7	enzyme
Saquinavir	ATP-dependent translocase ABCB1	transporter
Saquinavir	Solute carrier family 22 member 1	transporter
Saquinavir	Solute carrier organic anion transporter family member 1A2	transporter
Saquinavir	Broad substrate specificity ATP-binding cassette transporter ABCG2	transporter
Saquinavir	Solute carrier organic anion transporter family member 1B1	transporter
Saquinavir	Multidrug resistance-associated protein 1	transporter
Saquinavir	ATP-binding cassette sub-family C member 2	transporter
Saquinavir	Cytochrome P450 2C8	enzyme
Saquinavir	Cytochrome P450 2D6	enzyme
Saquinavir	Solute carrier organic anion transporter family member 2B1	transporter
Saquinavir	Bile salt export pump	transporter
Saquinavir	Gag-Pol polyprotein	target
Aripiprazole	D(2) dopamine receptor	target
Aripiprazole	5-hydroxytryptamine receptor 1A	target
Aripiprazole	5-hydroxytryptamine receptor 2A	target
Aripiprazole	Cytochrome P450 3A4	enzyme
Aripiprazole	Cytochrome P450 2D6	enzyme
Aripiprazole	5-hydroxytryptamine receptor 1B	target
Aripiprazole	5-hydroxytryptamine receptor 1D	target
Aripiprazole	5-hydroxytryptamine receptor 1E	target
Aripiprazole	D(1A) dopamine receptor	target
Aripiprazole	D(1B) dopamine receptor	target
Aripiprazole	D(3) dopamine receptor	target
Aripiprazole	D(4) dopamine receptor	target
Aripiprazole	5-hydroxytryptamine receptor 2C	target
Aripiprazole	5-hydroxytryptamine receptor 3A	target
Aripiprazole	5-hydroxytryptamine receptor 6	target
Aripiprazole	5-hydroxytryptamine receptor 7	target
Aripiprazole	Histamine H1 receptor	target
Aripiprazole	Alpha-1A adrenergic receptor	target
Aripiprazole	Alpha-1B adrenergic receptor	target
Aripiprazole	Alpha-2A adrenergic receptor	target
Aripiprazole	Alpha-2B adrenergic receptor	target
Aripiprazole	Alpha-2C adrenergic receptor	target
Aripiprazole	Cytochrome P450 3A5	enzyme
Aripiprazole	Cytochrome P450 3A7	enzyme
Aripiprazole	Albumin	carrier
Aripiprazole	5-hydroxytryptamine receptor 2B	target
Aripiprazole	5-hydroxytryptamine receptor 5A	target
Aripiprazole	Beta-1 adrenergic receptor	target
Aripiprazole	Beta-2 adrenergic receptor	target
Aripiprazole	Histamine H2 receptor	target
Aripiprazole	Histamine H3 receptor	target
Aripiprazole	Histamine H4 receptor	target
Aripiprazole	Muscarinic acetylcholine receptor M1	target
Aripiprazole	Muscarinic acetylcholine receptor M2	target
Aripiprazole	Muscarinic acetylcholine receptor M3	target
Aripiprazole	Muscarinic acetylcholine receptor M4	target
Aripiprazole	Muscarinic acetylcholine receptor M5	target
Aripiprazole	Kappa-type opioid receptor	target
Aripiprazole	Mu-type opioid receptor	target
Aripiprazole	Delta-type opioid receptor	target
Aripiprazole	Glutamate (NMDA) receptor	target
Aripiprazole	Sodium-dependent dopamine transporter	target
Aripiprazole	Sodium-dependent serotonin transporter	target
Aripiprazole	ATP-dependent translocase ABCB1	transporter
Aripiprazole	Broad substrate specificity ATP-binding cassette transporter ABCG2	transporter
Erythromycin	23S ribosomal RNA	target
Erythromycin	Cytochrome P450 3A4	enzyme
Erythromycin	Cytochrome P450 3A7	enzyme
Erythromycin	ATP-dependent translocase ABCB1	transporter
Erythromycin	Solute carrier organic anion transporter family member 1B1	transporter
Erythromycin	Motilin receptor	target
Erythromycin	Potassium voltage-gated channel subfamily H member 2	target
Erythromycin	Cytochrome P450 3A5	enzyme
Erythromycin	Solute carrier organic anion transporter family member 1B3	transporter
Erythromycin	Bile salt export pump	transporter
Erythromycin	ATP-binding cassette sub-family C member 2	transporter
Erythromycin	Solute carrier organic anion transporter family member 1A2	transporter
Carbamazepine	Voltage-gated sodium channel alpha subunit	target
Carbamazepine	Cytochrome P450 2C8	enzyme
Carbamazepine	Cytochrome P450 2B6	enzyme
Carbamazepine	Cytochrome P450 3A4	enzyme
Carbamazepine	Cytochrome P450 1A2	enzyme
Carbamazepine	Cytochrome P450 2C19	enzyme
Carbamazepine	Cytochrome P450 2C9	enzyme
Carbamazepine	ATP-dependent translocase ABCB1	transporter
Carbamazepine	Cytochrome P450 3A5	enzyme
Carbamazepine	UDP-glucuronosyltransferase 2B7	enzyme
Carbamazepine	RalA-binding protein 1	transporter
Carbamazepine	ATP-binding cassette sub-family C member 2	transporter
Carbamazepine	Neuronal acetylcholine receptor subunit alpha-4	target
Carbamazepine	Nuclear receptor subfamily 1 group I member 2	target
Carbamazepine	UDP-glucuronosyltransferase 1A1	enzyme
Carbamazepine	UDP-glucuronosyltransferase 1-6	enzyme
Carbamazepine	UDP-glucuronosyltransferase 1A7	enzyme
Sildenafil	cGMP-specific 3',5'-cyclic phosphodiesterase	target
Sildenafil	Cytochrome P450 2C9	enzyme
Sildenafil	Retinal rod rhodopsin-sensitive cGMP 3',5'-cyclic phosphodiesterase subunit gamma	target
Sildenafil	Retinal cone rhodopsin-sensitive cGMP 3',5'-cyclic phosphodiesterase subunit gamma	target
Sildenafil	Cytochrome P450 3A4	enzyme
Sildenafil	Cytochrome P450 3A5	enzyme
Sildenafil	Cytochrome P450 3A7	enzyme
Sildenafil	ATP-binding cassette sub-family C member 4	transporter
Sildenafil	ATP-binding cassette sub-family C member 5	transporter
Sildenafil	ATP-binding cassette sub-family C member 10	transporter
Sildenafil	Cytochrome P450 2C19	enzyme
Sildenafil	Cytochrome P450 2D6	enzyme
Sildenafil	Cytochrome P450 2E1	enzyme
Sildenafil	Solute carrier organic anion transporter family member 1B1	transporter
Sildenafil	ATP-dependent translocase ABCB1	transporter
Sildenafil	Ornithine decarboxylase	target
Sildenafil	Programmed cell death 1 ligand 1	target
Sildenafil	Plasma protease C1 inhibitor	target
Quinidine	Sodium channel protein type 5 subunit alpha	target
Quinidine	Alpha-1-acid glycoprotein 1	carrier
Quinidine	Potassium voltage-gated channel subfamily H member 2	target
Quinidine	Potassium channel subfamily K member 1	target
Quinidine	Potassium channel subfamily K member 6	target
Quinidine	Cytochrome P450 1A2	enzyme
Quinidine	Cytochrome P450 2E1	enzyme
Quinidine	Cytochrome P450 1A1	enzyme
Quinidine	Cytochrome P450 2D6	enzyme
Quinidine	Cytochrome P450 3A4	enzyme
Quinidine	Cytochrome P450 3A7	enzyme
Quinidine	Solute carrier family 22 member 2	transporter
Quinidine	Solute carrier family 22 member 1	transporter
Quinidine	Organic cation/carnitine transporter 2	transporter
Quinidine	ATP-dependent translocase ABCB1	transporter
Quinidine	Solute carrier organic anion transporter family member 1A2	transporter
Quinidine	Organic anion transporter 3	transporter
Quinidine	ATP-binding cassette sub-family C member 2	transporter
Quinidine	Solute carrier family 22 member 4	transporter
Quinidine	Solute carrier organic anion transporter family member 1B1	transporter
Quinidine	Cytochrome P450 2B6	enzyme
Quinidine	Cytochrome P450 2C9	enzyme
Quinidine	Alpha-1A adrenergic receptor	target
Quinidine	Alpha-1B adrenergic receptor	target
Quinidine	Alpha-1D adrenergic receptor	target
Quinidine	Bile salt export pump	transporter
Quinidine	Cytochrome P450 2C8	enzyme
Quinidine	Albumin	carrier
Trazodone	5-hydroxytryptamine receptor 2A	target
Trazodone	Sodium-dependent serotonin transporter	target
Trazodone	Alpha-1A adrenergic receptor	target
Trazodone	Alpha-2A adrenergic receptor	target
Trazodone	Histamine H1 receptor	target
Trazodone	5-hydroxytryptamine receptor 1A	target
Trazodone	Cytochrome P450 2D6	enzyme
Trazodone	Cytochrome P450 3A4	enzyme
Trazodone	5-hydroxytryptamine receptor 2C	target
Trazodone	Cytochrome P450 3A5	enzyme
Trazodone	Cytochrome P450 3A7	enzyme
Trazodone	ATP-dependent translocase ABCB1	transporter
Trazodone	5-hydroxytryptamine receptor 2C	target
Cyclosporine	Guided entry of tail-anchored proteins factor CAMLG	target
Cyclosporine	Peptidyl-prolyl cis-trans isomerase A	target
Cyclosporine	Calcineurin subunit B type 2	target
Cyclosporine	Cytochrome P450 3A5	enzyme
Cyclosporine	Cytochrome P450 3A4	enzyme
Cyclosporine	ATP-dependent translocase ABCB1	transporter
Cyclosporine	Bile salt export pump	transporter
Cyclosporine	Ileal sodium/bile acid cotransporter	transporter
Cyclosporine	Hepatic sodium/bile acid cotransporter	transporter
Cyclosporine	Solute carrier family 22 member 6	transporter
Cyclosporine	ATP-binding cassette sub-family C member 10	transporter
Cyclosporine	ATP-binding cassette sub-family C member 2	transporter
Cyclosporine	Broad substrate specificity ATP-binding cassette transporter ABCG2	transporter
Cyclosporine	Solute carrier organic anion transporter family member 1B1	transporter
Cyclosporine	Cytochrome P450 2C19	enzyme
Cyclosporine	Cytochrome P450 2D6	enzyme
Cyclosporine	Peptidyl-prolyl cis-trans isomerase F, mitochondrial	target
Cyclosporine	Solute carrier organic anion transporter family member 1B3	transporter
Cyclosporine	Protein phosphatase 3 catalytic subunit alpha	target
Verapamil	ATP-sensitive inward rectifier potassium channel 11	target
Verapamil	Voltage-dependent T-type calcium channel subunit alpha-1G	target
Verapamil	Potassium voltage-gated channel subfamily H member 2	target
Verapamil	Voltage-dependent L-type calcium channel subunit alpha-1C	target
Verapamil	Cytochrome P450 1A2	enzyme
Verapamil	Cytochrome P450 3A5	enzyme
Verapamil	Voltage-dependent N-type calcium channel subunit alpha-1B	target
Verapamil	Voltage-dependent P/Q-type calcium channel subunit alpha-1A	target
Verapamil	Sodium-dependent serotonin transporter	target
Verapamil	Cytochrome P450 3A4	enzyme
Verapamil	ATP-dependent translocase ABCB1	transporter
Verapamil	Solute carrier family 22 member 1	transporter
Verapamil	ATP-binding cassette sub-family C member 3	transporter
Verapamil	ATP-binding cassette sub-family C member 4	transporter
Verapamil	Organic cation/carnitine transporter 2	transporter
Verapamil	Solute carrier organic anion transporter family member 1A2	transporter
Verapamil	ATP-binding cassette sub-family C member 10	transporter
Verapamil	Solute carrier family 22 member 4	transporter
Verapamil	Solute carrier organic anion transporter family member 1B1	transporter
Verapamil	Cytochrome P450 2C8	enzyme
Verapamil	Cytochrome P450 2C9	enzyme
Verapamil	Cytochrome P450 2B6	enzyme
Verapamil	Cytochrome P450 2C19	enzyme
Verapamil	Cytochrome P450 2D6	enzyme
Verapamil	Alpha-1A adrenergic receptor	target
Verapamil	Alpha-1B adrenergic receptor	target
Verapamil	Alpha-1D adrenergic receptor	target
Verapamil	Albumin	carrier
Verapamil	Alpha-1-acid glycoprotein 1	carrier
Verapamil	Cytochrome P450 2C18	enzyme
Verapamil	Cytochrome P450 2E1	enzyme
Verapamil	Multidrug resistance-associated protein 1	transporter
Verapamil	Multidrug and toxin extrusion protein 1	transporter
Verapamil	Multidrug and toxin extrusion protein 2	transporter
Verapamil	Voltage-dependent T-type calcium channel subunit alpha-1H	target
Verapamil	Voltage-dependent calcium channel	target
Verapamil	ATP-dependent translocase ABCB1	target
Haloperidol	D(2) dopamine receptor	target
Haloperidol	Glutamate receptor ionotropic, NMDA 2B	target
Haloperidol	D(1A) dopamine receptor	target
Haloperidol	Cytochrome P450 1A2	enzyme
Haloperidol	Cytochrome P450 2D6	enzyme
Haloperidol	5-hydroxytryptamine receptor 2A	target
Haloperidol	D(3) dopamine receptor	target
Haloperidol	Cytochrome P450 3A4	enzyme
Haloperidol	Cytochrome P450 3A5	enzyme
Haloperidol	Cytochrome P450 3A7	enzyme
Haloperidol	ATP-dependent translocase ABCB1	transporter
Haloperidol	Carbonyl reductase [NADPH] 1	enzyme
Haloperidol	UDP-glucuronosyltransferase 1A9	enzyme
Haloperidol	Cytochrome P450 2C19	enzyme
Haloperidol	Cytochrome P450 2C9	enzyme
Haloperidol	Melanin-concentrating hormone receptor 1	target
Haloperidol	Synaptic vesicular amine transporter	target
Haloperidol	5-hydroxytryptamine receptor 2C	target
Haloperidol	Sigma non-opioid intracellular receptor 1	target
Haloperidol	Histamine H1 receptor	target
Haloperidol	Muscarinic acetylcholine receptor M3	target
Haloperidol	Alpha-1A adrenergic receptor	target
Haloperidol	Alpha-2A adrenergic receptor	target
Haloperidol	Alpha-2B adrenergic receptor	target
Haloperidol	Alpha-2C adrenergic receptor	target
Haloperidol	5-hydroxytryptamine receptor 1A	target
Haloperidol	5-hydroxytryptamine receptor 6	target
Haloperidol	5-hydroxytryptamine receptor 7	target
Haloperidol	Cytochrome P450 1A1	enzyme
Azithromycin	23S ribosomal RNA	target
Azithromycin	ATP-dependent translocase ABCB1	transporter
Azithromycin	Cytochrome P450 3A4	enzyme
Azithromycin	Protein-arginine deiminase type-4	target
Azithromycin	ATP-binding cassette sub-family C member 2	transporter
Rosuvastatin	3-hydroxy-3-methylglutaryl-coenzyme A reductase	target
Rosuvastatin	Cytochrome P450 2C9	enzyme
Rosuvastatin	ATP-binding cassette sub-family C member 4	transporter
Rosuvastatin	Solute carrier organic anion transporter family member 1A2	transporter
Rosuvastatin	Solute carrier organic anion transporter family member 1B3	transporter
Rosuvastatin	Solute carrier organic anion transporter family member 2B1	transporter
Rosuvastatin	Cystine/glutamate transporter	transporter
Rosuvastatin	Solute carrier organic anion transporter family member 1B1	transporter
Rosuvastatin	Bile salt export pump	transporter
Rosuvastatin	Broad substrate specificity ATP-binding cassette transporter ABCG2	transporter
Rosuvastatin	Albumin	carrier
Rosuvastatin	ATP-binding cassette sub-family C member 2	transporter
Rosuvastatin	Organic anion transporter 3	transporter
Rosuvastatin	Hepatic sodium/bile acid cotransporter	transporter
Rosuvastatin	Integrin alpha-L	target
Telaprevir	Cytochrome P450 3A4	enzyme
Telaprevir	Genome polyprotein	target
Telaprevir	ATP-dependent translocase ABCB1	transporter
Telaprevir	Albumin	carrier
Telaprevir	Alpha-1-acid glycoprotein 1	carrier
Telaprevir	Solute carrier organic anion transporter family member 1B1	target
Telaprevir	Solute carrier organic anion transporter family member 2B1	target
Telaprevir	Genome polyprotein	target
Boceprevir	Cytochrome P450 3A4	enzyme
Boceprevir	Cytochrome P450 3A5	enzyme
Boceprevir	ATP-dependent translocase ABCB1	transporter
Boceprevir	Genome polyprotein	target
Boceprevir	Genome polyprotein	target
Ritonavir	Pol polyprotein	target
Ritonavir	Cytochrome P450 2D6	enzyme
Ritonavir	Cytochrome P450 2C9	enzyme
Ritonavir	Cytochrome P450 2C19	enzyme
Ritonavir	Cytochrome P450 2B6	enzyme
Ritonavir	Cytochrome P450 2C8	enzyme
Ritonavir	ATP-dependent translocase ABCB1	transporter
Ritonavir	Multidrug resistance-associated protein 1	transporter
Ritonavir	ATP-binding cassette sub-family C member 2	transporter
Ritonavir	Solute carrier organic anion transporter family member 1A2	transporter
Ritonavir	Broad substrate specificity ATP-binding cassette transporter ABCG2	transporter
Ritonavir	Solute carrier organic anion transporter family member 1B1	transporter
Ritonavir	Cytochrome P450 1A2	enzyme
Ritonavir	Nuclear receptor subfamily 1 group I member 2	target
Ritonavir	Albumin	carrier
Ritonavir	Cytochrome P450 3A4	enzyme
Ritonavir	Cytochrome P450 3A5	enzyme
Ritonavir	Cytochrome P450 3A7	enzyme
Ritonavir	UDP-glucuronosyltransferases (UGTs)	enzyme
Ritonavir	Solute carrier organic anion transporter family member 2B1	transporter
Ritonavir	Bile salt export pump	transporter
Ritonavir	Alpha-1-acid glycoprotein 1	carrier
Ritonavir	Solute carrier organic anion transporter family member 1B3	transporter
Ritonavir	Gag-Pol polyprotein	target
Amiodarone	Beta adrenergic receptor	target
Amiodarone	HERG human cardiac K+ channel	target
Amiodarone	Cytochrome P450 2C8	enzyme
Amiodarone	Cytochrome P450 2C9	enzyme
Amiodarone	Cytochrome P450 2D6	enzyme
Amiodarone	Voltage-dependent T-type calcium channel subunit alpha-1I	target
Amiodarone	Voltage gated L-type calcium channel	target
Amiodarone	Cytochrome P450 3A4	enzyme
Amiodarone	Cytochrome P450 1A2	enzyme
Amiodarone	Cytochrome P450 1A1	enzyme
Amiodarone	ATP-dependent translocase ABCB1	transporter
Amiodarone	Cytochrome P450 2C19	enzyme
Amiodarone	Cytochrome P450 2A6	enzyme
Amiodarone	Thyroid hormone receptor	target
Amiodarone	Peroxisome proliferator-activated receptor gamma	target
Amiodarone	Bile salt export pump	transporter
Amiodarone	Solute carrier family 22 member 2	transporter
Amiodarone	Cytochrome P450 2J2	enzyme
Amiodarone	Peroxisome proliferator-activated receptor alpha	target
Amiodarone	Peroxisome proliferator-activated receptor gamma coactivator 1-beta	target
Amiodarone	Albumin	carrier
Isavuconazole	Cytochrome P450 3A4	enzyme
Isavuconazole	Cytochrome P450 3A5	enzyme
Isavuconazole	Cytochrome P450 2C8	enzyme
Isavuconazole	Cytochrome P450 2C9	enzyme
Isavuconazole	Cytochrome P450 2C19	enzyme
Isavuconazole	Cytochrome P450 2D6	enzyme
Isavuconazole	Cytochrome P450 2B6	enzyme
Isavuconazole	UDP-glucuronosyltransferase 1A9	enzyme
Isavuconazole	UDP-glucuronosyltransferase 1A8	enzyme
Isavuconazole	ATP-dependent translocase ABCB1	transporter
Isavuconazole	Broad substrate specificity ATP-binding cassette transporter ABCG2	transporter
Isavuconazole	Solute carrier family 22 member 2	transporter
Isavuconazole	Lanosterol 14-alpha demethylase	target
Isavuconazole	Potassium voltage-gated channel subfamily H member 2	target
Isavuconazole	Voltage-dependent L-type calcium channel subunit alpha-1C	target
Isavuconazole	G protein-activated inward rectifier potassium channel 2	target
Isavuconazole	G protein-activated inward rectifier potassium channel 3	target
Isavuconazole	ATP-sensitive inward rectifier potassium channel 11	target
Isavuconazole	Potassium voltage-gated channel subfamily A member 5	target
Isavuconazole	A-type voltage-gated potassium channel KCND3	target
Isavuconazole	Potassium voltage-gated channel subfamily KQT member 1	target
Isavuconazole	Sodium channel protein type 5 subunit alpha	target
Atazanavir	Pol polyprotein	target
Atazanavir	Cytochrome P450 3A4	enzyme
Atazanavir	Cytochrome P450 2C9	enzyme
Atazanavir	ATP-dependent translocase ABCB1	transporter
Atazanavir	Multidrug resistance-associated protein 1	transporter
Atazanavir	Albumin	carrier
Atazanavir	UDP-glucuronosyltransferase 1A1	enzyme
Atazanavir	Solute carrier organic anion transporter family member 1B1	transporter
Atazanavir	Solute carrier organic anion transporter family member 1B3	transporter
Atazanavir	Cytochrome P450 2C8	enzyme
Atazanavir	Bile salt export pump	transporter
Atazanavir	alpha1-acid glycoprotein	carrier
Atazanavir	Cytochrome P450 1A2	enzyme
Atazanavir	Solute carrier organic anion transporter family member 2B1	transporter
Atazanavir	Cytochrome P450 3A5	enzyme
Atazanavir	Cytochrome P450 3A7	enzyme
Atazanavir	Gag-Pol polyprotein	target
Etravirine	Cytochrome P450 2C19	enzyme
Etravirine	Cytochrome P450 2C9	enzyme
Etravirine	Cytochrome P450 3A4	enzyme
Etravirine	Gag-Pol polyprotein	target
Etravirine	Gag-Pol polyprotein	target
Etravirine	ATP-dependent translocase ABCB1	transporter
Etravirine	Phosphatidylcholine translocator ABCB4	transporter
Etravirine	Reverse transcriptase/RNaseH	target
Amprenavir	Pol polyprotein	target
Amprenavir	Cytochrome P450 3A4	enzyme
Amprenavir	ATP-dependent translocase ABCB1	transporter
Amprenavir	Multidrug resistance-associated protein 1	transporter
Amprenavir	Cytochrome P450 2B6	enzyme
Amprenavir	Cytochrome P450 2C19	enzyme
Amprenavir	Cytochrome P450 2C9	enzyme
Amprenavir	Cytochrome P450 2D6	enzyme
Amprenavir	Cytochrome P450 3A5	enzyme
Amprenavir	Solute carrier organic anion transporter family member 1B1	transporter
Amprenavir	Gag-Pol polyprotein	target
Nelfinavir	HIV-1 protease	target
Nelfinavir	Cytochrome P450 2C19	enzyme
Nelfinavir	Cytochrome P450 3A4	enzyme
Nelfinavir	Cytochrome P450 2B6	enzyme
Nelfinavir	Cytochrome P450 3A5	enzyme
Nelfinavir	Cytochrome P450 3A7	enzyme
Nelfinavir	ATP-dependent translocase ABCB1	transporter
Nelfinavir	Solute carrier family 22 member 1	transporter
Nelfinavir	Solute carrier organic anion transporter family member 1A2	transporter
Nelfinavir	Broad substrate specificity ATP-binding cassette transporter ABCG2	transporter
Nelfinavir	Solute carrier organic anion transporter family member 1B1	transporter
Nelfinavir	Cytochrome P450 2D6	enzyme
Nelfinavir	Albumin	carrier
Nelfinavir	UDP-glucuronosyltransferase 1A1	enzyme
Nelfinavir	Solute carrier organic anion transporter family member 1B3	transporter
Nelfinavir	Solute carrier organic anion transporter family member 2B1	transporter
Nelfinavir	Bile salt export pump	transporter
Nelfinavir	Cytochrome P450 2C9	enzyme
Nelfinavir	Alpha-1-acid glycoprotein 1	carrier
Fosamprenavir	Pol polyprotein	target
Fosamprenavir	Cytochrome P450 3A4	enzyme
Fosamprenavir	Gag-Pol polyprotein	target
Nefazodone	5-hydroxytryptamine receptor 2A	target
Nefazodone	Sodium-dependent serotonin transporter	target
Nefazodone	Sodium-dependent noradrenaline transporter	target
Nefazodone	Alpha-1A adrenergic receptor	target
Nefazodone	Alpha-1B adrenergic receptor	target
Nefazodone	Cytochrome P450 3A4	enzyme
Nefazodone	Cytochrome P450 2D6	enzyme
Nefazodone	Sodium-dependent dopamine transporter	target
Nefazodone	Alpha-2A adrenergic receptor	target
Nefazodone	5-hydroxytryptamine receptor 1A	target
Nefazodone	CYP2B protein	enzyme
Nefazodone	ATP-dependent translocase ABCB1	transporter
Nefazodone	5-hydroxytryptamine receptor 2C	target
Nefazodone	Potassium voltage-gated channel subfamily H member 2	target
Nefazodone	Cytochrome P450 3A Subfamily	enzyme
Nefazodone	Solute carrier organic anion transporter family member 1B3	transporter
Nefazodone	Solute carrier organic anion transporter family member 2B1	transporter
Nefazodone	Bile salt export pump	transporter
Riociguat	Albumin	carrier
Riociguat	Alpha-1-acid glycoprotein 1	carrier
Riociguat	Guanylate cyclase soluble subunit alpha-2	target
Riociguat	Broad substrate specificity ATP-binding cassette transporter ABCG2	transporter
Riociguat	Cytochrome P450 1A1	enzyme
Riociguat	Cytochrome P450 3A4	enzyme
Riociguat	Cytochrome P450 2C8	enzyme
Riociguat	Cytochrome P450 2J2	enzyme
Riociguat	ATP-dependent translocase ABCB1	transporter
Simeprevir	NS3 protease	target
Simeprevir	Albumin	carrier
Simeprevir	Cytochrome P450 1A2	enzyme
Simeprevir	ATP-dependent translocase ABCB1	transporter
Simeprevir	Solute carrier organic anion transporter family member 1B1	transporter
Simeprevir	Solute carrier organic anion transporter family member 1B3	transporter
Simeprevir	Cytochrome P450 3A4	enzyme
Simeprevir	ATP-binding cassette sub-family C member 2	transporter
Simeprevir	Broad substrate specificity ATP-binding cassette transporter ABCG2	transporter
Simeprevir	Solute carrier organic anion transporter family member 2B1	transporter
Simeprevir	Hepatic sodium/bile acid cotransporter	transporter
Simeprevir	Bile salt export pump	transporter
Simeprevir	Genome polyprotein	target
Simeprevir	Genome polyprotein	target
Temsirolimus	Serine/threonine-protein kinase mTOR	target
Temsirolimus	Cytochrome P450 3A4	enzyme
Temsirolimus	Cytochrome P450 3A5	enzyme
Temsirolimus	Cytochrome P450 3A7	enzyme
Temsirolimus	Cytochrome P450 2D6	enzyme
Temsirolimus	ATP-dependent translocase ABCB1	transporter
Asunaprevir	Genome polyprotein	target
Asunaprevir	Cytochrome P450 3A4	enzyme
Asunaprevir	Cytochrome P450 3A5	enzyme
Asunaprevir	Cytochrome P450 2A6	enzyme
Asunaprevir	Cytochrome P450 2B6	enzyme
Asunaprevir	Cytochrome P450 2C9	enzyme
Asunaprevir	Cytochrome P450 2C19	enzyme
Asunaprevir	Cytochrome P450 2D6	enzyme
Asunaprevir	Solute carrier organic anion transporter family member 1B1	transporter
Asunaprevir	Solute carrier organic anion transporter family member 1B3	transporter
Asunaprevir	Solute carrier organic anion transporter family member 2B1	transporter
Asunaprevir	ATP-dependent translocase ABCB1	transporter
Asunaprevir	Gag-Pol polyprotein	target
Amitriptyline	Sodium-dependent serotonin transporter	target
Amitriptyline	Sodium-dependent noradrenaline transporter	target
Amitriptyline	Potassium voltage-gated channel subfamily KQT member 2	target
Amitriptyline	Alpha-2A adrenergic receptor	target
Amitriptyline	Cytochrome P450 1A2	enzyme
Amitriptyline	Cytochrome P450 2C19	enzyme
Amitriptyline	Cytochrome P450 2D6	enzyme
Amitriptyline	Albumin	carrier
Amitriptyline	Alpha-1-acid glycoprotein 1	carrier
Amitriptyline	Histamine H1 receptor	target
Amitriptyline	5-hydroxytryptamine receptor 2A	target
Amitriptyline	5-hydroxytryptamine receptor 1A	target
Amitriptyline	Alpha-1A adrenergic receptor	target
Amitriptyline	Cytochrome P450 3A4	enzyme
Amitriptyline	Cytochrome P450 3A5	enzyme
Amitriptyline	Potassium voltage-gated channel subfamily A member 1	target
Amitriptyline	Alpha-1D adrenergic receptor	target
Amitriptyline	Delta-type opioid receptor	target
Amitriptyline	Kappa-type opioid receptor	target
Amitriptyline	High affinity nerve growth factor receptor	target
Amitriptyline	BDNF/NT-3 growth factors receptor	target
Amitriptyline	Cytochrome P450 2C9	enzyme
Amitriptyline	Cytochrome P450 2B6	enzyme
Amitriptyline	Cytochrome P450 2C8	enzyme
Amitriptyline	Histamine H2 receptor	target
Amitriptyline	Histamine H4 receptor	target
Amitriptyline	Sigma non-opioid intracellular receptor 1	target
Amitriptyline	5-hydroxytryptamine receptor 2C	target
Amitriptyline	Alpha-1B adrenergic receptor	target
Amitriptyline	5-hydroxytryptamine receptor 7	target
Amitriptyline	5-hydroxytryptamine receptor 1D	target
Amitriptyline	Mu-type opioid receptor	target
Amitriptyline	5-hydroxytryptamine receptor 1B	target
Amitriptyline	5-hydroxytryptamine receptor 6	target
Amitriptyline	Potassium voltage-gated channel subfamily KQT member 3	target
Amitriptyline	UDP-glucuronosyltransferase 2B10	enzyme
Amitriptyline	5-hydroxytryptamine receptor 2C	target
Amitriptyline	Muscarinic acetylcholine receptor	target
Amitriptyline	HERG human cardiac K+ channel	target
Amitriptyline	ATP-dependent translocase ABCB1	transporter
Amitriptyline	UDP-glucuronosyltransferase 1A4	enzyme
Amitriptyline	Glutathione S-transferases (Cytosolic)	enzyme
Clomipramine	Sodium-dependent serotonin transporter	target
Clomipramine	Sodium-dependent noradrenaline transporter	target
Clomipramine	Glutathione S-transferase P	target
Clomipramine	5-hydroxytryptamine receptor 2A	target
Clomipramine	Cytochrome P450 1A2	enzyme
Clomipramine	Cytochrome P450 2D6	enzyme
Clomipramine	Cytochrome P450 2C19	enzyme
Clomipramine	ATP-dependent translocase ABCB1	transporter
Clomipramine	Cytochrome P450 3A4	enzyme
Clomipramine	5-hydroxytryptamine receptor 2B	target
Clomipramine	5-hydroxytryptamine receptor 2C	target
Clomipramine	Albumin	carrier
Cyclobenzaprine	5-hydroxytryptamine receptor 2A	target
Cyclobenzaprine	Cytochrome P450 1A2	enzyme
Cyclobenzaprine	Cytochrome P450 3A4	enzyme
Cyclobenzaprine	Cytochrome P450 2D6	enzyme
Cyclobenzaprine	Albumin	carrier
Cyclobenzaprine	UDP-glucuronosyltransferase 1A4	enzyme
Cyclobenzaprine	UDP-glucuronosyltransferase 2B10	enzyme
Cyclobenzaprine	5-hydroxytryptamine receptor 2B	target
Cyclobenzaprine	5-hydroxytryptamine receptor 2C	target
Cyclobenzaprine	5-hydroxytryptamine receptor 7	target
Cyclobenzaprine	5-hydroxytryptamine receptor 6	target
Cyclobenzaprine	Sodium-dependent serotonin transporter	target
Cyclobenzaprine	Sodium-dependent noradrenaline transporter	target
Cyclobenzaprine	Toll-like receptor 4	target
Cyclobenzaprine	Aldehyde oxidase	target
Cyclobenzaprine	Alpha-2C adrenergic receptor	target
Doxepin	Sodium-dependent serotonin transporter	target
Doxepin	Sodium-dependent noradrenaline transporter	target
Doxepin	Histamine H1 receptor	target
Doxepin	Histamine H2 receptor	target
Doxepin	Cytochrome P450 2D6	enzyme
Doxepin	Muscarinic acetylcholine receptor M1	target
Doxepin	Muscarinic acetylcholine receptor M2	target
Doxepin	Muscarinic acetylcholine receptor M3	target
Doxepin	Muscarinic acetylcholine receptor M4	target
Doxepin	Muscarinic acetylcholine receptor M5	target
Doxepin	Alpha-1A adrenergic receptor	target
Doxepin	5-hydroxytryptamine receptor 1A	target
Doxepin	5-hydroxytryptamine receptor 2A	target
Doxepin	Cytochrome P450 2C19	enzyme
Doxepin	Cytochrome P450 2C9	enzyme
Doxepin	Cytochrome P450 1A2	enzyme
Doxepin	ATP-dependent translocase ABCB1	transporter
Doxepin	5-hydroxytryptamine receptor 2B	target
Doxepin	5-hydroxytryptamine receptor 2C	target
Doxepin	Alpha-1B adrenergic receptor	target
Doxepin	Alpha-1D adrenergic receptor	target
Doxepin	Cytochrome P450 3A4	enzyme
Doxepin	5-hydroxytryptamine receptor 6	target
Doxepin	Histamine H4 receptor	target
Doxepin	Potassium voltage-gated channel subfamily H member 2	target
Doxepin	Albumin	carrier
Doxepin	Alpha-1-acid glycoprotein 1	carrier
Imipramine	Sodium-dependent noradrenaline transporter	target
Imipramine	Sodium-dependent serotonin transporter	target
Imipramine	Cytochrome P450 1A2	enzyme
Imipramine	Cytochrome P450 2C19	enzyme
Imipramine	Cytochrome P450 2D6	enzyme
Imipramine	Histamine H1 receptor	target
Imipramine	Alpha-1A adrenergic receptor	target
Imipramine	5-hydroxytryptamine receptor 2A	target
Imipramine	Muscarinic acetylcholine receptor M1	target
Imipramine	Muscarinic acetylcholine receptor M2	target
Imipramine	Muscarinic acetylcholine receptor M3	target
Imipramine	Muscarinic acetylcholine receptor M4	target
Imipramine	Muscarinic acetylcholine receptor M5	target
Imipramine	A-type voltage-gated potassium channel KCND2	target
Imipramine	A-type voltage-gated potassium channel KCND3	target
Imipramine	Alpha-1D adrenergic receptor	target
Imipramine	Alpha-1-acid glycoprotein 1	carrier
Imipramine	Solute carrier family 22 member 2	transporter
Imipramine	Solute carrier family 22 member 3	transporter
Imipramine	ATP-dependent translocase ABCB1	transporter
Imipramine	Solute carrier family 22 member 4	transporter
Imipramine	Cytochrome P450 3A4	enzyme
Imipramine	Cytochrome P450 2B6	enzyme
Imipramine	Cytochrome P450 2C18	enzyme
Imipramine	Cytochrome P450 2E1	enzyme
Imipramine	Cytochrome P450 3A7	enzyme
Imipramine	5-hydroxytryptamine receptor 2C	target
Imipramine	Alpha-1B adrenergic receptor	target
Imipramine	5-hydroxytryptamine receptor 7	target
Imipramine	D(1) dopamine receptor	target
Imipramine	D(2) dopamine receptor	target
Imipramine	Potassium voltage-gated channel subfamily H member 2	target
Imipramine	Sodium-dependent dopamine transporter	target
Imipramine	5-hydroxytryptamine receptor 1A	target
Imipramine	5-hydroxytryptamine receptor 6	target
Imipramine	Potassium voltage-gated channel subfamily H member 1	target
Imipramine	Albumin	carrier
Imipramine	Alpha-1-acid glycoprotein 2	target
Nortriptyline	Sodium-dependent serotonin transporter	target
Nortriptyline	Sodium-dependent noradrenaline transporter	target
Nortriptyline	Cytochrome P450 1A2	enzyme
Nortriptyline	Cytochrome P450 2D6	enzyme
Nortriptyline	Albumin	carrier
Nortriptyline	Alpha-1-acid glycoprotein 1	carrier
Nortriptyline	Histamine H1 receptor	target
Nortriptyline	5-hydroxytryptamine receptor 2A	target
Nortriptyline	Alpha-1A adrenergic receptor	target
Nortriptyline	5-hydroxytryptamine receptor 1A	target
Nortriptyline	Cytochrome P450 3A4	enzyme
Nortriptyline	Cytochrome P450 3A5	enzyme
Nortriptyline	Alpha-1D adrenergic receptor	target
Nortriptyline	Cytochrome P450 2C19	enzyme
Nortriptyline	Cytochrome P450 2E1	enzyme
Nortriptyline	5-hydroxytryptamine receptor 2C	target
Nortriptyline	Alpha-1B adrenergic receptor	target
Nortriptyline	Alpha-2 adrenergic receptors	target
Nortriptyline	Beta adrenergic receptor	target
Nortriptyline	D(2) dopamine receptor	target
Nortriptyline	Sigma receptor	target
Nortriptyline	5-hydroxytryptamine receptor 2C	target
Nortriptyline	Sodium-dependent noradrenaline transporter	transporter
Nortriptyline	Muscarinic acetylcholine receptor	target
Nortriptyline	ATP-dependent translocase ABCB1	transporter
Avanafil	cGMP-specific 3',5'-cyclic phosphodiesterase	target
Avanafil	Cytochrome P450 3A4	enzyme
Avanafil	Albumin	carrier
Avanafil	Alpha-1-acid glycoprotein 1	carrier
Avanafil	ATP-dependent translocase ABCB1	transporter
Avanafil	Broad substrate specificity ATP-binding cassette transporter ABCG2	transporter
Avanafil	Cytochrome P450 2C9	enzyme
Conivaptan	Vasopressin V1a receptor	target
Conivaptan	Vasopressin V2 receptor	target
Conivaptan	Cytochrome P450 3A4	enzyme
Conivaptan	ATP-dependent translocase ABCB1	transporter
Darifenacin	Muscarinic acetylcholine receptor M3	target
Darifenacin	Cytochrome P450 3A4	enzyme
Darifenacin	Cytochrome P450 2D6	enzyme
Darifenacin	Muscarinic acetylcholine receptor M1	target
Darifenacin	Muscarinic acetylcholine receptor M2	target
Darifenacin	Muscarinic acetylcholine receptor M4	target
Darifenacin	Muscarinic acetylcholine receptor M5	target
Darunavir	Pol polyprotein	target
Darunavir	Cytochrome P450 3A4	enzyme
Darunavir	Solute carrier organic anion transporter family member 1B1	transporter
Darunavir	ATP-dependent translocase ABCB1	transporter
Darunavir	Albumin	carrier
Darunavir	Alpha-1-acid glycoprotein 1	carrier
Darunavir	Cytochrome P450 2D6	enzyme
Darunavir	Gag-Pol polyprotein	target
Ebastine	Cytochrome P450 3A4	enzyme
Ebastine	Cytochrome P450 3A Subfamily	enzyme
Everolimus	Serine/threonine-protein kinase mTOR	target
Everolimus	Cytochrome P450 3A4	enzyme
Everolimus	Solute carrier organic anion transporter family member 1B1	transporter
Everolimus	Solute carrier organic anion transporter family member 1B3	transporter
Everolimus	Solute carrier organic anion transporter family member 1A2	transporter
Everolimus	Cytochrome P450 2D6	enzyme
Everolimus	ATP-dependent translocase ABCB1	transporter
Ibrutinib	Tyrosine-protein kinase BTK	target
Ibrutinib	Cytochrome P450 3A4	enzyme
Ibrutinib	Cytochrome P450 3A5	enzyme
Ibrutinib	Albumin	carrier
Ibrutinib	alpha1-acid glycoprotein	carrier
Ibrutinib	Cytochrome P450 2D6	enzyme
Lomitapide	Microsomal triglyceride transfer protein large subunit	target
Lomitapide	Cytochrome P450 3A4	enzyme
Lomitapide	ATP-dependent translocase ABCB1	transporter
Naloxegol	Cytochrome P450 3A4	enzyme
Naloxegol	Cytochrome P450 2D6	enzyme
Naloxegol	Cytochrome P450 2C19	enzyme
Naloxegol	Mu-type opioid receptor	target
Budesonide	Glucocorticoid receptor	target
Budesonide	Cytochrome P450 3A4	enzyme
Budesonide	Cytochrome P450 3A5	enzyme
Budesonide	Bile salt export pump	transporter
Budesonide	ATP-dependent translocase ABCB1	transporter
Budesonide	Annexin A1	target
Budesonide	Cytochrome P450 3A Subfamily	enzyme
Budesonide	Cytochrome P450 2A6	enzyme
Budesonide	Cytochrome P450 1B1	enzyme
Budesonide	Cytochrome P450 2B6	enzyme
Budesonide	Cytochrome P450 2C8	enzyme
Budesonide	Cytochrome P450 2C9	enzyme
Budesonide	Cytochrome P450 2C19	enzyme
Budesonide	Corticosteroid-binding globulin	carrier
Budesonide	Solute carrier organic anion transporter family member 1A2	transporter
Budesonide	Organic anion transporter 3	transporter
Budesonide	Albumin	carrier
Dasatinib	Tyrosine-protein kinase ABL1	target
Dasatinib	Tyrosine-protein kinase ABL2	target
Dasatinib	Proto-oncogene tyrosine-protein kinase Src	target
Dasatinib	Tyrosine-protein kinase Fyn	target
Dasatinib	Tyrosine-protein kinase Lck	target
Dasatinib	Tyrosine-protein kinase Yes	target
Dasatinib	Mast/stem cell growth factor receptor Kit	target
Dasatinib	Platelet-derived growth factor receptor beta	target
Dasatinib	Ephrin type-A receptor 2	target
Dasatinib	Signal transducer and activator of transcription 5B	target
Dasatinib	Cytochrome P450 3A4	enzyme
Dasatinib	ATP-dependent translocase ABCB1	transporter
Dasatinib	Broad substrate specificity ATP-binding cassette transporter ABCG2	transporter
Dasatinib	Cytochrome P450 1A1	enzyme
Dasatinib	Cytochrome P450 1A2	enzyme
Dasatinib	Cytochrome P450 1B1	enzyme
Dasatinib	Cytochrome P450 3A5	enzyme
Dasatinib	Flavin-containing monooxygenase 3	enzyme
Dasatinib	Tyrosine-protein kinase BTK	target
Dasatinib	Nuclear receptor subfamily 4 group A member 3	target
Dasatinib	Breakpoint cluster region protein	target
Dasatinib	Tyrosine-protein kinase CSK	target
Dasatinib	Ephrin type-A receptor 5	target
Dasatinib	Ephrin type-B receptor 4	target
Dasatinib	Tyrosine-protein kinase Fgr	target
Dasatinib	Tyrosine-protein kinase FRK	target
Dasatinib	Heat shock cognate 71 kDa protein	target
Dasatinib	Tyrosine-protein kinase Lyn	target
Dasatinib	Mitogen-activated protein kinase kinase kinase 20	target
Dasatinib	Mitogen-activated protein kinase 14	target
Dasatinib	Amidophosphoribosyltransferase	target
Dronedarone	Alpha-1A adrenergic receptor	target
Dronedarone	Beta-1 adrenergic receptor	target
Dronedarone	Alpha-1B adrenergic receptor	target
Dronedarone	Alpha-1D adrenergic receptor	target
Dronedarone	Alpha-2A adrenergic receptor	target
Dronedarone	Alpha-2B adrenergic receptor	target
Dronedarone	Alpha-2C adrenergic receptor	target
Dronedarone	Potassium voltage-gated channel subfamily H member 2	target
Dronedarone	Voltage-dependent L-type calcium channel subunit alpha-1C	target
Dronedarone	Voltage-dependent L-type calcium channel subunit alpha-1D	target
Dronedarone	Voltage-dependent L-type calcium channel subunit alpha-1F	target
Dronedarone	Voltage-dependent L-type calcium channel subunit alpha-1S	target
Dronedarone	Voltage-dependent L-type calcium channel subunit beta-1	target
Dronedarone	Voltage-dependent L-type calcium channel subunit beta-2	target
Dronedarone	Voltage-dependent L-type calcium channel subunit beta-3	target
Dronedarone	Voltage-dependent L-type calcium channel subunit beta-4	target
Dronedarone	Cytochrome P450 2D6	enzyme
Dronedarone	Cytochrome P450 3A4	enzyme
Dronedarone	ATP-dependent translocase ABCB1	transporter
Dronedarone	Potassium channel subfamily K member 2	target
Dronedarone	Albumin	carrier
Dronedarone	Solute carrier family 22 member 2	transporter
Dronedarone	Solute carrier family 22 member 1	transporter
Dronedarone	Solute carrier organic anion transporter family member 1B1	transporter
Dronedarone	Solute carrier organic anion transporter family member 1B3	transporter
Dronedarone	Organic anion transporter 3	transporter
Dronedarone	Cytochrome P450 3A5	enzyme
Dronedarone	Cytochrome P450 2J2	enzyme
Dronedarone	Thyroid hormone receptor alpha	target
Dronedarone	Sodium channel protein type 5 subunit alpha	target
Dronedarone	G protein-activated inward rectifier potassium channel 1	target
Dronedarone	Potassium voltage-gated channel subfamily KQT member 1	target
Dronedarone	Inward rectifier potassium channel	target
Dronedarone	Sodium/calcium exchanger 1	target
Dronedarone	A-type voltage-gated potassium channel KCND3	target
Dronedarone	Potassium voltage-gated channel subfamily A member 5	target
Eletriptan	5-hydroxytryptamine receptor 1D	target
Eletriptan	5-hydroxytryptamine receptor 1A	target
Eletriptan	5-hydroxytryptamine receptor 1F	target
Eletriptan	5-hydroxytryptamine receptor 1B	target
Eletriptan	Cytochrome P450 3A4	enzyme
Eletriptan	Cytochrome P450 2D6	enzyme
Eletriptan	Cytochrome P450 2C9	enzyme
Eletriptan	Cytochrome P450 2C19	enzyme
Eletriptan	Prostaglandin G/H synthase 1	enzyme
Eletriptan	Cytochrome P450 2A6	enzyme
Eletriptan	ATP-dependent translocase ABCB1	transporter
Eplerenone	Mineralocorticoid receptor	target
Eplerenone	Cytochrome P450 3A4	enzyme
Eplerenone	Cytochrome P450 3A5	enzyme
Eplerenone	Cytochrome P450 11B2, mitochondrial	enzyme
Lurasidone	Cytochrome P450 3A4	enzyme
Lurasidone	D(2) dopamine receptor	target
Lurasidone	5-hydroxytryptamine receptor 2A	target
Lurasidone	5-hydroxytryptamine receptor 7	target
Lurasidone	5-hydroxytryptamine receptor 1A	target
Lurasidone	Alpha-2C adrenergic receptor	target
Lurasidone	Alpha-2A adrenergic receptor	target
Maraviroc	C-C chemokine receptor type 5	target
Maraviroc	Cytochrome P450 3A4	enzyme
Quetiapine	5-hydroxytryptamine receptor 2A	target
Quetiapine	5-hydroxytryptamine receptor 2C	target
Quetiapine	D(2) dopamine receptor	target
Quetiapine	5-hydroxytryptamine receptor 1A	target
Quetiapine	Histamine H1 receptor	target
Quetiapine	Cytochrome P450 3A4	enzyme
Quetiapine	Alpha-1 adrenergic receptors	target
Quetiapine	Alpha-2A adrenergic receptor	target
Quetiapine	Alpha-2B adrenergic receptor	target
Quetiapine	Alpha-2C adrenergic receptor	target
Quetiapine	5-hydroxytryptamine receptor 1D	target
Quetiapine	Muscarinic acetylcholine receptor M1	target
Quetiapine	Muscarinic acetylcholine receptor M2	target
Quetiapine	Muscarinic acetylcholine receptor M3	target
Quetiapine	Muscarinic acetylcholine receptor M4	target
Quetiapine	Muscarinic acetylcholine receptor M5	target
Quetiapine	5-hydroxytryptamine receptor 1B	target
Quetiapine	5-hydroxytryptamine receptor 1E	target
Quetiapine	5-hydroxytryptamine receptor 3A	target
Quetiapine	5-hydroxytryptamine receptor 6	target
Quetiapine	5-hydroxytryptamine receptor 7	target
Quetiapine	D(1B) dopamine receptor	target
Quetiapine	D(1A) dopamine receptor	target
Quetiapine	D(3) dopamine receptor	target
Quetiapine	D(4) dopamine receptor	target
Quetiapine	Cytochrome P450 3A5	enzyme
Quetiapine	ATP-dependent translocase ABCB1	transporter
Quetiapine	Cytochrome P450 2C19	enzyme
Quetiapine	Cytochrome P450 2D6	enzyme
Quetiapine	Cytochrome P450 3A7	enzyme
Ticagrelor	Cytochrome P450 3A4	enzyme
Ticagrelor	P2Y purinoceptor 12	target
Ticagrelor	ATP-dependent translocase ABCB1	transporter
Ticagrelor	Cytochrome P450 2C9	enzyme
Ticagrelor	Albumin	carrier
Ticagrelor	Cytochrome P450 3A5	enzyme
Ticagrelor	Cytochrome P450 2B6	enzyme
Tolvaptan	Vasopressin V2 receptor	target
Tolvaptan	Cytochrome P450 3A4	enzyme
Tolvaptan	ATP-dependent translocase ABCB1	transporter
Tolvaptan	Vasopressin V1a receptor	target
Aprepitant	Substance-P receptor	target
Aprepitant	Cytochrome P450 3A4	enzyme
Aprepitant	Cytochrome P450 2C9	enzyme
Aprepitant	Cytochrome P450 2C19	enzyme
Colchicine	Tubulin beta chain	target
Colchicine	Cytochrome P450 3A4	enzyme
Colchicine	ATP-dependent translocase ABCB1	transporter
Colchicine	Cytochrome P450 2B6	enzyme
Colchicine	Cytochrome P450 2C8	enzyme
Colchicine	Cytochrome P450 2E1	enzyme
Colchicine	Albumin	carrier
Eliglustat	Ceramide glucosyltransferase	target
Eliglustat	Cytochrome P450 2D6	enzyme
Eliglustat	Cytochrome P450 3A4	enzyme
Eliglustat	ATP-dependent translocase ABCB1	transporter
Rilpivirine	Cytochrome P450 3A4	enzyme
Rilpivirine	Reverse transcriptase/RNaseH	target
Rilpivirine	Nuclear receptor subfamily 1 group I member 2	target
Rilpivirine	Cytochrome P450 2C19	enzyme
Rilpivirine	Cytochrome P450 2B6	enzyme
Rilpivirine	ATP-dependent translocase ABCB1	transporter
Rilpivirine	Broad substrate specificity ATP-binding cassette transporter ABCG2	transporter
Rilpivirine	Solute carrier organic anion transporter family member 1B1	transporter
Rilpivirine	Solute carrier organic anion transporter family member 1B3	transporter
Rilpivirine	Albumin	carrier
Rilpivirine	Cytochrome P450 2D6	enzyme
Rilpivirine	Cytochrome P450 2C9	enzyme
Rilpivirine	Cytochrome P450 2C8	enzyme
Rilpivirine	Cytochrome P450 2E1	enzyme
Rilpivirine	Gag-Pol polyprotein	target
Rilpivirine	Sodium channel protein type 10 subunit alpha	target
Rivaroxaban	Coagulation factor X	target
Rivaroxaban	Cytochrome P450 3A4	enzyme
Rivaroxaban	Cytochrome P450 2J2	enzyme
Rivaroxaban	ATP-dependent translocase ABCB1	transporter
Rivaroxaban	Cytochrome P450 3A5	enzyme
Rivaroxaban	Broad substrate specificity ATP-binding cassette transporter ABCG2	transporter
Methysergide	5-hydroxytryptamine receptor 2A	target
Methysergide	5-hydroxytryptamine receptor 1A	target
Methysergide	5-hydroxytryptamine receptor 7	target
Methysergide	5-hydroxytryptamine receptor 2C	target
Methysergide	5-hydroxytryptamine receptor 2B	target
Methysergide	5-hydroxytryptamine receptor 1B	target
Methysergide	5-hydroxytryptamine receptor 1F	target
Methysergide	5-hydroxytryptamine receptor 1E	target
Methysergide	Cytochrome P450 3A4	enzyme
Tianeptine	Glutamate receptor 1	target
Tianeptine	Mu-type opioid receptor	target
Tianeptine	5-hydroxytryptamine receptor 1A	target
Tianeptine	D(3) dopamine receptor	target
Tianeptine	Cytochrome P450 3A4	enzyme
Tianeptine	Sodium-dependent serotonin transporter	target
Estradiol	Estrogen receptor	target
Estradiol	Nuclear receptor subfamily 1 group I member 2	target
Estradiol	Sex hormone-binding globulin	carrier
Estradiol	Estrogen receptor beta	target
Estradiol	Cytochrome P450 1A2	enzyme
Estradiol	UDP-glucuronosyltransferase 1A1	enzyme
Estradiol	Albumin	carrier
Estradiol	Fatty acid-binding protein, intestinal	carrier
Estradiol	Cytochrome P450 3A4	enzyme
Estradiol	Cytochrome P450 3A5	enzyme
Estradiol	Cytochrome P450 3A7	enzyme
Estradiol	Solute carrier family 22 member 2	transporter
Estradiol	Solute carrier family 22 member 3	transporter
Estradiol	ATP-binding cassette sub-family C member 10	transporter
Estradiol	Solute carrier family 22 member 11	transporter
Estradiol	Broad substrate specificity ATP-binding cassette transporter ABCG2	transporter
Estradiol	Solute carrier organic anion transporter family member 1B1	transporter
Estradiol	ATP-dependent translocase ABCB1	transporter
Estradiol	Cytochrome P450 1A1	enzyme
Estradiol	Cytochrome P450 1B1	enzyme
Estradiol	Cytochrome P450 2C19	enzyme
Estradiol	Cytochrome P450 2C8	enzyme
Estradiol	Cytochrome P450 2C9	enzyme
Estradiol	Organic anion transporter 3	transporter
Estradiol	Solute carrier organic anion transporter family member 1B3	transporter
Estradiol	Solute carrier organic anion transporter family member 1C1	transporter
Estradiol	Neuronal acetylcholine receptor subunit alpha-4	target
Estradiol	G-protein coupled estrogen receptor 1	target
Estradiol	ATP synthase subunit a	target
Estradiol	Beclin-1	target
Estradiol	UDP-glucuronosyltransferase 2B15	enzyme
Estradiol	Catechol O-methyltransferase	enzyme
Estradiol	UDP-glucuronosyltransferases (UGTs)	enzyme
Estradiol	Aromatase	enzyme
Estradiol cypionate	Estrogen receptor	target
Estradiol cypionate	Nuclear receptor subfamily 1 group I member 2	target
Estradiol cypionate	Sex hormone-binding globulin	carrier
Estradiol cypionate	Estrogen receptor beta	target
Estradiol cypionate	Cytochrome P450 1A2	enzyme
Estradiol cypionate	UDP-glucuronosyltransferase 1A1	enzyme
Estradiol cypionate	Albumin	carrier
Estradiol cypionate	Fatty acid-binding protein, intestinal	carrier
Estradiol cypionate	Cytochrome P450 3A4	enzyme
Estradiol cypionate	Cytochrome P450 3A5	enzyme
Estradiol cypionate	Cytochrome P450 3A7	enzyme
Estradiol cypionate	Solute carrier family 22 member 2	transporter
Estradiol cypionate	Solute carrier family 22 member 1	transporter
Estradiol cypionate	Solute carrier family 22 member 3	transporter
Estradiol cypionate	Solute carrier organic anion transporter family member 2B1	transporter
Estradiol cypionate	Solute carrier organic anion transporter family member 1A2	transporter
Estradiol cypionate	ATP-binding cassette sub-family C member 10	transporter
Estradiol cypionate	Solute carrier family 22 member 11	transporter
Estradiol cypionate	Broad substrate specificity ATP-binding cassette transporter ABCG2	transporter
Estradiol cypionate	Solute carrier organic anion transporter family member 1B1	transporter
Estradiol cypionate	ATP-dependent translocase ABCB1	transporter
Estradiol cypionate	Cytochrome P450 1A1	enzyme
Estradiol cypionate	Cytochrome P450 1B1	enzyme
Estradiol cypionate	Cytochrome P450 2C19	enzyme
Estradiol cypionate	Cytochrome P450 2C8	enzyme
Estradiol cypionate	Cytochrome P450 2C9	enzyme
Estradiol cypionate	Organic anion transporter 3	transporter
Estradiol cypionate	Solute carrier organic anion transporter family member 1B3	transporter
Estradiol cypionate	Solute carrier organic anion transporter family member 1C1	transporter
Estradiol cypionate	Solute carrier organic anion transporter family member 4A1	transporter
Estradiol cypionate	Neuronal acetylcholine receptor subunit alpha-4	target
Estradiol cypionate	Nuclear receptor coactivator 2	target
Estradiol cypionate	G-protein coupled estrogen receptor 1	target
Estradiol cypionate	ATP synthase subunit a	target
Estradiol cypionate	Beclin-1	target
Estradiol cypionate	17-beta-hydroxysteroid dehydrogenase type 2	target
Estradiol cypionate	Estrogen-related receptor gamma	target
Estradiol valerate	Estrogen receptor	target
Estradiol valerate	Nuclear receptor subfamily 1 group I member 2	target
Estradiol valerate	Sex hormone-binding globulin	carrier
Estradiol valerate	Estrogen receptor beta	target
Estradiol valerate	Cytochrome P450 1A2	enzyme
Estradiol valerate	UDP-glucuronosyltransferase 1A1	enzyme
Estradiol valerate	Albumin	carrier
Estradiol valerate	Fatty acid-binding protein, intestinal	carrier
Estradiol valerate	Cytochrome P450 3A4	enzyme
Estradiol valerate	Cytochrome P450 3A5	enzyme
Estradiol valerate	Cytochrome P450 3A7	enzyme
Estradiol valerate	Solute carrier family 22 member 2	transporter
Estradiol valerate	Solute carrier family 22 member 1	transporter
Estradiol valerate	Solute carrier family 22 member 3	transporter
Estradiol valerate	Solute carrier organic anion transporter family member 2B1	transporter
Estradiol valerate	Solute carrier organic anion transporter family member 1A2	transporter
Estradiol valerate	ATP-binding cassette sub-family C member 10	transporter
Estradiol valerate	Solute carrier family 22 member 11	transporter
Estradiol valerate	Broad substrate specificity ATP-binding cassette transporter ABCG2	transporter
Estradiol valerate	Solute carrier organic anion transporter family member 1B1	transporter
Estradiol valerate	ATP-dependent translocase ABCB1	transporter
Estradiol valerate	Cytochrome P450 1A1	enzyme
Estradiol valerate	Cytochrome P450 1B1	enzyme
Estradiol valerate	Cytochrome P450 2C19	enzyme
Estradiol valerate	Cytochrome P450 2C8	enzyme
Estradiol valerate	Cytochrome P450 2C9	enzyme
Estradiol valerate	Organic anion transporter 3	transporter
Estradiol valerate	Solute carrier organic anion transporter family member 1B3	transporter
Estradiol valerate	Solute carrier organic anion transporter family member 1C1	transporter
Estradiol valerate	Solute carrier organic anion transporter family member 4A1	transporter
Estradiol valerate	Neuronal acetylcholine receptor subunit alpha-4	target
Estradiol valerate	Nuclear receptor coactivator 2	target
Estradiol valerate	G-protein coupled estrogen receptor 1	target
Estradiol valerate	ATP synthase subunit a	target
Estradiol valerate	Beclin-1	target
Estradiol valerate	17-beta-hydroxysteroid dehydrogenase type 2	target
Estradiol valerate	Estrogen-related receptor gamma	target
Ethinylestradiol	Estrogen receptor	target
Ethinylestradiol	Nuclear receptor subfamily 1 group I member 2	target
Ethinylestradiol	Cytochrome P450 3A4	enzyme
Ethinylestradiol	Cytochrome P450 2C8	enzyme
Ethinylestradiol	Bile salt export pump	transporter
Ethinylestradiol	Hepatic sodium/bile acid cotransporter	transporter
Ethinylestradiol	ATP-binding cassette sub-family C member 2	transporter
Ethinylestradiol	ATP-dependent translocase ABCB1	transporter
Ethinylestradiol	UDP-glucuronosyltransferase 1A1	enzyme
Ethinylestradiol	Cytochrome P450 2C19	enzyme
Ethinylestradiol	UDP-glucuronosyltransferase 1A4	enzyme
Ethinylestradiol	UDP-glucuronosyltransferase 1A9	enzyme
Ethinylestradiol	Cytochrome P450 2C9	enzyme
Ethinylestradiol	Cytochrome P450 1A2	enzyme
Ethinylestradiol	Sulfotransferase 1E1	enzyme
Ethinylestradiol	Sulfotransferase 1A3	enzyme
Ethinylestradiol	Cytochrome P450 3A5	enzyme
Ethinylestradiol	UDP-glucuronosyltransferase 2B7	enzyme
Ethinylestradiol	UDP-glucuronosyltransferase 1A3	enzyme
Ethinylestradiol	Catechol O-methyltransferase	enzyme
Ethinylestradiol	Solute carrier organic anion transporter family member 1A2	transporter
Ethinylestradiol	Albumin	carrier
Ethinylestradiol	Sex hormone-binding globulin	carrier
Mestranol	Estrogen receptor	target
Mestranol	Cytochrome P450 2C9	enzyme
Mestranol	Cytochrome P450 3A4	enzyme
Mestranol	Cytochrome P450 2C8	enzyme
Aminophylline	cGMP-inhibited 3',5'-cyclic phosphodiesterase 3A	target
Aminophylline	Adenosine receptor A3	target
Aminophylline	Adenosine receptor A1	target
Aminophylline	Cytochrome P450 1A2	enzyme
Aminophylline	Cytochrome P450 2E1	enzyme
Aminophylline	Cytochrome P450 3A4	enzyme
Aminophylline	Histone deacetylase 2	target
Theophylline	cGMP-inhibited 3',5'-cyclic phosphodiesterase 3A	target
Theophylline	3',5'-cyclic-AMP phosphodiesterase 4B	target
Theophylline	Adenosine receptor A2b	target
Theophylline	3',5'-cyclic-AMP phosphodiesterase 4A	target
Theophylline	cGMP-specific 3',5'-cyclic phosphodiesterase	target
Theophylline	Adenosine receptor A1	target
Theophylline	Adenosine receptor A2a	target
Theophylline	Cytochrome P450 1A2	enzyme
Theophylline	Adenosine deaminase	enzyme
Theophylline	Cytochrome P450 2E1	enzyme
Theophylline	Cytochrome P450 3A4	enzyme
Theophylline	Solute carrier family 22 member 7	transporter
Theophylline	Cytochrome P450 1A1	enzyme
Theophylline	Cytochrome P450 1B1	enzyme
Theophylline	Cytochrome P450 2D6	enzyme
Theophylline	Histone deacetylase 2	target
Theophylline	Copine-1	target
Theophylline	Minor histocompatibility antigen H13	target
Theophylline	BOS complex subunit NOMO1	target
Theophylline	Poly [ADP-ribose] polymerase 1	target
Theophylline	Protein RIC-3	target
Theophylline	Tubulin monoglycylase TTLL3	target
Theophylline	5'-nucleotidase	target
Bromocriptine	D(2) dopamine receptor	target
Bromocriptine	Cytochrome P450 3A4	enzyme
Bromocriptine	5-hydroxytryptamine receptor 1D	target
Bromocriptine	Alpha-2A adrenergic receptor	target
Bromocriptine	D(3) dopamine receptor	target
Bromocriptine	5-hydroxytryptamine receptor 1A	target
Bromocriptine	Alpha-2C adrenergic receptor	target
Bromocriptine	Alpha-2B adrenergic receptor	target
Bromocriptine	5-hydroxytryptamine receptor 2B	target
Bromocriptine	D(4) dopamine receptor	target
Bromocriptine	5-hydroxytryptamine receptor 2A	target
Bromocriptine	5-hydroxytryptamine receptor 1B	target
Bromocriptine	5-hydroxytryptamine receptor 2C	target
Bromocriptine	D(1B) dopamine receptor	target
Bromocriptine	D(1A) dopamine receptor	target
Bromocriptine	Alpha-1A adrenergic receptor	target
Bromocriptine	Alpha-1B adrenergic receptor	target
Bromocriptine	Alpha-1D adrenergic receptor	target
Bromocriptine	5-hydroxytryptamine receptor 7	target
Bromocriptine	ATP-dependent translocase ABCB1	transporter
Cabergoline	D(2) dopamine receptor	target
Cabergoline	5-hydroxytryptamine receptor 2B	target
Cabergoline	D(3) dopamine receptor	target
Cabergoline	5-hydroxytryptamine receptor 2A	target
Cabergoline	Alpha-2B adrenergic receptor	target
Cabergoline	5-hydroxytryptamine receptor 1D	target
Cabergoline	D(4) dopamine receptor	target
Cabergoline	Alpha-2A adrenergic receptor	target
Cabergoline	5-hydroxytryptamine receptor 1A	target
Cabergoline	Alpha-2C adrenergic receptor	target
Cabergoline	D(1B) dopamine receptor	target
Cabergoline	D(1A) dopamine receptor	target
Cabergoline	5-hydroxytryptamine receptor 1B	target
Cabergoline	5-hydroxytryptamine receptor 2C	target
Cabergoline	Cytochrome P450 3A4	enzyme
Cabergoline	5-hydroxytryptamine receptor 7	target
Cabergoline	Alpha-1A adrenergic receptor	target
Cabergoline	Alpha-1B adrenergic receptor	target
Cabergoline	Alpha-1D adrenergic receptor	target
Cabergoline	Beta-1 adrenergic receptor	target
Cabergoline	Beta-2 adrenergic receptor	target
Cabergoline	D(1) dopamine receptor	target
Cabergoline	ATP-dependent translocase ABCB1	transporter
Dihydroergocornine	Serotonin Receptors	target
Dihydroergocornine	Beta adrenergic receptor	target
Dihydroergocornine	Alpha adrenergic receptor	target
Dihydroergocornine	Cytochrome P450 3A4	enzyme
Dihydroergocristine	Serotonin Receptors	target
Dihydroergocristine	Beta adrenergic receptor	target
Dihydroergocristine	Alpha adrenergic receptor	target
Dihydroergocristine	Dopamine receptor	target
Dihydroergocristine	Bile salt export pump	transporter
Dihydroergocristine	Cytochrome P450 3A4	enzyme
Dihydroergocristine	Alpha-2C adrenergic receptor	target
Dihydroergocryptine	Cytochrome P450 3A4	enzyme
Dihydroergotamine	5-hydroxytryptamine receptor 1D	target
Dihydroergotamine	5-hydroxytryptamine receptor 1B	target
Dihydroergotamine	Cytochrome P450 3A4	enzyme
Dihydroergotamine	Alpha-2A adrenergic receptor	target
Dihydroergotamine	5-hydroxytryptamine receptor 2B	target
Dihydroergotamine	ATP-dependent translocase ABCB1	transporter
Dihydroergotamine	5-hydroxytryptamine receptor 1A	target
Dihydroergotamine	5-hydroxytryptamine receptor 1E	target
Dihydroergotamine	5-hydroxytryptamine receptor 2A	target
Dihydroergotamine	5-hydroxytryptamine receptor 2C	target
Dihydroergotamine	Alpha-1 adrenergic receptors	target
Dihydroergotamine	Alpha-2 adrenergic receptors	target
Dihydroergotamine	D(2) dopamine receptor	target
Dihydroergotamine	D(3) dopamine receptor	target
Dihydroergotamine	D(4) dopamine receptor	target
Dihydroergotamine	5-hydroxytryptamine receptor 1F	target
Dihydroergotamine	5-hydroxytryptamine receptor 4	target
Dihydroergotamine	Beta-3 adrenergic receptor	target
Ergoloid mesylate	Dopamine receptor	target
Ergoloid mesylate	Alpha adrenergic receptor	target
Ergoloid mesylate	Beta adrenergic receptor	target
Ergoloid mesylate	Serotonin Receptors	target
Ergoloid mesylate	Cytochrome P450 3A4	enzyme
Ergometrine	Cytochrome P450 3A4	enzyme
Ergometrine	ATP-dependent translocase ABCB1	transporter
Ergometrine	Alpha-1A adrenergic receptor	target
Ergometrine	D(2) dopamine receptor	target
Ergotamine	Alpha-1A adrenergic receptor	target
Ergotamine	5-hydroxytryptamine receptor 1D	target
Ergotamine	5-hydroxytryptamine receptor 1B	target
Ergotamine	5-hydroxytryptamine receptor 2A	target
Ergotamine	Alpha-2A adrenergic receptor	target
Ergotamine	D(2) dopamine receptor	target
Ergotamine	Cytochrome P450 3A4	enzyme
Ergotamine	Alpha-1B adrenergic receptor	target
Ergotamine	Alpha-1D adrenergic receptor	target
Ergotamine	ATP-dependent translocase ABCB1	transporter
Ergotamine	D(1) dopamine receptor	target
Ergotamine	5-hydroxytryptamine receptor 1A	target
Ergotamine	5-hydroxytryptamine receptor 1F	target
Ergotamine	5-hydroxytryptamine receptor 2C	target
Ergotamine	5-hydroxytryptamine receptor 2B	target
Ergotamine	Alpha-2C adrenergic receptor	target
Lisuride	D(1A) dopamine receptor	target
Lisuride	5-hydroxytryptamine receptor 1A	target
Lisuride	D(2) dopamine receptor	target
Lisuride	Alpha-2A adrenergic receptor	target
Lisuride	Alpha-2B adrenergic receptor	target
Lisuride	Alpha-2C adrenergic receptor	target
Lisuride	D(3) dopamine receptor	target
Lisuride	5-hydroxytryptamine receptor 1D	target
Lisuride	5-hydroxytryptamine receptor 2B	target
Lisuride	5-hydroxytryptamine receptor 2A	target
Lisuride	D(4) dopamine receptor	target
Lisuride	5-hydroxytryptamine receptor 2C	target
Lisuride	D(1B) dopamine receptor	target
Lisuride	5-hydroxytryptamine receptor 1B	target
Lisuride	Cytochrome P450 3A4	enzyme
Lisuride	5-hydroxytryptamine receptor 7	target
Lysergic acid diethylamide	5-hydroxytryptamine receptor 1A	target
Lysergic acid diethylamide	5-hydroxytryptamine receptor 2B	target
Lysergic acid diethylamide	5-hydroxytryptamine receptor 6	target
Lysergic acid diethylamide	Cytochrome P450 3A4	enzyme
Lysergic acid diethylamide	Cytochrome P450 2D6	enzyme
Lysergic acid diethylamide	5-hydroxytryptamine receptor 2A	target
Methylergometrine	D(1A) dopamine receptor	target
Methylergometrine	Cytochrome P450 3A4	enzyme
Methylergometrine	5-hydroxytryptamine receptor 2B	target
Terguride	Cytochrome P450 3A4	enzyme
Triamcinolone	Corticosteroid-binding globulin	carrier
Triamcinolone	Glucocorticoid receptor	target
Triamcinolone	Cytochrome P450 3A4	enzyme
Triamcinolone	Prostaglandin G/H synthase 2	enzyme
Triamcinolone	Cholinesterase	enzyme
Triamcinolone	Cytochrome P450 3A5	enzyme
Triamcinolone	Cytochrome P450 3A7	enzyme
Triamcinolone	Albumin	carrier
Voriconazole	Cytochrome P450 2C19	enzyme
Voriconazole	Cytochrome P450 3A4	enzyme
Voriconazole	Cytochrome P450 2C9	enzyme
Voriconazole	Flavin-containing monooxygenase 1	enzyme
Voriconazole	Flavin-containing monooxygenase 3	enzyme
Voriconazole	Cytochrome P450 3A5	enzyme
Voriconazole	Cytochrome P450 3A7	enzyme
Voriconazole	Prostaglandin G/H synthase 1	enzyme
Voriconazole	Lanosterol 14-alpha demethylase	target
Voriconazole	Cytochrome P450 2B6	enzyme
Esomeprazole	Potassium-transporting ATPase alpha chain 1	target
Esomeprazole	Cytochrome P450 2C19	enzyme
Esomeprazole	Cytochrome P450 3A4	enzyme
Esomeprazole	N(G),N(G)-dimethylarginine dimethylaminohydrolase 1	target
Esomeprazole	ATP-dependent translocase ABCB1	transporter
Esomeprazole	Organic anion transporter 3	transporter
Esomeprazole	Potassium-transporting ATPase subunit beta	target
Omeprazole	Potassium-transporting ATPase alpha chain 1	target
Omeprazole	Cytochrome P450 2C19	enzyme
Omeprazole	Cytochrome P450 3A4	enzyme
Omeprazole	Cytochrome P450 2C9	enzyme
Omeprazole	Cytochrome P450 1A2	enzyme
Omeprazole	ATP-binding cassette sub-family C member 3	transporter
Omeprazole	ATP-dependent translocase ABCB1	transporter
Omeprazole	Broad substrate specificity ATP-binding cassette transporter ABCG2	transporter
Omeprazole	Cytochrome P450 1A1	enzyme
Omeprazole	Cytochrome P450 1B1	enzyme
Omeprazole	Cytochrome P450 2C18	enzyme
Omeprazole	Cytochrome P450 2C8	enzyme
Omeprazole	Cytochrome P450 2D6	enzyme
Omeprazole	Aryl hydrocarbon receptor	target
Omeprazole	Potassium-transporting ATPase subunit beta	target
Propafenone	Sodium channel protein type 5 subunit alpha	target
Propafenone	Potassium voltage-gated channel subfamily H member 2	target
Propafenone	Cytochrome P450 1A2	enzyme
Propafenone	Cytochrome P450 2D6	enzyme
Propafenone	Cytochrome P450 3A4	enzyme
Propafenone	ATP-dependent translocase ABCB1	transporter
Propafenone	Beta-1 adrenergic receptor	target
Propafenone	Beta-2 adrenergic receptor	target
Lopinavir	Pol polyprotein	target
Lopinavir	Cytochrome P450 3A4	enzyme
Lopinavir	Cytochrome P450 2D6	enzyme
Lopinavir	Cytochrome P450 2C19	enzyme
Lopinavir	ATP-dependent translocase ABCB1	transporter
Lopinavir	Cytochrome P450 2B6	enzyme
Lopinavir	Cytochrome P450 2C9	enzyme
Lopinavir	Cytochrome P450 3A Subfamily	enzyme
Lopinavir	Solute carrier organic anion transporter family member 1B1	transporter
Lopinavir	Solute carrier organic anion transporter family member 1B3	transporter
Lopinavir	Bile salt export pump	transporter
Lopinavir	Cytochrome P450 1A2	enzyme
Lopinavir	Alpha-1-acid glycoprotein 1	carrier
Lopinavir	Albumin	carrier
Tipranavir	Pol polyprotein	target
Tipranavir	Cytochrome P450 3A4	enzyme
Tipranavir	Cytochrome P450 2D6	enzyme
Tipranavir	Cytochrome P450 2C19	enzyme
Tipranavir	Bile salt export pump	transporter
Tipranavir	UDP-glucuronosyltransferase 1A1	enzyme
Tipranavir	Solute carrier organic anion transporter family member 2B1	transporter
Tipranavir	Solute carrier organic anion transporter family member 1B1	transporter
Tipranavir	Solute carrier organic anion transporter family member 1B3	transporter
Tipranavir	ATP-dependent translocase ABCB1	transporter
Tipranavir	Gag-Pol polyprotein	target
Phenprocoumon	Vitamin K epoxide reductase complex subunit 1	target
Phenprocoumon	Alpha-1-acid glycoprotein 1	carrier
Phenprocoumon	Albumin	carrier
Phenprocoumon	Cytochrome P450 2C9	enzyme
Phenprocoumon	Cytochrome P450 3A4	enzyme
Phenprocoumon	Cytochrome P450 2C8	enzyme
Teniposide	DNA topoisomerase 2-alpha	target
Teniposide	Cytochrome P450 2C19	enzyme
Teniposide	Cytochrome P450 2C9	enzyme
Teniposide	Cytochrome P450 3A4	enzyme
Teniposide	ATP-binding cassette sub-family C member 6	transporter
Teniposide	Broad substrate specificity ATP-binding cassette transporter ABCG2	transporter
Teniposide	Cytochrome P450 3A5	enzyme
Teniposide	DNA topoisomerase 2-beta	target
Ulipristal	Progesterone receptor	target
Ulipristal	Glucocorticoid receptor	target
Ulipristal	Androgen receptor	target
Ulipristal	Cytochrome P450 3A4	enzyme
Ulipristal	Cytochrome P450 1A2	enzyme
Ulipristal	Albumin	carrier
Ulipristal	Alpha-1-acid glycoprotein 1	carrier
Disopyramide	Sodium channel protein type 5 subunit alpha	target
Disopyramide	Alpha-1-acid glycoprotein 1	carrier
Disopyramide	Cytochrome P450 3A4	enzyme
Disopyramide	Muscarinic acetylcholine receptor M1	target
Disopyramide	Muscarinic acetylcholine receptor M2	target
Disopyramide	Muscarinic acetylcholine receptor M3	target
Disopyramide	A-type voltage-gated potassium channel KCND2	target
Disopyramide	A-type voltage-gated potassium channel KCND3	target
Disopyramide	Solute carrier family 22 member 2	transporter
Disopyramide	Solute carrier family 22 member 1	transporter
Disopyramide	Potassium voltage-gated channel subfamily H member 2	target
Disopyramide	Alpha-1-acid glycoprotein 2	target
Disopyramide	Cytochrome P450 1A2	enzyme
Methadone	NMDA receptor	target
Methadone	Mu-type opioid receptor	target
Methadone	Cytochrome P450 2B6	enzyme
Methadone	Cytochrome P450 3A4	enzyme
Methadone	Cytochrome P450 2C19	enzyme
Methadone	Delta-type opioid receptor	target
Methadone	Cytochrome P450 3A7	enzyme
Methadone	Cytochrome P450 2D6	enzyme
Methadone	ATP-dependent translocase ABCB1	transporter
Methadone	Cytochrome P450 2C8	enzyme
Methadone	Aromatase	enzyme
Methadone	Cytochrome P450 1A2	enzyme
Methadone	Cytochrome P450 2C18	enzyme
Methadone	Cytochrome P450 2C9	enzyme
Methadone	5-hydroxytryptamine receptor 3A	target
Methadone	Alpha-1-acid glycoprotein 1	carrier
Methadone	Albumin	carrier
Methadone	Neuronal acetylcholine receptor subunit alpha-7	target
Methadone	Neuronal acetylcholine receptor subunit alpha-3	target
Methadone	Neuronal acetylcholine receptor subunit alpha-4	target
Methadone	Neuronal acetylcholine receptor subunit beta-2	target
Methadone	Cytochrome P450 3A Subfamily	enzyme
Methadone	UDP-glucuronosyltransferase 2B4	enzyme
Alfuzosin	Alpha-1A adrenergic receptor	target
Alfuzosin	Alpha-1B adrenergic receptor	target
Alfuzosin	Alpha-1D adrenergic receptor	target
Alfuzosin	Cytochrome P450 3A4	enzyme
Alfuzosin	ATP-dependent translocase ABCB1	transporter
Alfuzosin	Alpha-1 adrenergic receptors	target
Alfuzosin	Albumin	carrier
Alfuzosin	Alpha-1-acid glycoprotein 1	carrier
Buprenorphine	Kappa-type opioid receptor	target
Buprenorphine	Mu-type opioid receptor	target
Buprenorphine	Cytochrome P450 3A4	enzyme
Buprenorphine	Cytochrome P450 2D6	enzyme
Buprenorphine	ATP-dependent translocase ABCB1	transporter
Buprenorphine	Broad substrate specificity ATP-binding cassette transporter ABCG2	transporter
Buprenorphine	Cytochrome P450 2C9	enzyme
Buprenorphine	Cytochrome P450 3A5	enzyme
Buprenorphine	Cytochrome P450 2C8	enzyme
Buprenorphine	Cytochrome P450 3A7	enzyme
Buprenorphine	Delta-type opioid receptor	target
Buprenorphine	Cytochrome P450 2C18	enzyme
Buprenorphine	Cytochrome P450 2C19	enzyme
Buprenorphine	Nociceptin receptor	target
Fostamatinib	Adenosine receptor A3	target
Fostamatinib	Synaptic vesicular amine transporter	target
Fostamatinib	Fatty-acid amide hydrolase 1	target
Fostamatinib	Equilibrative nucleoside transporter 1	target
Fostamatinib	UDP-glucuronosyltransferase 1A1	target
Fostamatinib	cGMP-specific 3',5'-cyclic phosphodiesterase	target
Fostamatinib	Polyunsaturated fatty acid 5-lipoxygenase	target
Fostamatinib	Cathepsin S	target
Fostamatinib	Procathepsin L	target
Fostamatinib	Tyrosine-protein kinase ABL1	target
Fostamatinib	Calcium-dependent protein kinase 1	target
Fostamatinib	Serine/threonine-protein kinase PknB	target
Fostamatinib	Ribosomal protein S6 kinase alpha-6	target
Fostamatinib	Non-receptor tyrosine-protein kinase TYK2	target
Fostamatinib	Atypical kinase COQ8A, mitochondrial	target
Fostamatinib	Tyrosine-protein kinase JAK1	target
Fostamatinib	Hepatocyte growth factor receptor	target
Fostamatinib	Serine/threonine-protein kinase NIM1	target
Fostamatinib	Serine/threonine-protein kinase 26	target
Fostamatinib	cAMP-dependent protein kinase catalytic subunit alpha	target
Fostamatinib	Serine/threonine-protein kinase 24	target
Fostamatinib	Serine/threonine-protein kinase 3	target
Fostamatinib	Tyrosine-protein kinase Tec	target
Fostamatinib	Tyrosine-protein kinase SYK	target
Fostamatinib	Serine/threonine-protein kinase 33	target
Fostamatinib	Serine/threonine-protein kinase 35	target
Fostamatinib	Serine/threonine-protein kinase 36	target
Fostamatinib	Serine/threonine-protein kinase 38	target
Fostamatinib	Serine/threonine-protein kinase 38-like	target
Fostamatinib	STE20/SPS1-related proline-alanine-rich protein kinase	target
Fostamatinib	Serine/threonine-protein kinase TAO1	target
Fostamatinib	Serine/threonine-protein kinase TAO2	target
Fostamatinib	Serine/threonine-protein kinase TAO3	target
Fostamatinib	Serine/threonine-protein kinase TBK1	target
Fostamatinib	Angiopoietin-1 receptor	target
Fostamatinib	Dual specificity testis-specific protein kinase 1	target
Fostamatinib	TGF-beta receptor type-1	target
Fostamatinib	TGF-beta receptor type-2	target
Fostamatinib	Tyrosine-protein kinase receptor Tie-1	target
Fostamatinib	Serine/threonine-protein kinase tousled-like 1	target
Fostamatinib	Serine/threonine-protein kinase tousled-like 2	target
Fostamatinib	TRAF2 and NCK-interacting protein kinase	target
Fostamatinib	Non-receptor tyrosine-protein kinase TNK1	target
Fostamatinib	Activated CDC42 kinase 1	target
Fostamatinib	Serine/threonine-protein kinase TNNI3K	target
Fostamatinib	Testis-specific serine/threonine-protein kinase 1	target
Fostamatinib	Dual specificity protein kinase TTK	target
Fostamatinib	Tyrosine-protein kinase TXK	target
Fostamatinib	Tyrosine-protein kinase receptor TYRO3	target
Fostamatinib	Serine/threonine-protein kinase ULK1	target
Fostamatinib	Serine/threonine-protein kinase ULK2	target
Fostamatinib	Serine/threonine-protein kinase ULK3	target
Fostamatinib	Wee1-like protein kinase	target
Fostamatinib	Tyrosine-protein kinase Yes	target
Fostamatinib	Mitogen-activated protein kinase kinase kinase 19	target
Fostamatinib	Mitogen-activated protein kinase kinase kinase 20	target
Fostamatinib	Tyrosine-protein kinase ZAP-70	target
Fostamatinib	AP2-associated protein kinase 1	target
Fostamatinib	Tyrosine-protein kinase ABL2	target
Fostamatinib	Activin receptor type-1	target
Fostamatinib	Activin receptor type-1B	target
Fostamatinib	Atypical kinase COQ8B, mitochondrial	target
Fostamatinib	ALK tyrosine kinase receptor	target
Fostamatinib	Ankyrin repeat and protein kinase domain-containing protein 1	target
Fostamatinib	Aurora kinase A	target
Fostamatinib	Aurora kinase B	target
Fostamatinib	Aurora kinase C	target
Fostamatinib	Tyrosine-protein kinase receptor UFO	target
Fostamatinib	Tyrosine-protein kinase Blk	target
Fostamatinib	BMP-2-inducible protein kinase	target
Fostamatinib	Bone morphogenetic protein receptor type-1B	target
Fostamatinib	Bone morphogenetic protein receptor type-2	target
Fostamatinib	Cytoplasmic tyrosine-protein kinase BMX	target
Fostamatinib	Serine/threonine-protein kinase B-raf	target
Fostamatinib	Tyrosine-protein kinase BTK	target
Fostamatinib	Calcium/calmodulin-dependent protein kinase type 1	target
Fostamatinib	Calcium/calmodulin-dependent protein kinase type 1D	target
Fostamatinib	Calcium/calmodulin-dependent protein kinase type 1G	target
Fostamatinib	Calcium/calmodulin-dependent protein kinase type II subunit alpha	target
Fostamatinib	Calcium/calmodulin-dependent protein kinase type II subunit beta	target
Fostamatinib	Calcium/calmodulin-dependent protein kinase type II subunit delta	target
Fostamatinib	Calcium/calmodulin-dependent protein kinase type II subunit gamma	target
Fostamatinib	Calcium/calmodulin-dependent protein kinase kinase 1	target
Fostamatinib	Calcium/calmodulin-dependent protein kinase kinase 2	target
Fostamatinib	Peripheral plasma membrane protein CASK	target
Fostamatinib	Kappa-casein	target
Fostamatinib	Cyclin-dependent kinase 1	target
Fostamatinib	Serine/threonine-protein kinase MRCK gamma	target
Fostamatinib	Cyclin-dependent kinase 4	target
Fostamatinib	Cyclin-dependent kinase-like 1	target
Fostamatinib	Cyclin-dependent kinase-like 2	target
Fostamatinib	Serine/threonine-protein kinase Chk1	target
Fostamatinib	Serine/threonine-protein kinase Chk2	target
Fostamatinib	Citron Rho-interacting kinase	target
Fostamatinib	Dual specificity protein kinase CLK1	target
Fostamatinib	Dual specificity protein kinase CLK2	target
Fostamatinib	Dual specificity protein kinase CLK3	target
Fostamatinib	Dual specificity protein kinase CLK4	target
Fostamatinib	Macrophage colony-stimulating factor 1 receptor	target
Fostamatinib	Tyrosine-protein kinase CSK	target
Fostamatinib	Casein kinase I isoform alpha	target
Fostamatinib	Casein kinase II subunit alpha	target
Fostamatinib	Casein kinase II subunit alpha'	target
Fostamatinib	Death-associated protein kinase 1	target
Fostamatinib	Death-associated protein kinase 2	target
Fostamatinib	Death-associated protein kinase 3	target
Fostamatinib	Serine/threonine-protein kinase DCLK1	target
Fostamatinib	Serine/threonine-protein kinase DCLK2	target
Fostamatinib	Serine/threonine-protein kinase DCLK3	target
Fostamatinib	Epithelial discoidin domain-containing receptor 1	target
Fostamatinib	Discoidin domain-containing receptor 2	target
Fostamatinib	Dual specificity tyrosine-phosphorylation-regulated kinase 1A	target
Fostamatinib	Dual specificity tyrosine-phosphorylation-regulated kinase 1B	target
Fostamatinib	Epidermal growth factor receptor	target
Fostamatinib	Eukaryotic translation initiation factor 2-alpha kinase 1	target
Fostamatinib	Interferon-induced, double-stranded RNA-activated protein kinase	target
Fostamatinib	eIF-2-alpha kinase GCN2	target
Fostamatinib	Ephrin type-A receptor 1	target
Fostamatinib	Ephrin type-A receptor 2	target
Fostamatinib	Ephrin type-A receptor 3	target
Fostamatinib	Ephrin type-A receptor 4	target
Fostamatinib	Ephrin type-A receptor 5	target
Fostamatinib	Ephrin type-A receptor 6	target
Fostamatinib	Ephrin type-A receptor 7	target
Fostamatinib	Ephrin type-A receptor 8	target
Fostamatinib	Ephrin type-B receptor 1	target
Fostamatinib	Ephrin type-B receptor 2	target
Fostamatinib	Ephrin type-B receptor 4	target
Fostamatinib	Ephrin type-B receptor 6	target
Fostamatinib	Receptor tyrosine-protein kinase erbB-2	target
Fostamatinib	Receptor tyrosine-protein kinase erbB-4	target
Fostamatinib	Serine/threonine-protein kinase/endoribonuclease IRE1	target
Fostamatinib	Tyrosine-protein kinase Fer	target
Fostamatinib	Tyrosine-protein kinase Fes/Fps	target
Fostamatinib	Fibroblast growth factor receptor 1	target
Fostamatinib	Fibroblast growth factor receptor 2	target
Fostamatinib	Fibroblast growth factor receptor 3	target
Fostamatinib	Tyrosine-protein kinase Fgr	target
Fostamatinib	Vascular endothelial growth factor receptor 1	target
Fostamatinib	Receptor-type tyrosine-protein kinase FLT3	target
Fostamatinib	Vascular endothelial growth factor receptor 3	target
Fostamatinib	Serine/threonine-protein kinase mTOR	target
Fostamatinib	Tyrosine-protein kinase FRK	target
Fostamatinib	Tyrosine-protein kinase Fyn	target
Fostamatinib	Cyclin-G-associated kinase	target
Fostamatinib	Glycogen synthase kinase-3 alpha	target
Fostamatinib	Glycogen synthase kinase-3 beta	target
Fostamatinib	Tyrosine-protein kinase HCK	target
Fostamatinib	Homeodomain-interacting protein kinase 2	target
Fostamatinib	Homeodomain-interacting protein kinase 3	target
Fostamatinib	Serine/threonine-protein kinase ICK	target
Fostamatinib	Inhibitor of nuclear factor kappa-B kinase subunit beta	target
Fostamatinib	Inhibitor of nuclear factor kappa-B kinase subunit epsilon	target
Fostamatinib	Insulin receptor	target
Fostamatinib	Insulin receptor-related protein	target
Fostamatinib	Interleukin-1 receptor-associated kinase 1	target
Fostamatinib	Interleukin-1 receptor-associated kinase 3	target
Fostamatinib	Interleukin-1 receptor-associated kinase 4	target
Fostamatinib	Tyrosine-protein kinase ITK/TSK	target
Fostamatinib	Tyrosine-protein kinase JAK2	target
Fostamatinib	Tyrosine-protein kinase JAK3	target
Fostamatinib	Vascular endothelial growth factor receptor 2	target
Fostamatinib	Serine/threonine-protein kinase SIK3	target
Fostamatinib	Mast/stem cell growth factor receptor Kit	target
Fostamatinib	Serine/threonine-protein kinase LATS1	target
Fostamatinib	Tyrosine-protein kinase Lck	target
Fostamatinib	LIM domain kinase 1	target
Fostamatinib	LIM domain kinase 2	target
Fostamatinib	Leucine-rich repeat serine/threonine-protein kinase 2	target
Fostamatinib	Leukocyte tyrosine kinase receptor	target
Fostamatinib	Tyrosine-protein kinase Lyn	target
Fostamatinib	Dual specificity mitogen-activated protein kinase kinase 2	target
Fostamatinib	Dual specificity mitogen-activated protein kinase kinase 3	target
Fostamatinib	Dual specificity mitogen-activated protein kinase kinase 5	target
Fostamatinib	Dual specificity mitogen-activated protein kinase kinase 6	target
Fostamatinib	Mitogen-activated protein kinase kinase kinase 1	target
Fostamatinib	Mitogen-activated protein kinase kinase kinase 10	target
Fostamatinib	Mitogen-activated protein kinase kinase kinase 11	target
Fostamatinib	Mitogen-activated protein kinase kinase kinase 12	target
Fostamatinib	Mitogen-activated protein kinase kinase kinase 13	target
Fostamatinib	Mitogen-activated protein kinase kinase kinase 15	target
Fostamatinib	Mitogen-activated protein kinase kinase kinase 2	target
Fostamatinib	Mitogen-activated protein kinase kinase kinase 3	target
Fostamatinib	Mitogen-activated protein kinase kinase kinase 4	target
Fostamatinib	Mitogen-activated protein kinase kinase kinase 6	target
Fostamatinib	Mitogen-activated protein kinase kinase kinase 9	target
Fostamatinib	Mitogen-activated protein kinase kinase kinase kinase 1	target
Fostamatinib	Mitogen-activated protein kinase kinase kinase kinase 2	target
Fostamatinib	Mitogen-activated protein kinase kinase kinase kinase 3	target
Fostamatinib	Mitogen-activated protein kinase kinase kinase kinase 4	target
Fostamatinib	Mitogen-activated protein kinase kinase kinase kinase 5	target
Fostamatinib	Mitogen-activated protein kinase 10	target
Fostamatinib	Mitogen-activated protein kinase 13	target
Fostamatinib	Mitogen-activated protein kinase 14	target
Fostamatinib	Mitogen-activated protein kinase 15	target
Fostamatinib	Mitogen-activated protein kinase 4	target
Fostamatinib	Mitogen-activated protein kinase 7	target
Fostamatinib	Mitogen-activated protein kinase 9	target
Fostamatinib	MAP kinase-activated protein kinase 5	target
Fostamatinib	Serine/threonine-protein kinase MARK1	target
Fostamatinib	Serine/threonine-protein kinase MARK2	target
Fostamatinib	MAP/microtubule affinity-regulating kinase 3	target
Fostamatinib	MAP/microtubule affinity-regulating kinase 4	target
Fostamatinib	CLIP-associating protein 1	target
Fostamatinib	Microtubule-associated serine/threonine-protein kinase 1	target
Fostamatinib	Megakaryocyte-associated tyrosine-protein kinase	target
Fostamatinib	Maternal embryonic leucine zipper kinase	target
Fostamatinib	Tyrosine-protein kinase Mer	target
Fostamatinib	Misshapen-like kinase 1	target
Fostamatinib	MAP kinase-interacting serine/threonine-protein kinase 1	target
Fostamatinib	MAP kinase-interacting serine/threonine-protein kinase 2	target
Fostamatinib	Macrophage-stimulating protein receptor	target
Fostamatinib	Muscle, skeletal receptor tyrosine-protein kinase	target
Fostamatinib	Myosin light chain kinase, smooth muscle	target
Fostamatinib	Myosin light chain kinase 2, skeletal/cardiac muscle	target
Fostamatinib	Myosin light chain kinase 3	target
Fostamatinib	Myosin light chain kinase family member 4	target
Fostamatinib	Myosin-IIIa	target
Fostamatinib	Serine/threonine-protein kinase Nek1	target
Fostamatinib	Serine/threonine-protein kinase Nek11	target
Fostamatinib	Serine/threonine-protein kinase Nek2	target
Fostamatinib	Serine/threonine-protein kinase Nek3	target
Fostamatinib	Serine/threonine-protein kinase Nek4	target
Fostamatinib	Serine/threonine-protein kinase Nek5	target
Fostamatinib	Serine/threonine-protein kinase Nek9	target
Fostamatinib	High affinity nerve growth factor receptor	target
Fostamatinib	BDNF/NT-3 growth factors receptor	target
Fostamatinib	NT-3 growth factor receptor	target
Fostamatinib	NUAK family SNF1-like kinase 1	target
Fostamatinib	NUAK family SNF1-like kinase 2	target
Fostamatinib	Serine/threonine-protein kinase OSR1	target
Fostamatinib	Serine/threonine-protein kinase PAK 1	target
Fostamatinib	Serine/threonine-protein kinase PAK 2	target
Fostamatinib	Serine/threonine-protein kinase PAK 3	target
Fostamatinib	Serine/threonine-protein kinase PAK 4	target
Fostamatinib	Serine/threonine-protein kinase PAK 6	target
Fostamatinib	Serine/threonine-protein kinase PAK 5	target
Fostamatinib	Cyclin-dependent kinase 16	target
Fostamatinib	Cyclin-dependent kinase 17	target
Fostamatinib	Platelet-derived growth factor receptor alpha	target
Fostamatinib	Platelet-derived growth factor receptor beta	target
Fostamatinib	3-phosphoinositide-dependent protein kinase 1	target
Fostamatinib	Cyclin-dependent kinase 15	target
Fostamatinib	Phosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoform	target
Fostamatinib	Phosphatidylinositol 4-kinase beta	target
Fostamatinib	Phosphatidylinositol 4-phosphate 3-kinase C2 domain-containing subunit beta	target
Fostamatinib	Phosphatidylinositol 3-kinase C2 domain-containing subunit gamma	target
Fostamatinib	Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform	target
Fostamatinib	Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform	target
Fostamatinib	Serine/threonine-protein kinase pim-1	target
Fostamatinib	Serine/threonine-protein kinase pim-3	target
Fostamatinib	Phosphatidylinositol 5-phosphate 4-kinase type-2 beta	target
Fostamatinib	Phosphatidylinositol 5-phosphate 4-kinase type-2 gamma	target
Fostamatinib	Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase	target
Fostamatinib	Serine/threonine-protein kinase N1	target
Fostamatinib	Serine/threonine-protein kinase N2	target
Fostamatinib	Serine/threonine-protein kinase PLK1	target
Fostamatinib	Serine/threonine-protein kinase PLK2	target
Fostamatinib	Serine/threonine-protein kinase PLK3	target
Fostamatinib	Serine/threonine-protein kinase PLK4	target
Fostamatinib	5'-AMP-activated protein kinase catalytic subunit alpha-1	target
Fostamatinib	5'-AMP-activated protein kinase	target
Fostamatinib	cAMP-dependent protein kinase catalytic subunit beta	target
Fostamatinib	Protein kinase C delta type	target
Fostamatinib	Protein kinase C epsilon type	target
Fostamatinib	Protein kinase C gamma type	target
Fostamatinib	Protein kinase C iota type	target
Fostamatinib	Protein kinase C theta type	target
Fostamatinib	Serine/threonine-protein kinase D1	target
Fostamatinib	cGMP-dependent protein kinase 2	target
Fostamatinib	Serine/threonine-protein kinase PRP4 homolog	target
Fostamatinib	Focal adhesion kinase 1	target
Fostamatinib	Protein-tyrosine kinase 2-beta	target
Fostamatinib	Protein-tyrosine kinase 6	target
Fostamatinib	RAF proto-oncogene serine/threonine-protein kinase	target
Fostamatinib	Proto-oncogene tyrosine-protein kinase receptor Ret	target
Fostamatinib	Serine/threonine-protein kinase RIO1	target
Fostamatinib	Serine/threonine-protein kinase RIO2	target
Fostamatinib	Serine/threonine-protein kinase RIO3	target
Fostamatinib	Receptor-interacting serine/threonine-protein kinase 1	target
Fostamatinib	Receptor-interacting serine/threonine-protein kinase 2	target
Fostamatinib	Receptor-interacting serine/threonine-protein kinase 4	target
Fostamatinib	Rho-associated protein kinase 2	target
Fostamatinib	Proto-oncogene tyrosine-protein kinase ROS	target
Fostamatinib	Ribosomal protein S6 kinase alpha-1	target
Fostamatinib	Ribosomal protein S6 kinase alpha-3	target
Fostamatinib	Serine/threonine-protein kinase SBK1	target
Fostamatinib	Uncharacterized serine/threonine-protein kinase SBK3	target
Fostamatinib	Serine/threonine-protein kinase Sgk3	target
Fostamatinib	Serine/threonine-protein kinase SIK1	target
Fostamatinib	Serine/threonine-protein kinase SIK2	target
Fostamatinib	STE20-like serine/threonine-protein kinase	target
Fostamatinib	SNF-related serine/threonine-protein kinase	target
Fostamatinib	Proto-oncogene tyrosine-protein kinase Src	target
Fostamatinib	Tyrosine-protein kinase Srms	target
Fostamatinib	Serine/threonine-protein kinase 10	target
Fostamatinib	Serine/threonine-protein kinase 16	target
Fostamatinib	Serine/threonine-protein kinase 17A	target
Fostamatinib	Serine/threonine-protein kinase 17B	target
Fostamatinib	Serine/threonine-protein kinase 32A	target
Fostamatinib	Cytochrome P450 3A4	enzyme
Fostamatinib	Broad substrate specificity ATP-binding cassette transporter ABCG2	transporter
Fostamatinib	ATP-binding cassette sub-family B member 5	transporter
Fostamatinib	UDP-glucuronosyltransferase 1A9	enzyme
Udenafil	cGMP-specific 3',5'-cyclic phosphodiesterase	target
Udenafil	Cytochrome P450 3A4	enzyme
Udenafil	Cytochrome P450 3A5	enzyme
Prednisone	Glucocorticoid receptor	target
Prednisone	Cytochrome P450 3A4	enzyme
Prednisone	ATP-dependent translocase ABCB1	transporter
Prednisone	Solute carrier organic anion transporter family member 1A2	transporter
Prednisone	Cytochrome P450 2C19	enzyme
Prednisone	Albumin	carrier
Prednisone	Cytochrome P450 3A5	enzyme
Prednisone	Corticosteroid-binding globulin	carrier
Prednisone	Cytochrome P450 3A Subfamily	enzyme
Prednisone	Cytochrome P450 2A6	enzyme
Prednisone	Cytochrome P450 1B1	enzyme
Prednisone	Cytochrome P450 2B6	enzyme
Prednisone	Cytochrome P450 2C8	enzyme
Prednisone	Cytochrome P450 2C9	enzyme
Prednisone	11-beta-hydroxysteroid dehydrogenase 1	enzyme
Fluticasone	Cytochrome P450 3A4	enzyme
Fluticasone	Cytochrome P450 2C8	enzyme
Fluticasone	ATP-dependent translocase ABCB1	carrier
Fluticasone	Solute carrier organic anion transporter family member 1B1	carrier
Fluticasone	ATP-dependent translocase ABCB1	transporter
Fluticasone	Solute carrier organic anion transporter family member 1B1	transporter
Fluticasone	Glucocorticoid receptor	target
Fluticasone	Corticosteroid-binding globulin	carrier
Fluticasone	Cytochrome P450 3A5	enzyme
Fluticasone	Cytochrome P450 3A7	enzyme
Fluticasone	Progesterone receptor	target
Fluticasone	Cytosolic phospholipase A2	target
Fluticasone	Mineralocorticoid receptor	target
Pantoprazole	Potassium-transporting ATPase alpha chain 1	target
Pantoprazole	Cytochrome P450 2C19	enzyme
Pantoprazole	Cytochrome P450 3A4	enzyme
Pantoprazole	ATP-dependent translocase ABCB1	transporter
Pantoprazole	Broad substrate specificity ATP-binding cassette transporter ABCG2	transporter
Pantoprazole	Organic anion transporter 3	transporter
Pantoprazole	N(G),N(G)-dimethylarginine dimethylaminohydrolase 1	target
Pantoprazole	Potassium-transporting ATPase subunit beta	target
Lansoprazole	Potassium-transporting ATPase alpha chain 1	target
Lansoprazole	Cytochrome P450 2C19	enzyme
Lansoprazole	Cytochrome P450 2C9	enzyme
Lansoprazole	Cytochrome P450 3A4	enzyme
Lansoprazole	ATP-dependent translocase ABCB1	transporter
Lansoprazole	Broad substrate specificity ATP-binding cassette transporter ABCG2	transporter
Lansoprazole	Cytochrome P450 1A1	enzyme
Lansoprazole	Cytochrome P450 1B1	enzyme
Lansoprazole	Cytochrome P450 2C18	enzyme
Lansoprazole	Cytochrome P450 2C8	enzyme
Lansoprazole	Cytochrome P450 2D6	enzyme
Lansoprazole	Microtubule-associated protein tau	target
Lansoprazole	Organic anion transporter 3	transporter
Lansoprazole	Solute carrier family 22 member 1	transporter
Lansoprazole	Solute carrier family 22 member 2	transporter
Lansoprazole	Solute carrier family 22 member 3	transporter
Dexlansoprazole	Potassium-transporting ATPase alpha chain 1	target
Dexlansoprazole	Cytochrome P450 2C19	enzyme
Dexlansoprazole	Cytochrome P450 3A4	enzyme
Dexlansoprazole	Potassium-transporting ATPase subunit beta	target
Dexlansoprazole	N(G),N(G)-dimethylarginine dimethylaminohydrolase 1	target
Rabeprazole	Potassium-transporting ATPase alpha chain 1	target
Rabeprazole	Cytochrome P450 3A4	enzyme
Rabeprazole	Cytochrome P450 2C19	enzyme
Rabeprazole	Broad substrate specificity ATP-binding cassette transporter ABCG2	transporter
Rabeprazole	Cytochrome P450 1A1	enzyme
Rabeprazole	Cytochrome P450 1A2	enzyme
Rabeprazole	Cytochrome P450 2C9	enzyme
Rabeprazole	Cytochrome P450 2D6	enzyme
Rabeprazole	Cytochrome P450 2C8	enzyme
Lacidipine	Cytochrome P450 3A4	enzyme
Lacidipine	Albumin	carrier
Lacidipine	Alpha-1-acid glycoprotein 1	carrier
Lacidipine	Voltage-dependent L-type calcium channel	target
Allylestrenol	Progesterone receptor	target
Allylestrenol	Estrogen receptor	target
Allylestrenol	Sodium- and chloride-dependent glycine transporter 1	target
Betamethasone	Glucocorticoid receptor	target
Betamethasone	Cytochrome P450 3A4	enzyme
Betamethasone	ATP-dependent translocase ABCB1	transporter
Betamethasone	Aromatase	enzyme
Betamethasone	Cytochrome P450 3A5	enzyme
Betamethasone	Cytochrome P450 3A7	enzyme
Betamethasone	Cytochrome P450 2A6	enzyme
Betamethasone	Cytochrome P450 1B1	enzyme
Betamethasone	Cytochrome P450 2B6	enzyme
Betamethasone	Cytochrome P450 2C8	enzyme
Betamethasone	Cytochrome P450 2C9	enzyme
Betamethasone	Cytochrome P450 2C19	enzyme
Betamethasone	Albumin	carrier
Betamethasone	Corticosteroid-binding globulin	carrier
Ciclesonide	Corticosteroid-binding globulin	carrier
Ciclesonide	Cytochrome P450 3A4	enzyme
Ciclesonide	Cytochrome P450 2D6	enzyme
Ciclesonide	Glucocorticoid receptor	target
Ciclesonide	Liver carboxylesterase 1	enzyme
Ciclesonide	Corticosteroid-binding globulin	target
Cortisone acetate	Glucocorticoid receptor	target
Cortisone acetate	Cytochrome P450 3A4	enzyme
Cortisone acetate	Cytochrome P450 3A5	enzyme
Cortisone acetate	Annexin A1	target
Cortisone acetate	Corticosteroid-binding globulin	carrier
Cortisone acetate	Albumin	carrier
Cortisone acetate	Solute carrier organic anion transporter family member 1A2	transporter
Cortisone acetate	ATP-dependent translocase ABCB1	transporter
Cortisone acetate	Organic anion transporter 3	transporter
Cortisone acetate	Steroid hormone receptor ERR1	target
Cortisone acetate	Steroid hormone receptor ERR2	target
Cortisone acetate	Estrogen-related receptor gamma	target
Deflazacort	Cytochrome P450 3A4	enzyme
Deflazacort	Glucocorticoid receptor	target
Deflazacort	Cytochrome P450 3A5	enzyme
Dienogest	Cytochrome P450 3A4	enzyme
Dienogest	Progesterone receptor	target
Dienogest	Androgen receptor	target
Dexamethasone	Glucocorticoid receptor	target
Dexamethasone	Annexin A1	target
Dexamethasone	Nitric oxide synthase, inducible	target
Dexamethasone	Nuclear receptor subfamily 0 group B member 1	target
Dexamethasone	Cytochrome P450 3A4	enzyme
Dexamethasone	Cytochrome P450 3A5	enzyme
Dexamethasone	Cytochrome P450 3A7	enzyme
Dexamethasone	Bile salt export pump	transporter
Dexamethasone	ATP-dependent translocase ABCB1	transporter
Dexamethasone	ATP-binding cassette sub-family C member 2	transporter
Dexamethasone	Solute carrier organic anion transporter family member 1A2	transporter
Dexamethasone	Broad substrate specificity ATP-binding cassette transporter ABCG2	transporter
Dexamethasone	Steroid 17-alpha-hydroxylase/17,20 lyase	enzyme
Dexamethasone	Cytochrome P450 1A1	enzyme
Dexamethasone	Cytochrome P450 2A6	enzyme
Dexamethasone	Cytochrome P450 2B6	enzyme
Dexamethasone	Cytochrome P450 2C19	enzyme
Dexamethasone	Cytochrome P450 2C8	enzyme
Dexamethasone	Cytochrome P450 2E1	enzyme
Dexamethasone	Cytochrome P450 3A43	enzyme
Dexamethasone	Cytochrome P450 4A11	enzyme
Dexamethasone	Nuclear receptor subfamily 1 group I member 2	target
Dexamethasone	Cytochrome P450 11B1, mitochondrial	enzyme
Dexamethasone	Albumin	carrier
Dexamethasone	11-beta-hydroxysteroid dehydrogenase type 2	enzyme
Dexamethasone	11-beta-hydroxysteroid dehydrogenase 1	enzyme
Dexamethasone	Organic anion transporter 3	transporter
Dexamethasone isonicotinate	Cytochrome P450 3A4	enzyme
Dexamethasone isonicotinate	Cytochrome P450 3A5	enzyme
Drospirenone	Progesterone receptor	target
Drospirenone	Mineralocorticoid receptor	target
Drospirenone	Androgen receptor	target
Drospirenone	Prostaglandin G/H synthase 2	enzyme
Drospirenone	Serum paraoxonase/arylesterase 1	enzyme
Drospirenone	Glucocorticoid receptor	target
Drospirenone	Cytochrome P450 3A4	enzyme
Estrone	Estrogen receptor	target
Estrone	Cytochrome P450 1A2	enzyme
Estrone	Cytochrome P450 1A1	enzyme
Estrone	Albumin	carrier
Estrone	Solute carrier organic anion transporter family member 2B1	transporter
Estrone	ATP-dependent translocase ABCB1	transporter
Estrone	Solute carrier organic anion transporter family member 1A2	transporter
Estrone	Broad substrate specificity ATP-binding cassette transporter ABCG2	transporter
Estrone	Solute carrier organic anion transporter family member 1B1	transporter
Estrone	Cytochrome P450 3A4	enzyme
Estrone	Cytochrome P450 1B1	enzyme
Estrone	Cytochrome P450 2B6	enzyme
Estrone	Cytochrome P450 2C9	enzyme
Estrone	Cytochrome P450 2E1	enzyme
Estrone	Cytochrome P450 3A5	enzyme
Estrone	Estrogen receptor beta	target
Estrone	Androgen receptor	target
Estrone	Aromatase	target
Estrone	Sex hormone-binding globulin	target
Estrone	Organic anion transporter 3	transporter
Estrone sulfate	Cytochrome P450 1A2	enzyme
Estrone sulfate	Cytochrome P450 3A4	enzyme
Estrone sulfate	Estrogen receptor	target
Estrone sulfate	Estrogen receptor beta	target
Estrone sulfate	Sex hormone-binding globulin	carrier
Estrone sulfate	Albumin	carrier
Estrone sulfate	Cytochrome P450 2C9	enzyme
Estrone sulfate	Multidrug and toxin extrusion protein 1	transporter
Estrone sulfate	Multidrug and toxin extrusion protein 2	transporter
Estrone sulfate	Hepatic sodium/bile acid cotransporter	transporter
Etonogestrel	Progesterone receptor	target
Etonogestrel	Cytochrome P450 3A4	enzyme
Etonogestrel	Albumin	carrier
Etonogestrel	Sex hormone-binding globulin	carrier
Flunisolide	Corticosteroid-binding globulin	carrier
Flunisolide	Glucocorticoid receptor	target
Flunisolide	Cytochrome P450 3A4	enzyme
Fluocortolone	Cytochrome P450 3A4	enzyme
Fluocortolone	Cytochrome P450 3A5	enzyme
Fluorometholone	Corticosteroid-binding globulin	carrier
Fluorometholone	Cytochrome P450 3A4	enzyme
Fluorometholone	Glucocorticoid receptor	target
Fluorometholone	Cytochrome P450 3A5	enzyme
Fluticasone furoate	Cytochrome P450 3A4	enzyme
Fluticasone furoate	Glucocorticoid receptor	target
Fluticasone furoate	ATP-dependent translocase ABCB1	transporter
Fluticasone furoate	Cytochrome P450 2C8	enzyme
Fluticasone furoate	Solute carrier organic anion transporter family member 1B1	transporter
Fluticasone furoate	Corticosteroid-binding globulin	carrier
Fluticasone furoate	Cytochrome P450 3A5	enzyme
Fluticasone furoate	Cytochrome P450 3A7	enzyme
Fluticasone furoate	Progesterone receptor	target
Fluticasone furoate	Mineralocorticoid receptor	target
Fluticasone furoate	Albumin	carrier
Fluticasone furoate	Alpha-1-acid glycoprotein 1	carrier
Fluticasone propionate	Corticosteroid-binding globulin	carrier
Fluticasone propionate	Cytosolic phospholipase A2	target
Fluticasone propionate	Glucocorticoid receptor	target
Fluticasone propionate	Cytochrome P450 3A4	enzyme
Fluticasone propionate	Progesterone receptor	target
Fluticasone propionate	Mineralocorticoid receptor	target
Fluticasone propionate	Cytochrome P450 3A5	enzyme
Fluticasone propionate	Cytochrome P450 3A7	enzyme
Fluticasone propionate	Cytochrome P450 2C8	enzyme
Fluticasone propionate	Solute carrier organic anion transporter family member 1B1	carrier
Fluticasone propionate	ATP-dependent translocase ABCB1	transporter
Fluticasone propionate	Solute carrier organic anion transporter family member 1B1	transporter
Hydrocortisone	Annexin A1	target
Hydrocortisone	Glucocorticoid receptor	target
Hydrocortisone	Sex hormone-binding globulin	carrier
Hydrocortisone	Cytochrome P450 3A4	enzyme
Hydrocortisone	Cytochrome P450 3A5	enzyme
Hydrocortisone	Cytochrome P450 3A7	enzyme
Hydrocortisone	ATP-dependent translocase ABCB1	transporter
Hydrocortisone	Solute carrier organic anion transporter family member 1A2	transporter
Hydrocortisone	Cytochrome P450 11B1, mitochondrial	enzyme
Hydrocortisone	Cytochrome P450 11B2, mitochondrial	enzyme
Hydrocortisone	Cytochrome P450 2C8	enzyme
Hydrocortisone	Corticosteroid-binding globulin	carrier
Hydrocortisone	Organic anion transporter 3	transporter
Hydrocortisone	Aldo-keto reductase family 1 member D1	enzyme
Hydrocortisone	3-oxo-5-alpha-steroid 4-dehydrogenase 2	enzyme
Hydrocortisone	11-beta-hydroxysteroid dehydrogenase type 2	enzyme
Hydrocortisone	11-beta-hydroxysteroid dehydrogenase 1	enzyme
Hydrocortisone	Cytochrome P450 2A6	enzyme
Hydrocortisone	Cytochrome P450 1B1	enzyme
Hydrocortisone	Cytochrome P450 2B6	enzyme
Hydrocortisone	Cytochrome P450 2C9	enzyme
Hydrocortisone	Cytochrome P450 2C19	enzyme
Hydrocortisone aceponate	Annexin A1	target
Hydrocortisone aceponate	Glucocorticoid receptor	target
Hydrocortisone aceponate	Sex hormone-binding globulin	carrier
Hydrocortisone aceponate	Cytochrome P450 3A4	enzyme
Hydrocortisone aceponate	Cytochrome P450 3A5	enzyme
Hydrocortisone aceponate	Cytochrome P450 3A7	enzyme
Hydrocortisone aceponate	ATP-dependent translocase ABCB1	transporter
Hydrocortisone aceponate	Solute carrier organic anion transporter family member 1A2	transporter
Hydrocortisone aceponate	Broad substrate specificity ATP-binding cassette transporter ABCG2	transporter
Hydrocortisone aceponate	Cytochrome P450 2C8	enzyme
Hydrocortisone aceponate	Corticosteroid-binding globulin	carrier
Hydrocortisone aceponate	11-beta-hydroxysteroid dehydrogenase type 2	target
Hydrocortisone aceponate	3 beta-hydroxysteroid dehydrogenase/Delta 5-->4-isomerase type 1	target
Hydrocortisone aceponate	Organic anion transporter 3	transporter
Hydrocortisone acetate	Annexin A1	target
Hydrocortisone acetate	Glucocorticoid receptor	target
Hydrocortisone acetate	Sex hormone-binding globulin	carrier
Hydrocortisone acetate	Cytochrome P450 3A4	enzyme
Hydrocortisone acetate	Cytochrome P450 3A5	enzyme
Hydrocortisone acetate	Cytochrome P450 3A7	enzyme
Hydrocortisone acetate	ATP-dependent translocase ABCB1	transporter
Hydrocortisone acetate	Solute carrier organic anion transporter family member 1A2	transporter
Hydrocortisone acetate	Broad substrate specificity ATP-binding cassette transporter ABCG2	transporter
Hydrocortisone acetate	Cytochrome P450 11B1, mitochondrial	enzyme
Hydrocortisone acetate	Cytochrome P450 11B2, mitochondrial	enzyme
Hydrocortisone acetate	Cytochrome P450 2C8	enzyme
Hydrocortisone acetate	Corticosteroid-binding globulin	carrier
Hydrocortisone acetate	11-beta-hydroxysteroid dehydrogenase type 2	target
Hydrocortisone acetate	3 beta-hydroxysteroid dehydrogenase/Delta 5-->4-isomerase type 1	target
Hydrocortisone acetate	Organic anion transporter 3	transporter
Hydrocortisone butyrate	Annexin A1	target
Hydrocortisone butyrate	Glucocorticoid receptor	target
Hydrocortisone butyrate	Sex hormone-binding globulin	carrier
Hydrocortisone butyrate	Cytochrome P450 3A4	enzyme
Hydrocortisone butyrate	Cytochrome P450 3A5	enzyme
Hydrocortisone butyrate	Cytochrome P450 3A7	enzyme
Hydrocortisone butyrate	ATP-dependent translocase ABCB1	transporter
Hydrocortisone butyrate	Solute carrier organic anion transporter family member 1A2	transporter
Hydrocortisone butyrate	Broad substrate specificity ATP-binding cassette transporter ABCG2	transporter
Hydrocortisone butyrate	Cytochrome P450 11B1, mitochondrial	enzyme
Hydrocortisone butyrate	Cytochrome P450 11B2, mitochondrial	enzyme
Hydrocortisone butyrate	Cytochrome P450 2C8	enzyme
Hydrocortisone butyrate	Corticosteroid-binding globulin	carrier
Hydrocortisone butyrate	11-beta-hydroxysteroid dehydrogenase type 2	target
Hydrocortisone butyrate	3 beta-hydroxysteroid dehydrogenase/Delta 5-->4-isomerase type 1	target
Hydrocortisone butyrate	Organic anion transporter 3	transporter
Hydrocortisone cypionate	Annexin A1	target
Hydrocortisone cypionate	Glucocorticoid receptor	target
Hydrocortisone cypionate	Sex hormone-binding globulin	carrier
Hydrocortisone cypionate	Cytochrome P450 3A4	enzyme
Hydrocortisone cypionate	Cytochrome P450 3A5	enzyme
Hydrocortisone cypionate	Cytochrome P450 3A7	enzyme
Hydrocortisone cypionate	ATP-dependent translocase ABCB1	transporter
Hydrocortisone cypionate	Solute carrier organic anion transporter family member 1A2	transporter
Hydrocortisone cypionate	Broad substrate specificity ATP-binding cassette transporter ABCG2	transporter
Hydrocortisone cypionate	Cytochrome P450 2C8	enzyme
Hydrocortisone cypionate	Corticosteroid-binding globulin	carrier
Hydrocortisone cypionate	11-beta-hydroxysteroid dehydrogenase type 2	target
Hydrocortisone cypionate	3 beta-hydroxysteroid dehydrogenase/Delta 5-->4-isomerase type 1	target
Hydrocortisone cypionate	Organic anion transporter 3	transporter
Hydrocortisone phosphate	Annexin A1	target
Hydrocortisone phosphate	Glucocorticoid receptor	target
Hydrocortisone phosphate	Sex hormone-binding globulin	carrier
Hydrocortisone phosphate	Cytochrome P450 3A4	enzyme
Hydrocortisone phosphate	Cytochrome P450 3A5	enzyme
Hydrocortisone phosphate	Cytochrome P450 3A7	enzyme
Hydrocortisone phosphate	ATP-dependent translocase ABCB1	transporter
Hydrocortisone phosphate	Solute carrier organic anion transporter family member 1A2	transporter
Hydrocortisone phosphate	Broad substrate specificity ATP-binding cassette transporter ABCG2	transporter
Hydrocortisone phosphate	Cytochrome P450 2C8	enzyme
Hydrocortisone phosphate	Corticosteroid-binding globulin	carrier
Hydrocortisone phosphate	11-beta-hydroxysteroid dehydrogenase type 2	target
Hydrocortisone phosphate	3 beta-hydroxysteroid dehydrogenase/Delta 5-->4-isomerase type 1	target
Hydrocortisone phosphate	Organic anion transporter 3	transporter
Hydrocortisone probutate	Annexin A1	target
Hydrocortisone probutate	Glucocorticoid receptor	target
Hydrocortisone probutate	Sex hormone-binding globulin	carrier
Hydrocortisone probutate	Cytochrome P450 3A4	enzyme
Hydrocortisone probutate	Cytochrome P450 3A5	enzyme
Hydrocortisone probutate	Cytochrome P450 3A7	enzyme
Hydrocortisone probutate	ATP-dependent translocase ABCB1	transporter
Hydrocortisone probutate	Solute carrier organic anion transporter family member 1A2	transporter
Hydrocortisone probutate	Broad substrate specificity ATP-binding cassette transporter ABCG2	transporter
Hydrocortisone probutate	Cytochrome P450 11B1, mitochondrial	enzyme
Hydrocortisone probutate	Cytochrome P450 11B2, mitochondrial	enzyme
Hydrocortisone probutate	Cytochrome P450 2C8	enzyme
Hydrocortisone probutate	Corticosteroid-binding globulin	carrier
Hydrocortisone probutate	11-beta-hydroxysteroid dehydrogenase type 2	target
Hydrocortisone probutate	3 beta-hydroxysteroid dehydrogenase/Delta 5-->4-isomerase type 1	target
Hydrocortisone probutate	Organic anion transporter 3	transporter
Hydrocortisone valerate	Annexin A1	target
Hydrocortisone valerate	Glucocorticoid receptor	target
Hydrocortisone valerate	Sex hormone-binding globulin	carrier
Hydrocortisone valerate	Cytochrome P450 3A4	enzyme
Hydrocortisone valerate	Cytochrome P450 3A5	enzyme
Hydrocortisone valerate	Cytochrome P450 3A7	enzyme
Hydrocortisone valerate	ATP-dependent translocase ABCB1	transporter
Hydrocortisone valerate	Solute carrier organic anion transporter family member 1A2	transporter
Hydrocortisone valerate	Broad substrate specificity ATP-binding cassette transporter ABCG2	transporter
Hydrocortisone valerate	Cytochrome P450 11B1, mitochondrial	enzyme
Hydrocortisone valerate	Cytochrome P450 11B2, mitochondrial	enzyme
Hydrocortisone valerate	Cytochrome P450 2C8	enzyme
Hydrocortisone valerate	Corticosteroid-binding globulin	carrier
Hydrocortisone valerate	11-beta-hydroxysteroid dehydrogenase type 2	target
Hydrocortisone valerate	3 beta-hydroxysteroid dehydrogenase/Delta 5-->4-isomerase type 1	target
Hydrocortisone valerate	Organic anion transporter 3	transporter
Hydroxyprogesterone caproate	Progesterone receptor	target
Hydroxyprogesterone caproate	Cytochrome P450 3A4	enzyme
Hydroxyprogesterone caproate	Cytochrome P450 3A5	enzyme
Hydroxyprogesterone caproate	Cytochrome P450 2C19	enzyme
Levonorgestrel	Progesterone receptor	target
Levonorgestrel	Estrogen receptor	target
Levonorgestrel	3-oxo-5-alpha-steroid 4-dehydrogenase 1	target
Levonorgestrel	Cytochrome P450 3A4	enzyme
Levonorgestrel	Androgen receptor	target
Levonorgestrel	Sex hormone-binding globulin	target
Levonorgestrel	Glucocorticoid receptor	target
Levonorgestrel	Cytochrome P450 3A5	enzyme
Medroxyprogesterone acetate	Progesterone receptor	target
Medroxyprogesterone acetate	Estrogen receptor	target
Medroxyprogesterone acetate	Cytochrome P450 3A4	enzyme
Medroxyprogesterone acetate	Cytochrome P450 2C8	enzyme
Medroxyprogesterone acetate	3 beta-hydroxysteroid dehydrogenase/Delta 5-->4-isomerase type 2	enzyme
Medroxyprogesterone acetate	Cytochrome P450 2C9	enzyme
Medroxyprogesterone acetate	Cytochrome P450 3A1	enzyme
Medroxyprogesterone acetate	Albumin	carrier
Medroxyprogesterone acetate	ATP-dependent translocase ABCB1	target
Medroxyprogesterone acetate	GABA(A) Receptor	target
Medroxyprogesterone acetate	ATP-dependent translocase ABCB1	transporter
Methylprednisolone	Glucocorticoid receptor	target
Methylprednisolone	Cytochrome P450 3A4	enzyme
Methylprednisolone	ATP-dependent translocase ABCB1	transporter
Methylprednisolone	Cytochrome P450 3A Subfamily	enzyme
Methylprednisolone	Cytochrome P450 2A6	enzyme
Methylprednisolone	Cytochrome P450 1B1	enzyme
Methylprednisolone	Cytochrome P450 2B6	enzyme
Methylprednisolone	Cytochrome P450 2C8	enzyme
Methylprednisolone	Cytochrome P450 2C9	enzyme
Methylprednisolone	Cytochrome P450 2C19	enzyme
Methylprednisolone	Annexin A1	target
Methylprednisolone	20-ketosteroid reductase (20-hydroxysteroid dehydrogenase)	enzyme
Methylprednisolone	11beta-hydroxysteroid dehydrogenase	enzyme
Methylprednisolone	Albumin	carrier
Norethisterone	Progesterone receptor	target
Norethisterone	ATP-dependent translocase ABCB1	transporter
Norethisterone	Cytochrome P450 2C19	enzyme
Norethisterone	Albumin	carrier
Norethisterone	Sex hormone-binding globulin	carrier
Norethisterone	Aldo-keto reductase family 1 member C4	enzyme
Norethisterone	3 beta-hydroxysteroid dehydrogenase/Delta 5-->4-isomerase type 2	enzyme
Norethisterone	3-oxo-5-alpha-steroid 4-dehydrogenase	enzyme
Norethisterone	Aldo-keto reductase family 1 member D1	enzyme
Norethisterone	Cytochrome P450 3A4	enzyme
Norethisterone	Cytochrome P450 1A2	enzyme
Norethisterone	Cytochrome P450 2A6	enzyme
Norethisterone	Glucocorticoid receptor	target
Norethisterone	Androgen receptor	target
Norgestimate	Progesterone receptor	target
Norgestimate	Estrogen receptor	target
Norgestimate	ATP-binding cassette sub-family C member 2	transporter
Norgestimate	Cytochrome P450 3A4	enzyme
Norgestimate	Androgen receptor	target
Norgestimate	Cytochrome P450 2B6	enzyme
Norgestimate	Cytochrome P450 2C9	enzyme
Norgestimate	UDP-glucuronosyltransferase 1A1	enzyme
Norgestimate	Albumin	carrier
Norgestimate	Sex hormone-binding globulin	carrier
Norgestimate	ATP-dependent translocase ABCB1	transporter
Norgestrel	Progesterone receptor	target
Norgestrel	3-oxo-5-alpha-steroid 4-dehydrogenase 1	target
Norgestrel	Androgen receptor	target
Norgestrel	Cytochrome P450 3A4	enzyme
Norgestrel	Aromatase	enzyme
Paramethasone	Corticosteroid-binding globulin	carrier
Paramethasone	Glucocorticoid receptor	target
Paramethasone	Cytochrome P450 3A4	enzyme
Paramethasone	Cytochrome P450 3A5	enzyme
Paramethasone	Corticosteroid-binding globulin	target
Prasterone	Cytochrome P450 3A7	enzyme
Prasterone	Peroxisome proliferator-activated receptor alpha	target
Prasterone	Estrogen receptor	target
Prasterone	Sigma non-opioid intracellular receptor 1	target
Prasterone	Estrogen receptor beta	target
Prasterone	Nuclear receptor subfamily 1 group I member 2	target
Prasterone	Nuclear receptor subfamily 1 group I member 3	target
Prasterone	GABA(A) Receptor	target
Prasterone	NMDA receptor	target
Prasterone	Androgen receptor	target
Prasterone	17-beta-hydroxysteroid dehydrogenase type 1	enzyme
Prasterone	Sulfotransferase 2A1	enzyme
Prasterone	Sulfotransferase 2B1	enzyme
Prasterone	3 beta-hydroxysteroid dehydrogenase/Delta 5-->4-isomerase type 1	enzyme
Prasterone	Cholesterol oxidase	enzyme
Prasterone	Steroid 17-alpha-hydroxylase/17,20 lyase	enzyme
Prasterone	Solute carrier organic anion transporter family member 1B3	transporter
Prasterone	Solute carrier organic anion transporter family member 2B1	transporter
Prasterone	Solute carrier organic anion transporter family member 1B1	transporter
Prasterone	Solute carrier organic anion transporter family member 1A2	transporter
Prasterone	Multidrug resistance-associated protein 1	transporter
Prasterone	Broad substrate specificity ATP-binding cassette transporter ABCG2	transporter
Prasterone	ATP-binding cassette sub-family C member 4	transporter
Prasterone	Glucose-6-phosphate 1-dehydrogenase	target
Prednisolone	Corticosteroid-binding globulin	carrier
Prednisolone	Cytochrome P450 3A4	enzyme
Prednisolone	Glucocorticoid receptor	target
Prednisolone	Solute carrier organic anion transporter family member 1A2	transporter
Prednisolone	ATP-dependent translocase ABCB1	transporter
Prednisolone	Albumin	carrier
Progesterone	Progesterone receptor	target
Progesterone	Estrogen receptor	target
Progesterone	Steroid 17-alpha-hydroxylase/17,20 lyase	target
Progesterone	Cytochrome P450 2C19	enzyme
Progesterone	Cytochrome P450 2C9	enzyme
Progesterone	Cytochrome P450 3A4	enzyme
Progesterone	Cytochrome P450 3A5	enzyme
Progesterone	Cytochrome P450 3A7	enzyme
Progesterone	ATP-dependent translocase ABCB1	transporter
Progesterone	Solute carrier family 22 member 2	transporter
Progesterone	Solute carrier family 22 member 1	transporter
Progesterone	Solute carrier family 22 member 3	transporter
Progesterone	Bile salt export pump	transporter
Progesterone	Multidrug resistance-associated protein 1	transporter
Progesterone	Hepatic sodium/bile acid cotransporter	transporter
Progesterone	Steroid 17-alpha-hydroxylase/17,20 lyase	enzyme
Progesterone	Cytochrome P450 1A1	enzyme
Progesterone	Cytochrome P450 1B1	enzyme
Progesterone	Cytochrome P450 2A6	enzyme
Progesterone	Cytochrome P450 2D6	enzyme
Progesterone	Mineralocorticoid receptor	target
Progesterone	Kappa-type opioid receptor	target
Progesterone	Alpha-1-acid glycoprotein 1	target
Progesterone	Glucocorticoid receptor	target
Progesterone	Androgen receptor	target
Progesterone	Sex hormone-binding globulin	target
Progesterone	Solute carrier organic anion transporter family member 1B1	transporter
Progesterone	Broad substrate specificity ATP-binding cassette transporter ABCG2	transporter
Progesterone	Estrogen receptor beta	target
Progesterone	Solute carrier organic anion transporter family member 1B3	transporter
Ramelteon	Melatonin receptor type 1B	target
Ramelteon	Melatonin receptor type 1A	target
Ramelteon	Cytochrome P450 1A2	enzyme
Ramelteon	Cytochrome P450 2C19	enzyme
Ramelteon	Cytochrome P450 3A4	enzyme
Ramelteon	Cytochrome P450 2C9	enzyme
Zolpidem	Gamma-aminobutyric acid receptor subunit alpha-1	target
Zolpidem	Cytochrome P450 3A4	enzyme
Zolpidem	Cytochrome P450 1A2	enzyme
Zolpidem	Gamma-aminobutyric acid receptor subunit alpha-2	target
Zolpidem	Gamma-aminobutyric acid receptor subunit alpha-3	target
Zolpidem	Cytochrome P450 2C9	enzyme
Zolpidem	Cytochrome P450 2C19	enzyme
Zolpidem	Cytochrome P450 2D6	enzyme
Zolpidem	Gamma-aminobutyric acid receptor subunit gamma-2	target
Zolpidem	Gamma-aminobutyric acid receptor subunit gamma-3	target
Zidovudine	Albumin	carrier
Zidovudine	Cytochrome P450 2A6	enzyme
Zidovudine	Cytochrome P450 2C9	enzyme
Zidovudine	Cytochrome P450 3A4	enzyme
Zidovudine	Reverse transcriptase/RNaseH	target
Zidovudine	Solute carrier family 22 member 2	transporter
Zidovudine	Solute carrier family 22 member 6	transporter
Zidovudine	Solute carrier family 22 member 7	transporter
Zidovudine	Organic anion transporter 3	transporter
Zidovudine	Solute carrier family 22 member 11	transporter
Zidovudine	Sodium/nucleoside cotransporter 1	transporter
Zidovudine	Equilibrative nucleoside transporter 2	transporter
Zidovudine	ATP-dependent translocase ABCB1	transporter
Zidovudine	ATP-binding cassette sub-family C member 4	transporter
Zidovudine	ATP-binding cassette sub-family C member 5	transporter
Zidovudine	Broad substrate specificity ATP-binding cassette transporter ABCG2	transporter
Zidovudine	Telomerase reverse transcriptase	target
Zidovudine	Thymidine kinase, cytosolic	enzyme
Zidovudine	UDP-glucuronosyltransferase 2B7	enzyme
Zidovudine	UDP-glucuronosyltransferase 1A1	enzyme
Zidovudine	Gag-Pol polyprotein	target
Zidovudine	Receptor-type tyrosine-protein kinase FLT3	target
Diethylstilbestrol	Estrogen receptor	target
Diethylstilbestrol	Estrogen-related receptor gamma	target
Diethylstilbestrol	Transthyretin	carrier
Diethylstilbestrol	Catechol O-methyltransferase	enzyme
Diethylstilbestrol	Aromatase	enzyme
Diethylstilbestrol	Broad substrate specificity ATP-binding cassette transporter ABCG2	transporter
Diethylstilbestrol	ATP-dependent translocase ABCB1	transporter
Diethylstilbestrol	Estrogen receptor beta	target
Diethylstilbestrol	Cytochrome P450 3A4	enzyme
Diethylstilbestrol	Cytochrome P450 2C8	enzyme
Diethylstilbestrol	Cytochrome P450 2C9	enzyme
Diethylstilbestrol	Cytochrome P450 2E1	enzyme
Diethylstilbestrol	Steroid hormone receptor ERR1	target
Diethylstilbestrol	Steroid hormone receptor ERR2	target
Diethylstilbestrol	Nuclear receptor coactivator 2	target
Diethylstilbestrol	Nuclear receptor subfamily 1 group I member 2	target
Diethylstilbestrol	Androgen receptor	target
Diethylstilbestrol	Sex hormone-binding globulin	target
Diethylstilbestrol	Solute carrier organic anion transporter family member 1B1	transporter
Diethylstilbestrol	Solute carrier organic anion transporter family member 2B1	transporter
Diethylstilbestrol	Bile salt export pump	transporter
Dapsone	Inactive dihydropteroate synthase 2	target
Dapsone	Dihydropteroate synthase	target
Dapsone	Cytochrome P450 2C9	enzyme
Dapsone	Cytochrome P450 2E1	enzyme
Dapsone	Cytochrome P450 3A4	enzyme
Dapsone	Flavin-containing monooxygenase 3	enzyme
Dapsone	Prostaglandin G/H synthase 1	enzyme
Dapsone	Prostaglandin G/H synthase 2	enzyme
Dapsone	Cytochrome P450 2C8	enzyme
Dapsone	Cytochrome P450 2C19	enzyme
Dapsone	Arylamine N-acetyltransferase 2	enzyme
Dapsone	Cytochrome P450 3A5	enzyme
Dapsone	Cytochrome P450 3A7	enzyme
Dapsone	Myeloperoxidase	enzyme
Dapsone	Cytochrome P450 2C18	enzyme
Morphine	Mu-type opioid receptor	target
Morphine	Delta-type opioid receptor	target
Morphine	Kappa-type opioid receptor	target
Morphine	ATP-dependent translocase ABCB1	transporter
Morphine	Cytochrome P450 2C8	enzyme
Morphine	Cytochrome P450 3A4	enzyme
Morphine	UDP-glucuronosyltransferase 2B7	enzyme
Morphine	UDP-glucuronosyltransferase 1A1	enzyme
Morphine	UDP-glucuronosyltransferase 1A8	enzyme
Morphine	UDP-glucuronosyltransferase 2B15	enzyme
Morphine	UDP-glucuronosyltransferase 2B4	enzyme
Morphine	UDP-glucuronosyltransferase 1A3	enzyme
Morphine	Lymphocyte antigen 96	target
Morphine	Albumin	carrier
Acenocoumarol	Vitamin K epoxide reductase complex subunit 1	target
Acenocoumarol	Cytochrome P450 2C9	enzyme
Acenocoumarol	Cytochrome P450 1A2	enzyme
Acenocoumarol	Albumin	carrier
Acenocoumarol	Alpha-1-acid glycoprotein 1	carrier
Acenocoumarol	Cytochrome P450 2C19	enzyme
Acenocoumarol	Cytochrome P450 3A4	enzyme
Acenocoumarol	ATP-dependent translocase ABCB1	transporter
Diphenadione	Cytochrome P450 3A4	enzyme
Ethyl biscoumacetate	Glutamine synthetase	enzyme
Ethyl biscoumacetate	Cytochrome P450 3A4	enzyme
Warfarin	Vitamin K epoxide reductase complex subunit 1	target
Warfarin	Cytochrome P450 2C8	enzyme
Warfarin	Cytochrome P450 1A2	enzyme
Warfarin	Cytochrome P450 2C9	enzyme
Warfarin	Alpha-1-acid glycoprotein 1	carrier
Warfarin	Albumin	carrier
Warfarin	Cytochrome P450 2C19	enzyme
Warfarin	Cytochrome P450 3A4	enzyme
Warfarin	Cytochrome P450 2C18	enzyme
Warfarin	Nuclear receptor subfamily 1 group I member 2	target
Azelnidipine	Cytochrome P450 3A4	enzyme
Azelnidipine	Voltage-dependent L-type calcium channel subunit beta-1	target
Barnidipine	Voltage-dependent L-type calcium channel subunit alpha-1C	target
Barnidipine	Cytochrome P450 3A4	enzyme
Barnidipine	Voltage-dependent T-type calcium channel subunit alpha-1G	target
Barnidipine	Voltage-dependent T-type calcium channel subunit alpha-1H	target
Bencyclane	Cytochrome P450 3A4	enzyme
Benidipine	Voltage-dependent L-type calcium channel	target
Benidipine	Voltage-dependent N-type calcium channel subunit alpha-1B	target
Benidipine	Voltage-dependent T-type calcium channel	target
Benidipine	Cytochrome P450 3A4	enzyme
Benidipine	Cytochrome P450 3A5	enzyme
Bepridil	Voltage-dependent P/Q-type calcium channel subunit alpha-1A	target
Bepridil	Sodium/potassium-transporting ATPase subunit alpha-1	target
Bepridil	Potassium voltage-gated channel subfamily KQT member 1	target
Bepridil	Troponin C, slow skeletal and cardiac muscles	target
Bepridil	Voltage-dependent T-type calcium channel subunit alpha-1H	target
Bepridil	Voltage-dependent calcium channel subunit alpha-2/delta-2	target
Bepridil	Dual specificity calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1B	target
Bepridil	Dual specificity calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1A	target
Bepridil	ATP-dependent translocase ABCB1	transporter
Bepridil	Cytochrome P450 2D6	enzyme
Bepridil	Potassium voltage-gated channel subfamily H member 2	target
Bepridil	Cytochrome P450 3A4	enzyme
Bepridil	Calmodulin	target
Bioallethrin	Voltage-gated sodium channel alpha subunit	target
Bioallethrin	Sodium channel protein	target
Bioallethrin	Voltage-dependent calcium channel	target
Bioallethrin	Voltage-dependent T-type calcium channel	target
Bioallethrin	Voltage-dependent P/Q-type calcium channel	target
Bioallethrin	Voltage-dependent L-type calcium channel	target
Bioallethrin	Cytochrome P450 2C8	enzyme
Bioallethrin	Cytochrome P450 2C9	enzyme
Bioallethrin	Cytochrome P450 2C19	enzyme
Bioallethrin	Cytochrome P450 3A4	enzyme
Bioallethrin	Cytochrome P450 2A1	enzyme
Bioallethrin	Cytochrome P450 1A1	enzyme
Bioallethrin	Cytochrome P450 2C6	enzyme
Bioallethrin	Cytochrome P450 2C11	enzyme
Bioallethrin	Cytochrome P450 3A1	enzyme
Bioallethrin	Cytochrome P450 3A2	enzyme
Carboxyamidotriazole	Cytochrome P450 3A4	enzyme
Carboxyamidotriazole	Muscarinic acetylcholine receptor M5	target
Caroverine	Cytochrome P450 3A4	enzyme
Cilnidipine	Voltage-dependent N-type calcium channel subunit alpha-1B	target
Cilnidipine	Voltage-dependent L-type calcium channel	target
Cilnidipine	Cytochrome P450 3A4	enzyme
Cinnarizine	Histamine H1 receptor	target
Cinnarizine	D(2) dopamine receptor	target
Cinnarizine	Voltage-dependent T-type calcium channel subunit alpha-1H	target
Cinnarizine	Cytochrome P450 2D6	enzyme
Cinnarizine	Cytochrome P450 2B6	enzyme
Cinnarizine	Cytochrome P450 2C9	enzyme
Cinnarizine	Cytochrome P450 1A1	enzyme
Cinnarizine	Cytochrome P450 1A2	enzyme
Cinnarizine	Cytochrome P450 2A6	enzyme
Cinnarizine	Voltage-dependent L-type calcium channel subunit alpha-1C	target
Cinnarizine	Voltage-dependent L-type calcium channel subunit alpha-1S	target
Cinnarizine	Voltage-dependent L-type calcium channel subunit alpha-1F	target
Cinnarizine	Voltage-dependent L-type calcium channel subunit alpha-1D	target
Cinnarizine	Voltage-dependent T-type calcium channel subunit alpha-1G	target
Cinnarizine	Voltage-dependent T-type calcium channel subunit alpha-1I	target
Cinnarizine	D(1) dopamine receptor	target
Cinnarizine	Muscarinic acetylcholine receptor	target
Cinnarizine	Cytochrome P450 3A4	enzyme
Cinnarizine	Albumin	carrier
Clevidipine	Voltage-dependent L-type calcium channel subunit alpha-1F	target
Clevidipine	Voltage-dependent L-type calcium channel subunit alpha-1S	target
Clevidipine	Voltage-dependent L-type calcium channel subunit alpha-1D	target
Clevidipine	Voltage-dependent L-type calcium channel subunit alpha-1C	target
Clevidipine	Cytochrome P450 2C9	enzyme
Clevidipine	Cytochrome P450 2D6	enzyme
Clevidipine	Cytochrome P450 2E1	enzyme
Clevidipine	Cytochrome P450 2C19	enzyme
Clevidipine	Cytochrome P450 3A4	enzyme
Clevidipine	Cholinesterase	enzyme
Cyclandelate	Voltage-dependent calcium channel subunit alpha-2/delta-1	target
Cyclandelate	Liver carboxylesterase 1	target
Cyclandelate	Cytochrome P450 3A4	enzyme
Darodipine	Cytochrome P450 3A4	enzyme
Dexniguldipine	ATP-dependent translocase ABCB1	target
Dexniguldipine	Cytochrome P450 3A4	enzyme
Dexniguldipine	Phosphatidylcholine translocator ABCB4	target
Dexverapamil	ATP-dependent translocase ABCB1	target
Dexverapamil	Cytochrome P450 3A4	enzyme
Dexverapamil	ATP-dependent translocase ABCB1	transporter
Dotarizine	5-hydroxytryptamine receptor 2A	target
Dotarizine	5-hydroxytryptamine receptor 1A	target
Dotarizine	Voltage-dependent P/Q-type calcium channel subunit alpha-1A	target
Dotarizine	5-hydroxytryptamine receptor 2C	target
Dotarizine	Cytochrome P450 3A4	enzyme
Efonidipine	Voltage-dependent T-type calcium channel subunit alpha-1I	target
Efonidipine	Voltage-dependent L-type calcium channel subunit alpha-1C	target
Efonidipine	Cytochrome P450 3A4	enzyme
Efonidipine	Voltage gated L-type calcium channel	target
Efonidipine	Voltage-dependent calcium channel	target
Efonidipine	Voltage-dependent T-type calcium channel	target
Efonidipine	Voltage-dependent T-type calcium channel subunit alpha-1G	target
Efonidipine	Voltage-dependent T-type calcium channel subunit alpha-1H	target
Emopamil	ATP-dependent translocase ABCB1	target
Emopamil	Cytochrome P450 3A4	enzyme
Emopamil	ATP-dependent translocase ABCB1	transporter
Eperisone	Cytochrome P450 3A4	enzyme
Ethosuximide	Voltage-dependent T-type calcium channel subunit alpha-1G	target
Ethosuximide	Cytochrome P450 3A4	enzyme
Ethosuximide	Cytochrome P450 2E1	enzyme
Ethosuximide	Cytochrome P450 3A Subfamily	enzyme
Fendiline	Cytochrome P450 3A4	enzyme
Fendiline	5-hydroxytryptamine receptor 2B	target
Fish oil	Diacylglycerol O-acyltransferase 2	target
Fish oil	Prostaglandin G/H synthase 2	target
Fish oil	Free fatty acid receptor 4	target
Fish oil	Voltage gated L-type calcium channel	target
Fish oil	Sodium channel protein	target
Fish oil	Free radicals	target
Fish oil	Nuclear factor NF-kappa-B	target
Fish oil	Sterol regulatory element-binding protein 1	target
Fish oil	Peroxisome proliferator-activated receptor alpha	target
Fish oil	Peroxisome proliferator-activated receptor gamma	target
Fish oil	Peroxisome proliferator-activated receptor delta	target
Fish oil	Cytochrome P450 3A4	enzyme
Flunarizine	Histamine H1 receptor	target
Flunarizine	Voltage-dependent T-type calcium channel subunit alpha-1G	target
Flunarizine	Voltage-dependent T-type calcium channel subunit alpha-1H	target
Flunarizine	Voltage-dependent T-type calcium channel subunit alpha-1I	target
Flunarizine	Cytochrome P450 2D6	enzyme
Flunarizine	Cytochrome P450 2C9	enzyme
Flunarizine	Cytochrome P450 1A1	enzyme
Flunarizine	Cytochrome P450 1A2	enzyme
Flunarizine	Cytochrome P450 2A6	enzyme
Flunarizine	Cytochrome P450 3A4	enzyme
Flunarizine	Voltage-dependent P/Q-type calcium channel subunit alpha-1A	target
Flunarizine	Calmodulin	target
Fluspirilene	D(2) dopamine receptor	target
Fluspirilene	5-hydroxytryptamine receptor 2A	target
Fluspirilene	Voltage-dependent calcium channel gamma-1 subunit	target
Fluspirilene	Cytochrome P450 3A4	enzyme
Gallopamil	Cytochrome P450 3A4	enzyme
Gallopamil	ATP-dependent translocase ABCB1	transporter
Gallopamil	Angiotensin-converting enzyme	target
Gallopamil	Neprilysin	target
Gallopamil	Sarcoplasmic/endoplasmic reticulum calcium ATPase 2	target
Isradipine	Voltage-dependent calcium channel subunit alpha-2/delta-1	target
Isradipine	Voltage-dependent L-type calcium channel subunit alpha-1C	target
Isradipine	Cytochrome P450 3A4	enzyme
Isradipine	Voltage-dependent T-type calcium channel subunit alpha-1H	target
Isradipine	Voltage-dependent calcium channel subunit alpha-2/delta-2	target
Isradipine	Voltage-dependent L-type calcium channel subunit beta-2	target
Isradipine	Voltage-dependent L-type calcium channel subunit alpha-1D	target
Isradipine	Voltage-dependent L-type calcium channel subunit alpha-1S	target
Isradipine	Bile salt export pump	transporter
Lercanidipine	Voltage-dependent calcium channel gamma-1 subunit	target
Lercanidipine	Cytochrome P450 3A4	enzyme
Lercanidipine	Cytochrome P450 3A5	enzyme
Lercanidipine	Cytochrome P450 3A7	enzyme
Lercanidipine	Cytochrome P450 2D6	enzyme
Lercanidipine	Voltage-dependent calcium channel subunit alpha-2/delta-1	target
Lidoflazine	Cytochrome P450 3A4	enzyme
Lidoflazine	Sodium channel protein type 3 subunit alpha	target
Lidoflazine	Equilibrative nucleoside transporter 1	target
Lomerizine	ATP-dependent translocase ABCB1	target
Lomerizine	Cytochrome P450 3A4	enzyme
Lomerizine	ATP-dependent translocase ABCB1	transporter
Lomerizine	Sodium channel protein type 5 subunit alpha	target
Lomerizine	Voltage-dependent N-type calcium channel subunit alpha-1B	target
Loperamide	Voltage-dependent P/Q-type calcium channel subunit alpha-1A	target
Loperamide	Mu-type opioid receptor	target
Loperamide	Pro-opiomelanocortin	target
Loperamide	Delta-type opioid receptor	target
Loperamide	Cytochrome P450 3A4	enzyme
Loperamide	ATP-dependent translocase ABCB1	transporter
Loperamide	Kappa-type opioid receptor	target
Loperamide	Cytochrome P450 2C8	enzyme
Loperamide	Cytochrome P450 2B6	enzyme
Loperamide	Cytochrome P450 2D6	enzyme
Loperamide	Potassium voltage-gated channel subfamily H member 2	target
Loperamide	Calmodulin	target
Manidipine	Voltage-dependent L-type calcium channel	target
Manidipine	Voltage-dependent T-type calcium channel	target
Manidipine	Cytochrome P450 2C9	enzyme
Manidipine	Cytochrome P450 2D6	enzyme
Manidipine	Cytochrome P450 1A1	enzyme
Manidipine	Cytochrome P450 2B6	enzyme
Manidipine	Cytochrome P450 2C19	enzyme
Manidipine	Cytochrome P450 3A4	enzyme
Manidipine	Voltage-dependent T-type calcium channel subunit alpha-1G	target
Manidipine	Voltage-dependent T-type calcium channel subunit alpha-1H	target
Manidipine	Voltage-dependent T-type calcium channel subunit alpha-1I	target
Manidipine	Voltage-dependent L-type calcium channel subunit alpha-1D	target
Manidipine	Voltage-dependent L-type calcium channel subunit alpha-1C	target
Manidipine	Cruzipain	target
Levomenthol	Transient receptor potential cation channel subfamily A member 1	target
Levomenthol	Transient receptor potential cation channel subfamily M member 8	target
Levomenthol	Transient receptor potential cation channel subfamily V member 3	target
Levomenthol	Kappa-type opioid receptor	target
Levomenthol	Voltage-dependent L-type calcium channel	target
Levomenthol	Cytochrome P450 3A4	enzyme
Mibefradil	Voltage-dependent T-type calcium channel subunit alpha-1G	target
Mibefradil	Voltage-dependent T-type calcium channel subunit alpha-1H	target
Mibefradil	Voltage-dependent L-type calcium channel subunit alpha-1C	target
Mibefradil	Voltage-dependent L-type calcium channel subunit beta-1	target
Mibefradil	Cytochrome P450 3A4	enzyme
Mibefradil	Cytochrome P450 1A2	enzyme
Mibefradil	Cytochrome P450 2D6	enzyme
Mibefradil	Cytochrome P450 3A5	enzyme
Mibefradil	Cytochrome P450 3A7	enzyme
Mibefradil	ATP-dependent translocase ABCB1	transporter
Mibefradil	Voltage-dependent T-type calcium channel subunit alpha-1I	target
Mibefradil	Voltage-dependent L-type calcium channel subunit alpha-1S	target
Mibefradil	Voltage-dependent L-type calcium channel subunit alpha-1F	target
Mibefradil	Voltage-dependent L-type calcium channel subunit alpha-1D	target
Mibefradil	Voltage-dependent L-type calcium channel subunit beta-2	target
Mibefradil	Voltage-dependent L-type calcium channel subunit beta-3	target
Mibefradil	Voltage-dependent L-type calcium channel subunit beta-4	target
Mibefradil	Cytochrome P450 11B1, mitochondrial	enzyme
Mibefradil	Cytochrome P450 11B2, mitochondrial	enzyme
Naftopidil	Cytochrome P450 3A4	enzyme
Naftopidil	Alpha-1A adrenergic receptor	target
Nicardipine	Voltage-dependent L-type calcium channel subunit alpha-1C	target
Nicardipine	Cytochrome P450 3A4	enzyme
Nicardipine	Cytochrome P450 2C19	enzyme
Nicardipine	Cytochrome P450 2C8	enzyme
Nicardipine	Cytochrome P450 2D6	enzyme
Nicardipine	Dual specificity calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1B	target
Nicardipine	Dual specificity calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1A	target
Nicardipine	Alpha-1A adrenergic receptor	target
Nicardipine	Alpha-1D adrenergic receptor	target
Nicardipine	Alpha-1B adrenergic receptor	target
Nicardipine	Muscarinic acetylcholine receptor M1	target
Nicardipine	Muscarinic acetylcholine receptor M2	target
Nicardipine	Muscarinic acetylcholine receptor M3	target
Nicardipine	Muscarinic acetylcholine receptor M4	target
Nicardipine	Muscarinic acetylcholine receptor M5	target
Nicardipine	Voltage-dependent calcium channel subunit alpha-2/delta-1	target
Nicardipine	Voltage-dependent L-type calcium channel subunit beta-2	target
Nicardipine	Voltage-dependent L-type calcium channel subunit alpha-1D	target
Nicardipine	ATP-dependent translocase ABCB1	transporter
Nicardipine	Cytochrome P450 2B6	enzyme
Nicardipine	Cytochrome P450 2E1	enzyme
Nicardipine	Cytochrome P450 3A5	enzyme
Nicardipine	Solute carrier organic anion transporter family member 1B1	transporter
Nicardipine	Bile salt export pump	transporter
Nicardipine	Cytochrome P450 2C9	enzyme
Nicardipine	Voltage-dependent calcium channel	target
Nicardipine	Voltage-dependent T-type calcium channel subunit alpha-1G	target
Nicardipine	Voltage-dependent T-type calcium channel subunit alpha-1H	target
Nicardipine	Voltage-dependent T-type calcium channel subunit alpha-1I	target
Nicardipine	Calmodulin	target
Niludipine	Cytochrome P450 3A4	enzyme
Nilvadipine	Cytochrome P450 3A4	enzyme
Nilvadipine	Cytochrome P450 2A6	enzyme
Nilvadipine	Cytochrome P450 2C19	enzyme
Nilvadipine	Cytochrome P450 2C8	enzyme
Nilvadipine	Cytochrome P450 2E1	enzyme
Nilvadipine	Voltage-dependent L-type calcium channel subunit alpha-1C	target
Nilvadipine	Voltage-dependent calcium channel subunit alpha-2/delta-1	target
Nilvadipine	Voltage-dependent L-type calcium channel subunit beta-2	target
Nilvadipine	Voltage-dependent L-type calcium channel subunit alpha-1D	target
Nilvadipine	Voltage-dependent L-type calcium channel subunit alpha-1S	target
Nilvadipine	Voltage-dependent calcium channel subunit alpha-2/delta-3	target
Nilvadipine	Voltage-dependent T-type calcium channel subunit alpha-1H	target
Nilvadipine	Voltage-dependent T-type calcium channel subunit alpha-1I	target
Nilvadipine	Voltage gated L-type calcium channel	target
Nilvadipine	Voltage-dependent T-type calcium channel	target
Nimesulide	Prostaglandin G/H synthase 2	target
Nimesulide	Group IIE secretory phospholipase A2	target
Nimesulide	Lactotransferrin	target
Nimesulide	Cytochrome P450 3A4	enzyme
Nimesulide	Tumor necrosis factor ligand superfamily member 10	target
Nimodipine	Cytochrome P450 3A4	enzyme
Nimodipine	Mineralocorticoid receptor	target
Nimodipine	Voltage-dependent L-type calcium channel subunit alpha-1D	target
Nimodipine	Voltage-dependent L-type calcium channel subunit alpha-1S	target
Nimodipine	Voltage-dependent L-type calcium channel subunit alpha-1C	target
Nimodipine	Voltage-dependent L-type calcium channel subunit beta-2	target
Nimodipine	Voltage-dependent L-type calcium channel subunit alpha-1F	target
Nimodipine	Voltage-dependent L-type calcium channel subunit beta-1	target
Nimodipine	Voltage-dependent L-type calcium channel subunit beta-3	target
Nimodipine	Voltage-dependent L-type calcium channel subunit beta-4	target
Nimodipine	Aryl hydrocarbon receptor	target
Nylidrin	Catechol O-methyltransferase	enzyme
Nylidrin	Voltage-dependent T-type calcium channel subunit alpha-1I	target
Nylidrin	Interferon alpha/beta receptor 2	target
Nylidrin	Cytochrome P450 3A4	enzyme
Niguldipine	Alpha-1A adrenergic receptor	target
Niguldipine	Cytochrome P450 3A4	enzyme
Niguldipine	ATP-dependent translocase ABCB1	transporter
Otilonium	Cytochrome P450 3A4	enzyme
Penfluridol	Cytochrome P450 3A4	enzyme
Penfluridol	Voltage-dependent T-type calcium channel subunit alpha-1G	target
Perhexiline	Carnitine O-palmitoyltransferase 1, liver isoform	target
Perhexiline	Carnitine O-palmitoyltransferase 2, mitochondrial	target
Perhexiline	Cytochrome P450 2D6	enzyme
Perhexiline	Cytochrome P450 2B6	enzyme
Perhexiline	Cytochrome P450 3A4	enzyme
Perhexiline	Potassium voltage-gated channel subfamily H member 2	target
Pinaverium	Voltage-dependent L-type calcium channel subunit alpha-1S	target
Pinaverium	Cytochrome P450 3A4	enzyme
Prenylamine	Myosin light chain kinase 2, skeletal/cardiac muscle	target
Prenylamine	Cytochrome P450 3A4	enzyme
Prenylamine	Calmodulin	target
Terodiline	Cytochrome P450 3A4	enzyme
Tetrahydropalmatine	D(1A) dopamine receptor	target
Tetrahydropalmatine	D(2) dopamine receptor	target
Tetrahydropalmatine	Cytochrome P450 3A4	enzyme
Tetrandrine	ATP-dependent translocase ABCB1	target
Tetrandrine	Cytochrome P450 3A4	enzyme
Tetrandrine	ATP-dependent translocase ABCB1	transporter
Tolfenamic acid	Prostaglandin G/H synthase 1	target
Tolfenamic acid	Prostaglandin G/H synthase 2	target
Tolfenamic acid	Cytochrome P450 3A4	enzyme
Tranilast	Hematopoietic prostaglandin D synthase	target
Tranilast	Cytochrome P450 3A4	enzyme
Tranilast	Cytochrome P450 2C9	enzyme
Tranilast	Histamine H1 receptor	target
Tranilast	Steryl-sulfatase	target
Trimebutine	Mu-type opioid receptor	target
Trimebutine	Voltage-dependent L-type calcium channel	target
Trimebutine	Calcium-activated potassium channel	target
Trimebutine	Voltage-dependent T-type calcium channel	target
Trimebutine	Muscarinic acetylcholine receptor M1	target
Trimebutine	Muscarinic acetylcholine receptor M2	target
Trimebutine	Muscarinic acetylcholine receptor M3	target
Trimebutine	Muscarinic acetylcholine receptor M4	target
Trimebutine	Cytochrome P450 3A4	enzyme
Trimethadione	Voltage-dependent T-type calcium channel subunit alpha-1G	target
Trimethadione	Cytochrome P450 2C19	enzyme
Trimethadione	Cytochrome P450 2C8	enzyme
Trimethadione	Cytochrome P450 2C9	enzyme
Trimethadione	Cytochrome P450 2E1	enzyme
Trimethadione	Cytochrome P450 3A4	enzyme
Seletracetam	Synaptic vesicle glycoprotein 2A	target
Seletracetam	Voltage-dependent N-type calcium channel subunit alpha-1B	target
Seletracetam	Glycine receptor (alpha-1/beta)	target
Seletracetam	Cytochrome P450 3A4	enzyme
Vinpocetine	Cytochrome P450 3A4	enzyme
WIN 55212-2	Cytochrome P450 3A4	enzyme
WIN 55212-2	Cannabinoid receptor 1	target
WIN 55212-2	Cannabinoid receptor 2	target
Zonisamide	Sodium channel protein type 1 subunit alpha	target
Zonisamide	Carbonic anhydrase 1	target
Zonisamide	Voltage-dependent T-type calcium channel subunit alpha-1G	target
Zonisamide	Cytochrome P450 3A4	enzyme
Zonisamide	Aldehyde oxidase	enzyme
Zonisamide	Amine oxidase [flavin-containing] B	target
Zonisamide	Carbonic anhydrase 2	target
Zonisamide	Carbonic anhydrase 3	target
Zonisamide	Carbonic anhydrase 4	target
Zonisamide	Carbonic anhydrase 5A, mitochondrial	target
Zonisamide	Carbonic anhydrase 5B, mitochondrial	target
Zonisamide	Carbonic anhydrase 6	target
Zonisamide	Carbonic anhydrase 7	target
Zonisamide	Carbonic anhydrase-related protein	target
Zonisamide	Carbonic anhydrase 9	target
Zonisamide	Carbonic anhydrase-related protein 10	target
Zonisamide	Carbonic anhydrase-related protein 11	target
Zonisamide	Carbonic anhydrase 12	target
Zonisamide	Carbonic anhydrase 13	target
Zonisamide	Carbonic anhydrase 14	target
Zonisamide	Voltage-dependent T-type calcium channel subunit alpha-1H	target
Zonisamide	Voltage-dependent T-type calcium channel subunit alpha-1I	target
Zonisamide	Sodium channel protein type 2 subunit alpha	target
Zonisamide	Sodium channel protein type 3 subunit alpha	target
Zonisamide	Sodium channel protein type 4 subunit alpha	target
Zonisamide	Sodium channel protein type 5 subunit alpha	target
Zonisamide	Sodium channel protein type 9 subunit alpha	target
Zonisamide	Sodium channel protein type 11 subunit alpha	target
Zonisamide	Sodium channel subunit beta-1	target
Zonisamide	Sodium channel subunit beta-2	target
Zonisamide	Sodium channel regulatory subunit beta-3	target
Zonisamide	Sodium channel subunit beta-4	target
Zonisamide	Amine oxidase [flavin-containing] A	target
Zonisamide	Cytochrome P450 2C19	enzyme
Zonisamide	UDP-glucuronosyltransferase 1A1	enzyme
Zonisamide	Cytochrome P450 3A5	enzyme
Zonisamide	ATP-dependent translocase ABCB1	transporter
Zonisamide	GABA(A) Receptor Benzodiazepine Binding Site	target
Ivermectin	ATP-dependent translocase ABCB1	transporter
Ivermectin	Multidrug resistance-associated protein 1	transporter
Ivermectin	ATP-binding cassette sub-family C member 2	transporter
Ivermectin	Broad substrate specificity ATP-binding cassette transporter ABCG2	transporter
Ivermectin	Cytochrome P450 3A4	enzyme
Ivermectin	Solute carrier organic anion transporter family member 1B1	transporter
Ivermectin	Solute carrier organic anion transporter family member 1B3	transporter
Ivermectin	Cytochrome P450 2D6	enzyme
Ivermectin	Cytochrome P450 2E1	enzyme
Ixabepilone	Tubulin beta-3 chain	target
Ixabepilone	Cytochrome P450 3A4	enzyme
Ixabepilone	ATP-dependent translocase ABCB1	transporter
Rifabutin	DNA-directed RNA polymerase subunit alpha	target
Rifabutin	Heat shock protein HSP 90-alpha	target
Rifabutin	Endoplasmin	target
Rifabutin	Cytochrome P450 3A4	enzyme
Rifabutin	DNA-directed RNA polymerase subunit beta	target
Rifabutin	DNA-directed RNA polymerase subunit beta'	target
Rifabutin	Cytochrome P450 2C19	enzyme
Rifabutin	Cytochrome P450 2B6	enzyme
Rifabutin	Cytochrome P450 2C8	enzyme
Rifabutin	Cytochrome P450 2C9	enzyme
Rifabutin	ATP-dependent translocase ABCB1	transporter
Rifapentine	DNA-directed RNA polymerase subunit beta'	target
Rifapentine	Cytochrome P450 2C8	enzyme
Rifapentine	Cytochrome P450 2C9	enzyme
Rifapentine	Cytochrome P450 3A4	enzyme
Rifapentine	Cytochrome P450 2C19	enzyme
Rifapentine	Cytochrome P450 2B6	enzyme
Rifapentine	Cytochrome P450 3A Subfamily	enzyme
Rifaximin	DNA-directed RNA polymerase subunit beta	target
Rifaximin	Nuclear receptor subfamily 1 group I member 2	target
Rifaximin	Cytochrome P450 3A4	enzyme
Rifaximin	Cytochrome P450 2C19	enzyme
Rifaximin	Cytochrome P450 2C8	enzyme
Regorafenib	Cytochrome P450 3A4	enzyme
Regorafenib	UDP-glucuronosyltransferase 1A9	enzyme
Regorafenib	Proto-oncogene tyrosine-protein kinase receptor Ret	target
Regorafenib	Vascular endothelial growth factor receptor 1	target
Regorafenib	Vascular endothelial growth factor receptor 2	target
Regorafenib	Vascular endothelial growth factor receptor 3	target
Regorafenib	Mast/stem cell growth factor receptor Kit	target
Regorafenib	Platelet-derived growth factor receptor alpha	target
Regorafenib	Platelet-derived growth factor receptor beta	target
Regorafenib	Fibroblast growth factor receptor 1	target
Regorafenib	Fibroblast growth factor receptor 2	target
Regorafenib	Angiopoietin-1 receptor	target
Regorafenib	Discoidin domain-containing receptor 2	target
Regorafenib	High affinity nerve growth factor receptor	target
Regorafenib	Ephrin type-A receptor 2	target
Regorafenib	RAF proto-oncogene serine/threonine-protein kinase	target
Regorafenib	Serine/threonine-protein kinase B-raf	target
Regorafenib	Cytochrome P450 2C8	enzyme
Regorafenib	Cytochrome P450 2C9	enzyme
Regorafenib	Cytochrome P450 2B6	enzyme
Regorafenib	Mitogen-activated protein kinase 11	target
Regorafenib	Tyrosine-protein kinase FRK	target
Regorafenib	Tyrosine-protein kinase ABL1	target
Regorafenib	ATP-dependent translocase ABCB1	transporter
Regorafenib	Broad substrate specificity ATP-binding cassette transporter ABCG2	transporter
Regorafenib	UDP-glucuronosyltransferase 1A1	enzyme
Regorafenib	Cytochrome P450 2C19	enzyme
Ivabradine	Cytochrome P450 3A4	enzyme
Ivabradine	Potassium/sodium hyperpolarization-activated cyclic nucleotide-gated channel 2	target
Vemurafenib	Albumin	carrier
Vemurafenib	Alpha-1-acid glycoprotein 1	carrier
Vemurafenib	Cytochrome P450 1A2	enzyme
Vemurafenib	Cytochrome P450 2D6	enzyme
Vemurafenib	Cytochrome P450 3A4	enzyme
Vemurafenib	Serine/threonine-protein kinase B-raf	target
Vemurafenib	Multidrug resistance-associated protein 1	transporter
Vemurafenib	Broad substrate specificity ATP-binding cassette transporter ABCG2	transporter
Vemurafenib	Cytochrome P450 2C9	enzyme
Vemurafenib	Cytochrome P450 2C8	enzyme
Vemurafenib	Cytochrome P450 2B6	enzyme
Vemurafenib	ATP-dependent translocase ABCB1	transporter
Vortioxetine	Sodium-dependent serotonin transporter	target
Vortioxetine	5-hydroxytryptamine receptor 3A	target
Vortioxetine	5-hydroxytryptamine receptor 7	target
Vortioxetine	5-hydroxytryptamine receptor 1B	target
Vortioxetine	5-hydroxytryptamine receptor 1A	target
Vortioxetine	Beta-1 adrenergic receptor	target
Vortioxetine	Sodium-dependent noradrenaline transporter	target
Vortioxetine	Cytochrome P450 2D6	enzyme
Vortioxetine	Cytochrome P450 3A4	enzyme
Vortioxetine	Cytochrome P450 3A5	enzyme
Vortioxetine	Cytochrome P450 2C19	enzyme
Vortioxetine	Cytochrome P450 2C9	enzyme
Vortioxetine	Cytochrome P450 2A6	enzyme
Vortioxetine	Cytochrome P450 2C8	enzyme
Vortioxetine	Cytochrome P450 2B6	enzyme
Pazopanib	Vascular endothelial growth factor receptor 1	target
Pazopanib	Vascular endothelial growth factor receptor 2	target
Pazopanib	Vascular endothelial growth factor receptor 3	target
Pazopanib	Platelet-derived growth factor receptor alpha	target
Pazopanib	Platelet-derived growth factor receptor beta	target
Pazopanib	Mast/stem cell growth factor receptor Kit	target
Pazopanib	Cytochrome P450 3A4	enzyme
Pazopanib	Cytochrome P450 2D6	enzyme
Pazopanib	Cytochrome P450 2C8	enzyme
Pazopanib	Cytochrome P450 1A2	enzyme
Pazopanib	ATP-dependent translocase ABCB1	transporter
Pazopanib	Broad substrate specificity ATP-binding cassette transporter ABCG2	transporter
Pazopanib	Solute carrier organic anion transporter family member 1B1	transporter
Pazopanib	UDP-glucuronosyltransferase 1A1	transporter
Pazopanib	Fibroblast growth factor receptor 3	target
Pazopanib	Tyrosine-protein kinase ITK/TSK	target
Pazopanib	Fibroblast growth factor 1	target
Pazopanib	SH2B adapter protein 3	target
Perampanel	Glutamate receptor 1	target
Perampanel	Cytochrome P450 3A4	enzyme
Perampanel	Cytochrome P450 3A5	enzyme
Perampanel	Cytochrome P450 1A2	enzyme
Perampanel	Cytochrome P450 2B6	enzyme
Perampanel	Glutamate receptor 2	target
Perampanel	Glutamate receptor 3	target
Perampanel	Glutamate receptor 4	target
Crizotinib	Cytochrome P450 3A4	enzyme
Crizotinib	Cytochrome P450 3A5	enzyme
Crizotinib	ATP-dependent translocase ABCB1	transporter
Crizotinib	ALK tyrosine kinase receptor	target
Crizotinib	Hepatocyte growth factor receptor	target
Crizotinib	Cytochrome P450 2B6	enzyme
Crizotinib	Cytochrome P450 3A Subfamily	enzyme
Crizotinib	Albumin	carrier
Crizotinib	alpha1-acid glycoprotein	carrier
Crizotinib	Proto-oncogene tyrosine-protein kinase ROS	target
Crizotinib	Macrophage-stimulating protein receptor	target
Cabozantinib	Cytochrome P450 3A4	enzyme
Cabozantinib	Cytochrome P450 2C9	enzyme
Cabozantinib	Hepatocyte growth factor receptor	target
Cabozantinib	Vascular endothelial growth factor receptor 2	target
Cabozantinib	Proto-oncogene tyrosine-protein kinase receptor Ret	target
Cabozantinib	Cytochrome P450 2C8	enzyme
Isavuconazonium	Cytochrome P450 3A4	enzyme
Isavuconazonium	ATP-dependent translocase ABCB1	transporter
Isavuconazonium	Cytochrome P450 3A5	enzyme
Isavuconazonium	Cholinesterase	enzyme
Isavuconazonium	Cytochrome P450 2C8	enzyme
Isavuconazonium	Cytochrome P450 2C9	enzyme
Isavuconazonium	Cytochrome P450 2C19	enzyme
Isavuconazonium	Cytochrome P450 2D6	enzyme
Isavuconazonium	Cytochrome P450 2B6	enzyme
Isavuconazonium	Broad substrate specificity ATP-binding cassette transporter ABCG2	transporter
Isavuconazonium	Solute carrier family 22 member 2	transporter
Isavuconazonium	Lanosterol 14-alpha demethylase	target
Isavuconazonium	Albumin	carrier
Axitinib	Vascular endothelial growth factor receptor 1	target
Axitinib	Vascular endothelial growth factor receptor 2	target
Axitinib	Vascular endothelial growth factor receptor 3	target
Axitinib	Cytochrome P450 3A4	enzyme
Axitinib	Cytochrome P450 3A5	enzyme
Axitinib	Cytochrome P450 1A2	enzyme
Axitinib	Cytochrome P450 2C19	enzyme
Axitinib	UDP-glucuronosyltransferase 1A1	enzyme
Axitinib	ATP-dependent translocase ABCB1	transporter
Axitinib	Solute carrier organic anion transporter family member 1B1	transporter
Axitinib	Tyrosine-protein kinase ABL1	target
Codeine	Mu-type opioid receptor	target
Codeine	Delta-type opioid receptor	target
Codeine	Kappa-type opioid receptor	target
Codeine	Cytochrome P450 2D6	enzyme
Codeine	Cytochrome P450 3A4	enzyme
Codeine	Solute carrier family 22 member 1	transporter
Codeine	UDP-glucuronosyltransferase 2B7	enzyme
Codeine	UDP-glucuronosyltransferase 2B4	enzyme
Apixaban	Coagulation factor X	target
Apixaban	Cytochrome P450 3A4	enzyme
Apixaban	Cytochrome P450 1A2	enzyme
Apixaban	Cytochrome P450 2C8	enzyme
Apixaban	Cytochrome P450 2C9	enzyme
Apixaban	Cytochrome P450 2C19	enzyme
Apixaban	Cytochrome P450 2J2	enzyme
Apixaban	ATP-dependent translocase ABCB1	transporter
Apixaban	Broad substrate specificity ATP-binding cassette transporter ABCG2	transporter
Apixaban	Cytochrome P450 3A5	enzyme
Pioglitazone	Peroxisome proliferator-activated receptor gamma	target
Pioglitazone	Cytochrome P450 2C8	enzyme
Pioglitazone	Cytochrome P450 3A4	enzyme
Pioglitazone	Solute carrier organic anion transporter family member 1B3	transporter
Pioglitazone	Solute carrier organic anion transporter family member 1B1	transporter
Pioglitazone	Amine oxidase [flavin-containing] B	target
Pioglitazone	Albumin	carrier
Pioglitazone	Cytochrome P450 1A1	enzyme
Lapatinib	Epidermal growth factor receptor	target
Lapatinib	Receptor tyrosine-protein kinase erbB-2	target
Lapatinib	Cytochrome P450 3A4	enzyme
Lapatinib	Cytochrome P450 2C8	enzyme
Lapatinib	ATP-dependent translocase ABCB1	transporter
Lapatinib	Antigen peptide transporter 1	transporter
Lapatinib	Cytochrome P450 3A5	enzyme
Lapatinib	Cytochrome P450 2C19	enzyme
Icotinib	Epidermal growth factor receptor	target
Icotinib	Cytochrome P450 3A4	enzyme
Icotinib	Cytochrome P450 1A2	enzyme
Icotinib	Cytochrome P450 3A5	enzyme
Cevimeline	Muscarinic acetylcholine receptor M1	target
Cevimeline	Muscarinic acetylcholine receptor M3	target
Cevimeline	Cytochrome P450 3A4	enzyme
Cevimeline	Cytochrome P450 2D6	enzyme
Cevimeline	Flavin-containing monooxygenase 1	enzyme
Bortezomib	Cytochrome P450 3A4	enzyme
Bortezomib	Cytochrome P450 2C19	enzyme
Bortezomib	Cytochrome P450 1A2	enzyme
Bortezomib	Cytochrome P450 2D6	enzyme
Bortezomib	Cytochrome P450 2C9	enzyme
Bortezomib	Proteasome subunit beta type-5	target
Bortezomib	Proteasome subunit beta type-1	target
Bortezomib	ATP-dependent translocase ABCB1	transporter
Bortezomib	Solute carrier organic anion transporter family member 1B3	transporter
Bortezomib	Serine protease 1	target
Dofetilide	Potassium channel subfamily K member 2	target
Dofetilide	Potassium voltage-gated channel subfamily H member 2	target
Dofetilide	ATP-sensitive inward rectifier potassium channel 12	target
Dofetilide	Cytochrome P450 3A4	enzyme
Dofetilide	Solute carrier family 22 member 2	transporter
Reboxetine	Sodium-dependent noradrenaline transporter	target
Reboxetine	Cytochrome P450 3A4	enzyme
Reboxetine	Cytochrome P450 2D6	enzyme
Reboxetine	ATP-dependent translocase ABCB1	transporter
Ranolazine	Cytochrome P450 3A4	enzyme
Ranolazine	Cytochrome P450 2D6	enzyme
Ranolazine	Bile salt export pump	transporter
Ranolazine	ATP-dependent translocase ABCB1	transporter
Ranolazine	Sodium channel protein	target
Ranolazine	Inward rectifier potassium channel	target
Ranolazine	Voltage gated L-type calcium channel	target
Ranolazine	Alpha-1 adrenergic receptors	target
Ranolazine	Beta-1 adrenergic receptor	target
Ranolazine	Fatty acid	target
Ranolazine	Alpha-1-acid glycoprotein 1	carrier
Ranolazine	Multidrug and toxin extrusion protein 1	transporter
Ranolazine	Multidrug and toxin extrusion protein 2	transporter
Ranolazine	Plasminogen	target
Ziprasidone	Alpha-1A adrenergic receptor	target
Ziprasidone	D(2) dopamine receptor	target
Ziprasidone	5-hydroxytryptamine receptor 2C	target
Ziprasidone	D(3) dopamine receptor	target
Ziprasidone	5-hydroxytryptamine receptor 1A	target
Ziprasidone	5-hydroxytryptamine receptor 1D	target
Ziprasidone	Histamine H1 receptor	target
Ziprasidone	5-hydroxytryptamine receptor 2A	target
Ziprasidone	D(4) dopamine receptor	target
Ziprasidone	5-hydroxytryptamine receptor 7	target
Ziprasidone	Cytochrome P450 3A4	enzyme
Ziprasidone	Alpha-2A adrenergic receptor	target
Ziprasidone	Alpha-1B adrenergic receptor	target
Ziprasidone	Alpha-2B adrenergic receptor	target
Ziprasidone	Alpha-2C adrenergic receptor	target
Ziprasidone	D(1A) dopamine receptor	target
Ziprasidone	D(1B) dopamine receptor	target
Ziprasidone	Muscarinic acetylcholine receptor M1	target
Ziprasidone	Muscarinic acetylcholine receptor M2	target
Ziprasidone	Muscarinic acetylcholine receptor M3	target
Ziprasidone	Muscarinic acetylcholine receptor M4	target
Ziprasidone	Muscarinic acetylcholine receptor M5	target
Ziprasidone	5-hydroxytryptamine receptor 1B	target
Ziprasidone	5-hydroxytryptamine receptor 1E	target
Ziprasidone	5-hydroxytryptamine receptor 6	target
Ziprasidone	Aldehyde oxidase	enzyme
Ziprasidone	Albumin	carrier
Ziprasidone	ATP-dependent translocase ABCB1	transporter
Ziprasidone	Alpha-1-acid glycoprotein 1	carrier
Ziprasidone	5-hydroxytryptamine 3 receptor	target
Ziprasidone	5-hydroxytryptamine receptor 5A	target
Ziprasidone	Neuronal acetylcholine receptor subunit alpha-7	target
Conjugated estrogens	Estrogen receptor	target
Conjugated estrogens	Cytochrome P450 3A4	enzyme
Conjugated estrogens	Cytochrome P450 1A2	enzyme
Conjugated estrogens	Catechol O-methyltransferase	enzyme
Conjugated estrogens	ATP-binding cassette sub-family C member 3	transporter
Conjugated estrogens	ATP-binding cassette sub-family C member 4	transporter
Conjugated estrogens	Multidrug resistance-associated protein 1	transporter
Conjugated estrogens	Solute carrier organic anion transporter family member 1A2	transporter
Conjugated estrogens	Hepatic sodium/bile acid cotransporter	transporter
Conjugated estrogens	Solute carrier family 22 member 10	transporter
Conjugated estrogens	Organic anion transporter 3	transporter
Conjugated estrogens	Solute carrier organic anion transporter family member 1C1	transporter
Conjugated estrogens	Solute carrier organic anion transporter family member 1B1	transporter
Conjugated estrogens	Solute carrier organic anion transporter family member 2B1	transporter
Conjugated estrogens	ATP-dependent translocase ABCB1	transporter
Conjugated estrogens	Solute carrier family 22 member 6	transporter
Conjugated estrogens	Organic solute transporter subunit alpha	transporter
Conjugated estrogens	Organic solute transporter subunit beta	transporter
Conjugated estrogens	ATP-binding cassette sub-family C member 2	transporter
Conjugated estrogens	Solute carrier organic anion transporter family member 4A1	transporter
Conjugated estrogens	ATP-binding cassette sub-family C member 11	transporter
Conjugated estrogens	Solute carrier organic anion transporter family member 1B3	transporter
Conjugated estrogens	Solute carrier family 22 member 11	transporter
Conjugated estrogens	Solute carrier organic anion transporter family member 3A1	transporter
Conjugated estrogens	Broad substrate specificity ATP-binding cassette transporter ABCG2	transporter
Conjugated estrogens	Thyroxine-binding globulin	carrier
Conjugated estrogens	Sex hormone-binding globulin	carrier
Conjugated estrogens	Albumin	carrier
Conjugated estrogens	Estrogen receptor beta	target
Bupivacaine	Sodium channel protein type 10 subunit alpha	target
Bupivacaine	Prostaglandin E2 receptor EP1 subtype	target
Bupivacaine	Cytochrome P450 3A4	enzyme
Bupivacaine	Cytochrome P450 2C19	enzyme
Bupivacaine	Cytochrome P450 2D6	enzyme
Bexarotene	Retinoic acid receptor RXR-beta	target
Bexarotene	Cytochrome P450 3A4	enzyme
Bexarotene	Retinoic acid receptor RXR-alpha	target
Bexarotene	Retinoic acid receptor RXR-gamma	target
Bexarotene	Cytochrome P450 2C8	enzyme
Vindesine	Tubulin beta-1 chain	target
Vindesine	Cytochrome P450 3A4	enzyme
Gefitinib	Epidermal growth factor receptor	target
Gefitinib	Cytochrome P450 3A4	enzyme
Gefitinib	Cytochrome P450 2D6	enzyme
Gefitinib	ATP-dependent translocase ABCB1	transporter
Gefitinib	Broad substrate specificity ATP-binding cassette transporter ABCG2	transporter
Gefitinib	Cytochrome P450 3A5	enzyme
Gefitinib	Cytochrome P450 1A1	enzyme
Gefitinib	Cytochrome P450 2C9	enzyme
Gefitinib	Cytochrome P450 2C19	enzyme
Gefitinib	Albumin	carrier
Gefitinib	Alpha-1-acid glycoprotein 1	carrier
Terfenadine	Histamine H1 receptor	target
Terfenadine	Potassium voltage-gated channel subfamily H member 2	target
Terfenadine	Cytochrome P450 3A4	enzyme
Terfenadine	Cytochrome P450 2D6	enzyme
Terfenadine	Muscarinic acetylcholine receptor M3	target
Terfenadine	Cytochrome P450 3A5	enzyme
Terfenadine	Cytochrome P450 3A7	enzyme
Terfenadine	ATP-dependent translocase ABCB1	transporter
Terfenadine	Cytochrome P450 2C8	enzyme
Terfenadine	Cytochrome P450 2J2	enzyme
Terfenadine	Muscarinic acetylcholine receptor M1	target
Terfenadine	Muscarinic acetylcholine receptor M5	target
Terfenadine	Muscarinic acetylcholine receptor M4	target
Terfenadine	Muscarinic acetylcholine receptor M2	target
Terfenadine	Bile salt export pump	transporter
Terfenadine	alpha1-acid glycoprotein	carrier
Terfenadine	Albumin	carrier
Vinorelbine	Tubulin beta chain	target
Vinorelbine	Cytochrome P450 3A4	enzyme
Vinorelbine	Cytochrome P450 2D6	enzyme
Grepafloxacin	DNA gyrase subunit A	target
Grepafloxacin	DNA topoisomerase 4 subunit A	target
Grepafloxacin	Cytochrome P450 3A4	enzyme
Grepafloxacin	Cytochrome P450 1A2	enzyme
Grepafloxacin	Solute carrier family 22 member 2	transporter
Grepafloxacin	Organic cation/carnitine transporter 2	transporter
Grepafloxacin	ATP-binding cassette sub-family C member 2	transporter
Grepafloxacin	ATP-dependent translocase ABCB1	transporter
Grepafloxacin	Multidrug resistance-associated protein 1	transporter
Grepafloxacin	Solute carrier family 22 member 6	transporter
Grepafloxacin	DNA gyrase subunit A	target
Grepafloxacin	DNA gyrase subunit B	target
Mirtazapine	5-hydroxytryptamine receptor 2A	target
Mirtazapine	5HT3 serotonin receptor	target
Mirtazapine	Alpha-2A adrenergic receptor	target
Mirtazapine	5-hydroxytryptamine receptor 2C	target
Mirtazapine	Kappa-type opioid receptor	target
Mirtazapine	Histamine H1 receptor	target
Mirtazapine	Cytochrome P450 1A2	enzyme
Mirtazapine	Cytochrome P450 3A4	enzyme
Mirtazapine	Cytochrome P450 2D6	enzyme
Mirtazapine	Alpha-1 adrenergic receptors	target
Mirtazapine	Sodium-dependent serotonin transporter	transporter
Sorafenib	Serine/threonine-protein kinase B-raf	target
Sorafenib	Receptor-type tyrosine-protein kinase FLT3	target
Sorafenib	RAF proto-oncogene serine/threonine-protein kinase	target
Sorafenib	Vascular endothelial growth factor receptor 3	target
Sorafenib	Platelet-derived growth factor receptor beta	target
Sorafenib	Mast/stem cell growth factor receptor Kit	target
Sorafenib	Vascular endothelial growth factor receptor 2	target
Sorafenib	Cytochrome P450 3A4	enzyme
Sorafenib	UDP-glucuronosyltransferase 1A9	enzyme
Sorafenib	Cytochrome P450 2B6	enzyme
Sorafenib	Cytochrome P450 2C8	enzyme
Sorafenib	Cytochrome P450 3A5	enzyme
Sorafenib	Cytochrome P450 3A7	enzyme
Sorafenib	Cytochrome P450 2C9	enzyme
Sorafenib	ATP-binding cassette sub-family C member 4	transporter
Sorafenib	ATP-dependent translocase ABCB1	transporter
Sorafenib	ATP-binding cassette sub-family C member 2	transporter
Sorafenib	Broad substrate specificity ATP-binding cassette transporter ABCG2	transporter
Sorafenib	Cytochrome P450 1A2	enzyme
Sorafenib	Cytochrome P450 2C19	enzyme
Sorafenib	Cytochrome P450 2D6	enzyme
Sorafenib	UDP-glucuronosyltransferase 1A1	enzyme
Sorafenib	RalA-binding protein 1	transporter
Sorafenib	Fibroblast growth factor receptor 1	target
Sorafenib	Proto-oncogene tyrosine-protein kinase receptor Ret	target
Sorafenib	Vascular endothelial growth factor receptor 1	target
Sorafenib	Solute carrier organic anion transporter family member 1B1	transporter
Sorafenib	Epidermal growth factor receptor	target
Eszopiclone	Cytochrome P450 3A4	enzyme
Eszopiclone	Gamma-aminobutyric acid receptor subunit alpha-1	target
Eszopiclone	Gamma-aminobutyric acid receptor subunit alpha-2	target
Eszopiclone	Gamma-aminobutyric acid receptor subunit alpha-3	target
Eszopiclone	Gamma-aminobutyric acid receptor subunit alpha-5	target
Eszopiclone	Cytochrome P450 2C8	enzyme
Eszopiclone	GABA(A) Receptor	target
Prochlorperazine	D(2) dopamine receptor	target
Prochlorperazine	Cytochrome P450 2D6	enzyme
Prochlorperazine	Histamine H1 receptor	target
Prochlorperazine	Alpha-1 adrenergic receptors	target
Prochlorperazine	Alpha-2 adrenergic receptors	target
Loratadine	Histamine H1 receptor	target
Loratadine	Cytochrome P450 3A4	enzyme
Loratadine	Cytochrome P450 2C19	enzyme
Loratadine	Cytochrome P450 2D6	enzyme
Loratadine	Cytochrome P450 2C8	enzyme
Loratadine	ATP-dependent translocase ABCB1	transporter
Loratadine	Potassium voltage-gated channel subfamily H member 2	target
Loratadine	Bile salt export pump	transporter
Loratadine	Cytochrome P450 1A1	enzyme
Loratadine	Cytochrome P450 1A2	enzyme
Loratadine	Cytochrome P450 2B6	enzyme
Loratadine	Cytochrome P450 2C9	enzyme
Loratadine	Cytochrome P450 3A5	enzyme
Loratadine	UDP-glucuronosyltransferase 2B10	enzyme
Loratadine	UDP-glucuronosyltransferase 1A1	enzyme
Loratadine	UDP-glucuronosyltransferase 1A3	enzyme
Loratadine	UDP-glucuronosyltransferase 2B15	enzyme
Dronabinol	Cannabinoid receptor 1	target
Dronabinol	Cytochrome P450 3A4	enzyme
Dronabinol	Cytochrome P450 2C9	enzyme
Dronabinol	Cannabinoid receptor 2	target
Dronabinol	ATP-dependent translocase ABCB1	transporter
Dronabinol	Broad substrate specificity ATP-binding cassette transporter ABCG2	transporter
Dronabinol	Prostaglandin G/H synthase 1	enzyme
Dronabinol	Cytochrome P450 2C19	enzyme
Dronabinol	Cytochrome P450 1A1	enzyme
Dronabinol	Cytochrome P450 1A2	enzyme
Dronabinol	Cytochrome P450 1B1	enzyme
Dronabinol	Cytochrome P450 2A6	enzyme
Dronabinol	Cytochrome P450 2B6	enzyme
Dronabinol	Cytochrome P450 2D6	enzyme
Dronabinol	Cytochrome P450 2J2	enzyme
Dronabinol	Cytochrome P450 3A5	enzyme
Dronabinol	Cytochrome P450 3A7	enzyme
Dronabinol	Multidrug resistance-associated protein 1	transporter
Dronabinol	Liver carboxylesterase 1	enzyme
Dronabinol	UDP-glucuronosyltransferase 1A1	enzyme
Dronabinol	UDP-glucuronosyltransferase 1A3	enzyme
Dronabinol	UDP-glucuronosyltransferase 1A9	enzyme
Dronabinol	UDP-glucuronosyltransferase 1A10	enzyme
Montelukast	Cysteinyl leukotriene receptor 1	target
Montelukast	Polyunsaturated fatty acid 5-lipoxygenase	target
Montelukast	Cytochrome P450 3A4	enzyme
Montelukast	Cytochrome P450 2C9	enzyme
Montelukast	Cytochrome P450 2C8	enzyme
Montelukast	Solute carrier organic anion transporter family member 2B1	transporter
Montelukast	Prostaglandin G/H synthase 1	enzyme
Montelukast	Cytochrome P450 2A6	enzyme
Albendazole	Tubulin alpha-1A chain	target
Albendazole	Tubulin beta-4B chain	target
Albendazole	Cytochrome P450 3A4	enzyme
Albendazole	Fumarate reductase flavoprotein subunit	target
Albendazole	Cytochrome P450 1A1	enzyme
Albendazole	Cytochrome P450 1A2	enzyme
Albendazole	Tubulin beta-2 chain	target
Albendazole	Cytochrome P450 2C19	enzyme
Albendazole	ATP-dependent translocase ABCB1	transporter
Erlotinib	Epidermal growth factor receptor	target
Erlotinib	Cytochrome P450 3A4	enzyme
Erlotinib	Broad substrate specificity ATP-binding cassette transporter ABCG2	transporter
Erlotinib	ATP-dependent translocase ABCB1	transporter
Erlotinib	Nuclear receptor subfamily 1 group I member 2	target
Erlotinib	Cytochrome P450 3A5	enzyme
Erlotinib	Cytochrome P450 1A1	enzyme
Erlotinib	Cytochrome P450 1A2	enzyme
Erlotinib	Cytochrome P450 1B1	enzyme
Erlotinib	Cytochrome P450 2D6	enzyme
Erlotinib	Cytochrome P450 2C8	enzyme
Erlotinib	UDP-glucuronosyltransferase 1A1	enzyme
Erlotinib	Albumin	carrier
Erlotinib	Alpha-1-acid glycoprotein 1	carrier
Erlotinib	Solute carrier organic anion transporter family member 2B1	transporter
Erlotinib	Epidermal growth factor receptor	enzyme
Rofecoxib	Prostaglandin G/H synthase 2	target
Rofecoxib	Elastin	target
Rofecoxib	Cytochrome P450 3A4	enzyme
Rofecoxib	Cytochrome P450 1A2	enzyme
Rofecoxib	ATP-binding cassette sub-family C member 4	transporter
Rofecoxib	Prostaglandin G/H synthase 1	enzyme
Rofecoxib	Cytochrome P450 2C8	enzyme
Rofecoxib	Cytochrome P450 2C9	enzyme
Toremifene	Estrogen receptor	target
Toremifene	Cytochrome P450 3A4	enzyme
Toremifene	ATP-dependent translocase ABCB1	transporter
Toremifene	Cytochrome P450 1A1	enzyme
Toremifene	Sex hormone-binding globulin	target
Bosentan	Endothelin receptor type B	target
Bosentan	Endothelin-1 receptor	target
Bosentan	Cytochrome P450 3A4	enzyme
Bosentan	Cytochrome P450 2C9	enzyme
Bosentan	Bile salt export pump	transporter
Vinblastine	Tubulin beta chain	target
Vinblastine	Transcription factor Jun	target
Vinblastine	Cytochrome P450 3A4	enzyme
Vinblastine	ATP-dependent translocase ABCB1	transporter
Vinblastine	Multidrug resistance-associated protein 1	transporter
Vinblastine	ATP-binding cassette sub-family C member 2	transporter
Vinblastine	ATP-binding cassette sub-family C member 6	transporter
Vinblastine	Bile salt export pump	transporter
Vinblastine	Tubulin alpha-1A chain	target
Vinblastine	Tubulin delta chain	target
Vinblastine	Tubulin epsilon chain	target
Vinblastine	Tubulin gamma-1 chain	target
Vinblastine	Cytochrome P450 2D6	enzyme
Vinblastine	Solute carrier organic anion transporter family member 1B1	transporter
Vinblastine	Tubulin beta-2A chain	target
Testosterone	Androgen receptor	target
Testosterone	Cytochrome P450 3A4	enzyme
Testosterone	Aromatase	enzyme
Testosterone	Amine oxidase [flavin-containing] A	enzyme
Testosterone	Cholesterol side-chain cleavage enzyme, mitochondrial	enzyme
Testosterone	Albumin	carrier
Testosterone	Sex hormone-binding globulin	carrier
Testosterone	Cytochrome P450 3A5	enzyme
Testosterone	Cytochrome P450 3A7	enzyme
Testosterone	Organic anion transporter 3	transporter
Testosterone	Solute carrier family 22 member 7	transporter
Testosterone	Hepatic sodium/bile acid cotransporter	transporter
Testosterone	Broad substrate specificity ATP-binding cassette transporter ABCG2	transporter
Testosterone	Cytochrome P450 1A1	enzyme
Testosterone	Cytochrome P450 1B1	enzyme
Testosterone	Cytochrome P450 2A13	enzyme
Testosterone	Cytochrome P450 2B6	enzyme
Testosterone	Cytochrome P450 2C19	enzyme
Testosterone	Cytochrome P450 2C8	enzyme
Testosterone	Cytochrome P450 2C9	enzyme
Testosterone	Cytochrome P450 3A43	enzyme
Testosterone	Estrogen receptor	target
Testosterone	Mineralocorticoid receptor	target
Testosterone	Solute carrier organic anion transporter family member 1B3	transporter
Efavirenz	Cytochrome P450 2B6	enzyme
Efavirenz	Cytochrome P450 3A4	enzyme
Efavirenz	Cytochrome P450 2C19	enzyme
Efavirenz	Cytochrome P450 2C9	enzyme
Efavirenz	Cytochrome P450 1A2	enzyme
Efavirenz	Cytochrome P450 2D6	enzyme
Efavirenz	Reverse transcriptase/RNaseH	target
Efavirenz	Cytochrome P450 2C8	enzyme
Efavirenz	Albumin	carrier
Efavirenz	Cytochrome P450 3A5	enzyme
Efavirenz	Cytochrome P450 3A7	enzyme
Efavirenz	UDP-glucuronosyltransferase 1A1	enzyme
Efavirenz	Bile salt export pump	transporter
Efavirenz	Solute carrier family 22 member 1	transporter
Efavirenz	Gag-Pol polyprotein	target
Clofibrate	Peroxisome proliferator-activated receptor alpha	target
Clofibrate	Cytochrome P450 3A4	enzyme
Clofibrate	Glutathione S-transferase A2	enzyme
Clofibrate	Cytochrome P450 2E1	enzyme
Clofibrate	Cytochrome P450 1A1	enzyme
Clofibrate	Cytochrome P450 4A11	enzyme
Clofibrate	Thyroxine-binding globulin	carrier
Clofibrate	Lipoprotein lipase	target
Galantamine	Acetylcholinesterase	target
Galantamine	Cytochrome P450 3A4	enzyme
Galantamine	Cytochrome P450 2D6	enzyme
Galantamine	Cholinesterase	target
Galantamine	ATP-dependent translocase ABCB1	transporter
Galantamine	Neuronal acetylcholine receptor subunit alpha-7	target
Galantamine	Muscle nicotinic acetylcholine receptor	target
Losartan	Type-1 angiotensin II receptor	target
Losartan	Cytochrome P450 3A4	enzyme
Losartan	Cytochrome P450 2C9	enzyme
Losartan	ATP-dependent translocase ABCB1	transporter
Losartan	Solute carrier family 22 member 6	transporter
Losartan	UDP-glucuronosyltransferase 1A1	enzyme
Losartan	UDP-glucuronosyltransferase 1A3	enzyme
Losartan	UDP-glucuronosyltransferase 1A10	enzyme
Losartan	UDP-glucuronosyltransferase 2B7	enzyme
Losartan	UDP-glucuronosyltransferase 2B17	enzyme
Losartan	Cytochrome P450 2C19	enzyme
Losartan	Albumin	carrier
Losartan	Solute carrier family 22 member 12	transporter
Losartan	Solute carrier family 2, facilitated glucose transporter member 9	transporter
Losartan	Bile salt export pump	transporter
Losartan	Cytochrome P450 2C8	enzyme
Losartan	Erythropoietin receptor	target
Delavirdine	Cytochrome P450 3A4	enzyme
Delavirdine	Cytochrome P450 2C9	enzyme
Delavirdine	Cytochrome P450 2D6	enzyme
Delavirdine	Cytochrome P450 3A5	enzyme
Delavirdine	Cytochrome P450 3A7	enzyme
Delavirdine	Cytochrome P450 2C19	enzyme
Delavirdine	Reverse transcriptase/RNaseH	target
Delavirdine	Gag-Pol polyprotein	target
Nateglinide	ATP-binding cassette sub-family C member 8	target
Nateglinide	Cytochrome P450 3A4	enzyme
Nateglinide	Cytochrome P450 2C9	enzyme
Nateglinide	Peroxisome proliferator-activated receptor gamma	target
Nateglinide	Cytochrome P450 3A5	enzyme
Nateglinide	Cytochrome P450 3A7	enzyme
Nateglinide	Solute carrier family 15 member 1	transporter
Nateglinide	Solute carrier family 15 member 2	transporter
Nateglinide	Solute carrier family 22 member 6	transporter
Nateglinide	Monocarboxylate transporter 1	transporter
Nateglinide	Prostaglandin G/H synthase 1	enzyme
Nateglinide	UDP-glucuronosyltransferase 1A9	enzyme
Nateglinide	Cytochrome P450 2D6	enzyme
Nateglinide	ATP-binding cassette sub-family C member 4	transporter
Nateglinide	Albumin	carrier
Nateglinide	Alpha-1-acid glycoprotein 1	carrier
Zileuton	Polyunsaturated fatty acid 5-lipoxygenase	target
Zileuton	Cytochrome P450 2C9	enzyme
Zileuton	Cytochrome P450 1A2	enzyme
Zileuton	Cytochrome P450 3A4	enzyme
Zileuton	Prostaglandin G/H synthase 1	enzyme
Zileuton	UDP-glucuronosyltransferase 1A9	enzyme
Zileuton	Albumin	carrier
Modafinil	Sodium-dependent dopamine transporter	target
Modafinil	Alpha-1B adrenergic receptor	target
Modafinil	Cytochrome P450 3A4	enzyme
Modafinil	Cytochrome P450 2C19	enzyme
Modafinil	Cytochrome P450 1A2	enzyme
Modafinil	Cytochrome P450 2B6	enzyme
Modafinil	Cytochrome P450 2C9	enzyme
Modafinil	Cytochrome P450 3A5	enzyme
Modafinil	Cytochrome P450 2D6	enzyme
Dolasetron	5-hydroxytryptamine receptor 3A	target
Dolasetron	Cytochrome P450 3A4	enzyme
Dolasetron	Cytochrome P450 2D6	enzyme
Dolasetron	Cytochrome P450 2C9	enzyme
Clopidogrel	P2Y purinoceptor 12	target
Clopidogrel	Cytochrome P450 3A4	enzyme
Clopidogrel	Cytochrome P450 2B6	enzyme
Clopidogrel	Cytochrome P450 3A5	enzyme
Clopidogrel	Cytochrome P450 2C19	enzyme
Clopidogrel	Cytochrome P450 2C9	enzyme
Clopidogrel	Cytochrome P450 1A2	enzyme
Clopidogrel	Cytochrome P450 2C8	enzyme
Clopidogrel	Liver carboxylesterase 1	enzyme
Clopidogrel	ATP-dependent translocase ABCB1	transporter
Clopidogrel	Solute carrier family 22 member 1	transporter
Clopidogrel	Solute carrier family 22 member 2	transporter
Clopidogrel	Albumin	carrier
Irinotecan	DNA topoisomerase I, mitochondrial	target
Irinotecan	DNA topoisomerase 1	target
Irinotecan	Cytochrome P450 3A4	enzyme
Irinotecan	Cytochrome P450 3A5	enzyme
Irinotecan	UDP-glucuronosyltransferase 1A1	enzyme
Irinotecan	UDP-glucuronosyltransferase 1A9	enzyme
Irinotecan	Cytochrome P450 3A7	enzyme
Irinotecan	Solute carrier family 22 member 3	transporter
Irinotecan	Solute carrier organic anion transporter family member 1B1	transporter
Irinotecan	Multidrug resistance-associated protein 1	transporter
Irinotecan	Broad substrate specificity ATP-binding cassette transporter ABCG2	transporter
Irinotecan	Albumin	carrier
Irinotecan	ATP-dependent translocase ABCB1	transporter
Irinotecan	ATP-binding cassette sub-family C member 2	transporter
Irinotecan	Human Carboxylesterases	enzyme
Etoposide	DNA topoisomerase 2-alpha	target
Etoposide	Cytochrome P450 3A4	enzyme
Etoposide	ATP-binding cassette sub-family C member 3	transporter
Etoposide	ATP-binding cassette sub-family C member 6	transporter
Etoposide	ATP-dependent translocase ABCB1	transporter
Etoposide	Multidrug resistance-associated protein 1	transporter
Etoposide	ATP-binding cassette sub-family C member 10	transporter
Etoposide	ATP-binding cassette sub-family C member 2	transporter
Etoposide	Broad substrate specificity ATP-binding cassette transporter ABCG2	transporter
Etoposide	Cytochrome P450 1A2	enzyme
Etoposide	Cytochrome P450 2E1	enzyme
Etoposide	Cytochrome P450 3A5	enzyme
Etoposide	UDP-glucuronosyltransferase 1A1	enzyme
Etoposide	DNA topoisomerase 2-beta	target
Etoposide	Glutathione S-transferase theta-1	enzyme
Etoposide	Glutathione S-transferase P	enzyme
Etoposide	Prostaglandin G/H synthase 2	enzyme
Etoposide	Prostaglandin G/H synthase 1	enzyme
Roxithromycin	50S ribosomal protein L10	target
Roxithromycin	ATP-dependent translocase ABCB1	target
Roxithromycin	Cytochrome P450 3A4	enzyme
Roxithromycin	Cytochrome P450 2B6	enzyme
Fentanyl	Mu-type opioid receptor	target
Fentanyl	Delta-type opioid receptor	target
Fentanyl	Cytochrome P450 3A4	enzyme
Fentanyl	Cytochrome P450 3A7	enzyme
Fentanyl	ATP-dependent translocase ABCB1	transporter
Fentanyl	Kappa-type opioid receptor	target
Fentanyl	ATP-dependent translocase ABCB1	target
Fentanyl	Albumin	carrier
Fentanyl	alpha1-acid glycoprotein	carrier
Mifepristone	Progesterone receptor	target
Mifepristone	Glucocorticoid receptor	target
Mifepristone	Cytochrome P450 3A4	enzyme
Mifepristone	Cytochrome P450 3A5	enzyme
Mifepristone	ATP-dependent translocase ABCB1	transporter
Mifepristone	Multidrug resistance-associated protein 1	transporter
Mifepristone	Cytochrome P450 2D6	enzyme
Mifepristone	Prostate-specific antigen	target
Mifepristone	Nuclear receptor subfamily 1 group I member 2	target
Mifepristone	Bile salt export pump	transporter
Mifepristone	Cytochrome P450 2C8	enzyme
Mifepristone	Cytochrome P450 2C9	enzyme
Mifepristone	Solute carrier organic anion transporter family member 1B1	transporter
Mifepristone	Solute carrier organic anion transporter family member 1B3	transporter
Donepezil	Acetylcholinesterase	target
Donepezil	5-hydroxytryptamine receptor 2A	target
Donepezil	Cytochrome P450 3A4	enzyme
Donepezil	Cytochrome P450 2D6	enzyme
Donepezil	Cytochrome P450 2C9	enzyme
Donepezil	Cholinesterase	target
Donepezil	Nitric oxide synthase 1	target
Donepezil	Tumor necrosis factor-inducible gene 6 protein	target
Donepezil	Interleukin-1 beta	target
Donepezil	Nuclear factor NF-kappa-B	target
Donepezil	Broad substrate specificity ATP-binding cassette transporter ABCG2	transporter
Donepezil	NMDA receptor	target
Granisetron	5-hydroxytryptamine receptor 3A	target
Granisetron	Cytochrome P450 3A4	enzyme
Granisetron	Cytochrome P450 1A1	enzyme
Ondansetron	5-hydroxytryptamine receptor 3A	target
Ondansetron	Cytochrome P450 3A4	enzyme
Ondansetron	Cytochrome P450 1A2	enzyme
Ondansetron	Cytochrome P450 2D6	enzyme
Ondansetron	Cytochrome P450 3A5	enzyme
Ondansetron	Cytochrome P450 3A7	enzyme
Ondansetron	5-hydroxytryptamine receptor 4	target
Ondansetron	5-hydroxytryptamine receptor 1A	target
Ondansetron	5-hydroxytryptamine receptor 1B	target
Ondansetron	Mu-type opioid receptor	target
Ondansetron	Cytochrome P450 2C9	enzyme
Ondansetron	Cytochrome P450 2E1	enzyme
Tiagabine	Sodium- and chloride-dependent GABA transporter 1	target
Tiagabine	Cytochrome P450 3A4	enzyme
Tiagabine	UDP-glucuronosyltransferase 1A1	enzyme
Cocaine	Sodium-dependent noradrenaline transporter	target
Cocaine	Sodium channel protein	target
Cocaine	Sodium-dependent serotonin transporter	target
Cocaine	Sodium-dependent dopamine transporter	target
Cocaine	Cytochrome P450 3A4	enzyme
Cocaine	Muscarinic acetylcholine receptor M1	target
Cocaine	Muscarinic acetylcholine receptor M2	target
Cocaine	Cytochrome P450 2D6	enzyme
Cocaine	Solute carrier family 22 member 2	transporter
Cocaine	Cytochrome P450 2C8	enzyme
Cocaine	Sigma non-opioid intracellular receptor 1	target
Cocaine	Liver carboxylesterase 1	target
Cocaine	Cholinesterase	enzyme
Cocaine	Sodium-dependent dopamine transporter	transporter
Cocaine	alpha1-acid glycoprotein	carrier
Cocaine	Liver carboxylesterase 1	enzyme
Paricalcitol	Vitamin D3 receptor	target
Paricalcitol	1,25-dihydroxyvitamin D(3) 24-hydroxylase, mitochondrial	enzyme
Paricalcitol	Cytochrome P450 3A4	enzyme
Paricalcitol	UDP-glucuronosyltransferase 1A4	enzyme
Tinidazole	Cytochrome P450 3A4	enzyme
Tinidazole	DNA	target
Tinidazole	Bile salt export pump	transporter
Almotriptan	5-hydroxytryptamine receptor 1D	target
Almotriptan	5-hydroxytryptamine receptor 1B	target
Almotriptan	Cytochrome P450 3A4	enzyme
Almotriptan	Cytochrome P450 2D6	enzyme
Almotriptan	Amine oxidase [flavin-containing] A	enzyme
Almotriptan	Flavin-containing monooxygenase 3	enzyme
Almotriptan	Cytochrome P450 2C19	enzyme
Almotriptan	Cytochrome P450 2E1	enzyme
Almotriptan	Cytochrome P450 2C8	enzyme
Salmeterol	Beta-2 adrenergic receptor	target
Salmeterol	Cytochrome P450 3A4	enzyme
Salmeterol	Cytochrome P450 2C8	enzyme
Salmeterol	Cytochrome P450 3A5	enzyme
Salmeterol	Cytochrome P450 3A7	enzyme
Salmeterol	Beta-1 adrenergic receptor	target
Salmeterol	Beta-3 adrenergic receptor	target
Salmeterol	Albumin	carrier
Salmeterol	alpha1-acid glycoprotein	carrier
Salmeterol	Solute carrier family 22 member 1	transporter
Salmeterol	Solute carrier family 22 member 2	transporter
Salmeterol	Solute carrier family 22 member 3	transporter
Hydrocodone	Mu-type opioid receptor	target
Hydrocodone	Delta-type opioid receptor	target
Hydrocodone	Cytochrome P450 3A4	enzyme
Hydrocodone	Cytochrome P450 2D6	enzyme
Hydrocodone	Cytochrome P450 2B6	enzyme
Hydrocodone	Cytochrome P450 2C19	enzyme
Hydrocodone	Sigma non-opioid intracellular receptor 1	target
Zaleplon	Gamma-aminobutyric acid receptor subunit alpha-1	target
Zaleplon	Cytochrome P450 3A4	enzyme
Zaleplon	Aldehyde oxidase	enzyme
Zaleplon	Cytochrome P450 3A5	enzyme
Zaleplon	Cytochrome P450 3A7	enzyme
Exemestane	Aromatase	target
Exemestane	Cytochrome P450 3A4	enzyme
Exemestane	Aromatase	enzyme
Doxorubicin	DNA topoisomerase 2-alpha	target
Doxorubicin	DNA	target
Doxorubicin	Cytochrome P450 3A4	enzyme
Doxorubicin	Cytochrome P450 2D6	enzyme
Doxorubicin	Cytochrome P450 2B6	enzyme
Doxorubicin	ATP-dependent translocase ABCB1	transporter
Doxorubicin	ATP-binding cassette sub-family C member 3	transporter
Doxorubicin	ATP-binding cassette sub-family C member 6	transporter
Doxorubicin	Multidrug resistance-associated protein 1	transporter
Doxorubicin	ATP-binding cassette sub-family C member 10	transporter
Doxorubicin	Broad substrate specificity ATP-binding cassette transporter ABCG2	transporter
Doxorubicin	Bile salt export pump	transporter
Doxorubicin	Solute carrier family 22 member 16	transporter
Doxorubicin	Mitochondrial potassium channel ATP-binding subunit	transporter
Doxorubicin	Cytochrome P450 1B1	enzyme
Doxorubicin	Carbonyl reductase [NADPH] 1	enzyme
Doxorubicin	Carbonyl reductase [NADPH] 3	enzyme
Doxorubicin	Aldo-keto reductase family 1 member A1	enzyme
Doxorubicin	Aldo-keto reductase family 1 member C3	enzyme
Doxorubicin	NAD(P)H dehydrogenase [quinone] 1	enzyme
Doxorubicin	Xanthine dehydrogenase/oxidase	enzyme
Doxorubicin	Nitric oxide synthase 3	enzyme
Doxorubicin	Nitric oxide synthase, inducible	enzyme
Doxorubicin	Nitric oxide synthase 1	enzyme
Doxorubicin	NADH dehydrogenase [ubiquinone] iron-sulfur protein 2, mitochondrial	enzyme
Doxorubicin	NADH dehydrogenase [ubiquinone] iron-sulfur protein 3, mitochondrial	enzyme
Doxorubicin	NADH dehydrogenase [ubiquinone] iron-sulfur protein 7, mitochondrial	enzyme
Doxorubicin	NADPH--cytochrome P450 reductase	enzyme
Doxorubicin	RalA-binding protein 1	transporter
Doxorubicin	ATP-binding cassette sub-family C member 2	transporter
Doxorubicin	Albumin	carrier
Doxorubicin	Nucleolar and coiled-body phosphoprotein 1	target
Doxorubicin	DNA topoisomerase 1	target
Doxorubicin	DNA topoisomerase 2-beta	target
Doxorubicin	Aldo-keto reductase family 1 member B1	enzyme
Doxorubicin	Aldo-keto reductase family 1 member B10	enzyme
Doxorubicin	Aldo-keto reductase family 1 member C4	enzyme
Doxorubicin	Telomerase reverse transcriptase	target
Levobupivacaine	Sodium channel protein type 10 subunit alpha	target
Levobupivacaine	Cytochrome P450 3A4	enzyme
Levobupivacaine	Cytochrome P450 1A2	enzyme
Letrozole	Aromatase	target
Letrozole	Cytochrome P450 3A4	enzyme
Letrozole	Cytochrome P450 2A6	enzyme
Letrozole	Aromatase	enzyme
Letrozole	Cytochrome P450 2C19	enzyme
Letrozole	UDP-glucuronosyltransferase 2B7	enzyme
Letrozole	Albumin	carrier
Letrozole	ATP-dependent translocase ABCB1	transporter
Busulfan	DNA	target
Busulfan	Cytochrome P450 3A4	enzyme
Busulfan	Glutathione S-transferase A2	enzyme
Busulfan	Glutathione S-transferase A1	enzyme
Busulfan	Glutathione S-transferase Mu 1	enzyme
Busulfan	Glutathione S-transferase P	enzyme
Busulfan	Microsomal glutathione S-transferase 2	enzyme
Cinacalcet	Extracellular calcium-sensing receptor	target
Cinacalcet	Cytochrome P450 3A4	enzyme
Cinacalcet	Cytochrome P450 2D6	enzyme
Cinacalcet	Cytochrome P450 1A2	enzyme
Ketoconazole	Cytochrome P450 3A4	enzyme
Ketoconazole	Cytochrome P450 2C9	enzyme
Ketoconazole	Cytochrome P450 2C19	enzyme
Ketoconazole	Cytochrome P450 3A5	enzyme
Ketoconazole	Cytochrome P450 1A2	enzyme
Ketoconazole	Cytochrome P450 2C8	enzyme
Ketoconazole	Cytochrome P450 1A1	enzyme
Ketoconazole	Cytochrome P450 2D6	enzyme
Ketoconazole	Bile salt export pump	transporter
Ketoconazole	ATP-dependent translocase ABCB1	transporter
Ketoconazole	Cytochrome P450 11B1, mitochondrial	enzyme
Ketoconazole	Cytochrome P450 1B1	enzyme
Ketoconazole	Cytochrome P450 2A6	enzyme
Ketoconazole	Cytochrome P450 2B6	enzyme
Ketoconazole	Lanosterol 14-alpha demethylase	target
Ketoconazole	Androgen receptor	target
Ketoconazole	Steroid 17-alpha-hydroxylase/17,20 lyase	target
Ketoconazole	Steroid 21-hydroxylase	target
Ketoconazole	Potassium voltage-gated channel subfamily H member 2	target
Ketoconazole	Nuclear receptor subfamily 1 group I member 2	target
Ketoconazole	Nuclear receptor subfamily 1 group I member 3	target
Ketoconazole	UDP-glucuronosyltransferase 1A1	enzyme
Ketoconazole	UDP-glucuronosyltransferase 2B7	enzyme
Ketoconazole	Solute carrier organic anion transporter family member 1B1	transporter
Ketoconazole	Cytochrome P450 4F12	enzyme
Ketoconazole	Cytochrome P450 4F2	enzyme
Ketoconazole	Albumin	carrier
Ketoconazole	Sex hormone-binding globulin	carrier
Ketoconazole	Aromatase	enzyme
Ketoconazole	UDP-glucuronosyltransferase 1A7	enzyme
Ketoconazole	Lanosterol 14-alpha demethylase	target
Oxybutynin	Muscarinic acetylcholine receptor M1	target
Oxybutynin	Muscarinic acetylcholine receptor M2	target
Oxybutynin	Muscarinic acetylcholine receptor M3	target
Oxybutynin	Cytochrome P450 3A4	enzyme
Oxybutynin	Cytochrome P450 2C8	enzyme
Oxybutynin	Cytochrome P450 2D6	enzyme
Oxybutynin	Cytochrome P450 3A5	enzyme
Oxybutynin	Alpha-1-acid glycoprotein 1	carrier
Oxybutynin	Albumin	carrier
Clonazepam	Cytochrome P450 3A4	enzyme
Clonazepam	Albumin	carrier
Clonazepam	Cytochrome P450 2E1	enzyme
Clonazepam	Arylamine N-acetyltransferase 2	enzyme
Clonazepam	GABA(A) Receptor	target
Clonazepam	Nuclear receptor subfamily 1 group I member 2	target
Clonazepam	GABA(A) Receptor Benzodiazepine Binding Site	target
Sibutramine	Sodium-dependent serotonin transporter	target
Sibutramine	Sodium-dependent noradrenaline transporter	target
Sibutramine	Cytochrome P450 3A4	enzyme
Sibutramine	Sodium-dependent dopamine transporter	target
Dutasteride	3-oxo-5-alpha-steroid 4-dehydrogenase 1	target
Dutasteride	3-oxo-5-alpha-steroid 4-dehydrogenase 2	target
Dutasteride	Sodium-dependent dopamine transporter	transporter
Dutasteride	Synaptic vesicular amine transporter	transporter
Dutasteride	Albumin	carrier
Dutasteride	Alpha-1-acid glycoprotein 1	carrier
Dutasteride	Cytochrome P450 3A5	enzyme
Dutasteride	Polyprenol reductase	target
Cilostazol	cGMP-inhibited 3',5'-cyclic phosphodiesterase 3A	target
Cilostazol	Cytochrome P450 2C19	enzyme
Cilostazol	Cytochrome P450 3A4	enzyme
Cilostazol	Cytochrome P450 3A5	enzyme
Cilostazol	Cytochrome P450 3A7	enzyme
Cilostazol	Cytochrome P450 1A2	enzyme
Cilostazol	Cytochrome P450 2D6	enzyme
Itraconazole	Cytochrome P450 3A4	enzyme
Itraconazole	Cytochrome P450 3A5	enzyme
Itraconazole	Cytochrome P450 3A7	enzyme
Itraconazole	Cytochrome P450 2B6	enzyme
Itraconazole	ATP-dependent translocase ABCB1	transporter
Itraconazole	Cytochrome P450 1A1	enzyme
Itraconazole	Cytochrome P450 2E1	enzyme
Itraconazole	Solute carrier organic anion transporter family member 2B1	transporter
Itraconazole	Cytochrome P450 3A Subfamily	enzyme
Itraconazole	Broad substrate specificity ATP-binding cassette transporter ABCG2	transporter
Itraconazole	Albumin	carrier
Itraconazole	Lanosterol 14-alpha demethylase	target
Itraconazole	Lanosterol 14-alpha demethylase	target
Escitalopram	Sodium-dependent serotonin transporter	target
Escitalopram	Cytochrome P450 3A4	enzyme
Escitalopram	Cytochrome P450 2D6	enzyme
Escitalopram	Sodium-dependent dopamine transporter	target
Escitalopram	Sodium-dependent noradrenaline transporter	target
Escitalopram	Muscarinic acetylcholine receptor M1	target
Escitalopram	Histamine H1 receptor	target
Escitalopram	Cytochrome P450 2C19	enzyme
Escitalopram	ATP-dependent translocase ABCB1	transporter
Escitalopram	5-hydroxytryptamine receptor 1A	target
Escitalopram	5-hydroxytryptamine receptor 2A	target
Escitalopram	5-hydroxytryptamine receptor 2C	target
Escitalopram	Alpha-1 adrenergic receptors	target
Escitalopram	Alpha-2 adrenergic receptors	target
Escitalopram	D(2) dopamine receptor	target
Escitalopram	Amine oxidase [flavin-containing] A	enzyme
Escitalopram	Amine oxidase [flavin-containing] B	enzyme
Escitalopram	Aldehyde oxidase	enzyme
Domperidone	D(2) dopamine receptor	target
Domperidone	Cytochrome P450 3A4	enzyme
Domperidone	Cytochrome P450 3A5	enzyme
Domperidone	Cytochrome P450 3A7	enzyme
Domperidone	ATP-dependent translocase ABCB1	transporter
Domperidone	Cytochrome P450 1A2	enzyme
Domperidone	Cytochrome P450 2B6	enzyme
Domperidone	Cytochrome P450 2C8	enzyme
Domperidone	Cytochrome P450 2D6	enzyme
Domperidone	D(3) dopamine receptor	target
Clindamycin	Cytochrome P450 3A4	enzyme
Clindamycin	Cytochrome P450 3A5	enzyme
Clindamycin	Alpha-1-acid glycoprotein 1	carrier
Clindamycin	ATP-dependent translocase ABCB1	transporter
Clindamycin	50S ribosomal protein L1	target
Estazolam	Cytochrome P450 3A4	enzyme
Estazolam	GABA(A) Receptor	target
Estazolam	GABA(A) Receptor Benzodiazepine Binding Site	target
Finasteride	3-oxo-5-alpha-steroid 4-dehydrogenase 1	target
Finasteride	Cytochrome P450 3A4	enzyme
Finasteride	3-oxo-5-alpha-steroid 4-dehydrogenase 2	target
Finasteride	Aldo-keto reductase family 1 member D1	target
Finasteride	Cytochrome P450 3A5	enzyme
Finasteride	Cytochrome P450 3A7	enzyme
Finasteride	Solute carrier family 12 member 5	transporter
Finasteride	Polyprenol reductase	target
Halofantrine	Fe(II)-protoporphyrin IX	target
Halofantrine	Potassium voltage-gated channel subfamily H member 2	target
Halofantrine	Cytochrome P450 3A4	enzyme
Halofantrine	Cytochrome P450 2D6	enzyme
Halofantrine	Plasmepsin-2	target
Halofantrine	Cytochrome P450 2C8	enzyme
Halofantrine	Cytochrome P450 3A5	enzyme
Halofantrine	Calmodulin-2	target
Halofantrine	Calmodulin-3	target
Levacetylmethadol	Mu-type opioid receptor	target
Levacetylmethadol	Cytochrome P450 3A4	enzyme
Levacetylmethadol	Neuronal acetylcholine receptor subunit beta-4	target
Levacetylmethadol	Neuronal acetylcholine receptor subunit alpha-3	target
Levacetylmethadol	Cytochrome P450 3A7	enzyme
Paclitaxel	Apoptosis regulator Bcl-2	target
Paclitaxel	Tubulin beta-1 chain	target
Paclitaxel	Cytochrome P450 2C8	enzyme
Paclitaxel	Cytochrome P450 3A4	enzyme
Paclitaxel	Cytochrome P450 3A5	enzyme
Paclitaxel	Cytochrome P450 3A7	enzyme
Paclitaxel	Bile salt export pump	transporter
Paclitaxel	ATP-dependent translocase ABCB1	transporter
Paclitaxel	Multidrug resistance-associated protein 1	transporter
Paclitaxel	ATP-binding cassette sub-family C member 10	transporter
Paclitaxel	Aromatase	enzyme
Paclitaxel	Cytochrome P450 1B1	enzyme
Paclitaxel	Solute carrier organic anion transporter family member 1B3	transporter
Paclitaxel	Nuclear receptor subfamily 1 group I member 2	target
Paclitaxel	Microtubule-associated protein 4	target
Paclitaxel	Microtubule-associated protein 2	target
Paclitaxel	Microtubule-associated protein tau	target
Paclitaxel	ATP-binding cassette sub-family C member 2	transporter
Retapamulin	50S ribosomal protein L3	target
Retapamulin	Cytochrome P450 3A4	enzyme
Sitagliptin	Dipeptidyl peptidase 4	target
Sitagliptin	Cytochrome P450 3A4	enzyme
Sitagliptin	Cytochrome P450 2C8	enzyme
Sitagliptin	ATP-dependent translocase ABCB1	transporter
Sitagliptin	Organic anion transporter 3	transporter
Sunitinib	Platelet-derived growth factor receptor beta	target
Sunitinib	Vascular endothelial growth factor receptor 1	target
Sunitinib	Vascular endothelial growth factor receptor 2	target
Sunitinib	Vascular endothelial growth factor receptor 3	target
Sunitinib	Mast/stem cell growth factor receptor Kit	target
Sunitinib	Receptor-type tyrosine-protein kinase FLT3	target
Sunitinib	Macrophage colony-stimulating factor 1 receptor	target
Sunitinib	Platelet-derived growth factor receptor alpha	target
Sunitinib	Cytochrome P450 3A4	enzyme
Sunitinib	Cytochrome P450 3A5	enzyme
Sunitinib	Cytochrome P450 3A7	enzyme
Sunitinib	ATP-binding cassette sub-family C member 4	transporter
Sunitinib	ATP-dependent translocase ABCB1	transporter
Sunitinib	ATP-binding cassette sub-family C member 2	transporter
Sunitinib	Broad substrate specificity ATP-binding cassette transporter ABCG2	transporter
Sunitinib	Hepatocyte growth factor receptor	target
Posaconazole	Cytochrome P450 3A4	enzyme
Posaconazole	ATP-dependent translocase ABCB1	transporter
Posaconazole	Lanosterol 14-alpha demethylase	target
Alosetron	5-hydroxytryptamine receptor 3A	target
Alosetron	Cytochrome P450 1A2	enzyme
Alosetron	Cytochrome P450 2C9	enzyme
Alosetron	Cytochrome P450 3A4	enzyme
Alosetron	Cytochrome P450 2E1	enzyme
Tiotropium	Muscarinic acetylcholine receptor M3	target
Tiotropium	Cytochrome P450 2D6	enzyme
Tiotropium	Cytochrome P450 3A4	enzyme
Tiotropium	Muscarinic acetylcholine receptor M1	target
Tiotropium	Muscarinic acetylcholine receptor M2	target
Tiotropium	Organic cation/carnitine transporter 2	transporter
Tiotropium	Solute carrier family 22 member 4	transporter
Tiotropium	Muscarinic acetylcholine receptor M4	target
Tiotropium	Muscarinic acetylcholine receptor M5	target
Solifenacin	Muscarinic acetylcholine receptor M3	target
Solifenacin	Muscarinic acetylcholine receptor M1	target
Solifenacin	Cytochrome P450 3A4	enzyme
Solifenacin	Muscarinic acetylcholine receptor M2	target
Solifenacin	Muscarinic acetylcholine receptor M4	target
Solifenacin	Muscarinic acetylcholine receptor M5	target
Solifenacin	alpha1-acid glycoprotein	carrier
Solifenacin	Cytochrome P450 1A1	enzyme
Solifenacin	Cytochrome P450 2D6	enzyme
Palonosetron	5-hydroxytryptamine receptor 3A	target
Palonosetron	Cytochrome P450 2D6	enzyme
Palonosetron	Cytochrome P450 3A4	enzyme
Palonosetron	Cytochrome P450 1A2	enzyme
Valdecoxib	Prostaglandin G/H synthase 2	target
Valdecoxib	Cytochrome P450 2C9	enzyme
Valdecoxib	Cytochrome P450 3A4	enzyme
Valdecoxib	UDP-glucuronosyltransferase 1A9	enzyme
Valdecoxib	Carbonic anhydrase 2	target
Valdecoxib	Carbonic anhydrase 3	target
Sertindole	5-hydroxytryptamine receptor 2A	target
Sertindole	5-hydroxytryptamine receptor 2C	target
Sertindole	D(2) dopamine receptor	target
Sertindole	Alpha-1A adrenergic receptor	target
Sertindole	Alpha-1B adrenergic receptor	target
Sertindole	Alpha-1D adrenergic receptor	target
Sertindole	Potassium voltage-gated channel subfamily H member 2	target
Sertindole	5-hydroxytryptamine receptor 6	target
Sertindole	Cytochrome P450 2D6	enzyme
Sertindole	Cytochrome P450 3A4	enzyme
Tesmilifene	ATP-dependent translocase ABCB1	target
Tesmilifene	Histamine H1 receptor	target
Tesmilifene	Cytochrome P450 3A4	enzyme
Tesmilifene	Cytochrome P450 2D6	enzyme
Tesmilifene	Cytochrome P450 1A1	enzyme
Etoricoxib	Prostaglandin G/H synthase 2	target
Etoricoxib	Cytochrome P450 3A4	enzyme
Etoricoxib	Cytochrome P450 2C9	enzyme
Etoricoxib	Cytochrome P450 2D6	enzyme
Etoricoxib	Cytochrome P450 1A2	enzyme
Etoricoxib	Cytochrome P450 2C19	enzyme
Etoricoxib	Cytochrome P450 2E1	enzyme
Rimonabant	Cannabinoid receptor 1	target
Rimonabant	Cytochrome P450 3A4	enzyme
Rimonabant	G-protein coupled receptor 55	target
Vicriviroc	C-C chemokine receptor type 5	target
Vicriviroc	Cytochrome P450 3A4	enzyme
Vicriviroc	Cytochrome P450 3A5	enzyme
Vicriviroc	Cytochrome P450 2C9	enzyme
Laquinimod	Cytochrome P450 3A4	enzyme
Laquinimod	C-X-C motif chemokine 2	target
Laquinimod	Nuclear factor NF-kappa-B p105 subunit	target
Laquinimod	Nuclear factor NF-kappa-B p100 subunit	target
Laquinimod	Transcription factor p65	target
Laquinimod	Proto-oncogene c-Rel	target
Fluvastatin	3-hydroxy-3-methylglutaryl-coenzyme A reductase	target
Fluvastatin	Cytochrome P450 2C9	enzyme
Fluvastatin	Cytochrome P450 3A4	enzyme
Fluvastatin	Cytochrome P450 2C8	enzyme
Fluvastatin	Cytochrome P450 2D6	enzyme
Fluvastatin	Cytochrome P450 2C19	enzyme
Fluvastatin	Cytochrome P450 1A1	enzyme
Fluvastatin	Solute carrier organic anion transporter family member 1B1	transporter
Fluvastatin	Solute carrier organic anion transporter family member 1B3	transporter
Fluvastatin	Solute carrier organic anion transporter family member 2B1	transporter
Fluvastatin	Solute carrier family 15 member 1	transporter
Fluvastatin	Cytochrome P450 3A5	enzyme
Fluvastatin	UDP-glucuronosyltransferase 1A1	enzyme
Fluvastatin	UDP-glucuronosyltransferase 1A3	enzyme
Fluvastatin	UDP-glucuronosyltransferase 2B7	enzyme
Fluvastatin	ATP-binding cassette sub-family C member 2	transporter
Fluvastatin	Cytochrome P450 2B6	enzyme
Fluvastatin	Histone deacetylase 2	target
Rotigotine	D(3) dopamine receptor	target
Rotigotine	D(1B) dopamine receptor	target
Rotigotine	D(4) dopamine receptor	target
Rotigotine	D(2) dopamine receptor	target
Rotigotine	5-hydroxytryptamine receptor 1A	target
Rotigotine	D(1A) dopamine receptor	target
Rotigotine	Cytochrome P450 2D6	enzyme
Rotigotine	Cytochrome P450 3A4	enzyme
Rotigotine	Alpha-2B adrenergic receptor	target
Rotigotine	Cytochrome P450 2C19	enzyme
Cerivastatin	3-hydroxy-3-methylglutaryl-coenzyme A reductase	target
Cerivastatin	Cytochrome P450 2C8	enzyme
Cerivastatin	Cytochrome P450 3A4	enzyme
Cerivastatin	Cytochrome P450 2D6	enzyme
Cerivastatin	Cytochrome P450 2C9	enzyme
Cerivastatin	Cytochrome P450 3A5	enzyme
Cerivastatin	Cytochrome P450 3A7	enzyme
Cerivastatin	ATP-dependent translocase ABCB1	transporter
Cerivastatin	ATP-binding cassette sub-family C member 2	transporter
Cerivastatin	Broad substrate specificity ATP-binding cassette transporter ABCG2	transporter
Cerivastatin	Solute carrier organic anion transporter family member 1B1	transporter
Cerivastatin	Cytochrome P450 2B6	enzyme
Cerivastatin	UDP-glucuronosyltransferase 1A1	enzyme
Cerivastatin	Bile salt export pump	transporter
Risperidone	Cytochrome P450 2D6	enzyme
Risperidone	Cytochrome P450 3A4	enzyme
Risperidone	ATP-dependent translocase ABCB1	transporter
Risperidone	Albumin	carrier
Risperidone	Alpha-1-acid glycoprotein 1	carrier